Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
04/2007
04/12/2007CA2624105A1 Phenyl-[1,2,4]-oxadiazol-5-one derivatives with phenyl group, processes for their preparation and their use as pharmaceuticals
04/12/2007CA2624102A1 Phenyl- and pyridinyl- 1, 2 , 4 - oxadiazolone derivatives, processes for their preparation and their use as pharmaceuticals
04/12/2007CA2624100A1 Derivatives of 2 -aminthiazoles and 2-aminooxazoles, processes for their preparation and their use as pharmaceuticals
04/12/2007CA2624093A1 Phenyl- and pyridyl-i,2,4 -oxadiazolone derivatives with phenyl group, processes for their preparation and their use as pharmaceuticals
04/12/2007CA2623813A1 Nitrogen-containing heterocyclic compound and pharmaceutical application thereof
04/12/2007CA2623348A1 Biaryl substituted heterocycle inhibitors of lta4h for treating inflammation
04/12/2007CA2623043A1 Isoxazolo derivatives as gaba a alpha5 inverse agonists
04/12/2007CA2623009A1 5- (phenylisoxazolylethoxy) -triazol- 3 -yl substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders
04/12/2007CA2622944A1 Diazine azole derivatives, their manufacture and use as pharmaceutical agents
04/11/2007EP1772453A1 Process to produce Oxazolidinones
04/11/2007EP1772452A2 Matrix metalloproteinase inhibitors and uses thereof
04/11/2007EP1771454A1 Hepatitis c inhibitor peptide analogs
04/11/2007EP1771453A1 Hepatitis c inhibitor dipeptide analogs
04/11/2007EP1771449A1 Histamine-3 receptor antagonists
04/11/2007EP1771441A1 Novel carboxamides for use as xa inhibitors
04/11/2007EP1771429A1 New benzoyl urea derivatives
04/11/2007EP1678164B1 Substituted pyrazinone compounds for the treatment of inflammation
04/11/2007EP1641756B1 4-arylsulphonylpiperidine derivatives for antagonism of the 5-ht2a receptor
04/11/2007EP1480972B1 Compounds possessing affinity at 5ht1-type receptors and use thereof in therapy of cns disorders
04/11/2007EP1351938B1 Phenyl derivatives
04/11/2007EP1313725B1 Tricyclic antitumor compounds being farnesyl protein transferase inhibitors
04/11/2007EP1147093B1 Substituted bicyclic derivatives useful as anticancer agents
04/11/2007EP0950656B1 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
04/11/2007CN1946717A Benzimidazole derivative and its use
04/11/2007CN1946716A Cyanopyrrole-containing cyclic carbamate and thiocarbamate biaryls and methods for preparing the same
04/11/2007CN1946714A Azabicyclo (3.1.0) hexane derivatives useful as modulators of dopamine d3 receptors
04/11/2007CN1946713A Chemokine receptor antagonists
04/11/2007CN1946699A Pyridazinone ureas as antagonists of alpha4 integrins
04/11/2007CN1946686A Method for preparing pyrrolidine oximes
04/11/2007CN1946685A Azetidine glycine transporter inhibitors
04/11/2007CN1946402A Piperdine derivatives useful as CCR3 antagonists
04/11/2007CN1944430A Anti-cancer active compound depside peptide as derivative of natural product
04/11/2007CN1944429A 2-oxazolinyl-benzo oxazinyl compound and its composition and preparing method
04/11/2007CN1309712C Precursor of key intermediate of AG 7088 class compound and its sythetic process
04/10/2007US7202381 Compounds as opioid receptor modulators
04/10/2007US7202368 Process for the preparation of 4-(benzimidazolymethylamino) benzamidines
04/10/2007US7202360 Reacting 2,4-difluorophenyl (4-piperidinyl) methanone oxime hydrochloride and 3-(2-haloethyl)-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one in an aqueous alkali solution: high yeild when alkali hydroxide concentration is in the range of 20 to 40%
