Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
08/2007
08/28/2007US7262299 Diels-Alder reaction; using zeolite y in exchanged with copper; separated from mixture for reuse
08/28/2007US7262296 Substituted aryl alkenoic acid heterocyclic amides
08/28/2007US7262215 N-carbacycle monosubstituted indolocarbazoles as protein kinase inhibitors
08/28/2007US7262207 Antidiabetic agents; hyperglycemic agents; obesity; atherosclerosis; immunomodulatory agents
08/28/2007US7262203 For therapy of hyperproliferative diseases such as cancer or retinopathy; pazopanib and salts
08/28/2007US7262199 Tyrosine kinase inhibitors
08/28/2007US7262196 Tri(cyclo) substituted amide glucokinase activator compounds
08/28/2007US7262195 Compounds useful as motilin agonists and method
08/28/2007US7262192 Such as 1-(2-ethoxyethyl)-3-methyl-5-[(3R)-3-methylpiperazin-1-yl]-N-pyrimidin-4-yl-1H-pyrazolo[4,3-d]pyrimidin-7-amine; cyclic-guanosine monophosphate phosphodiesterase inhibitors
08/28/2007US7262187 Substituted oxazolo- and thizaolopyrimidinones as a mitotic kinesin inhibitor
08/28/2007US7262186 Kinesin spindle protein inhibitor; antiproliferative agents; anticancer agents; 4-(2,5-difluorophenyl0-N-3-fluoropyrrolidin-3-yl)-2-hydroxymethyl-2-phenyl-2,5-dihydro-1N-pyrrol-1-carboxamide
08/23/2007WO2007094513A2 Cyclic amine compound and use thereof for the prophylaxis or treatment of hypertension
08/23/2007WO2007093904A1 Benzoxazinone and benzoxazepinone oxazolidinones as antibacterial agents
08/23/2007WO2007093827A1 Thiophene and thiazole substituted trifluoroethanone derivatives as histone deacetylase (hdac) inhibitors
08/23/2007WO2007093540A1 Benzoyl-piperidine derivatives as 5ht2/d3 modulators
08/23/2007WO2007093507A1 Heterobicyclic sulfonamide derivatives for the treatment of diabetes
08/23/2007WO2007093402A1 Pesticides containing a bicyclic bisamide structure
08/23/2007WO2007093364A1 Azacyclyl-substituted aryldihydroisoquinolinones, process for their preparation and their use as medicaments
08/23/2007WO2007093328A1 Aminoacyl prodrug derivatives and medicaments for the treatment of thromboembolitic disorders
08/23/2007WO2007071396A3 Pyrazinoylguanidine compounds useful in the treatment of inflammatory or allergic conditions
08/23/2007WO2007061741A3 Modulators of the h3 receptor useful for the treatment of disorders related thereto
08/23/2007WO2007059257A3 N4-phenyl-quinaz0line-4 -amine derivatives and related compounds as erbb type i receptor tyrosine kinase inhibitors for the treatment of hyperproliferative diseases
08/23/2007WO2007029062A3 Novel pyridine derivatives
08/23/2007US20070197794 Method for preparing pyrrolidine oximes
08/23/2007US20070197788 Method for the preparation of enantiomer forms of cis-configured 3-hydroxycyclohexane carboxylic acid derivatives using hydrolases
08/23/2007US20070197783 Compositions and methods of treating cell proliferation disorders
08/23/2007US20070197782 N4-[2,2-Dimethyl-3-oxo-benzo[1,4]thiazin-6-yl]-5-fluoro-N2-(3-hydroxy-4,5-dimethoxyphenyl)-2,4-pyrimidinediamine;5-Fluoro-N2-(3-hydroxy-4,5-dimethoxyphenyl)-N4-[3-oxo-benzo[1,4]thiazin-6-yl]-2,4-pyrimidinediamine; autoimmune diseases
08/23/2007US20070197775 Cytotoxic agents comprising taxanes and their therapeutic use
08/23/2007US20070197615 Process for the preparation of the PPAR alpha agonist NS-220
08/23/2007US20070197610 Benzisoxazoles
08/23/2007US20070197605 2-[3-(5-Methyl-2-m-tolyloxazol-4-ylmethoxymethyl)cyclohexylcarbamoyl]cyclobutanecarboxylic acid; modulation and control lipid and/or carbohydrate metabolism
