Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
02/2006
02/09/2006US20060030559 Diazole derivatives
02/09/2006US20060030558 use as pain relievers, gastrointestinal disorders; 2-Amino-3-aryl-1-[3-((hetero)aryl)piperidin-1-yl]-propan-1-one compounds
02/09/2006US20060030557 Substituted pyridines having antiangiogenic activity
02/09/2006US20060030553 Cell adhesion inhibitors
02/09/2006US20060030543 Multicyclic sulfonamide compounds as inhibitors of histone deacetylase for the treatment of disease
02/09/2006DE69717294C5 Chinazolin derivate und diese enthaltende pharmazeutische zusammenstellungen Quinazoline derivatives and those containing pharmaceutical assortments
02/09/2006CA2578261A1 Pyrazole derivative
02/09/2006CA2575417A1 Chiral pyrrolidine derivatives, and methods for preparing compounds thereof
02/09/2006CA2575018A1 Benzyloxy derivatives as maob inhibitors
02/09/2006CA2573124A1 Anti-inflammatory medicaments
02/09/2006CA2571937A1 Pyrimidine derivatives useful as inhibitors of pkc-theta
02/08/2006EP1622894A1 Antitumoral antiadrogenic pyrrolidines
02/08/2006EP1622893A1 New alicyclic-amine-substituted 4-carboxamido-benzimidazoles as parp-inhibitors and antioxidants
02/08/2006EP1622876A1 Cannabinoid receptor ligands and uses thereof
02/08/2006EP1622872A1 1,2,4-substituerte 1,2,3,4-tetrahydro-and 1,2 dihydro-quinoline and 1,2,3,4-tetrahydro-quinoxaline derivatives as cetp inhibitors for the treatment of atherosclerosis and obesity
02/08/2006EP1622870A2 Glutaminyl based dp iv-inhibitors
02/08/2006EP1622620A1 Quinazoline derivatives and their use in the treatment of cancer
02/08/2006EP1622618A1 Melanocortin receptor-specific compounds
02/08/2006EP1622615A2 Naphthyridine integrase inhibitors
02/08/2006EP1622611A1 Imidazolin-2-ylaminophenyl amides as ip antagonists
02/08/2006EP1187815B1 4-phenyl-pyrimidine derivatives
02/08/2006EP1183243B1 Short-acting benzodiazepines
02/08/2006CN1732165A 1-acyl-pyrrolidine derivatives for the treatment of viral infections
02/08/2006CN1732161A 1,3-diamino-2-hydroxypropane pro-drug derivatives
02/08/2006CN1732159A 2-oxopyrimidine derivatives and their use as human leukocyte elastase inhibitors
02/08/2006CN1732154A Alkyne compounds with MCH antagonistic activity and medicaments comprising these compounds
02/08/2006CN1732002A Derivatives of aryl-quinazoline/aryl-2amino-phenyl methanone which promote the release of parathyroid hormone
02/08/2006CN1731994A Prophylactic and therapeutic agent for neuropathy
02/08/2006CN1240688C Quinazoline compounds
02/08/2006CN1240681C Nitrile derivatives as cathepsin K inhibitors
02/08/2006CN1240680C 1,4-pentadiene-3-ketone compound containing halogenoindyl, and method for preparing same and medicinal use thereof
02/08/2006CN1240679C 2- and 2,5-substituted phenylketoenols
02/07/2006US6995274 Cyanine dyes
02/07/2006US6995263 Indolyl and dihydroindolyl derivatives, their manufacture and use as pharmaceutical agents
02/07/2006US6995262 Use of acylsulfonamido-substituted polymethine dyes as fluorescene dyes and/or markers
02/07/2006US6995261 Treatment of meningitis, septic shock, infections, reperfusion injuries, hepatitis, pancreatitis; bone, autoimmune, viral, and respiratory system disorders; antiinflammatory, antiarthritic, and antitumor agents
02/07/2006US6995182 1-sulfonyl pyrrolidine derivatives
02/07/2006US6995176 1-heterocyclylalkyl-3-sulfonyl-indole or -indazole derivatives as 5-hydroxytryptamine-6 ligands
02/07/2006US6995174 for inhibiting proteases
02/07/2006US6995172 Lactam-containing compounds and derivatives thereof as factor Xa inhibitors
