Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
09/2006
09/13/2006EP1218358B1 Therapeutic quinazoline compounds
09/13/2006EP1087951B9 Carbon substituted aminothiazole inhibitors of cyclin dependent kinases
09/13/2006EP0917462B1 Cell adhesion inhibitors
09/13/2006CN1832947A Thiazole derivatives as npy antagonists
09/13/2006CN1832946A Process for producing imide compound
09/13/2006CN1832941A Halogenated quinazolinyl nitrofurans as antibacterial agents
09/13/2006CN1832934A Benzoxazepine-based compound
09/13/2006CN1832932A Biaryl heterocyclic compounds and methods of making and using the same
09/13/2006CN1832930A Amide derivative
09/13/2006CN1832927A Novel gamma-secretase inhibitors
09/13/2006CN1832925A New p2x7 receptor avtagonists and their use
09/13/2006CN1832921A Tetrahydrocarbazole derivatives and their pharmaceutical use
09/13/2006CN1832740A Indol-5 sulfonamide derivatives, their preparation and their use 5-ht-6 as modulators
09/13/2006CN1830977A Novel process for preparation of 2-aminothiazolecarboxamide derivatives
09/13/2006CN1274686C Suitable industrialized method of preparing Lamivudine
09/13/2006CN1274675C Novel cyclobutene diketone compound and its producing process, and pharmaceutical composition containing the same compound
09/13/2006CN1274305C Pharmaceutical composition with combined active agents and methods for using the same
09/12/2006US7105701 Multibinding compounds for agonists for phenolic derivatives for adrenergic receptors with carriers
09/12/2006US7105682 Substituted amine derivatives and methods of use
09/12/2006US7105671 2-Substituted phenyl,3-polar ring,N-heroaromatic propion-amides, e.g., 1-(2-(3,4-Dichlorophenyl)-3-(tetrahydro-furan-2-yl)-propionyl)-3- methylurea; antidiabetic agents; increase the flux of glucose metabolism in beta-cells and hepatocytes
09/12/2006US7105670 Intermediates useful in the preparation of diaminothiazoles
09/12/2006US7105667 Fused heterocyclic compounds and use thereof
09/12/2006US7105564 7-(3-{[5-(Pyrrole-1-sulfonyl)-thiophene-2-carbonyl]-amino}-bicyclo[2.2.1]hept-2-yl)-hept-5-enoic acid; thromboxane A2 receptor and a prostaglandin D2 receptor; for all of eosinophilic infiltration, advance of respiratory anaphylaxis and respiratory contraction
09/12/2006US7105554 Benzylidene thiazolidinediones and their use as antimycotic agents
09/12/2006US7105553 Thiazolyl amide derivatives
09/12/2006US7105550 2,4-disubstituted thiazolyl derivatives
09/12/2006US7105544 N-{3-[1-(3-{[BIS(4-FLUOROPHENYL)ACETYL]AMINO}PROPYL)-4-PIPERIDINYL]PHENYL}-2-METHYLPROPANAMIDE; antagonists for melanin concentrating hormone-1 (MCH1) receptors; treating depression, anxiety, obesity
09/12/2006US7105537 For enhancing bone formation; for therapy of diseases or disorders associated with abnormal bone or mineral homeostasis
09/12/2006US7105529 A novel compound for treating alopecia induced by cancer chemotherapy or radiotherapy
09/12/2006US7105519 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
09/12/2006US7105517 N-{4-[2-(1-Dimethylamino-ethylimino)-4-phenyl-thiazol-5-yl]-pyrimidin-2-yl}-N-phenyl-amine; fungicides against infestation by phytopathogenic organisms, nematodes, insects, fungi, bacteria, viruses
09/12/2006US7105515 Such as N-[3-(2-diethylaminoethyl)-1H-indol-5-yl]-5-chloro-3-methylbenzo[b]thiophene-2-sulphonamide for treating anxiety, depression, cognitive memory disorders and senile dementia, psychosis, infant hyperkinesia (ADHD, attention deficit/hyperactivity disorder)
09/12/2006US7105514 2-methyl-3-(4,5,7-trifluorobenzothiazol-2-yl)methyl-indole-N-acetic; acidinhibit aldose reductase; treating diabetes mellitus, including, diabetic cataracts, retinopathy, nephropathy, and neuropathy