04/10/2007US7202350 (1S)-1,5-anhydro-1-[3-(1-benzothiene-2-ylmethyl)phenyl-D-glucitol and derivatives, are Na+-glucose cotransporter inhibitors and are used to treat diabetes and related diseases such as insulin-resistance and obesity
04/10/2007US7202262 E.g., 3-(5-p-tolyl-[1,2,4]oxadiazol-3-yl)-benzoic acid; translation of mRNA is allowed to continue past a nonsense mutation point, resulting in the production of a full length protein; genetic disorders
04/10/2007US7202254 N-(p-(substituted 1,2,3-triazol-1-yl)phenyl) derivatives of cycloazaalkanes; particularly useful for treating methicillin-resistant Staphylococcus aureas infections
04/10/2007US7202253 Cycloalkyl inhibitors of potassium channel function
04/10/2007US7202248 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
04/10/2007US7202244 Chk-1 inhibitors
04/10/2007US7202241 8-substituted by an optionally substituted and optionally fused piperidine or piperazine ring and 4 substituted by a (heteo)aryl-methyl-or sulfonyl- group, e.g., 4-(2-Fluoro-benzenesulfonyl)-2,2-dimethyl-8-piperazin-1-yl-3,4-dihydro-2H-benzo[1,4]oxazine; 5-HT6 modulators
04/10/2007CA2307068C Bicyclic compounds, process for their preparation and pharmaceutical compositions containing them
04/10/2007CA2204200C Phenyl alkyl ketone substituted by cyclic amine and a process for the preparation thereof
04/05/2007WO2007037534A1 2-heteroaryl-substituted indole derivative
04/05/2007WO2007037187A1 Sulfonamide derivative having pgd2 receptor antagonistic activity
04/05/2007WO2007037010A1 Phenoxyacetic acid derivatives and drugs using the same
04/05/2007WO2007036477A1 2-substituted hydroxylaminopyrimidine, method for the production and the use thereof in the form of pesticides
04/05/2007WO2007036306A1 2-aminoethoxyacetic acid derivatives and their use in treating thromboembolic disorders
04/05/2007WO2007014934A3 Quinoline derivatives as antibacterial agents
04/05/2007WO2007014934A2 Quinoline derivatives as antibacterial agents
04/05/2007WO2006124874A3 Inhibitors of b-raf kinase
04/05/2007WO2006058338A3 4 - piperidinecarboxamide derivatives as modulators of vanilloid vr1 receptor
04/05/2007WO2006041635A3 Arylthiobenzylpiperidine derivatives
04/05/2007US20070078263 Biaryl substituted heterocycle inhibitors of lta4h for treating inflammation
04/05/2007US20070078154 Quinoline potassium channel inhibitors
04/05/2007US20070078146 Antiinflamamtory agents; antiarthritic agents; inflammatory bowel disorders; multiple sclerosis; asthma
04/05/2007US20070078145 sodium channel modulators such as 4-{4-[3-(2,4-Dichloro-phenoxy)-propyl]-1H-imidazol-2-yl}-N-thiazol-2-yl-benzenesulfonamide; central or peripheral nervous system disorders, pain; neuropathy, inflammation
04/05/2007US20070078138 Analogs of dehydrophenylahistins and their therapeutic use
04/05/2007US20070078134 Treating sleep disorders insomnia; 1-[3-(4-Bromo-2-methyl-2H-pyrazol-3-yl)-4-methoxy-phenyl]-3-(4-chloro-phenyl)-urea; restless leg syndrome, cardiovascular disorders, reducing blood clot
04/05/2007US20070078133 Useful in treating conditions or disorders prevented by or ameliorated by histamine-3 receptor ligands; for example, 5-{4-[3-({2R}-2-methyl-pyrrolidin-1-yl)-cis-cyclobutyl]-phenyl}-pyrimidine
04/05/2007US20070078130 Dual alanyl aminopeptidase and dipeptidyl peptidase iv inhibitors for functionally influencing different cells and for treating immunological inflammatory, neuronal and other diseases
04/05/2007US20070078127 Control of arthropods in animals