02/07/2006US6995161 Central nervous system disorders
02/07/2006US6995160 Sodium channel blockers
02/07/2006US6995159 4-piperazin-1-yl-2-(pyridin-2-ylmethoxy)-pyrimidine, 2-(6-methyl-pyridin-2-ylmethoxy)-4-piperazin-1-yl-pyrimidine, and 2-(6-chloro-pyridin-2-ylmethoxy)-4-piperazin-1-yl-pyrimidine; for treatment of seizure and eating disorders; reduced side effects
02/07/2006US6995155 Imines such as 4-(3-((3-(2,4-dichlorophenyl)propanoyl)amino)-1-(3-(morpholin-4-yl)propyl)-2-oxo-2,3-dihydro-1H-1,4-benzodiazepin-5-yl)benzamide, administered for prophylaxis of Alzheimer's disease
02/07/2006US6995154 Catalyst for joining, breaking of Dna; antitumor, anticancer agents
02/07/2006US6995144 for example, 6-[2-[4-(2-fluorophenoxymethyl)piperidino]ethyl]-1H-pyrazin-2-one; therapeutic or prophylactic agent for diabetic neuralgia, HIV neuralgia, postherpetic neuralgia, nerve system disorders
02/07/2006CA2311344C 5-(2-imidazolinylamino)-benzimidazole derivatives, their preparation and their use as .alpha.-adrenoceptor agonists with improved metabolic stability
02/02/2006WO2006012395A2 Peptidase inhibitors
02/02/2006WO2006012374A1 Substituted aryl-amine derivatives and methods of use
02/02/2006WO2006011859A2 Preparation of hydrochloride salts of tetrazole derivative
02/02/2006WO2006011035A1 Novel dipeptidyl peptidase iv inhibitors; process for their preparation and compositions containing them
02/02/2006WO2006010749A2 Substituted propenyl piperazine derivatives as novel inhibitors of histone deacetylase
02/02/2006WO2006010591A2 Quinazoline derivatives
02/02/2006WO2005115392A3 3-(4-heteroarylcyclohexylamino) cyclopentanecarboxamides as modulators of chemokine receptors
02/02/2006WO2005105789A3 Novel pyrrole derivatives with angiotensin ii antagonist activity
02/02/2006US20060025599 Benzyloxy derivatives
02/02/2006US20060025597 4-(Aminomethyl)-2-(2,6-dioxo(3-piperidyl))isoindoline-1,3-dione hydrochloride; cytokines level reduced; tumor necrosis factor inhibitors; nontoxic; anticarcinogenic agents; antitumor agents (solid/blood-borne); cardiovascular disorders; osteoporosis; antiinflammatory agents; autoimmune diseases
02/02/2006US20060025591 New uracils having a herbicidal activity
02/02/2006US20060025589 2-Thiohydantoine derivative compounds and use thereof for the treatment of diabetes
02/02/2006US20060025468 Chiral pyrrolidine derivatives, and methods for preparing compounds thereof
02/02/2006US20060025461 Triazole derivative
02/02/2006US20060025459 Having Asp2 ( beta -secretase, BACE1 or Memapsin) inhibitory activity, for therapy of diseases characterised by elevated beta -amyloid levels or beta -amyloid deposits
02/02/2006US20060025454 Prenylation inhibitors and methods of their synthesis and use
02/02/2006US20060025451 Novel pyrazole compounds as transforming growth factor (TGF) inhibitors
02/02/2006US20060025433 Pyrimidine derivatives useful as inhibitors of PKC-theta
02/02/2006US20060025432 N-[2-[(3-Chloro-2-fluorobenzyl)thio]-6-[(2-hydroxy-1-methylethyl)amino]-4-pyrimidinyl]- 4-morpholinesulfonamide; asthma, antiallergens; rhinitis, chronic obstructive pulmonary disease, inflammatory bowel disease, irritable bowel syndrome, osteoarthritis, osteoporosis, rheumatoid arthritis, psoriasis
02/02/2006US20060025425 Benzimidazole and pyridylimidazole derivatives
02/02/2006US20060025424 topoisomerase inhibitors such as [5-(4-Cyclopropylcarbamoyl-imidazol-1-yl)-7-pyrimidin-2-yl-1H-benzoimidazol-2-yl]-carbamic acid ethyl ester, used for prophylaxis of bacterial infections in mammals
