Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
03/1996
03/26/1996US5502062 2-amino-4-quinolyl-dihydropyridines, processes for their preparation, and their use
03/26/1996US5502059 Substituted 1-naphthyl-3-pyrazolecarboxamides which are active on neurotensin, their preparation and pharmaceutical compositions containing them
03/26/1996US5502051 Central nervous system, antispasmodic
03/26/1996US5502048 Cns, strokes, hypoglycemic agents and antiischemic agents
03/26/1996US5502028 Herbicidal pyrimidinyl or triazinyl haloacetic acid derivatives
03/26/1996US5502027 Algicides
03/26/1996CA1338191C Herbicidal benzotriazole derivatives
03/21/1996WO1996008485A1 Quinoxalinedione nmda receptor antagonists
03/21/1996WO1996008480A1 Neurokinin antagonists
03/21/1996WO1996008475A1 Pesticidal pyridine derivatives
03/21/1996CA2200083A1 Neurokinin antagonists
03/20/1996EP0702011A1 Water soluble piperidine-triazine compounds for use as stabilizers for polyamide fibers
03/20/1996EP0702004A2 2,9-diamino- and 2-amino-8-carbamoyl-4-hydroxy-alkanoic acid amid derivatives
03/20/1996EP0702003A2 Process for preparing 2-halogenpyridinaldehydes and new 2-halogenpyridinaldehydes
03/20/1996EP0701819A2 Novel compositions containing sertraline and a 5-HT1D receptor agonist or antagonist
03/20/1996EP0701555A1 Indazole derivatives
03/20/1996EP0701553A1 Arylpyrazole fungicides
03/20/1996EP0701439A1 Stable copper(i) complexes and methods related thereto
03/20/1996EP0690867A4 Taxanes having furyl or thienyl substituted side-chain
03/20/1996EP0556332B1 Substituted tetrahydropyridines and hydroxypiperidines as central nervous system agents
03/20/1996EP0505465B1 4-Heterocyclyl-piperidine derivatives, their preparation and their use as inhibitors of calcium overload in brain cells
03/20/1996CN1118990A Medicament for treating or preventing cerebrovascular diseases
03/19/1996US5500426 Administered to improve glucose tolerance
03/19/1996US5500423 Analgesics
03/19/1996CA2014208C Selective blocking of spontaneously-active dopamine neurones in ventral tegmental area
03/16/1996CA2158227A1 2,9-diamino- and 2-amino-8-carbamoyl-4-hydroxy-alkanoic acid amide derivatives
03/14/1996WO1996007973A1 A method of preparing chemical compounds
03/14/1996WO1996007691A2 Thermosetting resin compositions containing maleimide and/or vinyl compounds
03/14/1996WO1996007641A1 Heterocyclic derivative and medicine
03/14/1996WO1996007633A1 Phenylacetic acid alkyl esters
03/14/1996WO1996007410A2 Depolarizing skeletal muscle relaxants
03/14/1996DE4426625A1 2-Phenylindole, Verfahren zu deren Herstellung, diese enthaltende pharmazeutische Präparate sowie deren Verwendung zur Herstellung von Arzneimitteln 2-phenylindoles, processes for their preparation, pharmaceutical compositions containing them and their use for the preparation of medicaments
03/14/1996CA2199518A1 Heterocyclic derivative and medicine
03/14/1996CA2199422A1 Alkyl phenylacetates
03/13/1996EP0700913A1 5,6-dihydro-4H-imidazo(4,5,1-ij)quinolines, processes for their preparation, their use as medicaments, and intermediate compounds
03/13/1996EP0700911A1 Imidazole derivatives having anti-HIV activity
03/13/1996EP0700907A1 Process for producing pyrimidine derivative
03/13/1996EP0700904A1 Heterocyclic-N-oxide substituted benzoylguanidines, process for their preparation, their use as medicament or diagnostic, medicaments containing them as well as intermediates for their preparation
03/13/1996EP0700396A1 Piperidine derivatives, their preparation and use
03/13/1996EP0700391A1 Herbicidal compounds
03/13/1996EP0700389A1 Anti-arrhythmic n-substituted 3-benzazepines or isoquinolines
03/13/1996EP0700388A1 Substituted beta-aryl and beta-heteroaryl-alpha-cyanoacrylamide derivatives as tyrosine kinase inhibitors
03/13/1996EP0700387A1 Salts of substituted heteroaromatic nitrogen compounds, method for their preparation and pharmaceutical compounds containing same
03/13/1996EP0700385A1 Novel compounds
03/13/1996EP0700292A1 Methods and compositions for treating gastric disorders using optically pure (+) pantoprazole
03/13/1996EP0690841A4 Synthetic matrix metalloprotease inhibitors and uses thereof
03/13/1996CN1118358A Compositions for the stabilization of synthetic polymers
03/13/1996CN1118347A Benzotoudened 5-ringneterocycl, preparation and phamaceutical and diagnostic use of same
03/13/1996CN1031265C Tetra hydro-pyrimidine compostion useful as pesticide
03/13/1996CN1031264C Preparation of 1,3-dihydro-4-pyridoyl-2H-imidazol-2-ones derivatives
