Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
05/2001
05/02/2001CN1293662A Novel sulfonamide derivatives as inhibitors of bone resorption and as inhibitors of cell adhesion
05/02/2001CN1293192A New benzothiophene, benzofuran and indole compounds, preparation method therefor and medicine composition containing same
05/01/2001US6225465 Process for the aminocarbonylation of benzazepines and benzodiazepines
05/01/2001US6225335 3-(4′-bromobenzylindenyl)-2-indolinone and analogues thereof for the treatment of disease
05/01/2001US6225324 Antidepressant heterocyclic compounds
05/01/2001US6225322 4-(6,11-dihydro-5h-cyclohepta(2,1-b:4, 5-b')dipyridin-11-yl)-1-piperidinecarboxylic or sulfonic acid derivatives
05/01/2001US6225318 4-aminoquinazolone derivatives
05/01/2001US6225316 3-phenyl-pyridine-derivatives
05/01/2001US6225312 Piperazine and piperidine compounds
05/01/2001US6225309 Aminoheterocyclic derivatives as antithrombotic or anticoagulant agents
05/01/2001CA2016664C Indole derivative and method of production thereof
04/2001
04/29/2001CA2324640A1 Method for preparing sodium-hydrogen exchanger type 1 inhibitor
04/26/2001WO2001029245A2 ENZYMATIC PROCESS FOR THE RESOLUTION OF ENANTIOMERIC MIXTURES OF β-LACTAMS
04/26/2001WO2001029030A1 N-substituted 1-(lactone) isoquinolones for treating nervous disorders
04/26/2001WO2001029029A1 Tetrahydrobenzindolone derivatives, their preparation and their use as 5-ht7 receptor antagonists
04/26/2001WO2001029028A1 9- (piperazinylalkyl) carbazoles as bax-modulators
04/26/2001WO2001029026A1 Phenyl- and pyridyl-tetrahydro-pyridines having tnf inhibiting activity
04/26/2001WO2001029025A2 Tyrosine kinase inhibitors
04/26/2001WO2001029021A1 Neuraminidase inhibitors
04/26/2001WO2001029012A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
04/26/2001WO2001029011A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
04/26/2001WO2001029009A1 4,5-disubstituted-2-aminopyrimidines
04/26/2001WO2001029005A1 Bicyclic vasopressin agonists
04/26/2001WO2001028996A2 Pyrrolidine derivatives, their preparation and their use as inhibitors of neuraminidases
04/26/2001WO2001028993A2 Tyrosine kinase inhibitors
04/26/2001WO2001028987A1 Benzylcycloalkyl amines as modulators of chemokine receptor activity
04/26/2001WO2001028559A1 Method for stabilizing benzimidazole compounds
04/26/2001WO2001028557A1 Cannabimimetic indole derivatives
04/26/2001WO2000055139A3 Heterocyclic urea and related compounds useful as anti-inflammatory agents
04/26/2001WO2000055125A3 N-cyanomethyl amides as protease inhibitors
04/26/2001DE19932621A1 Neue substituerte alpha, beta-anellierte Butyrolactone New substituerte alpha, beta-fused butyrolactones
04/26/2001CA2388859A1 Inhibitors of neuraminidases
04/26/2001CA2388782A1 Method and system for assay and removal of harmful toxins during processing of tobacco products
04/26/2001CA2387972A1 N-substituted 1-(lactone) isoquinolones for treating nervous disorders
04/26/2001CA2387886A1 Bicyclic vasopressin agonists
04/26/2001CA2387840A1 Tyrosine kinase inhibitors
04/26/2001CA2387138A1 Cannabimimetic indole derivatives
04/26/2001CA2387034A1 4,5-disubstituted-2-aminopyrimidines
04/26/2001CA2386487A1 Enzymatic process for the resolution of enantiomeric mixtures of .beta.-lactams
04/26/2001CA2384240A1 Benzylcycloalkyl amines as modulators of chemokine receptor activity
04/25/2001EP1094064A1 5-arylindolederivatives and their use as serotonin(5-ht1)agonists
04/25/2001EP1094063A1 9-(Piperazinylalkyl)carbazoles as Bax-modulators
04/25/2001EP1093372A1 CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING $g(b)-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS
04/25/2001CN1292698A Glycine transport inhibitors
04/25/2001CN1292694A New use
04/25/2001CN1292379A Preparation method of pyrazolzo [4,3-d] pyrimidine-7-ketone-3-pyridyl sulfonyl compound and its intermediate
04/25/2001CN1064965C Novel sulfonamides compound and its use as medicine
04/24/2001US6222039 Reacting lactone compound containing nitrogen heterocycle with cyclic amine; oxidizing to form carboxylic acid group; introducing hydroxylamine group at hydroxyl of carboxylic acid group
04/24/2001US6222037 Reacting 4,6-dimethoxypyrimidin-2-isocyante with 2-sulfonamido-pyridine compound in aprotic solvent to form potassium or sodium n-pyridylsulfonyl-n'-pyrimidinylurea compound
04/24/2001US6222036 Reacting 2-thio-4-dimethyoxymethyl-pyrimidine with acetic acid and catalytic amount of concetrated sulfuric acid to produce 2-thiopyrimidine aldehyde
04/24/2001US6221937 Mixtures; photostability, heat and oxidation resistance; for polymers
04/24/2001US6221886 Thio acid derived monocyclic N-heterocyclics as anticoagulants
04/24/2001US6221884 Carboxamides useful as 5-HT1F agonists
04/24/2001US6221881 Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
04/24/2001US6221871 Treating schizophrenia, depression or parkinson's disease
04/24/2001US6221865 Inhibitors of protein farnesyltransferase and protein geranylgeranyltransferase.
