Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
06/2004
06/24/2004US20040122079 (R)-thiophene-2,5-dicarboxylic acid 2-hydroxyamide 5-[(1-thiophen-2-yl-ethyl)-amide], e.g.: antiproliferative agents; anticarcinogenic agents; enzyme inhibitors of histonedeacetylases; colon, breast, lung, prostate, rectal, stomach, bladder cancers
06/24/2004US20040122074 1-[5-(4-chloro-phenyl)-1-(2-chloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-2-piperidin-1-yl-ethanone,e.g. as antagonist or inverse agonists; nicotine partial agonist; an opioid antagonist; a dopaminergic agent; an attention deficit disorder agent
06/24/2004US20040122070 Substituted 3-carbonyl-1H-indol-1-yl acetic acid derivatives for treating conditions resulting from fibrinolytic disorders, such as deep vein thrombosis and coronary heart disease, and pulmonary fibrosis; Alzheimer's disease
06/24/2004US20040122066 Oxadiazole derivatives having anticancer effects
06/24/2004US20040122063 Ethylenediamine derivatives
06/24/2004US20040122055 C10 carbonate taxane compositions
06/24/2004US20040122053 2-(substituted-phenyl)amino-imidazoline derivatives
06/24/2004US20040122026 N-[2-Methyl-3-(piperidinomethyl)phenyl]-3-[3-(3,5-dichlorobenzyl)-2-dicyanomethylidene imidazolidin-1-yl]propionamide for example; autoimmune or allergic diseases
06/24/2004US20040122017 Melanin concentrating hormone (MCH) modulators; metabolic and eating disorders
06/24/2004US20040122016 Compositions useful as inhibitors of rock and other protein kinases
06/24/2004US20040122015 Dicationic 2,5-diarylfuran aza-analogs as anti-protozoan agents
06/24/2004US20040122001 Pharmaceutical compounds
06/24/2004DE69233189T2 Heteroarylpiperidine-pyrrolidine und piperazine und ihre anwendung als antipsychotisches und analgetisches mittel Heteroarylpiperidines-pyrrolidine and piperazine and its application as an antipsychotic and analgesic medium
06/24/2004CA2509238A1 Substituted 3-carbonyl-1h-indol-1-yl acetic acid derivatives as inhibitors of plasminogen activator inhibitor-1 (pai-1)
06/24/2004CA2509170A1 Substituted 3-alkyl and 3-arylalkyl 1h-indol-1-yl acetic acid derivatives as inhibitors of plasminogen activator inhibitor-1 (pai-1)
06/24/2004CA2508990A1 Compounds and methods for the treatment or prevention of flavivirus infections
06/24/2004CA2508792A1 Heterocyclic compounds, methods of making them and their use in therapy
06/24/2004CA2508699A1 Crystalline derivative of 2- (5-chlorothien-2-yl)-n- ((3s)-1((1s)-1-methyl-2-morpholin-4-yl)-2-oxoethyl)-2-oxopyrrolidin-3-yl) ethensulfonamide
06/24/2004CA2506164A1 Anthranilic acid amide derivatives and their pharmaceutical use
06/24/2004CA2505887A1 Pyrazole and imidazole compounds and uses thereof
06/23/2004EP1431285A1 Reverse hydroxamic acid derivatives
06/23/2004EP1430120A1 Inhibitors of glycogen synthase kinase-3 (gsk-3) for treating glaucoma
06/23/2004EP1430043A1 Benzofuran and dihydrobenzofuran derivatives useful as beta-3 adrenoreceptor agonists
06/23/2004EP1430042A2 Bicyclic heterocycles as rxr ligands
06/23/2004EP1429765A2 Inhibitors of histone deacetylase
06/23/2004EP1429762A1 4,5-dihydro-1h-pyrazole derivatives having potent cb1-antagonistic activity
06/23/2004EP1429761A1 Novel 4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic activity
06/23/2004EP1429759A2 Compounds useful for treating hepatitus c virus
06/23/2004EP1429607A1 Delta 1-pyrrolines used as pesticides
