Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
01/2010
01/06/2010CN101622247A Cyclized derivatives as eg-5 inhibitors
01/06/2010CN101622246A Polycyclic heteroaryl substituted triazoles useful as AXL inhibitors
01/06/2010CN100577742C Cyanine dye labelling reagents
01/06/2010CN100577659C Processes for producing indole compound
01/06/2010CN100577658C 喹唑啉衍生物 Quinazoline derivatives
01/06/2010CN100577163C Compounds effecting glucokinase
01/06/2010CN100577160C Novel azabicyclic derivatives, preparation method thereof and pharmaceutical compositions containing same
01/05/2010US7642359 Pyrazolyl-substituted heterocycles and their use as phytosanitary products
01/05/2010US7642358 Antidiabetic agents; modulate insulin drug resistance
01/05/2010US7642354 Polycyclic pyrazines as potassium ion channel modulators
01/05/2010US7642352 Process for preparing 2,3-disubstituted indoles
01/05/2010US7642351 2,4-Pyrimidinediamine compounds and their uses
01/05/2010US7642278 Nitrogen compounds such as 3-(5-morpholin-4-yl-1H-benz-imidazol-2-yl)-1H-indazole and/or isomers, used as immunology modulators, antidiabetic agents, antiogenesis inhibitors or for prophylaxis of Alzheimer's disease
01/05/2010US7642277 Non-nucleoside reverse transcriptase inhibitors
01/05/2010US7642276 N-[4-methyl-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)phenyl]-2-pyrrolidin-1-ylisonicotinamide; rheumatoid arthritis
01/05/2010US7642267 Benzimidazole and pyridylimidazole derivatives
01/05/2010US7642265 Benzimidazoles and analogs thereof as antivirals
01/05/2010US7642253 Histone deacetylase inhibitors
01/05/2010US7642245 bactericide for treating drug resistant bacteria
01/05/2010CA2545999C 1,2-di(cyclic)substituted benzene compounds
01/05/2010CA2426457C Aryl or heteroaryl fused imidazole compounds as anti-inflammatory and analgesic agents
01/05/2010CA2392081C Pharmaceutically active isoindoline derivatives
01/05/2010CA2383769C Indole derivatives
01/05/2010CA2318192C .beta.2-adrenergic receptor agonists
01/05/2010CA2185397C Arylalkyl-diazinones
12/2009
12/31/2009US20090326220 Tetrazole-Substituted Arylamides as P2X3 and P2X2/3 Antagonists
12/31/2009US20090326024 Salts of imidazole-5-carboxylic acid derivatives, a method for preparing same and pharmaceutical compositions comprising same
12/31/2009US20090326015 Compounds with embedded benzopyran motif for core structures and preparation method thereof
12/31/2009US20090326011 Azab i cyclo [3 . 1 . 0] hexane derivatives as dopamin d3 receptor modulators
12/31/2009US20090325979 Novel imidazolylalkylcarbonyl derivatives as calcium channel modulators and preparation method thereof
12/31/2009US20090325974 1,5-diphenylpyrazoles ii as hsp90 inhibitors
12/31/2009US20090325973 Formulations containing pyridazine compounds
12/31/2009US20090325955 Gyrase inhibitors and uses thereof
12/31/2009US20090325935 Gyrase inhibitors and uses thereof
12/31/2009US20090325209 Method and reagent for measuring nitroreductase enzyme activity
12/31/2009US20090324720 Biocompatible crosslinked hydrogels, drug-loaded hydrogels and methods of using the same
12/31/2009US20090324569 Biaryl pde4 inhibitors for treating inflammatory, cardiovascular and cns disorders
12/31/2009US20090324540 Compounds and compositions for delivering active agents
12/30/2009WO2009158571A1 Heteroaryl compounds and uses thereof
12/30/2009WO2009158375A1 Aza-cylic indole- 2 -carboxamides and methods of use thereof
12/30/2009WO2009157860A1 New heterocyclic carboxamides for use as thrombin inhibitors
12/30/2009WO2009157428A1 Phosphorescent light-emitting composition and light-emitting element comprising the composition
12/30/2009WO2009157425A1 Composition, and light-emission element produced by using the composition
12/30/2009WO2009157011A1 Process for the preparation of high purity sunitinib and its pharmaceutically acceptable salt
12/30/2009WO2009157001A2 Process for preparation of candesartan cilexetil
12/30/2009WO2009156837A2 Amorphous form of a 3-pyrrole substituted 2-indolinone malate salt
12/30/2009WO2009156339A1 Isoquinolinone derivatives as nk3 antagonists
12/30/2009WO2009156128A1 Pharmaceutical composition comprising n-[2-(diethylamino)ethyl]-5-[(5-fluoro-1,2- dihydro-2-oxo-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1 h-pyrrole-3-carboxamide
12/30/2009WO2009137270A3 Azetidine derivatives
12/30/2009WO2009136995A3 2, 6-diamino- pyrimidin- 5-yl-carboxamides as syk or jak kinases inhibitors
12/30/2009WO2008142623A3 Tumor necrosis factor - alpha inhibitors
12/30/2009EP2138490A1 New method for synthesis of fluoroquinolones
12/30/2009EP2138489A1 Novel pyrimidine compound having benzyl(heterocyclicmethyl)amine structure and pharmaceutical product containing the same
