Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
10/1996
10/30/1996CN1134423A Adhesion receptor antagonists
10/30/1996CN1134422A Improved process for large-scale production of BMS 180048 and analogs
10/30/1996CN1134418A 1-cycloalkenyltetrazolinones
10/29/1996US5569768 Angiotensin II antagonists
10/29/1996US5569659 4-arylpiperazines and 4-arylpiperidines
10/29/1996US5569654 Benzodiazepinones
10/29/1996US5569653 N-[(4-(heteroaryl)-1-pyrrolidinyl)alkyl]-10,11-dihydro-5H-dibenz[B,F]azepines and related compounds and their therapeutic utility
10/29/1996CA2053863C Pyridazinone derivatives
10/24/1996WO1996033196A1 Indole-3-carbonyl and indole-3-sulfonyl derivatives as platelet activating factor antagonists
10/24/1996WO1996033194A1 Benzimidazole compounds and their use as modulators of the gaba a receptor complex
10/24/1996WO1996033192A1 Benzimidazole compounds and their use as modulators of the gabaa receptor complex
10/24/1996WO1996033191A1 Benzimidazole compounds and their use as modulators of the gabaa receptor complex
10/24/1996WO1996033184A1 Thf-containing sulfonamide inhibitors of aspartyl protease
10/24/1996WO1996033176A1 Novel hydroxamic acid and amino-carboxylate compounds as metalloprotease and tnf inhibitors
10/24/1996WO1996033175A1 Cyclic amidino agents useful as nitric oxide synthase inhibitors
10/24/1996WO1996033172A1 Arylsulfonyl hydroxamic acid derivatives as mmp and tnf inhibitors
10/24/1996WO1996032939A1 USE OF α1L AGONISTS IN THE TREATMENT OF INCONTINENCE
10/24/1996DE19514579A1 Verwendung von alpha¶1¶¶L¶-Agonisten zur Behandlung der Harninkontinenz Using alpha¶1¶¶L¶ agonists for treating urinary incontinence
10/24/1996CA2218345A1 Novel hydroxamic acid and amino-carboxylate compounds as metalloprotease and tnf inhibitors
10/24/1996CA2218020A1 Indole-3-carbonyl and indole-3-sulfonyl derivatives as platelet activating factor antagonists
10/24/1996CA2216882A1 Cyclic amidino agents useful as nitric oxide synthase inhibitors
10/23/1996EP0738716A2 Dihydropyridazinones and pyridazinones and their use as fungicides and insecticides
10/23/1996EP0738262A1 Novel heterocyclic compounds
10/23/1996EP0600950B1 Amide tetrazole acat inhibitors
10/23/1996EP0530264B1 Arthropodicidal tetrahydropyridazines
10/23/1996CN1134151A Pyrazine carboxamide derivs., their production and their use in medicaments
10/23/1996CN1134146A Benzoyl guanidines, their production and their use in medicaments
10/23/1996CN1033089C Process for preparation of aryl piperazinyl-heterocyclic compounds
10/22/1996US5567827 4-Hydroxyphenylthio derivatives, their preparation and their use for the preparation of aminoalkoxyphenylsulphonyl derivatives
10/22/1996US5567824 Catalyzing the cyclization in presence of a solvent and a proton acceptor
10/22/1996US5567819 From 4-amino-1,2,4-triazole and nitrobenzene derivative
10/22/1996US5567817 Triazole antifungal agents
10/22/1996US5567726 Selective agonists of 5-hydroxytryptamine-like receptors; useful in treatment of migraine and associated disorders
10/22/1996US5567725 Antidiabetic agent
10/22/1996US5567717 Heterocycle substituted phenoxyalkylheterocycles and their use as antiviral agents
10/22/1996US5567711 Indole-3-carbonyl and indole-3-sulfonyl derivatives as platelet activating factor antagonists
10/22/1996CA2174296A1 Dihydropyridazinones and pyridazinones and their use as fungicides and insecticides
10/22/1996CA1338670C .beta.-lactam antibiotics
10/17/1996WO1996032395A1 Benzimidazole derivatives
10/17/1996WO1996032385A1 Novel substituted piperazine derivatives having tachykinin receptor antagonists activity
10/17/1996WO1996032384A1 Novel 4,6-diarylpyrimidine derivatives and salts thereof
10/17/1996WO1996032383A1 Acetamide derivatives, process for producing the same, and medicinal composition containing the same
10/17/1996WO1996032382A1 1-phenylpyrazole-3-carboxamides acting on neurotensin receptors
10/17/1996WO1996032379A1 INDOLE DERIVATIVES AS cGMP-PDE INHIBITORS
10/17/1996WO1996026728A3 Use of moxonidine for the treatment of atherosclerosis
10/17/1996DE19513990A1 Benzimidazol-Derivate Benzimidazole derivatives
10/17/1996CA2220827A1 1-phenylpyrazole-3-carboxamides acting on neurotensin receptors
10/17/1996CA2218033A1 Acetamide derivative, process for preparing the same, and a pharmaceutical composition containing the same
