Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
12/2010
12/08/2010CN101910164A Diamido thiazole derivatives as protein kinase inhibitors
12/08/2010CN101910163A Heterocyclic urea and thiourea derivatives and methods of use thereof
12/08/2010CN101910162A Cyclic pyridyl-N-(1,3,4)-thiadiazol-2-yl-benzene sulfonamides, processes for their preparation and their use as pharmaceuticals
12/08/2010CN101910158A Pyridine and pyrazine derivatives useful in the treatment of cell proliferative disorders
12/08/2010CN101910152A 4-pyrazolyl-N-arylpyrimidin-2-amines and 4-pyrazolyl-N-heteroarylpyrimidin-2-amines as janus kinase inhibitors
12/08/2010CN101910145A Heterocyclic antiviral compounds
12/08/2010CN101910143A Condensed aminodihydrothiazine derivative
12/08/2010CN101910142A Modulators for amyloid beta
12/08/2010CN101910133A Heterocycle phenyl amide T-type calcium channel antagonists
12/08/2010CN101910121A Bis-(sulfonylamino) derivatives in therapy 066
12/08/2010CN101906099A Method for biochemically synthesizing epothilone D-lactam derivatives
12/07/2010USRE41990 epothilone derivatives used for the treatment of cancer and cancers which have developed a multidrug-resistant phenotype; anticarcinogenic agents
12/07/2010US7847101 such as (4-Benzothiazol-2-yl-1H-pyrazol-3-yl)-[2-(1H-imidazol-4-yl)-ethyl]-amine, used in the treatment of disorders associated with hyperproliferation and tissue remodelling or repair, inflammation, cell migration and invasion, and renal diseases, or as protein kinase inhibitors
12/07/2010US7846962 3-(5-tert-Butyl-2-Hydroxy-phenyl)-3-phenyl-1,3-dihydro-indol-2-one and/or its derivatives, used for the treatment of cellular proliferative disorders, non-proliferative, degenerative disorders, viral infections, and/or disorders associated with viral infections
12/07/2010US7846952 epothilone derivatives in combination with carriers or diluents, used for plant protection in agriculture, forestry or horticulture; plant safening agents
12/07/2010US7846951 treating cystic fibrosis, emphysema, or chronic obstructive pulmonary disease, comprising administering to a patient azole-4-carboxamide derivatives such as N,N-dibenzyl-2-[(2,6-dichlorophenyl)methyl]-1,3-thiazole-4-carboxamide
12/07/2010US7846950 Histamine H3 receptor inhibitors, preparation and therapeutic uses
12/07/2010US7846945 2-[4-Chloro-3-(4-hydroxy-benzyl)-phenyl]-6-methoxy-tetrahydro-pyran-3,4,5-triol; 2-[4-Chloro-3-(4-ethoxy-benzyl)-phenyl]-3,4,5-trihydroxy-piperidine-1-carboxylic acid methyl ester; (2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6-methoxytetrahydro-2H-thiopyran-3,4,5-triol; antidibetic, antiobesity agents
12/07/2010US7846925 such as 5-(1,3-benzodioxol-5-ylmethylene)-1,3-thiazolidine-2,4-dione, used for the treatment and/or prophylaxis of autoimmune, cardiovascular or neurodegenerative disorders, inflammatory or kidney diseases, bacterial or viral infections, platelet aggregation, cancer, transplant rejection or lung injuries
12/07/2010US7846922 1-(isopropyl)-4-{[4-(tetrahydro-2H-pyran4-yloxy)phenyl]carbonyl}hexahydro-1H-1,4-diazepine, used in the treatment of nervous system and psychological disorders such as Alzheimer's disease or as cognition activators
12/07/2010CA2583084C 7,8-bicycloalkyl-chroman derivatives
12/07/2010CA2440111C Combinations comprising an antidiarrheal agent and an epothilone or an epothilone derivative
12/07/2010CA2434203C 2-arylimino-2,3-dihydrothiazole derivatives, methods for preparing them and therapeutic use thereof
