Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979) |
---|
01/07/1998 | EP0816356A1 1-(2-(1-piperidinyl)-1-ethyl)-1,3-dihydro-2H-benzimidazole derivatives and their pharmaceutical use |
01/07/1998 | EP0816355A1 Heterocyclic spiro derivatives |
01/07/1998 | EP0816342A2 Process for producing 1-substituted-hydantoins |
01/07/1998 | EP0816341A1 Process for the preparation of chiral succinic acid derivatives |
01/07/1998 | EP0816338A1 3-(bis-substituted-phenylmethylene)oxindole derivatives |
01/07/1998 | EP0815859A1 Intimal thickening inhibitors |
01/07/1998 | EP0815856A2 Retroviral protease inhibitors |
01/07/1998 | EP0815120A1 17-difluoromethylene-oestratrienes |
01/07/1998 | EP0815108A1 Cyclic urea hiv protease inhibitors |
01/07/1998 | EP0815104A1 3-benzylamino-2-phenylpiperidines as neurokinin antagonists |
01/07/1998 | EP0815103A1 Trypsin and thrombin inhibitors |
01/07/1998 | EP0815102A1 REDUCTIVE ALKYLATION PROCESS FOR THE PREPARATION N-(2-(R)-HYDROXY-1-(S)-INDANYL)-2(R)-PHENYLMETHYL-4(S)-HYDROXY-5-(1-(4-(3-PYRIDYLMETHYL)-2(S)-N'-(t-BUTYLCARBOXAMIDO)-PIPERAZINYL))-PENTANEAMIDE (=COMPOUND J OR L-735,524) |
01/07/1998 | EP0815101A1 PROCESS TO MAKE HIV PROTEASE INHIBITOR FROM 2(S)-4-PICOLYL-2-PIPERAZINE-t-BUTYLCARBOXAMIDE |
01/07/1998 | EP0815100A1 Tricyclic amide and urea compounds useful for inhibition of g-protein function and for treatment of proliferative diseases |
01/07/1998 | EP0815099A1 Tricyclic amide and urea compounds useful for inhibition of g-protein function and for treatment of proliferative diseases |
01/07/1998 | EP0815089A1 Biphenyl-substituted triazines as light stabilizer |
01/07/1998 | EP0815080A1 Di-substituted 1,4-piperidine esters and amides having 5-ht 4? antagonistic activity |
01/07/1998 | EP0814840A1 Oral pharmaceutical dosage forms comprising a proton pump inhibitor and a prokinetic agent |
01/07/1998 | EP0814839A1 Oral pharmaceutical dosage forms comprising a proton pump inhibitor and a nsaid |
01/07/1998 | EP0814807A1 Tricyclic compounds useful for inhibition of g-protein function and for treatment of proliferative diseases |
01/07/1998 | EP0690846B1 Herbicidal heterocyclic-substituted pyridines |
01/07/1998 | EP0613458B1 Acyclic ethylenediamine derivatives as substance p receptor antagonists |
01/07/1998 | EP0565396B1 1-[2-(arylsulfonylamino)-1-oxoethyl]piperidine derivatives, their preparation and use in therapy |
01/07/1998 | EP0542795B1 Tnf inhibitors |
01/07/1998 | CN1169730A Aromatic heterocyclic derivatives as enzyme inhibitors |
01/07/1998 | CN1169723A Sulfamidyl (thio) carbonyl-1,2,4-triazolineone derivative and preparation method and application as weed killer |
01/07/1998 | CN1169426A Novel pyridajinone derivatives |
01/07/1998 | CN1036920C Heterocycle-containing carbonic acid derivatives |
01/06/1998 | US5705647 Intermediates for making HIV-protease inhibitors |
01/06/1998 | US5705646 Substituted pyrazoles as CRF antagonists |
01/06/1998 | US5705523 Thromboxane a2 synthetase inhibitors |
01/06/1998 | US5705515 Having reduced side effects |
01/06/1998 | US5705512 Modulators of acetylcholine receptors |
01/06/1998 | US5705506 Pharmaceutical compositions of alkylsulphonamides 5HT1 agonists for rectal administration |
01/06/1998 | US5705505 3-piperidinyl-alkyl-2h-isoquinolin-1-(thi)one derivatives; neurokinin antagonists |
01/06/1998 | US5705502 Pharmacologically active pyrimidineamine derivatives and processes for the preparation thereof |
01/06/1998 | US5705453 Indazole compounds and the use thereof |
01/02/1998 | DE19625263A1 Substituierte N-(4-Pyridyl)-thioamide Substituted N- (4-pyridyl) thioamides |
12/31/1997 | WO1997049704A1 N-[4-(heteroarylmethyl)phenyl]-heteroarylamines |
12/31/1997 | WO1997049700A1 Derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one and their use as farnesyl protein transferase inhibitors |
12/31/1997 | WO1997049699A1 Piperidine acetic acid derivatives and their use in the treatment of thrombotic disorders |
12/31/1997 | WO1997049698A1 Piperidine acetic acid derivatives and their use in the treatment of thrombotic disorders |
12/31/1997 | WO1997049697A1 Pyridylaminopyrimidines as fungicides |
12/31/1997 | WO1997049696A1 Pyridylaminopyrimidines as fungicides |
12/31/1997 | WO1997049695A1 Sulfonamide derivatives as 5ht7 receptor antagonists |
12/31/1997 | WO1997049690A1 A method for treating meniere's disease |
12/31/1997 | WO1997049683A1 Substituted n-(4-pyridyl)-thioamides with pesticide activity |
12/31/1997 | WO1997049682A1 Fibrinogen receptor antagonists and medicinal preparations containing the same as the active ingredient |
12/31/1997 | WO1997049404A1 Anticoagulant agents |
