Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
08/2001
08/16/2001EP1123274A1 Substituted phenyl derivatives, their preparation and use
08/16/2001EP1123272A1 (substituted)acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
08/16/2001EP0944388A4 Inhibitors of farnesyl-protein transferase
08/16/2001EP0684820B1 Biologically active 3-substituted oxindole derivatives useful as anti-angiogenic agents
08/16/2001EP0677050B1 Novel pyridone carboxylic acid derivatives
08/16/2001DE10006297A1 Substituierte Benzimidazole Substituted benzimidazoles
08/16/2001DE10006139A1 Indol-3-yl-Derivate Indol-3-yl derivatives
08/16/2001CA2399791A1 Cannabinoid receptor modulators, their processes of preparation, and use of cannabinoid receptor modulators in treating respiratory and non-respiratory diseases
08/16/2001CA2398822A1 Piperazine and piperidine derivatives
08/16/2001CA2397993A1 Dehydroamino acids
08/15/2001CN1308631A Heterocyclic derivatives which inhibit factor xa
08/15/2001CN1308628A Method for preparing 4-(3-pyridinyl)-1H-imidazole and the inter medicates used
08/15/2001CN1308617A Antiviral macrocyclic compounds
08/15/2001CN1308616A Non-peptidyl inhibitors and VLA-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory disease
08/15/2001CN1308614A Benzimidazoles, production thereof and use thereof medicaments
08/15/2001CN1308606A Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use pharmaceutical preparations comprising them
08/15/2001CN1308536A Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
08/15/2001CN1308535A Farnesyl protein transferase inhibitors for treating arthropathies
08/15/2001CN1308066A Preparation of chiral succinic acid derivative
08/15/2001CN1308065A 2-[(dihydro)pyrazole-3'-oxymethylene] aniline amide and its preparation and use
08/15/2001CN1069638C Azolyl oxybenzyl alkoxyachrylic acdid esters, prepn. method and use thereof
08/14/2001US6274610 Applying compounds such as 2-(1-chloro-cyclopropyl)-1-(2-chlorophenyl)-3-(5-(n-methyl-car bamoylthio)-1,2,4-triazol-1-yl)-propanol-2-ol to crops to prevent the growth of undesirable microorganisms
08/14/2001US6274607 N-linked ureas and carbamates of heterocyclic thioesters
08/14/2001US6274602 Administering compostitions such as 3,3-dimethyl-1-((2s)-2-(5-(3-pyridyl) pentanoyl)-1-pyrrolidine)-1, 2-pentanedione to treat alopecia or promoting hair growth in animals
08/14/2001US6274598 Methods for treating antibiotic-resistant infections
08/14/2001US6274595 Compositions for treating infection using optically pure (S)-lomefloxacin
08/14/2001US6274594 Isoquinoline derivatives and their therapeutical use
08/14/2001US6274593 Treating psychological disorders, schizophrenia, and parkinson*s disease
08/14/2001US6274588 4-phenyl-pyrimidine derivatives
08/14/2001US6274585 Benign prostatic hyperplasia treatment
08/14/2001US6274577 Autoimmune diseases; antiinflammatory agents
08/14/2001US6274536 Pyrazole derivatives as herbicides
08/14/2001US6274336 Producing three-dimensional structure of active site using computer program, displaying and superimposing three-dimensional representation of test compound onto active site, preparing test compound, and testing in biological assay
08/14/2001US6274173 Oral pharmaceutical composition with delayed release of active ingredient for pantoprazole
08/14/2001CA2226406C Novel pyridone carboxylic acid derivatives
08/14/2001CA2148380C 5-arylindole derivatives
08/09/2001WO2001057037A1 Platelet adp receptor inhibitors
08/09/2001WO2001057036A1 Nicotinamide benzofused-heterocyclyl derivatives useful as selective inhibitors of pde4 isozymes
08/09/2001WO2001057025A1 Pyrimidine carboxamides useful as inhibitors of pde4 isozymes
08/09/2001WO2001057024A1 Blockade of voltage dependent sodium channels
08/09/2001WO2001057023A1 Heterocyclic amide derivatives
08/09/2001WO2001057022A2 Pyrazole compositions useful as inhibitors of erk
08/09/2001WO2001057021A2 2-[1H]-QUINOLONE AND 2-[1H]-QUINOXALONE INHIBITORS OF FACTOR Xa
08/09/2001WO2001057019A1 INDALONE AND BENZIMIDAZOLONE INHIBITORS OF FACTOR Xa
08/09/2001WO2001056996A1 Hydantoin c-proteinase inhibitors
08/09/2001WO2001056995A1 Substituted imidazoles as selective modulators of bradykinin b2 receptors
08/09/2001WO2001056993A2 Pyrazole compositions useful as inhibitors of erk
08/09/2001WO2001056989A2 Inhibitors of factor xa
08/09/2001WO2001056988A1 Nitrogen-containing compounds having kinase inhibitory activity and drugs containing the same
