Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
09/2007
09/07/2007WO2007100066A1 17β HSD type 5 INHIBITOR
09/07/2007WO2007099852A1 Method of testing sensitivity of solid cancer against tyrosine kinase inhibitor and test kit therefor
09/07/2007WO2007099082A1 Novel method for the preparation of stavudine polymorphic form i and form ii
09/07/2007WO2007029156A3 Isoindoledione derivatives as adrenergic receptor antagonists
09/07/2007WO2007011760A3 Inhibitors of mitotic kinesin
09/07/2007WO2006110476A3 Cytotoxic compounds and conjugates comprising duocarmycins with cleavable substrates
09/07/2007CA2644809A1 17 .beta. hsd type 5 inhibitor
09/07/2007CA2644069A1 Therapeutic piperazines as pde4 inhibitors
09/07/2007CA2643044A1 Cinnoline and quinazoline derivates as phosphodiesterase 10 inhibitors
09/07/2007CA2640754A1 Pyrazole derivatives as sigma receptors antagonists
09/06/2007US20070208182 Zwitterionic Non-Linear Optophores And Devices Incorporating Same
09/06/2007US20070208176 Biphenyl derivatives
09/06/2007US20070208172 Process for Preparing Cephalosporin Intermediates Using Alpha-Iodo-1-Azetidineacetic Acid Esters and Trialkylphosphites
09/06/2007US20070208166 Tao Kinase Modulators And Method Of Use
09/06/2007US20070208049 e.g. 1-(2,6-Difluorobenzyl)-5-(3-Mehthoxyphenyl)-6-Methyl-3-[N-Methyl -N -(2-Pyridylethyl)Aminoethyl]Uracil; anticarcinoganic agent; prostate cancer, benign prostatic hypertrophy, breast cancer and endometriosis
09/06/2007US20070208048 New Aryl Imidazoles and Related Compounds as C5a Receptor Modulators
09/06/2007US20070208046 such as 4-benzyloxy-1-{4-[2-(dimethylamino)ethoxy]phenyl}-1H-pyridin-2-one, that as antagonists to melanin concentrating hormone receptors, used for treating cardiovascular, nervous system, metabolic, reproductive system, respiratory system and gatrointestinal disorders
09/06/2007US20070208044 Compounds and therapeutical use thereof
09/06/2007US20070208036 Arylalkanes, arylalkenes and aryl-azaalkanes, pharmaceutical compositions containing these compounds and processes for preparing them
09/06/2007US20070208034 4,6-disubstituted pyrimidines and their use as protein kinase inhibitors
09/06/2007US20070208033 Amine compound and use thereof
09/06/2007US20070208024 (3-Fluoro-4'-methanesulfonyl-biphenyl-4-yl)-[2-(S)-(2-(R)-methyl-pyrrolidin-1-ylmethyl)-pyrrolidin-1-yl]-methanone; treatment of obesity, cognitive deficiencies, narcolepsy, and other histamine H3 receptor-related diseases
09/06/2007US20070208019 Vasculostatic agents and methods of use thereof
09/06/2007US20070208008 Substituted sulfonamides and ureas useful for inhibiting kinase activity
09/06/2007US20070208007 Amine-Based Compound and Use Thereof
09/06/2007US20070208005 Tetrahydrobenzazepines as antagonists and/or reverse agonists of the histamine h3 receptor
09/06/2007US20070207991 Substituted N-aryl Heterocycles, Process For Their Preparation and Their Use As Medicaments
09/05/2007EP1829873A1 Pyrrazole derivatives as sigma receptors antagonists
09/05/2007EP1829865A2 Chemical compounds
09/05/2007EP1828172A1 Pyrrole derivatives having crth2 receptor antagonist activity
09/05/2007EP1828171A2 Heterocycle derivatives as histone deacetylase (hdac) inhibitors
09/05/2007EP1828169A2 Urea inhibitors of map kinases
09/05/2007EP1828167A2 Acrylamide derivatives as antibiotic agents
09/05/2007EP1828148A1 Triazole substituted aminobenzophenone compounds
09/05/2007EP1828146A1 Substituted n-heterocyclic compounds and their use as dopamine d3 receptor ligands
09/05/2007EP1828144A2 Integrin antagonists useful as anticancer agents