03/13/1996CN1031263C Method for preparing of quinoline, quinazoline, and cinnoline derivativos
03/12/1996US5498720 Antiinflammatory agent using 4h-1,2,4-triazol-3-thiol derivatives
03/12/1996US5498717 6,7-dialkoxy-3,4-diydroisoquinolin-8-yl compounds
03/12/1996US5498626 Acylaminoindole derivatives as 5-ht1 agonists
03/12/1996US5498612 4-phenethylaminopyrimidine derivative, and agricultural and horticultural chemical for controlling noxious organisms containing the same
03/12/1996US5498610 Blocking agent for n-methyl aspartic acid receptor sites
03/12/1996US5498609 Benzoazepinyl compounds as oxytocin and vasopressin antagonists
03/07/1996WO1996006841A1 Quinazoline derivative
03/07/1996WO1996006832A1 Novel 4-aminopyridazines, method of preparing them and drugs containing these compounds
03/07/1996WO1996006829A1 1,4-dihydropyridine derivative
03/07/1996WO1996006616A1 Quinazolinone pharmaceuticals and use thereof
03/07/1996WO1996006610A1 Use of 5-substituted pyridine and hexahydroquinoline-3 carboxylic acid derivatives for treating diseases of the central nervous system
03/07/1996WO1996006609A1 Inhibitors of farnesyl-protein transferase
03/07/1996DE4430757A1 Neue 4-Aminopyridazine, Verfahren zu ihrer Herstellung sowie diese Verbindungen enthaltende Arzneimittel New 4-Aminopyridazine, process for their preparation and pharmaceutical compositions containing them
03/07/1996DE4430639A1 Verwendung von 5-substituierten Pyridin- und Hexahydrochinolin-3-carbonsäurederivaten Use of 5-substituted pyridine and hexahydroquinoline-3-carboxylic acid derivatives
03/07/1996DE19531995A1 Photochemical and thermal stabilisation of polyamide fibre material
03/07/1996CA2198726A1 Inhibitors of farnesyl-protein transferase
03/07/1996CA2198495A1 Use of 5-substituted pyridine and hexahydroquinoline-3 carboxylic acid derivatives for treating diseases of the central nervous system
03/07/1996CA2198366A1 Novel 4-aminopyridazines, processes for their production as well as pharmaceutical agents
03/06/1996EP0699674A1 1-Aryl-2-acetylamidopentanone derivatives for use as tachykinin receptor antagonists
03/06/1996EP0699665A1 Imidazoline derivatives, their preparation and their use as tachykinin receptor antagonists
03/06/1996EP0699196A1 Carbazole derivatives with 17,20-lyase-inhibiting activity
03/06/1996EP0699195A1 Thioindole pyperidinyl derivatives used as antalgics
03/06/1996EP0699194A1 5-ht4 receptor antagonists
03/06/1996EP0699188A1 Quinoline derivatives as leukotriene antagonists
03/06/1996EP0699187A1 DERIVATIVES OF -g(b), -g(b)-DIMETHYL-4-PIPERIDINEETHANAMINE AS INHIBITORS OF THE CHOLESTEROL BIOSYNTHESIS
03/06/1996EP0699185A1 GUANIDINE DERIVATIVES AS INHIBITORS OF Na+ /H+ EXCHANGE IN CELLS
03/06/1996EP0515638B1 Novel preorganized hexadentate ligands useful in radiographic imaging agents
03/06/1996EP0440670B1 Heterocyclic acetylenic amines having central nervous system activity
03/06/1996CN1118165A Ortho-substituted 2-methoxyiminophenylacetic acid methylamides
03/06/1996CN1118138A Substituted azolone derivatives for treating diseases caused by helicobacter
03/06/1996CN1031190C Process for preparation of quinoline carboxylic acid derivatives
03/05/1996US5496956 By esterification of carboxy substitution with alcohols in the presence of mineral acid
03/05/1996US5496951 4-oxoquinoline-3-carboxylic acid derivatives their preparation and their use
03/05/1996US5496947 Quinolone carboxylic acid derivatives
03/05/1996US5496944 Process for preparing tris-pyrrolidonyl triazine crosslinker
03/05/1996US5496942 5-ht3-receptor antagonists
03/05/1996US5496844 Indole derivatives
03/05/1996US5496833 Piperidine tachykinin receptor antagonists
02/1996
02/29/1996WO1996006137A1 Naphtholactam dyes
02/29/1996WO1996006097A1 New multimerizing agents
02/29/1996WO1996006096A1 Pyridine derivative
02/29/1996WO1996006095A1 Endothelin antagonists
02/29/1996WO1996006094A1 Novel substituted piperidines useful for the treatment of allergic diseases
02/29/1996WO1996006087A1 Bicyclic compounds
02/29/1996WO1996006083A1 2-(piperazinyl-1-carbonylmethyl)-1,4-dihydropyridines as bradykinin antagonists
02/29/1996WO1996006082A1 Dihydropyridine derivatives as bradykinin antagonists
02/29/1996WO1996006078A1 N-(2-(pyrrolidinyl-1)-1-phenylethyl)acetamides as kappa receptor antagonists
02/29/1996WO1996006077A1 N-[2-(pyrrolidinyl-1)-1-phenylethyl]acetamides as kappa receptor antagonists
02/29/1996CA2517691A1 Endothelin antagonists