08/09/2001WO2001056974A2 Inha inhibitors and their use as antibacterials
08/09/2001WO2001056607A1 Integrin expression inhibitors
08/09/2001WO2001056571A1 Treating allergic and inflammatory conditions
08/09/2001WO2001056564A1 C10 heterosubstituted acetate taxanes as antitumor agents
08/09/2001WO2001056552A2 Farnesyl protein transferase inhibitors for treating breast cancer
08/09/2001WO2001056358A2 Enhanced propertied pesticides
08/09/2001WO2001019788A3 BENZAMIDES AND RELATED INHIBITORS OF FACTOR Xa
08/09/2001WO2001010834A9 Antibacterial agents
08/09/2001WO2000071511A3 INHIBITORS OF FACTOR Xa
08/09/2001WO2000047554A3 INHIBITORS OF FACTOR Xa
08/09/2001US20010012846 A diagnostic tool for assessing the degree to which neurokinin-2 and neurokinin-3 receptor activity(normal, over or underactivity) is implicated in a patient's symptoms
08/09/2001US20010012842 Lomefloxacin, or a pharmaceutically acceptable salt free of its (R)-stereoismomer is useful for treating infections, but insufficient to cause adverse effect associated with administration of racemic lomefloxacin
08/09/2001DE10005150A1 Verfahren zur Herstellung von 5-Arylnicotinaldehyden A process for the preparation of 5-Arylnicotinaldehyden
08/09/2001CA2399214A1 Novel heterocyclic amide derivatives
08/09/2001CA2398261A1 Treating allergic and inflammatory conditions
08/09/2001CA2369076A1 Pyrazole compositions useful as inhibitors of erk
08/09/2001CA2368502A1 C10 heterosubstituted acetate taxanes as antitumor agents
08/08/2001EP1122257A1 Benzimidazole compounds as ORL1-receptor agonists
08/08/2001EP1122254A2 4-Sulfonamide piperidine derivatives, method for their preparation and phamaceutical compositions containing them
08/08/2001EP1122253A1 Quinazolinone derivatives
08/08/2001EP1122252A1 Nitrogenous fused heterocycle compounds, process for the preparation thereof and agents containing the same
08/08/2001EP1122244A1 Uracil compounds and their use
08/08/2001EP1122243A1 Novel imidazoles with anti-inflammatory activity
08/08/2001EP1121357A1 2-hetaryl-3,4-dihydro-2h-pyrrole derivatives
08/08/2001EP1121356A1 3-tetrahydropyridin-4-yl indoles for treatment of psychotic disorders
08/08/2001EP1121355A1 Quinoline derivatives and their use as antibacterial agents
08/08/2001EP1121354A1 N-(imidazolylalkyl)substituted cyclic amines as histamine-h 3? agonists or antagonists
08/08/2001EP1121353A1 Benzazine derivatives as phosphodiesterase 4 inhibitors
08/08/2001EP1121342A1 Diaminopropionic acid derivatives
08/08/2001EP1121108A2 Novel therapeutic use of compounds with beta-3-agonist activity
08/08/2001CN1307576A Serotongergic agents
08/08/2001CN1307575A New hydroxyindoles, their use as phosphodiesterase 4 inhibitors and method for producing same
08/08/2001CN1307574A Indolyl derivatives as serotonergic agents
08/08/2001CN1307573A Indolyl derivatives and serotonergic agents
08/08/2001CN1307565A Quinolones used as MRS inhibitor and bactericides
08/08/2001CN1307564A Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them
08/08/2001CN1307560A Amidino and guanidino beta-azetidinone tryptase inhibitors
08/08/2001CN1069316C Substituted 5-ring heterocycles, their preparation and use
08/08/2001CN1069314C 2-oxoindoline derivative
08/08/2001CN1069167C Insecticide for preserving technical materials
08/07/2001US6271416 O-(hydrocarbonoxyacetamido)benzoic acid derivatives as intermediates
08/07/2001US6271390 Suppression of the IgE-dependent allergic response by benzimidazole analogs
08/07/2001US6271378 Process for preparing tricyclic compounds having antihistaminic activity
08/07/2001US6271373 Compounds, compositions and methods for treating influenza
08/07/2001US6271372 Process for the preparation of arylamides of heteroaromatic carboxylic acids
08/07/2001US6271342 Sugar-modified cytostatics
08/07/2001US6271253 Cyclooxygenase inhibitors
08/07/2001US6271247 Binding to neuropeptide receptors
08/07/2001US6271244 N-linked urea or carbamate of heterocyclic thioester hair growth compositions and uses
08/07/2001US6271238 Useful in treating and preventing diseases involving chymotrypsin type proteases which are related to asthma, allergy, inflammations, rheumatism, hypertension, heart failure, myocardial infarction, and cardiac hypertrophy
08/07/2001US6271237 Nitrogen containing heteromatics with ortho-substituted P1s as factor Xa inhabitors