Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
08/2005
08/17/2005EP1562934A1 Amino-heterocycles as vr-1 antagonists for treating pain
08/17/2005EP1562931A2 Anti-infective biaryl compounds
08/17/2005EP1562925A1 Phenylalanine derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
08/17/2005EP1562898A1 Indole derivatives as somatostatin agonists or antagonists
08/17/2005EP1562589A2 Diaminotriazoles useful as inhibitors of protein kinases
08/17/2005EP1282418B1 Use of pyrazole derivatives for treating infertility
08/17/2005EP0991638B1 NOVEL GUANIDINE MIMICS AS FACTOR Xa INHIBITORS
08/17/2005EP0989982B1 Barbituric acid derivatives with antimetastatic and antitumor activity
08/17/2005EP0894085B1 Benzyl(idene)-lactam derivatives, their preparation and their use as selective (ant)agonists of 5-ht1a- and/or 5-ht1d receptors
08/17/2005CN1656109A Non nucleoside reverse transcriptase inhibitors
08/17/2005CN1656090A Heterocyclic compounds which inhibit leukocyte adhesion mediated by alpha4 integrins
08/17/2005CN1656082A Protein kinase inhibitors
08/17/2005CN1656081A 4-anilino quinazoline derivatives as antiproliferative agents
08/17/2005CN1656079A Pyrazole compounds and pharmaceutical compositions comprising the compound
08/17/2005CN1656073A Diaryl urea derivatives useful for the treatment of protein kinase dependent diseases
08/17/2005CN1656069A 1-(aminoalkyl)-3-sulfonylindole and-indazole derivatives as 5-hydroxytryptamine-6 ligands
08/17/2005CN1656066A Pharmaceutical combination
08/17/2005CN1656046A Process for producing cyclic compound
08/17/2005CN1215067C 哒嗪酮醛糖还原酶抑制剂 Pyridazinone aldose reductase inhibitors
08/17/2005CN1215061C Process for preparing anticancer compound, and intermediate
08/16/2005US6930136 For use on metal substrates or in adhesive, sealant or coating compositions for use in proximity to metal substrates
08/16/2005US6930124 Drug for detaching tumor
08/16/2005US6930116 Such as 4-chloro-5-(2-phenyl-thiazol-5-yl)-2H-pyrazole-3-carboxylic acid ethyl amide; for inhibiting topoisomerases; treating bacterial infections in mammals
08/16/2005US6930113 For therapy and prophylaxis of sexual dysfunctios; hypertension, pulmonary hypertension, congestive heart failure, renal failure, myocardial infraction, stable, unstable and variant (Prinzmetal) angina, atherosclerosis
08/16/2005US6930110 Nitrogen compounds such as 5-chloro-4-{4-[4-(2,3-dihydrobenzo[1,4]dioxine-5-yl)-piperazine-1-yl]-butylamino}-2H-piridazin-3-one, used as anxiolytic and hypotensive agents; side effect reduction
08/16/2005US6930107 treating obesity, overweight condition, hyperlipidemia, thyroid disease, hypothyroidism, thyroid cancer and related disorders
08/16/2005CA2342974C Methods and compositions for inhibition of angiogenesis
08/16/2005CA2323703C New cyano-indole serotonin reuptake inhibitors, the procedure for preparing them and the pharmaceutical formulations that contain them
08/16/2005CA2106642C Carbazolone derivatives and process for preparing the same
08/11/2005WO2005073221A1 HETEROCYCLIC MODULATORS OF THE GLUCOCORTICOID RECEPTOR, AP-1, AND/OR NF-κB ACTIVITY AND USE THEREOF
08/11/2005WO2005073220A1 Remedy for irritable bowel syndrome with diarrhea
08/11/2005WO2005073219A1 Fused heteroaryl derivatives for use as p38 kinase inhibitors in the treatment of i.a. rheumatoid arthritis
08/11/2005WO2005073189A1 Fused heteroyral derivatives for use as p38 kinase inhibitors
08/11/2005WO2005072733A1 Dyarylurea compounds as chk-1 inhibitors
08/11/2005WO2005072730A1 Therapeutic agent for diarrhea-type irritable bowel syndrome
08/11/2005WO2005051302A3 Bicyclic inhibitors of mek and methods of use thereof
08/11/2005WO2005044807A3 Benzoimidazole compounds
