Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
02/2010
02/18/2010US20100041889 Processes and intermediates for preparing a macrocyclic protease inhibitor of hcv
02/18/2010US20100041711 Urea Glucokinase Activators
02/18/2010US20100041708 N-phenylarylsulfonamide compound, pharmaceutical composition comprising the compound as active ingredient, synthetic intermediate for the compound and process for it's preparation
02/18/2010US20100041707 Inhibitors of ion channels
02/18/2010US20100041700 Substituted 1-(Azolin-2-yl)-Amino-1,2-Heterocyclyl-Ethane Compounds For Combating Pests
02/18/2010US20100041660 Novel 2-pyridinecarboxamide derivatives
02/18/2010US20100041656 Novel amide derivatives and medicinal use thereof
02/18/2010US20100041649 viricides used for for treating a human papillomavirus (HPV) viral infections, for inhibiting HPV DNA replication or for preventing prenatal transmission of HPV from mother to baby by administering to the mother prior to giving birth
02/18/2010US20100041645 Rho kinase inhibitors
02/18/2010US20100041555 3-Phenoxy-4-pyridazinol derivatives and herbicidal composition containing the same
02/18/2010CA2733966A1 Benzoxazoles, benzthiazoles and related analogs as sirtuin modulators
02/18/2010CA2733397A1 Azetidine polysubstituted compounds, preparation thereof, and therapeutic application thereof
02/18/2010CA2731102A1 Imine derivatives as cannabinoid receptor ligands
02/17/2010EP2153832A2 Heterocyclic aspartyl protease inhibitors
02/17/2010EP2152717A1 Processes for making epothilone compounds and analogs
02/17/2010EP2152702A1 Amino-thiazolyl- pyrimidine derivatives and their use for the treatment of cancer
02/17/2010EP2152701A1 Phenyl amino pyrimidine compounds and uses thereof
02/17/2010EP2152700A1 Csf-1r inhibitors, compositions, and methods of use
02/17/2010EP2152696A1 Aminopyrimidines useful as kinase inhibitors
02/17/2010EP2152694A2 Thiazoles and pyrazoles useful as kinase inhibitors
02/17/2010EP2152690A1 Pyridyl piperidine orexin receptor antagonists
02/17/2010EP2152688A1 Compounds and compositions as c-kit and pdgfr kinase inhibitors
02/17/2010EP2152674A1 Benzimidazolone chymase inhibitors
02/17/2010EP2152664A1 Dipeptide analogs as coagulation factor inhibitors
02/17/2010EP1902026B1 Tetrahydrocarbazole derivatives useful as androgen receptor modulators (sarm)
02/17/2010EP1773827B1 Benzothiazole derivatives
02/17/2010EP1549318B1 Crystal structure of aurora-2 protein and binding pockets thereof
02/17/2010EP1377263B1 Novel dyeing composition for dyeing keratinous fibres comprising a particular dicationic diazo dye
02/17/2010CN101652363A Thiazolyl compounds useful as kinase inhibitors
02/17/2010CN101652362A Method for producing epothilone derivatives by means of selective catalytic epoxidation
02/17/2010CN101648949A inhibitors of phosphatidylinositol 3-kinase
02/17/2010CN101648944A 病毒聚合酶抑制剂 Viral polymerase inhibitors
02/17/2010CN100590123C 2,4-disubstituted thiazolines derivatives, preparing method and application thereof
02/16/2010US7662972 Insecticidal and acaricidal activity for many agricultural insect pests, spider mites; endo- or ecto-parasiticide for mammals or birds; veterinary medicine; environmentally friendly
02/16/2010US7662971 enzyme inhibitor for treating sleep disorders
02/16/2010US7662958 e.g. N-[3-{1-[(cyclobutyl)amino]-4-hydroxy-2-oxo-1,2-dihydro-quinolin -3-yl}-1,1-dioxo-1,4-dihydro-1 lambda 6-thieno[2,3-e][1,2,4]thiadiazin-7-yl)methyl]methane-sulfonamide; viricides for infections caused by an RNA-containing virus; hepatitis C virus (HCV) polymerase inhibitor; liver cirrhosis