08/23/2007US20070197604 3-Methyl-6-(4-{5-methyl-4-[2-(2-methyl-pyrrolidin-1-yl)-ethyl]-oxazol-2-yl}-phenyl)-pyridazine; for treatment of obesity, cognitive deficiencies, narcolepsy
08/23/2007US20070197595 Benzisoxazoles
08/23/2007US20070197587 Quinoline Derivatives as CRTH2 Antagonists
08/23/2007US20070197570 Indanol derivative
08/23/2007US20070197551 such as 3-amino-5,6-dimethyl-2-[3-(4-quinolin-2-ylpiperazin-1-yl)propylthio]-3H-thieno[2,3-d]pyrimidin-4-one, having serotonin receptor modulatory activity, used for treating irritable bowel syndrome
08/23/2007US20070197547 4-(1-piperazinyl)-2(1H)-quinolone and 4-(1-piperazinyl)quinoline derivatives, e.g., 4-(1-piperazinyl)-1-methyl-3-nitro-2(1H)-quinolone
08/23/2007US20070197541 Biaryl heterocyclic amines,amides, and sulfur-containing compounds and methods of making and using the same
08/23/2007US20070197536 Pyridazin-3(2)-one derivatives and their use as pde4 inhibitors
08/23/2007US20070197532 Glucokinase activators
08/23/2007US20070197531 Benzoyl-piperidine derivatives as dual modulators of the 5-HT2A and D3 receptors
08/23/2007US20070197530 Cycloalkylcarbonyl-3H-spiro[2-benzofuran-1,3'-pyrrolidin]-3-ones: 1'-{[1-(4-Chlorophenyl)cyclo-pentyl]carbonyl}-3H-spiro[2-benzofuran-1,3'-pyrrolidin]-3-one; 11- beta hydroxyl steroid dehydrogenase type 1 inhibitors; mineralcorticoid receptor antagonists; antidiabetic agents
08/23/2007US20070197529 Isolated desfluoro-linezolid, preparation thereof and its use as a reference marker and standard
08/23/2007US20070197526 Pyrazoles for the treatment of obesity and other CNS disorders
08/23/2007US20070197525 Novel tetracyclic tetrahydrofuran derivatives
08/23/2007US20070197513 calcium channel modulator; [[1-(4-{2-[1-(4-Chloro-phenyl)-2-(2-methoxy-phenyl)-1H-imidazol-4-yl]-ethyl}-(4-fluoro-phenyl)-methyl-amine; analgesic, antidiabetic agent; angina, hypertension, myocardial ischemia, arrhythmia, diabetes, urinary incontinence, stroke, pain, brain injury, or neuronal disorders
08/23/2007US20070197509 Compositions and methods for modulating gated ion channels
08/23/2007US20070197508 Novel processes for the preparation of piperazinyl and diazapanyl benzamide derivatives
08/23/2007US20070197504 tert-butyl 4-{[3-({[(6-methyl-3-pyridyl)amino]carbonylamino}methyl)phenyl]methyl}-piperazinecarboxylate; selectively modulates the cardiac sarcomere, for example by potentiating cardiac myosin, and may be useful in the treatment of systolic heart failure including congestive heart failure
08/23/2007US20070197492 Modulation of Pathogenicity
08/23/2007US20070197472 N-Alkynyl-2-Heteroaryloxyalkylamides For Use As Fungicides
08/23/2007US20070197393 Tricyclic benzoylpyrazole derivatives
08/23/2007US20070196332 Cytotoxic agents comprising taxanes and their therapeutic use
08/23/2007DE102006007146A1 Aminoacyl-Prodrugs Aminoacyl prodrugs
08/23/2007CA2642406A1 Benzoxazinone and benzoxazepinone oxazolidinones as antibacterial agents
08/23/2007CA2641933A1 Thiophene and thiazole substituted trifluoroethanone derivatives as histone deacetylase (hdac) inhibitors
08/23/2007CA2641734A1 Acetyl-coa carboxylase (acc) inhibitors and their use in diabetes, obesity and metabolic syndrome
08/23/2007CA2640807A1 Benzoyl-piperidine derivatives as 5ht2/d3 modulators
08/23/2007CA2640307A1 Pesticides containing a bicyclic bisamide structure
08/23/2007CA2638787A1 Cyclic amine compound and use thereof for the prophylaxis or treatment of hypertension
08/23/2007CA2636873A1 Azacyclyl-substituted aryldihydroisoquinolinones, process for their preparation and their use as medicaments