09/05/2007EP1828140A1 5-aminopyrazole derivatives as pesticidal compounds
09/05/2007EP1828135A2 Compounds and compositions as modulators of steroidal receptors and calcium channel activities
09/05/2007EP1828127A2 INSECTICIDAL BIS(SUBSTITUTED PHENYL)-1-äÝ4-(SATURATED HETEROCYCLYL-SUBSTITUTED)PHENYLMETHYL¨-(4-PIPERIDYL)üMETHANE DERIVATIVES
09/05/2007EP1828125A1 Arylpiperazine derivatives and their use as ligangs selective of the dopamine d3 receptor
09/05/2007EP1828123A1 Indolinones and their use as antiproliferative agents
09/05/2007EP1828092A1 Process and intermediate compounds useful in the preparation of statins
09/05/2007EP1730116B1 4-carbox pyrazole derivates useful as anti-viral agents
09/05/2007EP1618094B1 Substituted heteroaryls as inhibitors of protein tyrosine phosphatases
09/05/2007EP1474419B1 Amides of aminoalkyl-substituted azetidines, pyrrolidines, piperidines and azepanes
09/05/2007EP1441724B1 Methods of increasing endogenous testosterone levels
09/05/2007EP1373233B1 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same
09/05/2007CN101031563A Benzimidazole derivatives, composition containing thereof and its preparation and application
09/05/2007CN101031558A HIV inhibiting 5-heterocyclyl pyrimidines
09/05/2007CN101031550A HIV inhibiting 5-carbo- or heterocyclic substituted pyrimidines
09/05/2007CN101031545A Isoindoline compounds and methods of their use
09/05/2007CN101031539A Substituted arylalkanoic acid derivatives and use thereof
09/05/2007CN101029042A Bicyclic androgen and progesterone receptor modulator compounds and methods
09/05/2007CN101029022A Process for the preparation of 4-phenoxy quinoline derivatives
09/04/2007US7265228 N-(alpha-methylolbenzyl)1-(aminoethyl)- or 1-(aminocarbonyl)-2-aryl(especially phenyl or benzodioxanyl)-2-hydroxyethylamine intermediates for enantiomeric synthesis of amino ceramide-like compounds
09/04/2007US7265226 Interact with opoid receptors; decreasing metabolic rates of the phenolic piperidines by amidation, imidation, or forming a formamide, a hydroxyamidine or a thioamide; analgesics, anticonvulsants, antitussive agents; diarrhea, drug addiction
09/04/2007US7265152 Benzofuran compounds, compositions and methods for treatment and prophylaxis of hepatitis C viral infections and associated diseases
09/04/2007US7265146 Administering small molecule compounds, especially acids or esters, that inhibit the interaction between alpha 4 integrins and ligands MAdCAM and/or VCAM for treatment of chronic inflammatory diseases such as arthritis, asthma, multiple sclerosis, Chrohn's disease, ulcerative colitis, and hepatitis C
09/04/2007US7265133 Biphenylylaminocarbonyl-amino- or -oxypiperidine derivatives, e.g., biphenyl-2-ylcarbamic acid 1-[2-({4-[(4-hydroxybenzylamino)methyl]benzoyl}methylamino)ethyl]piperidin-4-yl ester; treating bronchodilation and COPD
09/04/2007US7265132 Peptidyl spiroheterocyclic, amidino and guanidino compounds; reversible inhibitors of the cysteine protease cathepsin S, K, F, L and B; useful in the treatment of autoimmune and other related diseases
09/04/2007US7265131 For therapy of disease-states associated with nuclear receptor activity
09/04/2007US7265123 Heterocyclic compounds
09/04/2007US7265120 Pyrazine derivatives and pharmaceutical use thereof
09/04/2007US7265116 Attention deficit disorders; hyperactivity; post-trauma stress disorders; anxiolytic agents; obsessive compulsive disorders; analgesics; Parkinson's disease
09/04/2007US7265114 Antiproliferative agents for smooth muscle cells; antiinflammatory agents for endothelial cells; restenosis, atherosclerosis
