Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
04/2002
04/30/2002US6380398 Compounds such as (s,s)1-(2-amino-3,3-dimethyl-butyryl)-2,5-dihydro-1h-pyrrole-2 -carbonitrile administered as antidiabetic agents; dipeptidyl peptidase-iv (dpp-iv)
04/30/2002US6380395 Anticancer agents
04/30/2002US6380394 Anticancer agents
04/30/2002US6380258 Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds
04/30/2002US6380246 For combating pests and weeds
04/30/2002US6380241 For therapy of coronary angina, cerebral vasospasm, acute and chronic renal failure, gastric ulceration, cyclosporin-induced nephrotoxicity, endotoxin-induced toxicity, asthma, lpl-related lipoprotein disorders, proliferative diseases
04/30/2002US6380230 For therapy of dyskinesia, obesity, irritable bowel syndrome, diseases whose treatment requires stimulation of the cholecystokinin cck-a receptors
04/30/2002US6380229 Useful for therapy and prophylaxis of hyperlipidemia and related complications
04/30/2002US6380225 Microbicidal benzotriazoles
04/30/2002US6380221 Ortho-anthranilamide derivatives as anti-coagulants
04/30/2002US6380218 For therapy of respiratory, allergic, and inflammatory disorders comprising asthma, chronic obstructive pulmonary disease, acute respiratory disease syndrome, pulmonary hypersensitivity, and allergic rhinitis in a mammal
04/30/2002US6380214 Thiophene-3-carboxylic acid amide derivatives
04/30/2002US6380213 Compounds useful as neuro-protective agents
04/30/2002US6380205 2-cyclohexyl quinazoline NMDA/NR2B antagonists
04/30/2002US6380204 Alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor antagonist activity
04/30/2002US6380189 2-amino benzoxazinones for the treatment of viral infections
04/30/2002US6380186 Psychotherapeutic agents
04/30/2002US6380180 Potassium channel blocking agents
04/30/2002US6379823 Electroluminescence device, cyclic azine compound and production process of cyclic azine dye
04/25/2002WO2002032900A2 Aryl or heteroaryl fused imidazole compounds as anti-inflammatory and analgesic agents
04/25/2002WO2002032897A1 Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists
04/25/2002WO2002032894A1 Substituted imidazoles useful in the treatment of inflammatory diseases
04/25/2002WO2002032893A2 Piperidine compounds as anti-allergic
04/25/2002WO2002032891A1 Flavan compounds, their preparation and their use in therapy
04/25/2002WO2002032889A1 Aromatic and heterocyclic thiazolyl thiourea compounds and use
04/25/2002WO2002032886A1 A process for the preparation of bis-benzazolyl compounds
04/25/2002WO2002032872A1 Nitrogenous aromatic ring compounds
04/25/2002WO2002032844A2 Epothilone synthesis components iii and iv: asymmetrically substituted acyloins and acyloin derivatives, method for the production thereof and method for the production of epithilone b, d and epothilone derivatives
04/25/2002WO2002032422A2 Ep4 receptor inhibitors to treat rheumatoid arthritis
04/25/2002WO2002010137A3 Indazole derivatives as JNK inhibitors
04/25/2002WO2001081341A3 9-oxa-epothilon derivatives, method for the production and use thereof in pharmaceutical preparations
04/25/2002WO2001058891A3 Piperazine and piperidine derivatives for treatment or prevention of neuronal damage
04/25/2002WO2001002369A3 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use
04/25/2002US20020049330 Such as 5-(N,N-dibenzyl)aminocarbonyl-2-pyridone; enzyme inhibitors; for treatment of Alzheimer's disease
04/25/2002US20020049329 Novel human NK3 receptor-selective antagonist compounds, method for obtaining them and pharmaceutical compositions containing them
04/25/2002US20020049316 Protease inhibitors
04/25/2002US20020049246 Benzimidazole compounds for treatment of asthma, vasospasm, memory loss, migraine and others diseases associated with potassium channels
04/25/2002US20020049240 Novel compounds
04/25/2002US20020049239 Novel indole and benzothiazole derivatives
04/25/2002US20020049231 S(-)-3-aminothalidomide; treating wide variety of diseases including diabetic retinopathy
04/25/2002US20020049223 Quinoline and naphthyridine carboxylic acid antibacterials
04/25/2002US20020049214 Aralkyl and aralkylidene heterocyclic lactams and imides as selective agonists and antagonists of serotonin 1 (5-HT1) recepor, used in treating hypertension and all forms of depression
04/25/2002US20020049210 Heteroaryl amines as novel acetylcholinesterase inhibitors
04/25/2002US20020049204 1,4-dihydro-benzo(d)oxazin-2-one derivatives useful for treating hormone-dependent neoplastic disease is selected from uterine myometrial fibroids, endometriosis, benign prostatic hypertrophy, carcinomas, and adenocarcinoma
04/25/2002US20020049201 Sulfonamide inhibitors of aspartyl protease
04/25/2002US20020049195 Urea compounds that are muscarinic receptor antagonists and agonists, administering to the mammal the urea compound to treat urinary incontinence, chronic pulmonary obstructive disease, asthma, hyper salivation, blurred vision etc.
04/25/2002US20020049194 A benzoazepin or benzodiazepin derivatives, shows excellent anti-vasopressin activity, vasopressin agonistic activity and oxytocin antagonistic activity, and are useful as antagonist
04/25/2002US20020049193 Inhibitors of the enzyme activity associated with immunophilin proteins, particularly peptidyl-prolyl isomerase, or rotamase, enzyme activity.