10/17/1996CA2217707A1 Indole derivatives as cgmp-pde inhibitors
10/16/1996EP0737682A1 Substituted thiophene derivative and agricultural and horticultural fungicide containing the same as active ingredient
10/16/1996EP0737677A1 4-Indolylpiperazinyl derivates
10/15/1996US5565562 Triaza macrocycles
10/15/1996US5565551 Non-azo naphthalimide dyes and uses for same
10/15/1996US5565488 Oxalylamino-benzofuran- and benzothienyl-derivatives
10/15/1996US5565480 Substituted histidines
10/15/1996US5565474 1-heteroarylazetidines and -pyrrolidines process for their preparation and pharmaceutical compositions containing them
10/15/1996US5565469 Benzimidazoles and pharmaceutical compositions containing them
10/15/1996US5565464 Compounds having angiotensine II antagonistic activity
10/15/1996US5565459 Insecticides
10/15/1996US5565456 Anxiolytic aroyl piperidinyl and piperazinylacyl pyrroles
10/15/1996US5565455 Method for treating substance abuse disorders
10/11/1996CA2173693A1 4-indolylpiperazinyl derivatives
10/10/1996WO1996031501A1 Carbonyl-piperazinyl and piperidinil compounds which inhibit farnesyl protein transferase
10/10/1996WO1996031498A1 Novel heterocyclic compounds
10/10/1996WO1996031111A1 Tricyclic compounds useful in the treatment of cell proliferative disorders
10/10/1996CA2217680A1 Tricyclic compounds useful in the treatment of cell proliferative disorders
10/10/1996CA2217197A1 Novel heterocyclic compounds
10/10/1996CA2216654A1 Inhibitors of farnesyl-protein transferase
10/09/1996EP0736525A1 Benzonitriles and -fluorides as 5-HT agonists and antagonists
10/09/1996EP0736022A1 5-(2-imidazolinylamino)benzimidazole derivatives, their preparation and their use as alpha-2 adrenoceptor agonists
10/09/1996EP0736021A1 Polymorphs of losartan and the process for the preparation of form ii of losartan
10/09/1996EP0736008A1 Indole derivatives as anti-estrogens
10/09/1996EP0735877A1 6-(2-imidazolinylamino)quinoxaline compounds useful as alpha-2 adrenoceptor agonists
10/09/1996EP0735872A1 A method of treating neurogenic inflammation
10/09/1996EP0678089B1 N-acyl pyrrolidines and drugs for the treatment or prevention of cholecystokinin and gastrin-related disorders
10/09/1996CN1133042A Indole derivatives as NMDA antagonists
10/09/1996CN1132751A Novel sulfonamides compound and its use as medicine
10/09/1996CN1132748A Tetrazolinones
10/09/1996CN1132625A NK-1 receptor antagonits and 5HT3 receptor antagonists for treatment of emesis
10/08/1996US5563278 Angiotensin II antagonists
10/08/1996US5563165 Prostaglandin inhibitor; fda orange book listed patent for celebrex
10/08/1996US5563162 Bradykinin antagonist quinolines
10/08/1996US5563142 Diaromatic substituted compounds as anti-HIV-1 agents
10/08/1996US5563136 3-Ureidobenzodiazepinones useful as antagonists of CCK or of gastrin
10/03/1996WO1996030364A1 Pharmaceutical compositions
10/03/1996WO1996030348A1 Synthesis of bis-indolylmaleimides
10/03/1996WO1996030347A1 Quinazoline derivatives
10/03/1996WO1996030346A1 Uracil derivatives, and antitumor effect potentiator and antitumor agent containing the same
10/03/1996WO1996030343A1 Inhibitors of farnesyl-protein transferase
10/03/1996WO1996030018A1 Tricyclic carbamate compounds useful for inhibition of g-protein function and for treatment of proliferative diseases
10/03/1996WO1996026196A3 Benzylpiperidines and piperazines as muscarinic antagonists
10/03/1996CA2216707A1 Inhibitors of farnesyl-protein transferase
10/02/1996EP0734386A1 Platelet activating factor antagonists: imidazopyridine indoles
10/02/1996EP0734384A1 3-substituted 1-arylindole compounds
10/02/1996EP0734378A1 Aminosulphonyl-phenyl-1h-pyrrole derivatives, method of their preparation and their use
10/02/1996CN1132509A Process for the prepn. of N-methyl-3-(1-methyl-4-piperidinyl)-14-idole-5-ethanesulfonamide
10/02/1996CN1132206A Pyrrole derivatives
10/01/1996US5561234 1-(7-chloroquinolin-4-yl)pyrazole-3-carboxamide N-oxide derivatives, method of preparing them, and their pharmaceutical compositions
10/01/1996US5561227 Chlorination a carboxylic acid; deprotonation a chiral (oxa or thia)zolidinone; enolizing; cyclization
10/01/1996US5561133 Thymidylate synthase inhibiting quinazolinones