08/11/2005WO2005041858A3 Mucin production inhibitor
08/11/2005US20050176966 Process for the preparation of pyrimidine derivative, intermediate therefor and process for the preparation thereof
08/11/2005US20050176905 Monomer with anti-microbial character, polymer using the same, and manufacturing method thereof
08/11/2005US20050176802 Pyrrole substituted 2-indolinone protein kinase inhibitors
08/11/2005US20050176799 drugs such as 1-Benzyl-3-(2-furyl)-5-trifluoromethylpyrazole, capable of modulating biosynthesis of cyclic guanosine monophosphate, used for therapy and prophylaxis of cardiovascular disorders such as hypertension, angina pectoris, cardiac insufficiency, thrombosis or atherosclerosis
08/11/2005US20050176796 Tricyclic pyrazole derivatives, process for their preparation and their use as antitumor agents
08/11/2005US20050176794 reacting 2-butyl-1,3-diazaspiro[4.4]non-1-ene-4-one and 5-(4'-bromomethylbiphenyl-2-yl)-1-trityl-1H-tetrazole in the presence of a phase transfer catalyst and immiscible solvents, to form 2-butyl-3-[2'-(triphenylmethyltetrazol-5-yl)-biphenyl-4-yl methyl]-1,3-diazaspiro[4.4]non-1-ene-4-one
08/11/2005US20050176793 formed by dissolving Irbesartan in a mixture of haloalkane and alcohol solvents, then distilling off the solvent from the solution and drying; non-peptide angiotensin antagonist, used for treatment of cardiovascular disorders such as hypertension and heart failure
08/11/2005US20050176771 4-fluoro-1-({[1-(methanesulfonyl)piperidin-4-yl]amino}acetyl)pyrrolidine-2-carbonitrile; insulin-dependent diabetes (type 1 diabetes), non insulin-dependent diabetes (type 2 diabetes), insulin-resistant disorders, obesity; dipeptidyl peptidase IV-inhibiting activity
08/11/2005US20050176770 Novel 1,3-dihydro-2H-indol-2-one derivatives, process for preparing them and pharmaceutical compositions containing them
08/11/2005US20050176760 and tumors; imino-, thiocarbonyl- or hydroxyimino-substituted N-heterocyclic amide compounds such as 2-(3-aminomethylphenylamino)-N-[3-chloro-4-(2-hydroxyiminopyrrolidin-1-yl)phenyl]-2-phenylacetamide
08/11/2005US20050176759 7-sulfonyl-3-benzazepine derivatives as modulators of the dopamine receptor and their use for the treatment cns disorders
08/11/2005US20050176733 Chk-1 inhibitors
08/11/2005US20050176727 Male erectile dysfunction; 1-(3-chlorophenyl)-3-(4-pyridin-2-yl-piperazin-1-yl)propan-1-one O-methyloxime
08/11/2005US20050176726 Pyrimidine ether derivatives; antiinflammatory; analgesic; antiarthritis; antirheumatic;diseases involving sensory nerve function; 2-((6-(4-((1S)-1-(4-fluorophenyl)ethyl)-1-piperazinyl)-4-pyrimidinyl)oxy)quinoline
08/11/2005US20050176721 2,5-Diarylpyrazines, 2,5-diarylpyridines and 2,5-diarylprimidines
08/11/2005US20050176716 (2,3-5,6 aryl-heteroaryl)-bicyclo(2,2,2,)octane-amide derivatives; antiinflammatory, obesity, antidiabetic agent, autoimmune disease, asthma, arthritis; non-steroidal; side effect reduction; pharmacokinetics
08/11/2005US20050176713 Amide derivatives as glycogen synthase kinase 3-beta inhibitors
08/11/2005US20050176712 Integrin expression inhibitor
08/11/2005US20050176709 Selective NPY (Y5) antagonists
08/11/2005US20050176705 5-Chloro-1-(3,5-dichloro-2-methoxy benzenesulfonyl)-4-piperazin-1-yl-1H-indole trifluoroacetic acid salt; 5-hydroxytryptamine (serotonin) HT6 receptor antagonists; antidepressant, anxiolytic agent, cognition activator; ADHD, Alzheimer's and Parkinson's disease, drug and nicotine abuse
08/11/2005US20050176699 Benzodiazepine derivatives, preparation thereof and use thereof