12/07/2010CA2374995C Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
12/02/2010WO2010138790A1 Antiviral compounds composed of three aligned aryl moieties to treat diseases such as hepatitis c
12/02/2010WO2010138578A1 Pyrimidine inhibitors of kinase activity
12/02/2010WO2010138490A1 Benzoxazepines as inhibitors of mtor and methods of their use and manufacture
12/02/2010WO2010138487A1 BENZOXAZEPINES AS INHIBITORS OF PI3K/m TOR AND METHODS OF THEIR USE AND MANUFACTURE
12/02/2010WO2010137351A1 Aryl substituted carboxamide derivatives as calcium or sodium channel blockers
12/02/2010WO2010137350A1 Agent for treatment or prevention of diseases associated with activity of neurotrophic factors
12/02/2010WO2010137349A1 Agent for treatment or prevention of diseases associated with activity of neurotrophic factors
12/02/2010WO2010137302A1 Nitrogen-containing heteroaryl derivatives and fungicides for agricultural and horticultural use
12/02/2010WO2010136138A1 Substituted piperidines
12/02/2010WO2010136128A1 Substituted piperidines
12/02/2010WO2010136109A1 Materials for organic electroluminescent devices
12/02/2010WO2009118596A3 Phthalimide derivatives as trpa1 modulators
12/02/2010US20100305174 Novel Heterocyclic Derivatives
12/02/2010US20100305133 Prolyl Hydroxylase Inhibitors
12/02/2010US20100305118 Pyrimidine inhibitors of kinase activity
12/02/2010US20100305112 Pyrimidine inhibitors of kinase activity
12/02/2010US20100305100 Methods for treating hepatitis c
12/02/2010US20100305097 N-benzyl-4-methyleneamino-3-hydroxy-2-pyridones
12/02/2010US20100305073 Amide compounds as boosters of antivirals
12/02/2010US20100305070 Treatment or prophylaxis of proliferative conditions
12/02/2010US20100305067 Antibacterial condensed thiazoles
12/02/2010CA2763633A1 Pyrimidine inhibitors of kinase activity
12/02/2010CA2763386A1 Substituted piperidines
12/02/2010CA2763370A1 Substituted piperidines
12/02/2010CA2763008A1 Benzoxazepines as inhibitors of pi3k/mtor and methods of their use and manufacture
12/02/2010CA2762885A1 Antiviral compounds composed of three aligned aryl moieties to treat diseases such as hepatitis c
12/02/2010CA2762620A1 Agent for treatment or prevention of diseases associated with activity of neurotrophic factors
12/02/2010CA2761639A1 Aryl substituted carboxamide derivatives as calcium or sodium channel blockers
12/01/2010EP2256119A1 Vasopressin V1a antagonists
12/01/2010EP2256115A1 Heteromonocyclic compound and use thereof
12/01/2010EP2256105A1 Novel tetrahydroisoquinoline derivative
12/01/2010EP2254888A1 Novel aminopyridine derivatives having aurora a selective inhibitory action
12/01/2010EP2254887A1 Oxazolidinone derivatives
12/01/2010EP2254886A2 3,4-dihydro-2h-pyrazinoý1,2-a¨indol-1-one derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
12/01/2010EP2254878A1 Aldh-2 inhibitors in the treatment of addiction
12/01/2010EP2254410A1 Methods for inhibiting drug degradation
12/01/2010EP1869020B1 Heteroaryl urea derivatives useful for inhibiting chk1
12/01/2010EP1487442B1 Thiazolidine carboxamide derivatives as modulators of the prostaglandin f receptor
12/01/2010EP1368342B3 Benzimidazole and pyridylimidazole derivatives as ligands for gaba receptors
12/01/2010CN101903380A 5-aminocyclylmethyl-oxazolidin-2-one derivatives
12/01/2010CN101903378A Aminotriazole derivatives
12/01/2010CN101903373A Functionally selective alpha2c adrenoreceptor agonists
12/01/2010CN101903372A Heteroaryl derivatives as orexin receptor antagonists