09/12/2006US7105513 Cardiovascular disorders; strokes; hypotensive agents
09/12/2006US7105512 Having anti- inflammatory effect, which is less irritant, which has high safety and storage stability
09/12/2006US7105509 Benzodiazepine derivatives as APP modulators
09/12/2006US7105508 Integrin receptors antagonists
09/12/2006US7105507 Cyclohexane derivatives and their use as therapeutic agents
09/12/2006US7105505 Benzimidazole derivatives useful as histamine H3 antagonists
09/12/2006US7105503 Pyrazole compounds
09/12/2006CA2235986C Inhibitors of protein isoprenyl transferases
09/12/2006CA2167004C Agent for treating mental disorders associated with cerebrovascular disorders
09/12/2006CA2140929C Hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
09/11/2006CA2500667A1 Preparation of acid addition salts of ziprasidone and intermediates thereof by solid phase-gas phase reactions
09/08/2006WO2006094235A1 Fused heterocyclic compounds and their use as sirtuin modulators
09/08/2006WO2006093801A1 Thiadiazine derivatives useful as anti-infective agents
09/08/2006WO2006093339A1 Use of cinnamoyl compound
09/08/2006WO2006093247A1 NOVEL AMINOPYRIDINE COMPOUND WITH Syk INHIBITORY ACTIVITY
09/08/2006WO2006092608A1 Tricyclic derivatives of azetidine and pyrrole with antibacterial activity
09/08/2006WO2006092599A2 Pyrrole derivatives as dna gyrase and topoisomerase inhibitors
09/08/2006WO2006092574A1 Indolylamino quinazoline derivatives as antitumor agents
09/08/2006WO2006092573A1 Indazolylamino qionazoline derivatives as antitumor agents
09/08/2006WO2006092395A1 9-amino-acridine derivatives and their use for eliminating misfolded proteins
09/08/2006WO2005086700A3 Hiv integrase inhibitors
09/08/2006WO2005035551A3 Inhibitors of proteins that bind phosphorylated molecules
09/08/2006CA2600287A1 Use of cinnamoyl compound
09/08/2006CA2599992A1 Acridine and quinoline dervatives as sirtuin modulators
09/08/2006CA2599987A1 Fused heterocyclic compounds and their use as sirtuin modulators
09/08/2006CA2599544A1 Novel aminopyridine compound with syk inhibitory activity
09/07/2006US20060199964 preparation of 6-haloalkyl-3-nicotinic acid esters and also to novel enamine intermediates
09/07/2006US20060199960 e.g. 6-Methyl-3-(pyridin-3-ylamino)-pyridine-2-carboxylic acid (4-methyl-thiazol-2-yl)-amide; metabotropic glutamate receptor antagonists (mGluR); central nervous system disorders, antidepressant, anxiolytc agent; psychosis, epilepsy, schizophrenia, Alzheimer's disease, cognitive disorders
09/07/2006US20060199958 Process and intermediates for the preparation of pyrrolidine carboxylic acids
09/07/2006US20060199949 Cyanine dyes as labeling reagents for detection of biological and other materials by luminescence methods
09/07/2006US20060199851 Novel compounds that are useful for improving pharmacokinetics
09/07/2006US20060199844 Inhibitors of raf-kinase; Hyperproliferative disorders
09/07/2006US20060199830 N-(4-(4-methylthiazol-5-yl) pyrimidin-2-yl)-N-phenylamines as antiproliferative compounds
09/07/2006US20060199828 Pyrazine-2-carboxyamide derivatives
09/07/2006US20060199827 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
09/07/2006US20060199826 Cyclopropane compounds and pharmaceutical use thereof
09/07/2006US20060199825 4-Aminating a 4-chloro-2-hydroxy-3-nitrodihydroquinoline with a N-(hetero)cyclylpiperazine, and alkylating the remaining amine group in the quinoline ring to produce a 4-(4-(hetero)cyclylpiperazinyl)-3-nitro-1-alkyldihydroquinolinone
