Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979) |
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10/28/2003 | CA2249786C Difluoro statone analogs |
10/28/2003 | CA2104268C Preparation of imidazoles |
10/25/2003 | CA2383390A1 Easily removalbe reagents for the mitsunobu reaction |
10/23/2003 | WO2003087304A2 Tri-substituted heteroaryls and methods of making and using the same |
10/23/2003 | WO2003087098A1 Nitrogen-containing bicyclic heterocycles for use as antibacterials |
10/23/2003 | WO2003087095A1 Quinolinone derivatives |
10/23/2003 | WO2003087092A2 Inhibitors of serine proteases, particularly hepatitis c virus ns3 - ns4 protease |
10/23/2003 | WO2003087090A2 Novel heteroaryl alkylamide derivatives useful as bradykinin receptor modulators |
10/23/2003 | WO2003087089A1 Piperidine derivatives having ccr3 antagonism |
10/23/2003 | WO2003087088A2 (condensed) pyrimidone and (condensed) pyridone compounds, processes for their preparation, and pharmaceutical compositions containing them |
10/23/2003 | WO2003087087A2 Heterocyclic compounds and their use as modulators of p38 map kinase |
10/23/2003 | WO2003087086A2 Substituted indoles |
10/23/2003 | WO2003087085A1 Heterocyclic amide derivatives as cytokine inhibitors |
10/23/2003 | WO2003087067A1 Aryl-alkyne compounds as herbicides |
10/23/2003 | WO2003087066A1 α,β-UNSATURATED HYDROXAMIC ACID DERIVATIVES AND THEIR USE AS HISTONE DEACETYLASE INHIBITORS |
10/23/2003 | WO2003087064A1 Chemical compounds with dual activity, processes for their preparation and pharmaceutical compositions |
10/23/2003 | WO2003087063A1 Imidazolidine compounds as chemokine receptor modulators |
10/23/2003 | WO2003087062A2 4-(heterocyclyl)-benzenesulfoximine compounds for the treatment of inflammation |
10/23/2003 | WO2003087061A1 Pyrazole compounds as anti-inflammatory and analgesic agents |
10/23/2003 | WO2003087060A1 Fredericamycin derivatives |
10/23/2003 | WO2003087057A1 Benzamide derivatives useful as histone deacetylase inhibitors |
10/23/2003 | WO2003087037A1 Substituted aryl amides |
10/23/2003 | WO2003086605A2 Functionalized ionic liquids, and methods of use thereof |
10/23/2003 | WO2003086467A1 Cancer treatment method comprising administering an erb-family inhibitor and a raf and/or ras inhibitor |
10/23/2003 | WO2003086404A1 Fused quinoxaline derivatives as inhibitors of akt activity |
10/23/2003 | WO2003086403A1 Inhibitors of akt activity |
10/23/2003 | WO2003086400A1 N-substituted pyridinone and pyrimidinone derivatives for use as lp-pla2 inhibitors in the treatment of artherosclerosis |
10/23/2003 | WO2003086398A1 Aminocarbonyl substituted pyridines, pyridazines, pyrimidines, pyrazines and triazines having antiangiogenic activity |
10/23/2003 | WO2003086397A1 Medicine for treating cancer |
10/23/2003 | WO2003086394A1 Inhibitors of akt activity |
10/23/2003 | WO2003086390A1 Imidazole compounds as anti-inflammatory and analgesic agents |
10/23/2003 | WO2003086385A1 Derivatives of 1-(oxoaminoacetyl) pentylcarbamate as cathepsin k inhibitors for the treatment of bone loss |
10/23/2003 | WO2003086373A1 Methods for identification of modulators of angiogenesis, compounds discovered thereby, and methods of treatment using the compounds |
10/23/2003 | WO2003086371A2 Use of ep4 receptor ligands in the treatment of il-6 involved diseases |
10/23/2003 | WO2003086318A2 Improved prodrugs of cc-1065 analogs |
10/23/2003 | WO2003086294A2 1h-benzo[f]indazol-5-yl derivatives as selective glucocorticoid receptor modulators |
