Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
01/1998
01/07/1998EP0816356A1 1-(2-(1-piperidinyl)-1-ethyl)-1,3-dihydro-2H-benzimidazole derivatives and their pharmaceutical use
01/07/1998EP0816355A1 Heterocyclic spiro derivatives
01/07/1998EP0816342A2 Process for producing 1-substituted-hydantoins
01/07/1998EP0816341A1 Process for the preparation of chiral succinic acid derivatives
01/07/1998EP0816338A1 3-(bis-substituted-phenylmethylene)oxindole derivatives
01/07/1998EP0815859A1 Intimal thickening inhibitors
01/07/1998EP0815856A2 Retroviral protease inhibitors
01/07/1998EP0815120A1 17-difluoromethylene-oestratrienes
01/07/1998EP0815108A1 Cyclic urea hiv protease inhibitors
01/07/1998EP0815104A1 3-benzylamino-2-phenylpiperidines as neurokinin antagonists
01/07/1998EP0815103A1 Trypsin and thrombin inhibitors
01/07/1998EP0815102A1 REDUCTIVE ALKYLATION PROCESS FOR THE PREPARATION N-(2-(R)-HYDROXY-1-(S)-INDANYL)-2(R)-PHENYLMETHYL-4(S)-HYDROXY-5-(1-(4-(3-PYRIDYLMETHYL)-2(S)-N'-(t-BUTYLCARBOXAMIDO)-PIPERAZINYL))-PENTANEAMIDE (=COMPOUND J OR L-735,524)
01/07/1998EP0815101A1 PROCESS TO MAKE HIV PROTEASE INHIBITOR FROM 2(S)-4-PICOLYL-2-PIPERAZINE-t-BUTYLCARBOXAMIDE
01/07/1998EP0815100A1 Tricyclic amide and urea compounds useful for inhibition of g-protein function and for treatment of proliferative diseases
01/07/1998EP0815099A1 Tricyclic amide and urea compounds useful for inhibition of g-protein function and for treatment of proliferative diseases
01/07/1998EP0815089A1 Biphenyl-substituted triazines as light stabilizer
01/07/1998EP0815080A1 Di-substituted 1,4-piperidine esters and amides having 5-ht 4? antagonistic activity
01/07/1998EP0814840A1 Oral pharmaceutical dosage forms comprising a proton pump inhibitor and a prokinetic agent
01/07/1998EP0814839A1 Oral pharmaceutical dosage forms comprising a proton pump inhibitor and a nsaid
01/07/1998EP0814807A1 Tricyclic compounds useful for inhibition of g-protein function and for treatment of proliferative diseases
01/07/1998EP0690846B1 Herbicidal heterocyclic-substituted pyridines
01/07/1998EP0613458B1 Acyclic ethylenediamine derivatives as substance p receptor antagonists
01/07/1998EP0565396B1 1-[2-(arylsulfonylamino)-1-oxoethyl]piperidine derivatives, their preparation and use in therapy
01/07/1998EP0542795B1 Tnf inhibitors
01/07/1998CN1169730A Aromatic heterocyclic derivatives as enzyme inhibitors
01/07/1998CN1169723A Sulfamidyl (thio) carbonyl-1,2,4-triazolineone derivative and preparation method and application as weed killer
01/07/1998CN1169426A Novel pyridajinone derivatives
01/07/1998CN1036920C Heterocycle-containing carbonic acid derivatives
01/06/1998US5705647 Intermediates for making HIV-protease inhibitors
01/06/1998US5705646 Substituted pyrazoles as CRF antagonists
01/06/1998US5705523 Thromboxane a2 synthetase inhibitors
01/06/1998US5705515 Having reduced side effects
01/06/1998US5705512 Modulators of acetylcholine receptors
01/06/1998US5705506 Pharmaceutical compositions of alkylsulphonamides 5HT1 agonists for rectal administration
01/06/1998US5705505 3-piperidinyl-alkyl-2h-isoquinolin-1-(thi)one derivatives; neurokinin antagonists
01/06/1998US5705502 Pharmacologically active pyrimidineamine derivatives and processes for the preparation thereof
01/06/1998US5705453 Indazole compounds and the use thereof
01/02/1998DE19625263A1 Substituierte N-(4-Pyridyl)-thioamide Substituted N- (4-pyridyl) thioamides
12/1997
12/31/1997WO1997049704A1 N-[4-(heteroarylmethyl)phenyl]-heteroarylamines
12/31/1997WO1997049700A1 Derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one and their use as farnesyl protein transferase inhibitors
12/31/1997WO1997049699A1 Piperidine acetic acid derivatives and their use in the treatment of thrombotic disorders
12/31/1997WO1997049698A1 Piperidine acetic acid derivatives and their use in the treatment of thrombotic disorders
12/31/1997WO1997049697A1 Pyridylaminopyrimidines as fungicides
12/31/1997WO1997049696A1 Pyridylaminopyrimidines as fungicides
12/31/1997WO1997049695A1 Sulfonamide derivatives as 5ht7 receptor antagonists
12/31/1997WO1997049690A1 A method for treating meniere's disease
12/31/1997WO1997049683A1 Substituted n-(4-pyridyl)-thioamides with pesticide activity
12/31/1997WO1997049682A1 Fibrinogen receptor antagonists and medicinal preparations containing the same as the active ingredient
12/31/1997WO1997049404A1 Anticoagulant agents