12/01/2010CN101903357A Cyclic amine substituted pyrimidinediamines as PKC inhibitors
12/01/2010CN101903351A 病毒聚合酶抑制剂 Viral polymerase inhibitors
12/01/2010CN101903349A 4-(4-pyridinyl)-benzamides and their use as ROCK activity modulators
12/01/2010CN101903347A Piperidinyl and piperazinyl modulators of gamma-secretase
12/01/2010CN101903339A Substituted n-phenyl-bipyrrolidine carboxamides and therapeutic use thereof
12/01/2010CN101902912A Fungicidal amines
12/01/2010CN101899042A 4-substituted-1,2,3-thiadiazole formoxyl ureide compound, preparation method and application thereof
12/01/2010CN101899039A Crystalline polymorph of a bisulfate salt of a thrombin receptor antagonist
12/01/2010CN101899010A Quinazol derivative, preparation method and application thereof
12/01/2010CN101898996A Organic material and application thereof to organic electroluminescent devices
11/2010
11/30/2010US7842816 Mitogen-activated protein kinase kinase inhibitors such as 2-amino-3-methylbutyric acid 2-{[6-(4-bromo-2-chlorophenylamino)-7-fluoro-3-methyl-3H -benzoimidazole-5-carbonyl]-aminooxy}-ethylester, used for the treatment of diseases, such as cancer and inflammation in mammals
11/30/2010US7842813 for synthesis of erythromycin derivatives; reacting thionyl chloride with 6-hydroxylmethyl-nicotinic acid methyl ester to provide 6-chloromethyl-nicotinic acid methyl ester, chlorinating, reacting with ammonia or ammonium hydroxide, sulfiding
11/30/2010US7842704 Biphenyl-2-ylcarbamic Acid 1-{9-[2-(4-Hydroxy-2-oxo-2,3-dihydrobenzothiazol-7-yl)-ethylamino]nonyl}piperidin-4-yl Ester Bis(trifluoroacetate) Salt; chronic obstructive pulmonary disease, asthma; bronchodilators
11/30/2010US7842686 Calcitonin gene-related peptide (CGRP) receptor antagonists, such as 2-(2-Butyl-3-oxo-2H-benzo[b][1,4]thiazin-4(3H)-yl)-N-(2,5-dioxo-1',3'-dihydrospiro[imidazolidine-4,2'-indene]-5'-yl)acetamide, used as analgesics
11/30/2010CA2607499C Histamine-3 receptor antagonists
11/30/2010CA2583492C Naphthalene and isoquinoline derivatives bearing a pyridyl group for the treatment of skin lesions
11/30/2010CA2519938C Prostaglandin analogs as ep4 receptor agonists
11/30/2010CA2482858C Tricyclic thrombin receptor antagonists
11/30/2010CA2432809C Heteroaryl urea neuropeptide y y5 receptor antagonists
11/30/2010CA2335477C Sulfonamide inhibitors of aspartyl protease
11/25/2010WO2010135568A1 Benzoxazepines as inhibitors of mtor and their use to treat cancer
11/25/2010WO2010135524A1 Benzoxazepines based p13k/mt0r inhibitors against proliferative diseases
11/25/2010WO2010135014A1 Tri-cyclic pyrazolopyridine kinase inhibitors
11/25/2010WO2010133534A1 Bicyclic amino substituted compounds as pi3k inhibitors
11/25/2010WO2010133312A1 Halogen-substituted compounds as pesticides
11/25/2010WO2010132999A1 Methyl sulfanyl pyrmidmes useful as antiinflammatories, analgesics, and antiepileptics
11/25/2010WO2010132951A1 Oligothiophenes and uses thereof in photovoltaic devices
11/25/2010WO2010106436A3 Novel anti-inflammatory agents
11/25/2010WO2010081036A3 Fluorine containing compounds and methods of use thereof
11/25/2010WO2009132202A3 Macrocyclic compounds and their use as kinase inhibitors
11/25/2010US20100298558 Substituted dihydroazole compound and pest control agent
11/25/2010US20100298390 Inhibition of lethal factor protease activity from anthrax toxin
11/25/2010US20100298389 Novel Imaging Tracers for Early Detection and Treatment of Amyloid Plaques Caused by Alzheimer's Disease and Related Disorders