10/23/2003 | WO2003086287A2 Compounds and methods for inducing apoptosis in proliferating cells |
10/23/2003 | WO2003086279A2 Inhibitors of akt activity |
10/23/2003 | WO2003086275A2 Preperation of desloratatine |
10/23/2003 | WO2003086271A2 Azole derivatives as antifungal agents |
10/23/2003 | WO2003057147A3 Useful aroyl pyrrole heteroaryl methanones and methanols |
10/23/2003 | WO2003051315A3 Heteroaryl substituted triazole modulators of metabotropic glutamate receptor-5 |
10/23/2003 | WO2003027094A3 Substituted 3-pyridyl indoles and indazoles as c17,20 lyase inhibitors |
10/23/2003 | WO2003016248A3 Bicyclic hydroxamates as inhibitors of matrix metalloproteinases and/or tnf-$g(a) converting enzyme (tace) |
10/23/2003 | WO2003007954A3 Sulfonyl aryl hydroxamates and their use as matrix metalloprotease inhibitors |
10/23/2003 | WO2003002064A3 Fused pyrimidine dhfr inhibitors as antibacterials |
10/23/2003 | WO2002042272A8 Substituted polycyclic aryl and heteroaryl pyridines useful for selective inhibition of the coagulation cascade |
10/23/2003 | WO2001079195A9 Pyridine and pyrazine derivatives as thrombin inhibitors |
10/23/2003 | US20030199696 Heterocyclic imines such as 3-(3-quinolyl)-2-propyn-1-ol morpholine carbamate, used as chemical intermediates for antibiotics such as clarithromycin |
10/23/2003 | US20030199689 Heterocyclic nitrogen compounds such as 1-(5-(5-Chlorothiophen -2-yl)-isoxazol-3-ylmethyl)-1H-indole-2-carboxylic acid (1-isopropyl-piperidin-4-yl)-amide, used as anticoagulants for prophylaxis of cardiovascular disorders |
10/23/2003 | US20030199569 Pyrrolidine derivatives |
10/23/2003 | US20030199561 Boronic ester and acid compounds, synthesis and uses |
10/23/2003 | US20030199555 Indoline compounds and to pharmaceutical compositions containing them |
10/23/2003 | US20030199554 2,3-Disubstituted pyridine derivative, process for the preparation thereof, pharmaceutical composition containing the same, and intermediate therefor |
10/23/2003 | US20030199552 Amide derivatives as NMDA receptor antagonists |
10/23/2003 | US20030199549 Novel piperidine based MCH antagonists for treatment of obesity and CNS disorders |
10/23/2003 | US20030199548 Administering quinolinyl-piperidin-4-ylidene-methyl-benzamide derivatives containing one of the ring selected from benzene, pyridine, thienyl, furanyl, imidazolyl and triazolyl for therapy in pain management |
10/23/2003 | US20030199547 Quinolinone derivatives containing imidazole rings is useful as anticarcinogenic agent |
10/23/2003 | US20030199546 6-(((2S)-2-(alkoxycabonyl)-4,4-difluoropyrrolidinyl)methyl)-1, 2, 3.4, 4a, 5, 6, 7, 8, 8a-decahydroisoquinoline-3-carboxylate, or acid derivatives, useful for treating migraine, and dural protein extravasation |
10/23/2003 | US20030199534 Kinase inhibitors |
10/23/2003 | US20030199530 New compounds derived from quinazoline |
10/23/2003 | US20030199526 Pyrimidine-based compounds useful as GSK-3 inhibitors |
10/23/2003 | US20030199522 Such as (2S)-(-)-2-(2-aminoethoxy)-3-(1-phenyl-1H-imidazol-4-yl)propanoic acid for treating thrombosis, atherosclerosis, adhesions, scarring, cancer, fibrosis, inflammation, and conditions which benefit from maintaining brandykinin levels |
10/23/2003 | US20030199519 Prodrugs of CC-1065 analogs |
10/23/2003 | US20030199516 Methods of treating infection by drug resistant bacteria |
10/23/2003 | US20030199513 Cinnoline derivatives and use as medicine |
