Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
06/2004
06/24/2004WO2004017922A3 Keto cannabinoids with therapeutic indications
06/24/2004WO2004011425A3 Indole, azaindole and related heterocyclic ureido and thioureido piperazine derivatives
06/24/2004WO2003099221A3 Methods for using jnk inhibitors for treating or preventing disease-related wasting
06/24/2004WO2003051841A3 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
06/24/2004US20040122237 Substituted benzazoles and methods of their use as inhibitors of Raf kinase
06/24/2004US20040122227 Cyclic guanidine derivatives and their use as pesticides
06/24/2004US20040122079 (R)-thiophene-2,5-dicarboxylic acid 2-hydroxyamide 5-[(1-thiophen-2-yl-ethyl)-amide], e.g.: antiproliferative agents; anticarcinogenic agents; enzyme inhibitors of histonedeacetylases; colon, breast, lung, prostate, rectal, stomach, bladder cancers
06/24/2004US20040122074 1-[5-(4-chloro-phenyl)-1-(2-chloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-2-piperidin-1-yl-ethanone,e.g. as antagonist or inverse agonists; nicotine partial agonist; an opioid antagonist; a dopaminergic agent; an attention deficit disorder agent
06/24/2004US20040122069 Diarylcycloalkyl derivatives, processes for their preparation and their use as pharmaceuticals
06/24/2004US20040122066 Oxadiazole derivatives having anticancer effects
06/24/2004US20040122049 heterocyclic derivatives containing N-substituted piperidine ring and an amide or urea group; useful for treating rheumatic arthritis
06/24/2004US20040122047 Substituted tetrahydroisoquinolines
06/24/2004US20040122025 4-(4-Fluorophenyl)-3-(2-methylsulfanyl-pyrimidin-4-yl)-2H-isoxazol-5-one for example; treating rheumatoid arthritis, osteoarthritis and congestive heart failure
06/24/2004US20040122017 Melanin concentrating hormone (MCH) modulators; metabolic and eating disorders
06/24/2004US20040122005 Isoxazoline derivatives as inhibitors of matrix metalloproteinases and/or TNF-alpha converting enzyme
06/24/2004US20040122001 Pharmaceutical compounds
06/24/2004US20040121996 Benzoxazin-3-ones and derivatives thereof as therapeutic agents
06/24/2004US20040121490 Metal chelate containing compositions for use in chemiluminescent assays
06/24/2004DE69233189T2 Heteroarylpiperidine-pyrrolidine und piperazine und ihre anwendung als antipsychotisches und analgetisches mittel Heteroarylpiperidines-pyrrolidine and piperazine and its application as an antipsychotic and analgesic medium
06/24/2004DE10256182A1 2-Oxadiazolchromonderivate 2-Oxadiazolchromonderivate
06/24/2004CA2508788A1 3-pyrrolyl urea derivatives and their use as antiviral agents
06/24/2004CA2508623A1 Benzomorpholine derivatives
06/24/2004CA2508608A1 Substituted piperazine compounds and their use as fatty acid oxidation inhibitors
06/24/2004CA2508601A1 Benzoxazin-3-ones and derivatives thereof as inhibitors of pi3k
06/24/2004CA2508170A1 Pyrazine-based tubulin inhibitors
06/24/2004CA2505887A1 Pyrazole and imidazole compounds and uses thereof
06/23/2004EP1430050A1 Piperidine derivatives and their use as modulators of chemokine (especially ccr3) activity
06/23/2004EP1430048A1 3-(arylamino)methylene-1, 3-dihydro-2h-indol-2-ones as kinase inhibitors
06/23/2004EP1430043A1 Benzofuran and dihydrobenzofuran derivatives useful as beta-3 adrenoreceptor agonists
06/23/2004EP1430032A2 Substituted amides for the treatment of neurological disorders
06/23/2004EP1429765A2 Inhibitors of histone deacetylase
06/23/2004EP1429759A2 Compounds useful for treating hepatitus c virus
06/23/2004EP1429607A1 Delta 1-pyrrolines used as pesticides
06/23/2004EP1251848B1 Gyrase inhibitors and uses thereof
06/23/2004EP1230227B1 Benzoxa-and benzothiazolyl sulfamates and their use as steroid sulfatase inhibitors
06/23/2004EP1036075B1 Substituted thiazolidinedione and oxazolidinedione having antidiabetic, hypolipidemia and antihypertensive properties
06/23/2004CN1507446A Broadspectrum 2-amino-benzoxazole sulfonamide HIV protease inhibitors
06/23/2004CN1507435A Novel cyano-substituted dihydropyrimidine compounds and their use to treat diseases
06/23/2004CN1507434A Novel 4-anilinoquinoline-3-carboxamides compound
06/23/2004CN1506359A Coumarin amide derivative and its prepn, medicinal composition and use
06/23/2004CN1154645C S-oxide and S,S-dioxide tetrahydrothiopyran phenyloxazolidinones
06/23/2004CN1154644C Oxazolidinone derivatives and pharmaceutical compositions
06/22/2004US6753432 Process for the preparation of thiazolidinedione derivatives
06/22/2004US6753342 2-(1h-indol-3-yl)-2-oxo-acetamides with antitumor activity
06/22/2004US6753331 Heterocyclic derivatives which inhibit factor Xa
06/22/2004CA2192596C 4-(6-fluoro-1,2-benzisoxazolyl)-1-piperidinyl-propoxy-chromen-4-one derivatives, their preparation and their use in the treatment of psychosis, schizophrenia and anxiety