04/24/2001CA2220055C Dipeptides which promote release of growth hormone
04/24/2001CA2044310C Piperidine-triazine co-oligomers for use as stabilizers for organic materials
04/19/2001WO2001027113A2 PYRAZOLO `4,3-d! PYRIMIDINE DERIVATIVES
04/19/2001WO2001027108A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF Aβ PROTEIN PRODUCTION
04/19/2001WO2001027107A2 Heterocyclic sodium/proton exchange inhibitors and method
04/19/2001WO2001027106A1 Substituted pyrroles as antiproliferative agents for the treatment of cancer
04/19/2001WO2001027105A1 Pyrimidine-5-carboxamide compounds, process for producing the same and use thereof
04/19/2001WO2001027104A1 Substituted imidazolidinone derivatives
04/19/2001WO2001027103A1 Fab i inhibitors
04/19/2001WO2001027102A1 Substituted diazepanes
04/19/2001WO2001027091A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF Aβ PROTEIN PRODUCTION
04/19/2001WO2001027090A1 m-SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING INTEGRINαvβ3 ANTAGONISM
04/19/2001WO2001027089A1 Pyrimidine derivatives
04/19/2001WO2001027087A2 Process for making boc-protected 3-aminohydantoins/thiohydantoins and 3-aminodihydrouracils/dihydrothiouracils
04/19/2001WO2001027085A1 Nicotinyl aspartyl ketones as inhibitors of caspase-3
04/19/2001WO2001027084A1 Beta disubstituted metalloprotease inhibitors
04/19/2001WO2001027082A1 3-AMINOPIPERIDINE DERIVATIVES AS INTEGRIN αvβ3 ANTAGONISTS
04/19/2001WO2001027081A1 6-position substituted indoline, production and use thereof as a medicament
04/19/2001WO2001027080A2 5-substituted indolinones and use thereof as kinase and cyclin/cdk complex inhibitors
04/19/2001WO2001026652A1 Fab i inhibitors
04/19/2001WO2000077008A3 Heteroaryl substituted piperidines as gaba brain receptor lingands
04/19/2001WO2000073274A3 Substituted phenylcyclohexane carboxylic acid amides and their use as adenosine uptake inhibitors
04/19/2001WO2000046198A8 Anti-inflammatory indole derivatives
04/19/2001WO2000045894A3 Use of pyrazole carboxamides
04/19/2001WO2000018767A9 2-piperazino alkylamino benzoazole derivatives: dopamine receptor subtype specific ligands
04/19/2001WO1999032448A8 Substituted pyridine and pyridazine compounds and their pharmaceutical use
04/19/2001DE19949209A1 In 5-Stellung substituierte Indolinone, ihre Herstellung und ihre Verwendung als Arzneimittel In the 5-position substituted indolinones, their preparation and their use as medicaments
04/19/2001DE19948417A1 Imidazol-Derivate und ihre Verwendung als Arzneimittel Imidazole derivatives and their use as medicaments
04/19/2001CA2392209A1 M-substituted benzoic acid derivatives having integrin .alpha.v.beta.3 antagonistic activity
04/19/2001CA2388813A1 Heterocyclic sodium/proton exchange inhibitors and method
04/19/2001CA2387535A1 Substituted imidazolidinone derivatives
04/19/2001CA2387493A1 Amino lactam sulfonamides as inhibitors of a.beta. protein production
04/19/2001CA2386821A1 3-aminopiperidine derivatives as integrin .alpha.v.beta.3 antagonists
04/19/2001CA2386485A1 Beta disubstituted metalloprotease inhibitors
04/19/2001CA2386411A1 Nicotinyl aspartyl ketones as inhibitors of caspase-3
04/19/2001CA2385071A1 Substituted pyrroles as antiproliferative agents for the treatment of cancer
04/19/2001CA2384544A1 Amino lactam sulfonamides as inhibitors of a.beta. protein production
04/19/2001CA2382605A1 Pyrimidine derivatives
04/18/2001EP1092720A2 Process for the preparation of pyrazolo [4,3-d] pyrimidin-7-ones-3-pyridylsulphonyl compounds and intermediates thereof
04/18/2001EP1092718A1 2-(2-Alkoxy-5-heterocyclylsulphonylphenyl)purin-6-ones as phosphodiesterase inhibitors
04/18/2001EP1092716A2 Derivatives of benzothiophenes, benzofurans and indoles, method for their preparation and pharmaceutical compositions containing them
04/18/2001EP1092715A2 Cyano-indole derivatives as inhibitors of serotonin reuptake, method for their preparation and pharmaceutical compositions containing the same
04/18/2001EP1091960A1 Bifunctional antagonists of cytokine-sensitive protein kinase activation cascades and methods for use as anti-inflammatory agents
04/18/2001EP1091957A1 Pyrimidin-aminomethyl-pyridine derivatives, their preparation and their use in the control of helicobacter bacteria