09/04/2007US7265112 Small molecule modulators of hepatocyte growth factor (scatter factor) activity
09/04/2007US7265110 Psychological disorders; antidepressants; anxiolytic agents; analgesics; antiinflammatory agents; central nervous system disorders
09/04/2007US7265108 For example, 6-[2-[4-(2-fluorophenoxymethyl)piperidino]ethyl]-1H-pyrazin-2-one; therapeutic or prophylactic agent for diabetic neuralgia, HIV neuralgia, postherpetic neuralgia, nerve system disorders
09/04/2007CA2283083C Use of 2,3,4,5-tetrahydro-1h-3-benzazepines for the manufacture of a pharmaceutical composition for the treatment of sleep disorders
09/04/2007CA2274063C Substituted pyrimidine compounds and their use
09/04/2007CA2258044C Muscarinic antagonists
09/04/2007CA2239174C Novel compounds with analgesic effect
08/2007
08/30/2007WO2007098418A1 Compounds having 5-ht6 receptor affinity
08/30/2007WO2007098356A1 Congeners of milnacipran as monoamine re-uptake
08/30/2007WO2007098214A1 Cinnoline derivatives as phosphodiesterase 10 inhibitors
08/30/2007WO2007098169A1 Cinnoline derivatives as phosphodiesterase 10 inhibitors
08/30/2007WO2007097937A1 Pyrrolidine derivatives as erk inhibitors
08/30/2007WO2007097403A1 Remedy or preventive for digestive ulcer
08/30/2007WO2007097197A1 Amide derivative or salt thereof
08/30/2007WO2007096751A1 Process for the preparation of atorvastatin calcium
08/30/2007WO2007096352A1 5-amino-6-bromo-n-{ [1- (tetrahydr0-2h-pyran-4-ylmethyl) -4-piperidinyl] methyl}-3, 4 -dihydro-2h-chromene-8-carboxamide as 5-ht4 receptor agonist
08/30/2007WO2007096072A2 New pyridin-3-amine derivatives
08/30/2007WO2007095789A1 Imidazol-5-carboxylic acid derivatives, preparation methods and use therrof
08/30/2007WO2007079163A3 Prokineticin 1 receptor antagonists
08/30/2007WO2007073303A3 Novel benzimidazole derivatives as vanilloid receptor 1 (vrl) inhibitors
08/30/2007WO2007071455B1 Sulfoximine-substituted pyrimidines , their preparation and use as drugs
08/30/2007WO2007070556A3 N-(6-membered aromatic ring)-amido anti-viral compounds
08/30/2007WO2007042912A3 Heterocyclic compounds as pstat3/il-6 inhibitors
08/30/2007WO2007034326A3 Imidazole compounds for the treatment of neurological disorders
08/30/2007US20070203338 2-((4,6-dimethoxy)pyrimidin-2-yl-),3-(methoxy-), 3,3-(diphenyl)propionic acid; antihypotensive agents; pulmonary hypertension, mycocardial necrosis; renal failure; brain disorders; antispasmodic agents; antiischemic agents; coagulants; asthma; atherosclerosis; restenosis; Raynaud's syndrome
08/30/2007US20070203221 Processes for preparing darifenacin hydrobromide
08/30/2007US20070203214 6-Hydroxy-2,2-dimethyl-chroman-4-one; anticancer agents; bioavailability
08/30/2007US20070203197 Phosphodiesterase 4 inhibitors
08/30/2007US20070203194 Calcium channel modulators comprising 3-thio-4H-1,2,4-triazoles or S-oxides thereof; angina, hypertension, congestive heart failure, myocardial ischemia, arrhythmia, diabetes, urinary incontinence, stroke, pain, brain injury, or neuronal disorders
08/30/2007US20070203193 Crystalline polymorph of a bisulfate salt of a thrombin receptor antagonist
08/30/2007US20070203192 Saturated and unsaturated 3-pyridyl-benzocycloalkylmethyl-amines for use in treating pain, depression and/or anxiety
08/30/2007US20070203184 Novel Indolin-2-one Derivatives, Their Preparation and the Pharmaceutical Compositions Comprising Them
08/30/2007US20070203179 Azadecalin Glucocorticoid Receptor Modulators
08/30/2007US20070203129 2-Pyridone Derivatives As Neutrophil Elastase Inhibitors And Their Use
08/30/2007US20070203101 Pyrazolyl-substituted heterocycles and their use as phytosanitary products