10/23/2003 | US20030199511 Such as N,N-dimethyl-N-(2-((5-((E)-2-pyridin-4-ylvinyl) pyridin-3-yl)oxy)ethyl)amine |
10/23/2003 | US20030199510 Geometrically restricted 2-indolinone derivatives as modulators of protein kinase activity |
10/23/2003 | US20030199506 An enzyme inhibitor of cysteine proteases, a morpholine-4-carboxyamide 1,3,4-oxadiazole derivatives; for treating arthritis, muscular dystrophy, inflammation, tumor, glomerulonephritis, malaria, periodontal disease |
10/23/2003 | US20030199505 Anticoagulants as inhibitors of factor Xa; treating thrombosis, or aftertreatment following angioplasty and coronary bypass operations |
10/23/2003 | US20030199504 Anticoagulants as inhibitors of factor Xa; treating thrombosis, or aftertreatment following angioplasty and coronary bypass operations |
10/23/2003 | US20030199499 Novel guanidinobenzamides |
10/23/2003 | US20030199498 Novel heterocyclic compounds, their preparation, pharmaceutical compositions containing them and their use in medicine |
10/23/2003 | US20030199491 Quinoline derivatives having vegf inhibiting activity |
10/23/2003 | US20030199482 Anticholesterol agents; a drug mixture for treating hypercholesterolemia comprising an apical sodium co-dependent bile acid transport inhibitor, enzyme inhibitors of a cyclooxygenase-2 |
10/23/2003 | US20030199478 For modulating tyrosine kinase signal transduction in order to regulate, modulate and/or inhibit abnormal cell proliferation |
10/23/2003 | EP1494675A2 Inhibitors of akt activity |
10/23/2003 | CA2485679A1 Compounds and methods for inducing apoptosis in proliferating cells |
10/23/2003 | CA2484261A1 Piperidine derivatives having ccr3 antagonism |
10/23/2003 | CA2482775A1 Fredericamycin derivatives |
10/23/2003 | CA2482382A1 Pyrazole compounds as anti-inflammatory and analgesic agents |
10/23/2003 | CA2481855A1 Novel heteroaryl alkylamide derivatives useful as bradykinin receptor modulators |
10/23/2003 | CA2481532A1 Imidazole compounds as anti-inflammatory and analgesic agents |
10/23/2003 | CA2481387A1 Methods for identification of modulators of angiogenesis, compounds discovered thereby, and methods of treatment using the compounds |
10/23/2003 | CA2481320A1 1h-benzo[f]indazol-5-yl derivatives as selective glucocorticoid receptor modulators |
10/23/2003 | CA2481240A1 Aminocarbonyl substituted pyridines, pyridazines, pyrimidines, pyrazines and triazines having antiangiogenic activity |
10/23/2003 | CA2481202A1 Functionalized ionic liquids, and methods of use thereof |
10/23/2003 | CA2481008A1 Aryl-alkyne compounds as herbicides |
10/23/2003 | CA2480860A1 Tri-substituted heteroaryls and methods of making and using the same |
10/23/2003 | CA2480856A1 Substituted aryl amides |
10/23/2003 | CA2480759A1 Improved prodrugs of cc-1065 analogs |
10/23/2003 | CA2448525A1 Nitrogen-containing bicyclic heterocycles for use as antibacterials |
10/22/2003 | EP1354887A1 Ligands for metals and improved metal-catalyzed processes based thereon |
10/22/2003 | EP1354882A1 Dipeptidyl peptidase iv inhibitor |
10/22/2003 | EP1353916A2 Pyrazole compounds useful as protein kinase inhibitors |
10/22/2003 | EP1353915A2 Therapeutic chroman compounds |
10/22/2003 | EP1353914A2 Therapeutic chromone compounds |
10/22/2003 | EP1353913A2 Therapeutic heterocyclic compounds |
10/22/2003 | EP1353911A1 Antiviral agents |
10/22/2003 | EP1353909A2 8-substituted-2,6-methano-3-benzazocines and 3-substituted morphinanes as opioidreceptor binding agents |