08/23/2007CA2618628A1 Triazole compounds that modulate hsp90 activity
08/22/2007EP1820799A1 2,3,4,5-tetrahydro-1h-1,5-benzodiazepine derivative and medicinal composition
08/22/2007EP1820798A1 7-membered ring compound, process for producing the same, and medicinal use thereof
08/22/2007EP1820503A2 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
08/22/2007EP1819701A1 Cyclic iminocarbamates and use thereof
08/22/2007EP1819700A2 Potassium salt of an hiv intergrase inhibitor
08/22/2007EP1819699A2 Diazepine oxazolidinones as antibacterial agents
08/22/2007EP1819690A2 Chroman compounds
08/22/2007EP1819683A2 Potassium salt of an hiv integrase inhibitor
08/22/2007EP1819341A2 Il-12 modulatory compounds
08/22/2007EP1572670B1 5-substituted-pyrazine or -pyridine glucokinase activators
08/22/2007EP1448523B1 Heterocyclic compounds and methods of use
08/22/2007EP1399433B1 Fluoropyrrolidines as dipeptidyl peptidase inhibitors
08/22/2007EP1379513B1 Prodrugs of cox-2 inhibitors
08/22/2007EP1359908B1 Quinolines and nitrogenated derivatives thereof substituted in 4-position by a piperidine-containing moiety and their use as antibacterial agents
08/22/2007EP1150970B1 (1-phenacy-3-phenyl-3-piperidylethyl)piperidine derivatives, method for the production thereof and pharmaceutical compositions containing the same
08/22/2007CN1332959C Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
08/22/2007CN101023074A Inhibitors of the interaction between MDM2 and P53
08/22/2007CN101023063A Azine-carboxamides as anti-cancer agent
08/21/2007US7259263 Method of synthesis of azole-containing amino acids
08/21/2007US7259262 Arylazole derivatives, their manufacture and use as pharmaceutical agents
08/21/2007US7259250 C-nitroso compounds and use thereof
08/21/2007US7259179 Kinase inhibitors
08/21/2007US7259177 Containing an oxazole ring 2-phenyl-, furanyl- or thiophenyl-substituted; e.g., 2,2-Dimethyl-4-[3-(5-methyl-2-p-tolyloxazol-4-ylmethoxy)cyclohexyl]-butyric acid; treating disorders of fatty acid metabolism, glucose utilization disorders, and also of disorders in which insulin resistance is involvolved
08/21/2007US7259175 Alkanoic acids substituted with a group containing pyridinyl-, pyrimidinyl- or pyrazinyl-phenyl linked through a thiazolyl- or oxazolyl- phenyl group; e.g., 3-[4-(2-{2-[6-(2-Fluoro-phenyl)-pyridin-3-yl]-5-methyl-thiazol-4-yl}-ethoxy)-2-methyl-phenyl]-propionic acid; treating diabetes and atherosclerosis
08/21/2007US7259162 Benzazole derivatives and their use as JNK modulators
08/21/2007US7259161 For therapy of immune response, an autoimmune disease, a neurodegenerative, or a solid or hematologic malignancy
08/21/2007US7259158 Naphthaline derivatives as H3 inverse agonists
08/21/2007US7259157 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists
08/21/2007US7259155 Phosphonic diester derivatives
08/21/2007US7259154 Pyrrolopyrimidines
08/21/2007CA2397270C Method for the preparation of 5-cyanophthalide
08/21/2007CA2304965C ((cyclo)alkyl substituted)-gamma-aminobutyric acid derivatives (=gaba analogues), their preparation and their use in the treatment of neurological disorders
08/16/2007WO2007092751A2 Compounds and methods for modulating fx-receptors
08/16/2007WO2007092531A2 Compounds and compositions as protein kinase inhibitors
08/16/2007WO2007091570A1 Binding inhibitor of sphingosine-1-phosphate
08/16/2007WO2007091147A1 Oxazolidinones containing oxindoles as antibacterial agents
08/16/2007WO2007091046A1 Chemical compounds
08/16/2007WO2007076460A3 Substituted thiazole ureas useful as inhibitors of protein kinases