04/05/2007US20070078121 Enzyme modulators and treatments
04/05/2007US20070077549 Violet laser excitable dyes and their method of use
04/05/2007DE102005047563A1 New modification of specific substituted thiophene carboxamide, useful for prevention and treatment of thrombo-embolic disease, has higher solubility than known modifications
04/05/2007CA2623958A1 2-heteroaryl-substituted indole derivative
04/05/2007CA2623294A1 2-aminoethoxyacetic acid derivatives and their use
04/05/2007CA2621967A1 2-substituted hydroxylaminopyrimidine, method for the production and the use thereof in the form of pesticides
04/05/2007CA2621310A1 Sulfonamide derivative having pgd2 receptor antagonistic activity
04/04/2007EP1770092A1 Process for the preparation of 5-(4-(2-(N-methyl-N-(2-pyridyl)amino)ethoxy)benzyl)-2,4-thiazolidinedione
04/04/2007EP1770091A1 CGRP-antagonists, process for their preparation as well as their use as medicaments
04/04/2007EP1768978A1 2,4,6-trisubstituted pyrimidines as phosphotidylinositol (pi) 3-kinase inhibitors and their use in the treatment of cancer
04/04/2007EP1768974A1 Substituted diketopiperazines as oxytocin antagonists
04/04/2007EP1768968A1 2-((hetero) aryl)-benzoxazole compounds and derivatives, compositions and methods for stabilizing transthyretin and inhibiting transthyretin misfolding
04/04/2007EP1768959A2 Hetero isonipecotic modulators of vanilloid vr1 receptor
04/04/2007EP1768957A2 Indole-2-carboxylic acid hydrazides as glycogen phosphorylase inhibitors
04/04/2007EP1536797B1 1-amido-4-phenyl-4-benzyloxymethyl-piperidine derivatives and related comounds as neurokinin-1 (nk-1) antagonsists for the treatment of emesis, depression, anxiety and cough
04/04/2007EP1472246B1 Oxadiazoles having antiproliferative activity
04/04/2007EP1429607B1 Delta 1-pyrrolines used as pesticides
04/04/2007EP1383501B1 Acylated piperidine derivatives as melanocortin-4 receptor agonists
04/04/2007EP1377556B1 Pyrazole derivatives for treating hiv
04/04/2007EP1219609B1 Aromatic nitrogenous six-membered ring compounds
04/04/2007CN1942467A 2, 4, 6-substituted pyridyl derivative compounds useful as beta-secretase inhibitors for the treatment of Alzheimer's disease
04/04/2007CN1942463A 2-aminopyridine derivative
04/04/2007CN1942457A 1,3,5-substituted phenyl derivative compounds useful as beta-secretase inhibitors for the treatment of alzheimer's disease
04/04/2007CN1942456A Benzoxazocines and their therapeutic use as monoamine reuptake inhibitors
04/04/2007CN1942445A Novel quinoline-carbaxamides as JACK3 kinase modulators
04/04/2007CN1942441A Sulfonyloxy derivatives
04/04/2007CN1942188A Pyrimidine derivatives and use thereof as agricultural and horticultural fungicides
04/04/2007CN1939917A Cannabinol derivatives and pharmaceutical use thereof
04/04/2007CN1939307A 2,4,6-triamino-1,3,5-triazine derivative
04/04/2007CN1308313C Fused azepine drivatives and their use as antidiuretic agents
04/04/2007CN1308310C Nitrogenous aromatic ring compounds
04/03/2007US7199248 Process
04/03/2007US7199244 Cyclic amine derivatives and methods of use
04/03/2007US7199143 3-[4-(3,6-dihydro-2H-thiopyran-4-yl) phenyl]-]5[1H or 2H-1,2,3-triazol-1 or 2-yl] oxazolidin-2-ones; grampositive bactericides for drug resistant bacteria, especially Staphylococcus, Enterococcus, and Streptococcus
04/03/2007US7199142 1-((5-aryl-1,2,4-oxadiazol-3-yl) benzyl)azetidine-3-carboxylates and 1-((5-aryl-1,2,4-oxadiazol-3-yl)benzyl) pyrrolidine-3-carboxylates as edg receptor agonists