12/30/2009EP2138486A1 Compound for organic electroluminescent device and organic electroluminescent device
12/30/2009EP2138482A1 Bicyclic heterocyclic compound
12/30/2009EP2138167A1 Pharmaceutical composition comprising N-[2-(Diethylamino)ethyl]-5-[(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene) methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
12/30/2009EP2137208A2 Compounds for diagnosing apoptosis
12/30/2009EP2137177A2 Aurora kinase modulators and method of use
12/30/2009EP2137166A1 4, 6-disubstituted aminopyrimidine derivatives as inhibitors of protein kinases
12/30/2009EP2137164A1 Inhibitors of protein kinases
12/30/2009EP2136635A1 Chemical compounds
12/30/2009EP2049525B1 N-(aminoheteroaryl)-1h-indole-2-carboxamide derivatives, and preparation and therapeutic application thereof
12/30/2009EP2004625B1 C-met protein kinase inhibitors for the treatment of proliferative disorders
12/30/2009EP1608632B1 Quinazolines useful as modulators of ion channels
12/30/2009CN101616911A Chemical linkers with single amino acids and conjugates thereof
12/30/2009CN101613321A Mono- and bicyclic azole derivatives that inhibit the interaction of ligands with rage
12/30/2009CN100575352C 1-(4- chloroanilino)-4-(4-methylpyridyl)-2,3-diazophenodiazine synthesis and uses
12/30/2009CN100575346C Pyrimidinone derivaties as therapeutic agents against acute and chronic inflammatory, ischaemic and remodelling processes
12/30/2009CN100575345C Pyridone derivative having affinity for cannabinoid 2-type receptor
12/30/2009CN100575341C Tetrahydro-indolone derivative and tetrahydro-indazolone derivatives and their use
12/30/2009CN100575330C Novel compounds
12/30/2009CA2766328A1 New therapeutic agents
12/30/2009CA2729546A1 Compounds and compositions as kinase inhibitors
12/30/2009CA2728852A1 Pharmaceutical composition comprising n-[2-(diethylamino)ethyl]-5-[(5-fluoro-1,2-dihydro-2-oxo-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide
12/30/2009CA2728283A1 Isoquinolinone derivatives as nk3 antagonists
12/30/2009CA2727925A1 New heterocyclic carboxamides for use as thrombin inhibitors
12/30/2009CA2727455A1 Heteroaryl compounds and uses thereof
12/30/2009CA2724310A1 Process for the preparation of high purity sunitinib and its pharmaceutically acceptable salt
12/29/2009USRE41065 Such as (6,7-dimethoxyquinazolin-4-yl)-(3-ethynylphenyl)-amine for treatment of hyperproliferative diseases
12/29/2009US7638549 Mitotic kinesin inhibitors
12/29/2009US7638546 Imidazolyl derivatives
12/29/2009US7638523 e.g. tert-butyl 2-(4-(2-(4-(2-(diethylamino)ethoxy)phenylamino)pyrimidin-5-yl)-2-fluorobenzamido)acetate; C-kit kinase receptor or stem cell factor inhibitors; asthma allergic sinusitis and rhinitis, atopic and allergic dermatitis, allergic contact rheumatoid arthritis, multiple sclerosis, lupus etc.
12/29/2009US7638521 3-guanidinocarbonyl-1-heteroaryl-indole derivatives, preparation process, their use as medicaments, and pharmaceutical compositions comprising them
12/29/2009US7638513 inhibitors of matrix metalloproteinases, aggrecanases, tumor necrosis factor-alpha converting enzyme, and tumor necrosis factors
12/29/2009CA2428133C Indolylmaleimide derivatives as protein kinase c inhibitors
12/29/2009CA2410311C Barbituric acid analogs as therapeutic agents
12/29/2009CA2387013C 6-position substituted indolinones, the preparation thereof and their use as pharmaceutical compositions
12/29/2009CA2370250C Di-aryl acid derivatives as ppar receptor ligands
12/29/2009CA2338543C Method of direct identification of compound efficacy at a g protein-coupled orphan receptor
12/24/2009US20090318706 Process for the Preparation of Candesartan Cilexetil
12/24/2009US20090318694 Cross-Linked Amine Compounds and Agents for Pest Control
12/24/2009US20090318692 Process of making imatinib
12/24/2009US20090318691 Novel Aromatic AZA Heterocycles, Method of Production and Use of the Material in Organic Electronics
12/24/2009US20090318687 Methods of Treating or Preventing Autoimmune Diseases With 2,4-Pyrimidinediamine Compounds
12/24/2009US20090318668 Water-Soluble CC-1065 Analogs and Their Conjugates
12/24/2009US20090318525 Process For Preparing A 3-Pyrrole Substituted 2-Indolinone Malate Salt
12/24/2009US20090318521 Synthesis of 4-Bromomethyl-2'-Formylbiphenyl and 4-Bromomethyl-2'-Hydroxymethylbiphenyl and Its Use in Preparation of Giotensin II Antagonists
12/24/2009US20090318518 Indole and indoline cyclopropyl amide derivatives as ep4 receptor antagonists
12/24/2009US20090318517 Novel Compounds 148
12/24/2009US20090318504 Use of GAL3 receptor antagonists for the treatment of depression and/or anxiety and compounds useful in such methods