02/16/2010US7662849 N-cyanomethyl-2R-[(benzenesulfonyliminomethyl)amino]-3-(2-difluoromethoxyphenylmethanesulfonyl)-propionamide; treating autoimmune disorders
02/16/2010US7662847 Myelodysplastic syndrome, Parkinson*s disease, multiple sclerosis, AIDS, chronic obstructive pulmonary disease, acquired respiratory distress; analgesics, angiogenesis inhibitors; anticarcinogenic and antitumor agents; phopshodiesterase, tumor necrosis factor and matrix metalloproteinase inhibitors
02/16/2010US7662842 (4R)-2-(4-methoxyphenyl)-N-octadecylthiazolidine-4-carboxamide; antiacarcinogenic agent for destroying a melanoma cell
02/16/2010US7662839 EP receptor (for which the endogenous ligand is prostaglandin E2, PGE2); dysmenorrhoea, preterm labour, glaucoma, immune disorders, inflammatory disorders; e.g. {4-[(5-Phenyl-furan-2-carbonyl)-amino]-phenyl}-acetic acid
02/16/2010US7662834 Methods of 1H-indol-3-yl-2-oxoacetamide compounds
02/16/2010US7662818 e.g. 4-[5-(piperidine-1-carbonyl)-furan-2-ylmethyl]-2H-phthalazin-1-one; enzyme poly(ADP-ribose)polymerase (synthase)-1 or poly ADP-ribosyltransferase (PARP-1) inhibitor; anticarcinogenic agent with BRCA2 deficient phenotype; septic shock; ischemic injury; hemorrhagic shock; and multiple sclerosis
02/16/2010US7662811 1,2,3,4-tetrahydropyrazin-2-yl acetamides and methods of use
02/16/2010CA2628224C Vinyl-pyrrolidinone cephalosporins with basic substituents
02/16/2010CA2571627C Substituted aryl-amine derivatives and methods of use
02/16/2010CA2479274C Thiazolidinedione derivatives and pharmaceutical composition comprising the same
02/16/2010CA2450922C Piperidines for use as orexin receptor antagonists
02/16/2010CA2385938C Cyclic amine compounds as ccr5 antagonists
02/16/2010CA2385081C Carboxylic acid compound and a medicament comprising it
02/16/2010CA2343883C An improved process for the preparation of thiazolidine-2,4-dione derivatives
02/11/2010WO2010017350A1 Aminopyridine kinase inhibitors
02/11/2010WO2010017079A1 Oxazole derivatives useful as inhibitors of faah
02/11/2010WO2010016612A1 Dye for dye-sensitized solar cell, semiconductor electrode, and dye-sensitized solar cell
02/11/2010WO2010015792A1 Nitrogen containing heterocyclic compounds useful as bifunctional modulators of m3 receptors and beta-2 receptors
02/11/2010WO2010015681A1 Fungicidal n-(2-pyridylpropyl)carboxamide derivatives and their oxa, aza and thia analogues
02/11/2010WO2010015652A2 Thiazole compounds as activators of soluble guanylate cyclase
02/11/2010WO2010015090A1 Functionalized pyrrolidines and use thereof as iap inhibitors
02/11/2010US20100036118 Fused Ring Heterocycle Kinase Modulators
02/11/2010US20100035929 Unnatural dispyrin analogues, preparation and uses thereof
02/11/2010US20100035899 5,7-DISUBSTITUTED[1.3]THIAZOLO[4,5-d]PYRIMIDIN-2(3H)-AMINE DERIVATIVES AND THEIR USE IN THERAPY
02/11/2010US20100035869 Targeted nitroxide agents
02/11/2010US20100035858 Novel Compositions and Methods for Binding and Inhibiting 5-HT4 Receptor
02/11/2010US20100034813 Substituted pyrazole and triazole compounds as ksp inhibitors
02/11/2010US20100032658 Novel organic electroluminescent compounds and organic electroluminescent device using the same
02/11/2010CA2732765A1 Aminopyridine kinase inhibitors
02/11/2010CA2732526A1 Oxazole derivatives useful as inhibitors of faah
02/10/2010EP2151438A1 Pharmaceutical containing ppar agonist
02/10/2010EP2151435A1 Pharmaceutical composition for treatment of alzheimer's disease
