Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
07/2003
07/08/2003US6589984 Blood cholesterol and triglycerides (TG) themselves are generally insoluble in blood, and they exist as lipoproteins by binding with apolipoproteins. In the body, triglycerides are biosynthesized primarily in the liver from acetyl CoA as
07/08/2003US6589978 Therapy for nervous system disorders
07/08/2003US6589969 Carboxylic acid derivatives and drugs containing the same as the active ingredient
07/08/2003US6589968 Epothilone compounds and methods for making and using the same
07/08/2003US6589963 Drug salt thereof show a hypoglycemic action, a blood hypolipidemic action, an insulin resistance-improving action and a PPAR activating action, and are useful as a hypoglycemic agent, a hypolipidemic agent, an insulin
07/08/2003US6589962 Certain alpha -hydroxy- gamma -(((carbocyclic- or heterocyclic- substituted)amino)carbonyl)alkanamide derivatives are described as inhibitors of HIV protease and inhibitors of HIV replication. These compounds are useful in
07/08/2003US6589956 Its enantiomers, diastereoisomers, and addition salts thereof with a pharmaceutically acceptable acid or base, and medicinal products containing the same which are useful as a TXA2 receptor antagonist and 5-HT2 receptor antagonist.
07/08/2003US6589953 Indole derivatives as 5-HT1B and 5-HT1D agonists
07/08/2003US6589949 3-oxo-2,1-benzisoxazol-1(3H)-carboxamides for treatment of CNS diseases
07/03/2003WO2003053960A2 Quinline derivates and their use as mek inhibitors
07/03/2003WO2003053959A1 Heterocyclylamino carbonyluracils
07/03/2003WO2003053958A1 Quinazolinedione derivatives
07/03/2003WO2003053955A1 Thiochromenones used to combat painful conditions and neurodegenerative diseases
07/03/2003WO2003053948A1 Isochroman compounds for treatment of cns disorders
07/03/2003WO2003053945A2 Urea derivatives and their use as vanilloid receptor antagonists
07/03/2003WO2003053939A1 Benzimidazole derivatives and their use as gnrh antagonists
07/03/2003WO2003053928A1 Serotonine reuptake inhibitor
07/03/2003WO2003053925A1 Pyrrolidine-2-ones as factor xa inhibitors
07/03/2003WO2003053915A2 Compounds for the treatment of inflammatory disorders
07/03/2003WO2003053912A1 α-(N-SULPHONAMIDO)ACETAMIDE DERIVATIVES AS β-AMYLOID INHIBITORS
07/03/2003WO2003053368A2 Chalcone derivatives and their use to treat diseases
07/03/2003WO2003053366A2 Pyrimidine a2b selective antagonist compounds, their synthesis and use
07/03/2003WO2003053352A2 Therapeutic compounds for treating dyslipidemic conditions
07/03/2003WO2003053344A2 Substituted 2-methyl-benzimidazole respiratory syncytial virus antiviral agents
07/03/2003WO2002101073A3 Aryl-benzimidazole compounds having antiinfective activity
07/03/2003WO2002016340A8 Aminoalkoxybenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same
07/03/2003US20030125551 Benzoxazines, thermosetting resins comprised thereof, and methods for use thereof
07/03/2003US20030125547 Cross coupling reaction of a 2-halopyridine derivative and a 4-halopyridine using a nickel complex catalyst
07/03/2003US20030125370 Treating or preventing protein kinase related disorders in a organism, such as cancer, diabetes, autoimmune disoders, hyperproliferation diosrders, osteoarthritis, rhematoid arthritis, angiogenesis, immunological disorders
07/03/2003US20030125367 Administering a patient with bacterial infections a oxazolidinones having a bicylcic/3.1.0/ hexane containing group as antibiotic
07/03/2003US20030125366 Phorboxazole derivatives for treating cancer
07/03/2003US20030125362 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
07/03/2003US20030125354 Aromatic compounds containing urea or thiourea groups are useful for terating cytokine mediated diseases
07/03/2003US20030125346 Amino-substituted pyrimidinyl derivatives and methods of use
07/03/2003US20030125344 Rho-kinase inhibitors
07/03/2003US20030125340 3-(Amino-or aminoalkyl) pyridinone derivatives and their use for the treatment of HIV related diseases
07/03/2003US20030125339 Substituted alkylamine derivatives and methods of use
07/03/2003US20030125336 Hydrohalide salts of an HIV protease inhibitor
07/03/2003US20030125325 Fungicides
07/03/2003US20030125324 Alpha 4 beta 1 integrin and CD49d/ CD29 (vla-4); antiinflammatory agents
07/03/2003CA2471461A1 Pyrrolidine-2-ones as factor xa inhibitors
07/03/2003CA2470931A1 Chalcone derivatives and their use to treat diseases
07/03/2003CA2470591A1 Therapeutic compounds for treating dyslipidemic conditions
07/03/2003CA2469278A1 Isochroman compounds for treatment of cns disorders
07/03/2003CA2448811A1 Thiochromenones used to combat painful conditions and neurodegenerative diseases
07/02/2003EP1323710A1 Nitrogenous five-membered ring compounds
07/02/2003EP1323420A1 Remedies for inflammatory bowel diseases
07/02/2003EP1323419A1 Airway mucus secretion inhibitors
07/02/2003EP1322646A1 2-(1h-indol-3-yl)-2-oxo-acetic acid amides with antitumor activity