06/17/2004WO2004050681A2 Kinase modulators
06/17/2004WO2004050651A1 Anilinopyrazole derivatives useful for the treatment of diabetes
06/17/2004WO2004050650A1 Anilinopyrazole derivatives useful for the treatment of diabetes
06/17/2004WO2004050636A2 IMIDAZOLE-DERIVATIVES AS FACTOR Xa INHIBITORS
06/17/2004WO2004050632A1 Pyrazole derivatives useful as cox-i inhibitors
06/17/2004WO2004050630A1 The use of aryl- and heteroaryl-substituted tetrahydroisoquinolines in the treatment of chronic and neuropathic pain, migraine headaches, and urge, stress and mixed urinary incontinence
06/17/2004WO2004050082A1 The novel coumarin-amide derivatives and its preparation, said drug composition and its use
06/17/2004WO2004050036A2 Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents
06/17/2004WO2004050024A2 3-aminopyrrolidine derivatives as modulators of chemokine receptors
06/17/2004WO2004031176A3 Delta1 pyrrolines used as pesticides
06/17/2004WO2004026794A3 Removal of aldehyde impurity by reactive polystyrene resin
06/17/2004WO2004021997A3 Inhibitors of fungal invasion
06/17/2004WO2004018414A3 Antibacterial agents
06/17/2004WO2003105781A3 Ophthalmic compositions for treating ocular hypertension
06/17/2004US20040116710 N3 alkylated benzimidazole derivatives as MEK inhibitors
06/17/2004US20040116706 Therapeutic ureas
06/17/2004US20040116530 Tissue fibrosis inhibitors
06/17/2004US20040116507 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
06/17/2004US20040116486 Metalloproteinase inhibitors
06/17/2004US20040116483 Glucagon antagonists/inverse agonists
06/17/2004US20040116475 Nitrogen compounds such as N-(2-{4-[3-chloro-1-(4-methoxyphenyl)-1-H-pyrazol-5-yl]-phenoxy}ethyl)urea, used as cyclooxygenase inhibitors; analgesics; antiinflammatory agents
06/17/2004US20040116474 Novel pyrazole compounds as transforming growth factor (TGF) inhibitors
06/17/2004US20040116473 useful in the treatment of TGF- beta related disease states including, for example, cancer and fibrotic diseases
06/17/2004US20040116471 Indolylpiperidine derivatives as antihistaminic aand antiallergic agents
06/17/2004US20040116465 Novel compounds
06/17/2004US20040116454 Pyrazole compounds useful as protein kinase inhibitors
06/17/2004US20040116445 Substituted thioacetamides
06/17/2004US20040116440 Useful for diagnosis, treatment of male or female sexual dysfunction
06/17/2004US20040116435 Benzimidazol derivatives modulate chemokine receptors
06/17/2004US20040116431 Substituted aryl compounds as novel cyclooxygenase-2 selective inhibitors, compositions and methods of use
06/17/2004US20040116427 Compounds for inhibition of HIV infection by blocking HIV entry
06/17/2004US20040116424 Aryl imidazoles and related compounds as C5a receptor modulators
06/17/2004US20040116421 Heterocyclic compounds as antitumor agents with benzimidazole group and morpholine group, triazoline or pyrimidine heterocycles
06/17/2004US20040116420 Remedial agent for viral infectious disease
06/17/2004US20040116417 Thiohydantoins and use thereof for treating diabetes
06/17/2004US20040116413 useful against a number of human and veterinary pathogens, including gram-positive aerobic bacteria such as multiply-resistant staphylococci and streptococci, anaerobic organisms such as bacteroides and clostridia species, and acid-fast organisms
06/17/2004US20040116388 triazine compoound inhibitors of enzymes that catalyze phosphoryl transfer and/or that bind ATP/GTP nucleotides
06/17/2004US20040116353 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same
06/17/2004US20040116330 Preventive/therapeutic method for cancer
06/17/2004DE10256405A1 New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens
06/17/2004DE10247233A1 New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens
06/17/2004CA2507624A1 Imidazole-derivatives as factor xa inhibitors
06/17/2004CA2507186A1 Anilinopyrazole derivatives useful for the treatment of diabetes
06/17/2004CA2506546A1 Kinase modulators
06/17/2004CA2505945A1 Pyrazole derivatives useful as cox-i inhibitors
06/16/2004EP1428534A1 Benzofurazan derivatives for enhancing glutamatergic synaptic responses
06/16/2004EP1428531A1 Oxyiminoalkanoic acid derivatives with hypoglycemic and hypolipidemic activity
06/16/2004EP1427723A1 Tetrahydropyran derivatives and their use as therapeutic agents
06/16/2004EP1427720A1 3-substituted-4-pyrimidone derivatives
06/16/2004EP1427711A1 Oxazolidinone and/or isoxazoline derivatives as antibacterial agents
06/16/2004EP1427709A1 3-substituted-4-pyrimidone derivatives
06/16/2004EP1427421A1 2,4-disubstituted pyrimidinyl derivatives for use as anticancer agents
06/16/2004EP1427416A2 3-glyoxlylamideindoles for treating cancer
06/16/2004EP1427415A1 Lactam-containing compounds and derivatives thereof as factor xa inhibitors