04/25/2002US20020049142 Fungicidal, insecticidal, acaricidal, molluscicidal or nematicidal composition
04/25/2002US20020048271 Methods and composition for restoring conformational stability of a protein of the p53 family
04/25/2002CA2426487A1 Ep4 receptor inhibitors to treat rheumatoid arthritis
04/25/2002CA2426337A1 Substituted imidazoles useful in the treatment of inflammatory diseases
04/25/2002CA2426148A1 Aromatic and heterocyclic thiazolyl thiourea compounds and use
04/25/2002CA2423792A1 Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists
04/24/2002EP1199307A1 Pharmaceutically active benzoquinazoline compounds
04/24/2002EP1199306A1 Biarylurea derivatives
04/24/2002EP0714299B1 Benzoxazinone and benzopyrimidinone piperidinyl tocolytic oxytocin receptor antagonists
04/24/2002CN1346355A Novel inhibitors of farnesyl-protein transferase
04/24/2002CN1346354A Substituted benzoylpyrazoles as herbicides
04/24/2002CN1346351A 1,2-benzothiazepines for the treatment of hyperlipidemic diseases
04/24/2002CN1346350A Compound which inhibiti leukocyte adhesion mediated by VLA-4
04/24/2002CN1346282A Use of a cyclooxygenase-2 inhibitor and one or more antineoplastic agents as combination therapy method in treating neoplasia
04/24/2002CN1346271A Quinazoline derivatives as angiogenesis inhibitors
04/24/2002CN1083446C Process for preparing 2-chlorothiazole compounds
04/24/2002CN1083431C Novel heterocyclic compounds
04/23/2002US6376675 Pyridyl-1,2,5-thiadiazole derivatives
04/23/2002US6376665 Antiarthritic agents, antiinflammatory agents
04/23/2002US6376507 NK-1 receptor antagonists for the treatment of neuronal injury and stroke
04/23/2002US6376503 Alpha 1a adrenergic receptor antagonists
04/23/2002US6376491 Benzofuran derivatives for treatment or prevention of mycosis in mammals
04/23/2002US6376490 Strong n-methyl-d-asparate receptor antagonists; useful in treating strokes, ischemia, and central nervous system injuries
04/23/2002US6376487 Oxadiazine derivatives
04/23/2002US6376484 For prevention and/or treatment of various kinds of inflammatory disease
04/23/2002CA2246727C Novel substituted n-methyl-n-(4-(piperidin-1-yl)-2-(aryl)butyl)benzamides useful for the treatment of allergic diseases
04/18/2002WO2002030927A1 Novel aminophenyl piperazine or aminophenyl piperidine derivatives inhibiting prenyl transferase proteins and methods for preparing same
04/18/2002WO2002030926A1 Quinazoline derivatives
04/18/2002WO2002030923A1 Novel aminotriazolone compounds, method for preparing same and pharmaceutical compositions containing same
04/18/2002WO2002030895A1 SUBSTITUTED INDOLES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH INDOLES AND THEIR USE AS PPAR-η BINDING AGENTS
04/18/2002WO2002030890A1 Nitrogenous five-membered ring compounds
04/18/2002WO2002030886A2 Heterocyclic angiogenesis inhibitors
04/18/2002WO2002030867A2 Drugs for diabetes
04/18/2002WO2002030358A2 Modulation of ccr4 function
04/18/2002WO2002030357A2 Compounds and methods for modulating ccr4 function
04/18/2002WO2002030356A2 Synthesis of epothilones and relates analogs
04/18/2002WO2002012210A9 Biphenyl derivatives and their use as ppar-gamma receptor activators
04/18/2002WO2002008217A3 COUMARIN DERIVATIVES USEFUL AS TNFα INHIBITORS
04/18/2002WO2001091732A3 Medicament for combating respiratory depression
04/18/2002WO2001087830A3 Substituted thioacetamides
04/18/2002WO2001058893A3 Indol-3-yl derivatives and their use as integrin inhibitors
04/18/2002WO2001026656A3 5-membered heterocycle derivatives and use thereof as monoamine oxidase inhibitors
04/18/2002US20020045654 Sulfonylbenzene compounds as anti-inflammatory/analgesic agents
04/18/2002US20020045652 Prophylactic or therapeutic drug for renal diseases
04/18/2002US20020045647 N-linked urea or carbamate of heterocyclic thioester hair growth compositons and uses
04/18/2002US20020045642 Antiinflammatory, -arthritic and -emetic agents; central nervous system disorders; Parkinson's disease; antidepressants; psychological disorders; anxiolytic agents; antagonists of substance P receptors
04/18/2002US20020045641 Multiple heteroatom containing heterocyclic ring compounds substituted with carboxylic acids and isosteres thereof
04/18/2002US20020045629 Sleep, eating and brain disorders, wakefulness promoters; Parkinson's disease, antiischemic agents, stroke, chronic fatigue syndrome; antidepressants; schizophrenia, nervous system disorders; multiple sclerosis, cognition activators
04/18/2002US20020045620 Readily metabolized by the metabolic drug detoxification systems; metabolized by serum or intracellular hydrolases and esterases; shorthalf-life; noninsulin-dependent diabetes mellitus (NIDDM) (Type II); side effect reduction
04/18/2002US20020045618 Heteroaryl diazacycloalkanes, their preparation and use
04/18/2002US20020045615 Benzothiazole derivatives with activity as adenosine receptor ligands
04/18/2002US20020045609 Epothilone derivatives and methods for making and using the same