Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979) |
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05/02/2001 | CN1293662A Novel sulfonamide derivatives as inhibitors of bone resorption and as inhibitors of cell adhesion |
05/02/2001 | CN1293192A New benzothiophene, benzofuran and indole compounds, preparation method therefor and medicine composition containing same |
05/01/2001 | US6225465 Process for the aminocarbonylation of benzazepines and benzodiazepines |
05/01/2001 | US6225335 3-(4′-bromobenzylindenyl)-2-indolinone and analogues thereof for the treatment of disease |
05/01/2001 | US6225324 Antidepressant heterocyclic compounds |
05/01/2001 | US6225322 4-(6,11-dihydro-5h-cyclohepta(2,1-b:4, 5-b')dipyridin-11-yl)-1-piperidinecarboxylic or sulfonic acid derivatives |
05/01/2001 | US6225318 4-aminoquinazolone derivatives |
05/01/2001 | US6225316 3-phenyl-pyridine-derivatives |
05/01/2001 | US6225312 Piperazine and piperidine compounds |
05/01/2001 | US6225309 Aminoheterocyclic derivatives as antithrombotic or anticoagulant agents |
05/01/2001 | CA2016664C Indole derivative and method of production thereof |
04/29/2001 | CA2324640A1 Method for preparing sodium-hydrogen exchanger type 1 inhibitor |
04/26/2001 | WO2001029245A2 ENZYMATIC PROCESS FOR THE RESOLUTION OF ENANTIOMERIC MIXTURES OF β-LACTAMS |
04/26/2001 | WO2001029030A1 N-substituted 1-(lactone) isoquinolones for treating nervous disorders |
04/26/2001 | WO2001029029A1 Tetrahydrobenzindolone derivatives, their preparation and their use as 5-ht7 receptor antagonists |
04/26/2001 | WO2001029028A1 9- (piperazinylalkyl) carbazoles as bax-modulators |
04/26/2001 | WO2001029026A1 Phenyl- and pyridyl-tetrahydro-pyridines having tnf inhibiting activity |
04/26/2001 | WO2001029025A2 Tyrosine kinase inhibitors |
04/26/2001 | WO2001029021A1 Neuraminidase inhibitors |
04/26/2001 | WO2001029012A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists |
04/26/2001 | WO2001029011A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists |
04/26/2001 | WO2001029009A1 4,5-disubstituted-2-aminopyrimidines |
04/26/2001 | WO2001029005A1 Bicyclic vasopressin agonists |
04/26/2001 | WO2001028996A2 Pyrrolidine derivatives, their preparation and their use as inhibitors of neuraminidases |
04/26/2001 | WO2001028993A2 Tyrosine kinase inhibitors |
04/26/2001 | WO2001028987A1 Benzylcycloalkyl amines as modulators of chemokine receptor activity |
04/26/2001 | WO2001028559A1 Method for stabilizing benzimidazole compounds |
04/26/2001 | WO2001028557A1 Cannabimimetic indole derivatives |
04/26/2001 | WO2000055139A3 Heterocyclic urea and related compounds useful as anti-inflammatory agents |
04/26/2001 | WO2000055125A3 N-cyanomethyl amides as protease inhibitors |
04/26/2001 | DE19932621A1 Neue substituerte alpha, beta-anellierte Butyrolactone New substituerte alpha, beta-fused butyrolactones |
04/26/2001 | CA2388859A1 Inhibitors of neuraminidases |
04/26/2001 | CA2388782A1 Method and system for assay and removal of harmful toxins during processing of tobacco products |
04/26/2001 | CA2387972A1 N-substituted 1-(lactone) isoquinolones for treating nervous disorders |
04/26/2001 | CA2387886A1 Bicyclic vasopressin agonists |
04/26/2001 | CA2387840A1 Tyrosine kinase inhibitors |
04/26/2001 | CA2387138A1 Cannabimimetic indole derivatives |
04/26/2001 | CA2387034A1 4,5-disubstituted-2-aminopyrimidines |
04/26/2001 | CA2386487A1 Enzymatic process for the resolution of enantiomeric mixtures of .beta.-lactams |
04/26/2001 | CA2384240A1 Benzylcycloalkyl amines as modulators of chemokine receptor activity |
04/25/2001 | EP1094064A1 5-arylindolederivatives and their use as serotonin(5-ht1)agonists |
04/25/2001 | EP1094063A1 9-(Piperazinylalkyl)carbazoles as Bax-modulators |
04/25/2001 | EP1093372A1 CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING $g(b)-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS |
04/25/2001 | CN1292698A Glycine transport inhibitors |
04/25/2001 | CN1292694A New use |
04/25/2001 | CN1292379A Preparation method of pyrazolzo [4,3-d] pyrimidine-7-ketone-3-pyridyl sulfonyl compound and its intermediate |
04/25/2001 | CN1064965C Novel sulfonamides compound and its use as medicine |
04/24/2001 | US6222039 Reacting lactone compound containing nitrogen heterocycle with cyclic amine; oxidizing to form carboxylic acid group; introducing hydroxylamine group at hydroxyl of carboxylic acid group |
04/24/2001 | US6222037 Reacting 4,6-dimethoxypyrimidin-2-isocyante with 2-sulfonamido-pyridine compound in aprotic solvent to form potassium or sodium n-pyridylsulfonyl-n'-pyrimidinylurea compound |
04/24/2001 | US6222036 Reacting 2-thio-4-dimethyoxymethyl-pyrimidine with acetic acid and catalytic amount of concetrated sulfuric acid to produce 2-thiopyrimidine aldehyde |
04/24/2001 | US6221937 Mixtures; photostability, heat and oxidation resistance; for polymers |