08/11/2005US20050176647 Having an alkylation site via a vinyl linker at the end of a pyrrole-imidazole polyamide; inhibits the expression of a specific gene; high anti-cancer activity
08/11/2005US20050175858 Blue light emitter with large triplet energy band gap; color purity, luminescence efficiency. reduced power consumption
08/11/2005US20050175856 Electroluminescent device
08/11/2005US20050172420 Based on diaminobenzanilides or, more specifically (aminobenzoylamino),(sulfo-),(methoxy)anilines; stable aqueous solutions;nonbleeding/colorfastness; excellent degrees of exhaustion with high colour strength; dyeing natural or synthetic materials, particularly, paper; neutral or greenish-yellow hues
08/11/2005DE102004003811A1 Substituierte N-Cyclohexylimidazolinone, Verfahren ihrer Herstellung und ihre Verwendung als Arzneimittel Substituted N-Cyclohexylimidazolinone, processes for their preparation and their use as medicaments
08/11/2005DE102004003493A1 5-Phenylpyrimidine 5-phenylpyrimidines
08/11/2005CA2555273A1 Heterocycle grafted monomers and related polymers and hybrid inorganic-organic polymer membranes
08/10/2005EP1560824A1 Compounds useful as inhibitors of jak and other protein kinases
08/10/2005EP1560823A1 4-substituted 1-aminocyclohexane derivatives for utilization as orl1-receptor and mu-opiate receptor ligands
08/10/2005EP1560822A1 4-imidazol-1-ylmethyl-pyrimidine derivatives as ligands for gabaa receptors
08/10/2005EP1560817A1 Methods and compositions of novel triazine compounds
08/10/2005EP1560816A1 Quinazoline derivatives
08/10/2005EP1560815A1 Novel pyrimidine-4,6-dicarboxamides for the selective inhibition of collagenases
08/10/2005EP1560811A2 Pharmaceutical compositions as inhibitors of dipeptidyl peptidase-iv (dpp-iv)
08/10/2005EP1560584A2 Fab i inhibitors
08/10/2005EP1507769A4 Copper-catalysed ligation of azides and acetylenes
08/10/2005EP1368340B1 Piperazine derivatives as melanocortin receptor agonists
08/10/2005CN1653073A Substituted phenylacetic acids
08/10/2005CN1653062A (imidazol-1-yl-methyl)-pyridazine as NMDA receptor blocker
08/10/2005CN1653025A NK1 antagonists
08/10/2005CN1652792A N3 alkylated benzimidazole derivatives as MEK inhibitors
08/10/2005CN1652776A N3 alkylated benzimidazole derivatives as MEK inhibitors
08/10/2005CN1651392A 2-and 2, 5-substituted phenylketoenols
08/10/2005CN1214026C Indol-3-yl derivatives
08/10/2005CN1214018C Morpholinones as light stabilizers
08/10/2005CN1214013C HIV replication inhibiting pyrimidines
08/09/2005US6927296 Improved preparation of alpha -polymorphic eletriptan hydrobromide, by salt formation in a solution of 2-butanone and water, distillation, dehydration, desolventizing; purity, white color crystals
08/09/2005US6927232 Phenylethynyl and styryl derivatives of imidazole and fused ring heterocycles
08/09/2005US6927230 Triazole derivatives
08/09/2005US6927227 Heterocyclic containing biphenyl aP2 inhibitors and method
08/09/2005US6927222 Compounds
08/09/2005US6927214 Non-peptide GLP-1 agonists
08/09/2005US6927193 And aryl sulfide derivatives
08/09/2005US6926885 In-vivo diagnostic method by means of near infrared radiation
08/09/2005CA2303217C Use of an angiotensin ii receptor antagonist for the preparation of drugs to increase the survival rate of renal transplant patients
08/04/2005WO2005070922A2 Bis-indole pyrroles useful as antimicrobials agents
08/04/2005WO2005070902A1 Therapeutic agents ii
08/04/2005WO2005070900A1 N-4-(6- (heteo) aryl-pyrimidin-4-ylaminophenyl) -bezenesulfonamides as kinase inhibitors
08/04/2005WO2005070899A1 5-phenylpyrimidines and their use as microbicides
08/04/2005WO2005070898A1 Substituted n-cyclohexyl imidazolinones having an mch-modulatory effect
08/04/2005WO2005070891A2 Compounds and methods of use