06/23/2004EP1252157B1 Pyrimidine carboxamides useful as inhibitors of pde4 isozymes
06/23/2004CN1507445A Chromenylmethyl pyrimidinediamines as antibacterial agents
06/23/2004CN1507444A 2,3-diazanaphthalene derivatives with angiogenesis inhibiting activity
06/23/2004CN1507442A Furan and thiophene derivatives that activate human peroxisome proliferator activated receptors
06/23/2004CN1507436A Aryl and heteroaryl urea CHK1 inhibitors for use as radiosensitizers and chamosensitizers
06/23/2004CN1507435A Novel cyano-substituted dihydropyrimidine compounds and their use to treat diseases
06/23/2004CN1507434A Novel 4-anilinoquinoline-3-carboxamides compound
06/23/2004CN1506366A Preparation of 2,2'-di(3,4-ethylenedioxy-thiophene)
06/23/2004CN1154642C Pyranone compounds useful to treat retroviral infections
06/23/2004CN1154636C Process for preparnig intermediate in preparation of substd. peperidines
06/22/2004US6753342 2-(1h-indol-3-yl)-2-oxo-acetamides with antitumor activity
06/22/2004US6753335 Delta agonists for nervous system pain
06/17/2004WO2004050653A2 Oxime ester photoinitiators with heteroaromatic groups
06/17/2004WO2004050643A2 Non-nucleoside reverse transcriptase inhibitors
06/17/2004WO2004050633A1 Pesticidal 1-ayl-3-amidoxime-pyrazole derivatives
06/17/2004WO2004050631A1 Substituted dihydrophenanthridinesul fonamides
06/17/2004WO2004050630A1 The use of aryl- and heteroaryl-substituted tetrahydroisoquinolines in the treatment of chronic and neuropathic pain, migraine headaches, and urge, stress and mixed urinary incontinence
06/17/2004WO2004050619A1 Hydroxyethylamine derivatives for the treatment of alzheimer's disease
06/17/2004WO2004050612A1 S-substituted n-1-[(hetero)aryl]alkyl-n′-[(hetero)aryl] alkylysothiocarbamides, method for the production thereof, physiologically active s-substituted n-1-[(hetero)aryl]alkyl-n′-[(hetero)aryl]alkylysothiocarbamides, a pharmaceutical compound and curing method
06/17/2004WO2004050610A2 Modulators of melanocortin receptor
06/17/2004WO2004050087A1 3-(2-hydroxy-phenyl)-1h-pyrazole-4-carboxylic acid amide derivatives as hsp90 inhibitors for the treatment of cancer
06/17/2004WO2004050084A2 Ace-inhibitors having antioxidant and nitricoxid-donor activity
06/17/2004WO2004050035A2 Benzimidazoles and analogs thereof as antivirals
06/17/2004WO2004050024A2 3-aminopyrrolidine derivatives as modulators of chemokine receptors
06/17/2004WO2004050018A2 Dicationic 2,5-diarylfuran aza-analogs as anti-protozoan agents
06/17/2004WO2004049797A2 Pesticidal sulphonylaminopyrazoles
06/17/2004WO2004043463A3 Sulfonamides
06/17/2004WO2004031176A3 Delta1 pyrrolines used as pesticides
06/17/2004WO2004018414A3 Antibacterial agents
06/17/2004WO2003105781A3 Ophthalmic compositions for treating ocular hypertension
06/17/2004US20040116706 Therapeutic ureas
06/17/2004US20040116695 2-Mercapto-4,5-diarylimidazole derivatives and the use thereof as cyclooxygenase inhibitors
06/17/2004US20040116509 Antiviral agent; reducing the activity of viral polymerase; 3-(4-Chloro-2,5-dimethyl-benzenesulfonylamino)-5-(4-chloro-phenyl)-thiophene-2-carboxylic acid for example
06/17/2004US20040116508 1-(N,N-bischloroethylaminoethoxy)-4-tert-butyldimethylsilyloxythioxanthone; administering first then sodium fluoride; tissue targeted therapy; administering in nontoxic, protodrug form which accumulates in neoplasm, followed by an activation drug