09/07/2006US20060199824 Treating or preventing pain, UI, an ulcer, IBD, IBS, an addictive disorder, Parkinson's disease, parkinsonism, anxiety, epilepsy, stroke, a seizure, a pruritic condition, psychosis, a cognitive disorder, a memory deficit, restricted brain function, Huntington's chorea, amyotrophic lateral sclerosis
09/07/2006US20060199822 Bis-sulfonamide hydroxyethylamino retroviral protease inhibitors
09/07/2006US20060199818 Inhibiting the activity of a 5-hydroxytryptamine 2A by administering a N-heterocyclyl (preferably 1,3-dioxan-5-yl)-4-[(N-substituted)(hetero)arylamino]piperidine in which the N-substituant is arylalkanoyl, arylthioalkanoyl, arylalkylaminocarbonyl or arylalkylaminothiocarbonyl group
09/07/2006US20060199813 Neurodegenerative diseases, psychological disorders; e.g. 1-[3-(4-Butyl-piperidin-1-yl)-propyl]-1,2,3,4-tetrahydroquinoline
09/07/2006US20060199810 Neurodegenerative diseases, psychological disorders; e.g. 1-[3-(4-Butyl-piperidin-1-yl)-propyl]-1,2,3,4-tetrahydro-quinoline
09/07/2006US20060199804 ATP-competitive inhibitors of serine/threonine kinase (mTOR); antifungal agents, anticancer agents, autoimmune diseases, inflammation, bone loss, bowel disorders, hepatic fibrosis/necrosis, rheumatoid arthritis, psoriasis
09/07/2006US20060199799 Benzimidazolidinone derivatives as muscarinic agents
09/07/2006US20060199242 Stain compounds containing fluorophore and reducible quenching unit; for detection of bacterial cells, monitoring electron transport chain function of bacterial cells, monitoring oxidation state of non-biological systems, and assaying the effectiveness of antibacterial or antimicrobial agents; kits
09/07/2006DE102005009909A1 Verbindungen geeignet zur Beseitigung fehlgefalteter Proteine Compounds suitable for the removal of misfolded proteins
09/06/2006EP1698696A1 Target protein of antidiabetic agent and novel antidiabetic agent insuful corresponding thereto
09/06/2006EP1698628A1 Hydroxypyrimidinone derivative having hiv integrase inhibitory activity
09/06/2006EP1698627A1 Pyrazole compounds useful as protein kinase inhibitors
09/06/2006EP1698626A1 Amidopyrazole derivative
09/06/2006EP1698624A1 Phenylpropanoic acid derivatives
09/06/2006EP1698375A1 Azetidine ring compounds and drugs comprising the same
09/06/2006EP1697355A2 Amidino compounds as cysteine protease inhibitors
09/06/2006EP1697354A1 Isothiazole dioxides as cxc- and cc- chemokine receptor ligands
09/06/2006EP1697352A2 4-azole substituted imidazole compositions useful as inhibitors or c-met receptor tyrosine kinase
09/06/2006EP1697351A1 2,6-bisheteroaryl-4-aminopyrimidines as adenosine receptor antagonists
09/06/2006EP1697348A1 Hiv protease inhibiting compounds
09/06/2006EP1697344A2 Hiv protease inhibiting compounds
09/06/2006EP1697334A1 Heterocyclic substituted indane derivatives and related compounds for the treatment of schizophrenia
09/06/2006EP1697333A1 (3,4-disubstituted)propanoic carboxylates as s1p (edg) receptor agonists
09/06/2006EP1697327A1 Insecticidal spiroindane derivatives
09/06/2006EP1697320A1 A synthetic methodology for the reductive alkylation at the c-3 position of indoles
09/06/2006EP1697312A2 Hydroxamic acid esters and pharmaceutical use thereof
09/06/2006EP1696924A1 Acidic quinoline derivatives and their use for the prevention and/or treatment of hyperglycaemia-related pathologies
09/06/2006EP1696919A2 3-cycloalkylaminopyrrolidine derivatives as modulators of chemokine receptors
09/06/2006EP1696915A1 Benzenesulfonylamino-pyridin-2-yl derivatives and related compounds as inhibitors of 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-hsd-1) for the treatment of diabetes and obesity
09/06/2006EP1458697B1 Biphenylmethyl-thiazolidinediones and analogues and their use as ppar-gamma activators