12/31/1997 | WO1997049395A1 Substituted 3,5-diphenyl-1,2,4-triazoles and their use as pharmaceutical metal chelators |
12/31/1997 | CN1168886A Process for production of amidinobenzofuran and amidionbenzothiophen derivatives and salt thereof |
12/31/1997 | CN1168885A Process for prodn. of amidinoindole derivatives and salts thereof |
12/31/1997 | CN1036849C Method for prepn. of anti-viral compounds |
12/31/1997 | CA2259222A1 Derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one and their use as farnesyl protein transferase inhibitors |
12/31/1997 | CA2258915A1 Anticoagulant agents |
12/31/1997 | CA2258753A1 Piperidine acetic acid derivatives and their use in the treatment of thrombotic disorders |
12/30/1997 | US5703243 Intermediates for pyrrolidylthiocarbapenem derivative |
12/30/1997 | US5703240 Analgesics; antiinflammatory agents; nervous system disorders; psychological disorders; gastrointestinal disorders |
12/30/1997 | US5703239 Indanylpiperidines as melatonergic agents |
12/30/1997 | US5703231 Process for making antimicrobial compounds |
12/30/1997 | US5703215 Water-soluble dyes which are polymerizable containing molecules which contain a nucleophilic group and an electrophilic group |
12/30/1997 | US5703107 Central nervous system disorders; analgesics; antiepileptic agents |
12/30/1997 | US5703100 Modulators of acetylcholine receptors |
12/30/1997 | US5703099 Treatment of thrombosis, arteriosclerosis, ischemic heart diseases, gastric ulcer or hypertension |
12/30/1997 | US5703098 Inhibitors of cytokines including tumor necrosis factor |
12/30/1997 | US5703097 Antiulcer agents |
12/30/1997 | US5703094 Quinolone- and naphthyridonecarboxylic acid derivatives |
12/30/1997 | US5703092 Hydroxamic acid compounds as metalloprotease and TNF inhibitors |
12/30/1997 | US5703090 Tricyclic compounds useful for inhibition of G-protein function and for treatment of proliferative diseases |
12/30/1997 | US5703087 Phenyl indole compounds |
12/30/1997 | US5703081 Cell adhesion inhibitors |
12/30/1997 | US5703077 Methods for using (2-imidazolin-2-ylamino) quinoxaline derivatives |
12/30/1997 | US5703076 Retroviral protease inhibitors |
12/30/1997 | US5703071 Tropolone derivatives and pharmaceutical composition thereof for preventing and treating ischemic diseases |
12/30/1997 | US5703017 3-(Het) arylcarboxylic acid derivatives, their preparation and intermediates for their preparation |
12/30/1997 | CA2142707C Benzo-fused lactams promote release of growth hormone |
12/29/1997 | EP0814084A1 Indole derivatives as 5-HT1A antagonists and as inhibitors of serotonine reuptake |
12/29/1997 | EP0813868A2 Retroviral protease inhibitors |
12/29/1997 | EP0813867A2 Retroviral protease inhibitors |
12/29/1997 | EP0813525A1 Benzamidine derivatives their preparation and their use as anti-coagulants |
12/29/1997 | EP0813524A1 Indole derivatives as eaa antagonists |
12/29/1997 | EP0813424A1 Oral pharmaceutical dosage forms comprising a proton pump inhibitor and an antacid agent or alginate |
12/29/1997 | EP0719264B1 Imidazolone and oxazolone derivatives as dopamine antagonists |
12/26/1997 | CA2208652A1 Pharmaceutical compounds |
12/24/1997 | WO1997048704A1 Process for preparing imidazoquinolinamines |
12/24/1997 | WO1997048700A1 Indoline derivatives useful as 5-ht-2c receptor antagonists |
12/24/1997 | WO1997048699A1 Indoline derivatives useful as 5-ht-2c receptor antagonists |
12/24/1997 | WO1997048698A1 Compounds having effects on serotonin-related systems |
12/24/1997 | WO1997048697A1 Substituted azabicylic compounds and their use as inhibitors of the production of tnf and cyclic amp phosphodiesterase |
12/24/1997 | WO1997048696A1 Pyridyl alkene- and pyridyl alkine- acid amides as cytostatics and immunosuppressives |
12/24/1997 | WO1997048695A1 New pyridyl alkane acid amides as cytostatics and immunosuppressives |
12/24/1997 | WO1997048694A1 Compounds and methods for providing pharmacologically active preparations and uses thereof |
12/24/1997 | WO1997048685A1 Metalloprotease inhibitors |
12/24/1997 | WO1997048683A1 Substituted benzamide derivatives and their use as anticonvulsants |
12/24/1997 | WO1997048681A1 Sulphonamide derivatives and their use in the treatment of cns disorders |
12/24/1997 | CN1168668A Sulfonylaminocarbonyltriazolinones with substituents bound by oxygen and sulphur |
12/24/1997 | CN1168667A Pyridopyrimidones, quinolines and fused N-heretocycles as bradykinin antagonists |
12/24/1997 | CN1168633A Boronic ester and acid compounds, synthesis and uses |
12/24/1997 | CN1168375A Process for preparation of substituted pyrimidines |
12/24/1997 | CA2258822A1 Compounds and methods for providing pharmacologically active preparations and uses thereof |