02/10/2010EP2150546A2 Pyrimidine derivatives as inhibitors of phosphatidylinositol-3-kinase
02/10/2010EP2150539A1 Pyridazinone derivatives
02/10/2010EP2150255A1 Quinoxaline derivatives as p13 kinase inhibitors
02/10/2010EP2150115A1 Cyclopropyl pyrrolidine orexin receptor antagonists
02/10/2010EP2086965B1 Aminopyridines and aminopyrimidines useful as inhibitors of protein kinases
02/10/2010EP1817287B1 Aromatic ether derivatives useful as thrombin inhibitors
02/10/2010EP1747196B1 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication
02/10/2010EP1411932B1 Substituted oxazolidinones for combinational therapy
02/09/2010US7659405 Protease inhibitor; viricides; purity; crystal structure; mixing tank
02/09/2010US7659404 Broad spectrum 2-(substituted-amino)-benzothiazole sulfonamide HIV protease inhibitors
02/09/2010US7659399 1-thia-2,4a-diaza-cyclopenta[b]napththalene-3,4-diones and related compounds as anti-infective agents
02/09/2010US7659394 Substituted morpholine compounds for the treatment of central nervous system disorders
02/09/2010US7659307 Heterocyclic carboxamides and their use as fungicides
02/09/2010US7659298 2-(3-Phenyl-5-chloro-1-methyl-1H-pyrazol-4-ylmethylsulphanyl)-N-quinolin-3-ylbenzamide; 2-(3-Phenyl-5-chloro-1-methyl-1H-pyrazol-4-ylmethoxy)-N-naphthalin-2-ylbenzamide; obesity, including obesity of the non-insuline-dependent diabetes patients, sleeping disorders, stroke, nausea and vomiting
02/09/2010US7659296 2-{1-[4-(3,3-dimethyl-2-oxo-butoxy)-3-methyl-phenyl]-1-ethyl-propyl}-benzooxazole-6-carboxylic acid; 1-[4-(3,3-Dimethyl-2-oxo-butoxy)-3-methyl-phenyl]-1-ethyl-propyl}-benzooxazole-6-carboxylic acid amide; stimulate bone formation, restore bone quality, acne, alopecia, Alzheimer's disease etc.
02/09/2010US7659280 2,4-pyrimidinediamine compounds for treating or preventing autoimmune diseases
02/09/2010US7659269 Substituted indolealkanoic acids
02/09/2010US7659266 N1-[(3S)-2-hydroxytetrahydrofuran-3-yl]-N2-[imino(10H-phenothiazin-2-yl)methyl]-L-leucinamide; (3S)-3-({N-[imino(10H-phenothiazin-2-yl)methyl]-L-leucyl}amino)tetrahydrofuran-2-yl acetate; hearing disorders, muscular dystrophy
02/09/2010US7659265 5-(4,4-dimethyl-2-thioxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)-1-methyl-1H-pyrrole-2-carbothioamide; menopause therapy; contraceptive; anticancer agents
02/09/2010CA2484954C 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as vla-4 inhibitors
02/09/2010CA2413061C Serine protease inhibitors
02/09/2010CA2291065C Raf kinase inhibitors
02/09/2010CA2274201C Di-or triaza-spiro[4,5]decane derivatives
02/04/2010WO2010014611A1 Cycloalkylidene and heterocycloalkylidene histone deacetylase inhibitor compounds
02/04/2010WO2010014240A2 Novel bioactive small molecules derived from sea sponges
02/04/2010WO2010013769A1 Crystal of thiazolidinedione compound, and process for production thereof
02/04/2010WO2010013768A1 Crystal of thiazolidinedione compound, and process for production thereof
02/04/2010WO2010013595A1 (5-membered)-(5-membered) or (5-membered)-(6-membered) fused ring cycloalkylamine derivative
02/04/2010WO2010013222A1 Pyrrole carboxylic acid derivatives as antibacterial agents
02/04/2010WO2010013161A1 Fluorinated heteroaryls
02/04/2010WO2010013078A2 Pyrrolidinyl-alkyl-amide derivatives their preparation and their therapeutic application as ccr3 receptor ligands
02/04/2010WO2010013037A1 1,2,4-oxadiazole substituted piperidine and piperazine derivatives as smo antagonists