06/17/2004US20040116507 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
06/17/2004US20040116497 Chromane derivatives, process for their preparation and their use as antitumor agents
06/17/2004US20040116495 Compounds and methods
06/17/2004US20040116490 Compounds and methods
06/17/2004US20040116488 Substituted 3-alkyl and 3-arylalkyl 1H-indol-1-yl acetic acid derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1)
06/17/2004US20040116486 Metalloproteinase inhibitors
06/17/2004US20040116480 Oxime ether compound and agricultural or horticultural bactericide
06/17/2004US20040116477 2-Heteroaryl-3,4-dihydro-2h-pyrrole derivatives and the use thereof as pesticides
06/17/2004US20040116471 Indolylpiperidine derivatives as antihistaminic aand antiallergic agents
06/17/2004US20040116465 Novel compounds
06/17/2004US20040116456 Remedies for psychoneurosis
06/17/2004US20040116455 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
06/17/2004US20040116454 Pyrazole compounds useful as protein kinase inhibitors
06/17/2004US20040116445 Substituted thioacetamides
06/17/2004US20040116440 Useful for diagnosis, treatment of male or female sexual dysfunction
06/17/2004US20040116439 Serine protease inhibitors
06/17/2004US20040116425 Prenylation inhibitors and methods of their synthesis and use
06/17/2004US20040116424 Aryl imidazoles and related compounds as C5a receptor modulators
06/17/2004US20040116423 5-Aryltetrazole compounds, compositions thereof, and uses therefor
06/17/2004US20040116420 Remedial agent for viral infectious disease
06/17/2004US20040116417 Thiohydantoins and use thereof for treating diabetes
06/17/2004US20040116399 for preventing or treating coagulation disorders
06/17/2004US20040116388 triazine compoound inhibitors of enzymes that catalyze phosphoryl transfer and/or that bind ATP/GTP nucleotides
06/17/2004US20040116387 thyroid receptor ligands, preferably antagonists for the treatment of cardiac and metabolic disorders, such as cardiac arrhythmias, thyrotoxicosis, subcllinical hyperthyrodism and liver diseases
06/17/2004US20040116353 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same
06/17/2004CA2508914A1 Modulators of melanocortin receptor
06/17/2004CA2508783A1 S-substituted n-1-¬(hetero) aryl|alkyl-n'-¬(hetero)aryl|alkylisothiocarbamides, a method for the preparation of these, physiologically active s-substituted n-1-¬(hetero)aryl|alkyl-n'-¬(hetero)aryl|alkylisothiocarbamides, a pharmaceutical composition and method of treatment
06/17/2004CA2508574A1 3-(2-hydroxy-phenyl)-1h-pyrazole-4-carboxylic acid amide derivatives as hsp90 inhibitors for the treatment of cancer
06/17/2004CA2508329A1 Substituted dihydrophenanthridinesul fonamides
06/17/2004CA2508325A1 Hydroxyethylamine derivatives for the treatment of alzheimer's disease
06/17/2004CA2505893A1 Oxime ester photoinitiators with heteroaromatic groups
06/17/2004CA2504740A1 Dicationic 2,5-diarylfuran aza-analogs as anti-protozoan agents
06/16/2004EP1428827A1 Derivatives of 2,2'-Di (3,4-alkylenedioxythiophen) their preparation and use
06/16/2004EP1427725A1 Pyrazolyl-substituted thienyloxypyridines
06/16/2004EP1427722A2 Pyrrole-type compounds, compositions, and methods for treating cancer, treating viral diseases and causing immunosuppression
06/16/2004EP1427719A1 4-alkyl-substitute thienyloxy-pyridines
06/16/2004EP1427718A1 Benzothiepine ileal bile acid transport inhibotors