02/02/2006US20060025423 2,3-Dichloro-N-(3-methoxy-5-methyl-2-pyrazinyl)-benzenesulphonamide; inflammatory diseases, such as asthma
02/02/2006US20060025421 Pyridyl piperazines for the treatment of CNS disorders
02/02/2006US20060025417 Substituted 2-(diaza-bicyclo-alkyl)-pyrimidone derivatives
02/02/2006US20060025415 Compositions useful as inhibitors of voltage-gated sodium channels
02/02/2006US20060025414 Poly-heterocyclic compounds and their use as metabotropic glutamate receptor antagonists
02/02/2006US20060025413 3-(arylamino)methylene-1,3-dihydro-2H-indol-2-ones as kinase inhibitors
02/02/2006US20060025410 2,4-Pyrimidinediamine compounds and their uses
02/02/2006US20060025409 e.g. N-{2-[3-(3,4-dimethoxy-phenyl)-propyl]-6-morpholin-4-yl-pyrimidin-4-yl}-N'-(1H-indol-3-ylmethylene)-hydrazine; interleukin-12 antagonist; antiinflammatory, antidiabetic agent; rheumatoid arthritis, sepsis, Crohn's disease, multiple sclerosis, psoriasis, or insulin-dependent diabetes mellitus
02/02/2006US20060025406 Modulators of hepatocyte growth factor/c- Met activity
02/02/2006US20060025405 1-Methyl,2,6-dioxo,4-(4-(ethyloxycarbony)piperazin-1-yl-),5-(3-trifluoromethylphenyl)methyl-)-1,2,3,6-tetrahydropyrimidine; antagonist, antagonism; psychoses; antidepressants; schizophrenia; psychological disorders; Alzheimer's disease; neurodegenerative diseases;drug abuse, drug dependence (cocaine)
02/02/2006US20060025403 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same
02/02/2006US20060025402 Benzimidazolidinone derivatives as muscarinic agents
02/02/2006US20060025400 1,2,3,4-Tetrahydropyrazin-2-yl acetamides and methods of use
02/02/2006US20060025347 IAP binding compounds
02/02/2006US20060022193 As sensitizers, optical brighteners and electroluminescent materials; monomers for the synthesis of polymeric light emitting materials of electroluminescent elements
02/02/2006DE112004000350T5 Organische Verbindung und organisches elektrolumineszierendes Element Organic compound and an organic electroluminescent element
02/02/2006DE102004033834A1 New 1-sulfonyl-2-oxo-dihydroindole derivatives are selective antagonists of vasopressin receptors useful e.g. for treating hypertension, cardiac insufficiency, unstable angina or affective disorders
02/02/2006CA2575254A1 Preparation of hydrochloride salts of tetrazole derivative
02/02/2006CA2574361A1 1, 3 substituted cycloamino derivatives and their use as histamine-3 receptor antagonists
02/02/2006CA2572971A1 Substituted propenyl piperazine derivatives as novel inhibitors of histone deacetylase
02/02/2006CA2571223A1 Quinazoline derivatives
02/01/2006EP1620445A2 Method and compositions for identifying anti-hiv therapeutic compounds
02/01/2006EP1620440A1 Synthesis of substituted heterocyclic compounds
02/01/2006EP1620434A1 Fused bicyclic-substituted amines as histamine-3 receptor ligands
02/01/2006EP1620428A1 Substituted pyrimidinones and pyrimidinthiones as crf antagonists
02/01/2006EP1620410A1 Use of derivatives of 2, 4-dihydro- 1,2,4 triazole-3-thione as inhibitors of the enzyme myeloperoxidase (mpo)
02/01/2006EP1620397A1 Hydroxamic acids useful in the treatment of hyper-proliferative disorders
02/01/2006EP1620108A2 Pyrazole-amine compounds useful as kinase inhibitors
02/01/2006EP1620092A2 Compounds, compositions, and methods
02/01/2006EP1620091A2 Inhibitors of glutaminyl cyclase
02/01/2006EP1620088A2 Indole acetic acid derivatives and their use as pharmaceutical agents
02/01/2006EP1620087A1 Azabicyclo derivatives as muscarinic receptor antagonists