12/31/1997WO1997049395A1 Substituted 3,5-diphenyl-1,2,4-triazoles and their use as pharmaceutical metal chelators
12/31/1997CN1168886A Process for production of amidinobenzofuran and amidionbenzothiophen derivatives and salt thereof
12/31/1997CN1168885A Process for prodn. of amidinoindole derivatives and salts thereof
12/31/1997CN1036849C Method for prepn. of anti-viral compounds
12/31/1997CA2259222A1 Derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one and their use as farnesyl protein transferase inhibitors
12/31/1997CA2258915A1 Anticoagulant agents
12/31/1997CA2258753A1 Piperidine acetic acid derivatives and their use in the treatment of thrombotic disorders
12/30/1997US5703243 Intermediates for pyrrolidylthiocarbapenem derivative
12/30/1997US5703240 Analgesics; antiinflammatory agents; nervous system disorders; psychological disorders; gastrointestinal disorders
12/30/1997US5703239 Indanylpiperidines as melatonergic agents
12/30/1997US5703231 Process for making antimicrobial compounds
12/30/1997US5703215 Water-soluble dyes which are polymerizable containing molecules which contain a nucleophilic group and an electrophilic group
12/30/1997US5703107 Central nervous system disorders; analgesics; antiepileptic agents
12/30/1997US5703100 Modulators of acetylcholine receptors
12/30/1997US5703099 Treatment of thrombosis, arteriosclerosis, ischemic heart diseases, gastric ulcer or hypertension
12/30/1997US5703098 Inhibitors of cytokines including tumor necrosis factor
12/30/1997US5703097 Antiulcer agents
12/30/1997US5703094 Quinolone- and naphthyridonecarboxylic acid derivatives
12/30/1997US5703092 Hydroxamic acid compounds as metalloprotease and TNF inhibitors
12/30/1997US5703090 Tricyclic compounds useful for inhibition of G-protein function and for treatment of proliferative diseases
12/30/1997US5703087 Phenyl indole compounds
12/30/1997US5703081 Cell adhesion inhibitors
12/30/1997US5703077 Methods for using (2-imidazolin-2-ylamino) quinoxaline derivatives
12/30/1997US5703076 Retroviral protease inhibitors
12/30/1997US5703071 Tropolone derivatives and pharmaceutical composition thereof for preventing and treating ischemic diseases
12/30/1997US5703017 3-(Het) arylcarboxylic acid derivatives, their preparation and intermediates for their preparation
12/30/1997CA2142707C Benzo-fused lactams promote release of growth hormone
12/29/1997EP0814084A1 Indole derivatives as 5-HT1A antagonists and as inhibitors of serotonine reuptake
12/29/1997EP0813868A2 Retroviral protease inhibitors
12/29/1997EP0813867A2 Retroviral protease inhibitors
12/29/1997EP0813525A1 Benzamidine derivatives their preparation and their use as anti-coagulants
12/29/1997EP0813524A1 Indole derivatives as eaa antagonists
12/29/1997EP0813424A1 Oral pharmaceutical dosage forms comprising a proton pump inhibitor and an antacid agent or alginate
12/29/1997EP0719264B1 Imidazolone and oxazolone derivatives as dopamine antagonists
12/26/1997CA2208652A1 Pharmaceutical compounds
12/24/1997WO1997048704A1 Process for preparing imidazoquinolinamines
12/24/1997WO1997048700A1 Indoline derivatives useful as 5-ht-2c receptor antagonists
12/24/1997WO1997048699A1 Indoline derivatives useful as 5-ht-2c receptor antagonists
12/24/1997WO1997048698A1 Compounds having effects on serotonin-related systems
12/24/1997WO1997048697A1 Substituted azabicylic compounds and their use as inhibitors of the production of tnf and cyclic amp phosphodiesterase
12/24/1997WO1997048696A1 Pyridyl alkene- and pyridyl alkine- acid amides as cytostatics and immunosuppressives
12/24/1997WO1997048695A1 New pyridyl alkane acid amides as cytostatics and immunosuppressives
12/24/1997WO1997048694A1 Compounds and methods for providing pharmacologically active preparations and uses thereof
12/24/1997WO1997048685A1 Metalloprotease inhibitors
12/24/1997WO1997048683A1 Substituted benzamide derivatives and their use as anticonvulsants
12/24/1997WO1997048681A1 Sulphonamide derivatives and their use in the treatment of cns disorders
12/24/1997CN1168668A Sulfonylaminocarbonyltriazolinones with substituents bound by oxygen and sulphur
12/24/1997CN1168667A Pyridopyrimidones, quinolines and fused N-heretocycles as bradykinin antagonists
12/24/1997CN1168633A Boronic ester and acid compounds, synthesis and uses
12/24/1997CN1168375A Process for preparation of substituted pyrimidines
12/24/1997CA2258822A1 Compounds and methods for providing pharmacologically active preparations and uses thereof