07/02/2003EP1322645A2 Quinazolines, medicaments, which contain these compounds and which are effective as tyrosine kinase inhibitors, their use, and methods for the production thereof
07/02/2003EP1322642A2 sHARMACEUTICALLY ACTIVE SULFONAMIDE DERIVATIVES BEARING BOTH LIPOPHILIC AND IONISABLE MOIETIES AS INHIBITORS OF PROTEIN JUNKINASES
07/02/2003EP1322640A1 Heteroaryl substituted hydroxyphenyltriazine uv-absorbers
07/02/2003EP1322636A1 Farnesyl transferase inhibiting 6- (substituted phenyl)methyl]-quinoline and quinazoline derivatives
07/02/2003EP1322619A1 Isoquinolinone potassium channel inhibitors
07/02/2003EP1322617A1 Compounds and methods for modulation of estrogen receptors
07/02/2003EP1322613A1 Spiroheterocyclic nitriles useful as reversible inhibitors of cysteine proteases
07/02/2003EP1322611A1 Chemical compounds
07/02/2003EP1224180B1 Substituted azoles
07/02/2003EP1218372B1 Novel heterocyclic compounds useful as reversible inhibitors of cysteine proteases
07/02/2003EP1070041B1 Phosphate-mediated cyclization
07/02/2003EP0991627B1 Pyrimidinone compounds, pharmaceutical compositions containing the compounds and the process for preparing the same
07/02/2003EP0913392B1 Ethylene derivatives and pest controlling agents
07/02/2003EP0740658B1 N-substituted azabicycloheptane derivatives used, for example, as neuroleptics
07/02/2003CN1427824A Indole derivatives, process for preparation of same and use thereof
07/02/2003CN1427823A Pyrrolecarboxamides and pyrrolethioamides as fungicides
07/02/2003CN1113059C Pipeazino derivatives as neurokinin antagonists
07/01/2003US6586471 Halogenated 2-amino-3, 4 heptenoic acid derivatives useful as nitric oxide synthase inhibitors
07/01/2003US6586441 Adenosine receptor ligands and their use in the treatment of disease
07/01/2003US6586431 3,3-Biarylpiperidine and 2,2-biarylmorpholine derivatives
07/01/2003US6586430 Administering azabicyclo compounds to treat human immunodeficiency virus infections and respiratory system disorders
07/01/2003US6586368 Condensed heterocylic compounds and herbicides containing them
06/2003
06/26/2003WO2003051870A1 Novel compounds
06/26/2003WO2003051869A1 3,4-dihydro-1h-isoquinoloin-2-yl-derivatives
06/26/2003WO2003051868A1 Lactams as tachykinin antagonists
06/26/2003WO2003051866A1 2-guanidino-4-heterocyclylquinazolines
06/26/2003WO2003051860A2 Substituted 2-phenyl benzofurans as estrogenic agents
06/26/2003WO2003051842A2 Compositions decreasing activity of hormone-sensitive lipase
06/26/2003WO2003051841A2 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
06/26/2003WO2003051840A1 Pyrrolidine and piperidine derivates as nk1 antagonists
06/26/2003WO2003051833A2 Heteroaryl substituted pyrazole modulators of metabotropic glutamate receptor-5
06/26/2003WO2003051359A1 Cis-2,4,5- triphenyl-imidazolines and their use in the treatment of tumors
06/26/2003WO2003051358A1 Hydroxyphenyl-pyrazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
06/26/2003WO2003051274A2 Benzodiazepine derivatives, preparation thereof and use thereof
06/26/2003WO2003040109A3 Quinazoline derivatives as antitumor agents
06/26/2003US20030120080 Such as (2S)-2-((4S)-4-(2,2-difluorovinyl)-2-oxopyrrolidinyl) butanamide; antiepileptic agents; anticonvulsants
06/26/2003US20030120072 Such as (4-(3,4-Difluoro-phenyl)-piperazin-1-yl)-((4S ,4aS,8aR)-2-((S)-3-(6-methoxy-pyridin-3-yl)-2-methyl-propyl)-decahydro -isoquinolin-4yl)-methanone for treatment of schizophrenia, depression, anxiety and bipolar disorders
06/26/2003US20030119895 Anticancer agents
06/26/2003US20030119878 A 1-arylalkyl-3-aminoalkyl-1,4-dihydropyrid-4-one derivative; sexual disorders; anticarcinogenic agents; benign prostatic hypertrophy/fibroids of the uterus; endometriosis, polycystic ovarian disease, precocious puberty; contraceptives
06/26/2003US20030119868 Gyrase inhibitors and uses thereof
06/26/2003US20030119857 Pyrimidinyl methyl indole derivatives with antibacterial activity
06/26/2003US20030119852 Pyridine or pyrimidine compounds containing C(=O or =S)-N-S(O)m=o,1,2 group, used as insecticides, fungicides, miticides and parasiticides
06/26/2003US20030119849 Piperazine and piperidine compounds
06/26/2003US20030119830 Monocyte chemoattractant protein-1 inhibitor compounds
06/26/2003US20030119817 Oxazolidinone derivatives as potential antimicrobials
06/26/2003US20030119816 Cycline-dependent kinase protein inhibitors; antiproliferative agents
06/26/2003US20030119811 Ion channel antagonists that are NMDA antagonists; treatment of migraine, depression, anxiety, schizophrenia, Parkinson's disease, or stroke.
06/26/2003US20030119754 Treating respiratory syncytial virus and human parainfluenza virus infections
06/26/2003US20030119670 Difluoromethyltriazolone compounds, use of the same and intermediates for the production thereof
06/26/2003US20030119029 Apoptosis, autoimmune diseases, antiproliferative agents, antiinflammatory agents, anticancer agents
06/26/2003CA2470723A1 3,4-dihydro-1h-isoquinolin-2-yl-derivatives