04/24/2001 | US6221886 Thio acid derived monocyclic N-heterocyclics as anticoagulants |
04/24/2001 | US6221884 Carboxamides useful as 5-HT1F agonists |
04/24/2001 | US6221881 Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses |
04/24/2001 | US6221871 Treating schizophrenia, depression or parkinson's disease |
04/24/2001 | US6221865 Inhibitors of protein farnesyltransferase and protein geranylgeranyltransferase. |
04/24/2001 | CA2220055C Dipeptides which promote release of growth hormone |
04/24/2001 | CA2044310C Piperidine-triazine co-oligomers for use as stabilizers for organic materials |
04/19/2001 | WO2001027113A2 PYRAZOLO `4,3-d! PYRIMIDINE DERIVATIVES |
04/19/2001 | WO2001027108A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF Aβ PROTEIN PRODUCTION |
04/19/2001 | WO2001027107A2 Heterocyclic sodium/proton exchange inhibitors and method |
04/19/2001 | WO2001027106A1 Substituted pyrroles as antiproliferative agents for the treatment of cancer |
04/19/2001 | WO2001027105A1 Pyrimidine-5-carboxamide compounds, process for producing the same and use thereof |
04/19/2001 | WO2001027104A1 Substituted imidazolidinone derivatives |
04/19/2001 | WO2001027103A1 Fab i inhibitors |
04/19/2001 | WO2001027102A1 Substituted diazepanes |
04/19/2001 | WO2001027091A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF Aβ PROTEIN PRODUCTION |
04/19/2001 | WO2001027090A1 m-SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING INTEGRINαvβ3 ANTAGONISM |
04/19/2001 | WO2001027089A1 Pyrimidine derivatives |
04/19/2001 | WO2001027087A2 Process for making boc-protected 3-aminohydantoins/thiohydantoins and 3-aminodihydrouracils/dihydrothiouracils |
04/19/2001 | WO2001027085A1 Nicotinyl aspartyl ketones as inhibitors of caspase-3 |
04/19/2001 | WO2001027084A1 Beta disubstituted metalloprotease inhibitors |
04/19/2001 | WO2001027082A1 3-AMINOPIPERIDINE DERIVATIVES AS INTEGRIN αvβ3 ANTAGONISTS |
04/19/2001 | WO2001027081A1 6-position substituted indoline, production and use thereof as a medicament |
04/19/2001 | WO2001027080A2 5-substituted indolinones and use thereof as kinase and cyclin/cdk complex inhibitors |
04/19/2001 | WO2001026652A1 Fab i inhibitors |
04/19/2001 | WO2000077008A3 Heteroaryl substituted piperidines as gaba brain receptor lingands |
04/19/2001 | WO2000073274A3 Substituted phenylcyclohexane carboxylic acid amides and their use as adenosine uptake inhibitors |
04/19/2001 | WO2000046198A8 Anti-inflammatory indole derivatives |
04/19/2001 | WO2000045894A3 Use of pyrazole carboxamides |
04/19/2001 | WO2000018767A9 2-piperazino alkylamino benzoazole derivatives: dopamine receptor subtype specific ligands |
04/19/2001 | WO1999032448A8 Substituted pyridine and pyridazine compounds and their pharmaceutical use |
04/19/2001 | DE19949209A1 In 5-Stellung substituierte Indolinone, ihre Herstellung und ihre Verwendung als Arzneimittel In the 5-position substituted indolinones, their preparation and their use as medicaments |
04/19/2001 | DE19948417A1 Imidazol-Derivate und ihre Verwendung als Arzneimittel Imidazole derivatives and their use as medicaments |
04/19/2001 | CA2392209A1 M-substituted benzoic acid derivatives having integrin .alpha.v.beta.3 antagonistic activity |
04/19/2001 | CA2388813A1 Heterocyclic sodium/proton exchange inhibitors and method |
04/19/2001 | CA2387535A1 Substituted imidazolidinone derivatives |
04/19/2001 | CA2387493A1 Amino lactam sulfonamides as inhibitors of a.beta. protein production |
04/19/2001 | CA2386821A1 3-aminopiperidine derivatives as integrin .alpha.v.beta.3 antagonists |
04/19/2001 | CA2386485A1 Beta disubstituted metalloprotease inhibitors |
04/19/2001 | CA2386411A1 Nicotinyl aspartyl ketones as inhibitors of caspase-3 |
04/19/2001 | CA2385071A1 Substituted pyrroles as antiproliferative agents for the treatment of cancer |
04/19/2001 | CA2384544A1 Amino lactam sulfonamides as inhibitors of a.beta. protein production |
04/19/2001 | CA2382605A1 Pyrimidine derivatives |
04/18/2001 | EP1092720A2 Process for the preparation of pyrazolo [4,3-d] pyrimidin-7-ones-3-pyridylsulphonyl compounds and intermediates thereof |
04/18/2001 | EP1092718A1 2-(2-Alkoxy-5-heterocyclylsulphonylphenyl)purin-6-ones as phosphodiesterase inhibitors |
04/18/2001 | EP1092716A2 Derivatives of benzothiophenes, benzofurans and indoles, method for their preparation and pharmaceutical compositions containing them |
04/18/2001 | EP1092715A2 Cyano-indole derivatives as inhibitors of serotonin reuptake, method for their preparation and pharmaceutical compositions containing the same |
04/18/2001 | EP1091960A1 Bifunctional antagonists of cytokine-sensitive protein kinase activation cascades and methods for use as anti-inflammatory agents |
04/18/2001 | EP1091957A1 Pyrimidin-aminomethyl-pyridine derivatives, their preparation and their use in the control of helicobacter bacteria |