Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
07/2004
07/13/2004US6762194 Quinolinone derivatives
07/13/2004US6762189 5-pyrimidinecarboxamide derivatives and the pharmaceutical compositions containing said derivatives
07/13/2004US6762187 Heterocyclic nitrogen compounds used as enzyme inhibitors for prophylaxis of human immunodeficiency virus(hiv)
07/13/2004US6762186 Use to treat allergy, nasal congestion, inflammatory and central nervous system-related diseases
07/13/2004US6762181 Broad antibacterial activity including drug resistant staphylococcus aureus (mrsa), pneumococcus (prsp) and enterococcus (vre); safely used in conjuction with nonsteroidal antiinflammatory drugs
07/13/2004US6762176 Inhibiting no-synthase enzymes producing nitrogen monoxide and/or trapping reactive forms of oxygen; inhibit lipidic peroxidation
07/13/2004CA2358479C 4-substituted-2-(4-fluorophenylamino)-5,6 dimethylpyrimidine
07/13/2004CA2313106C Tetrazolylalkyl indole compounds as anti-inflammatory and analgesic agents
07/13/2004CA2272690C Process for making 2-amino-2-imidazoline, guanidine, and 2-amino-3,4,5,6-tetrahydropyrimidine derivatives
07/13/2004CA2255333C Quinolinone derivative, method for preparing the same, and anti-allergic agent
07/13/2004CA2244771C Substituted 3-aryl-3-carboxyalkyl glutaramides, method for preparing same, and use thereof
07/09/2004CA2676216A1 Aripiprazole
07/08/2004WO2004056998A1 The gene cluster involved in safracin biosynthesis and its uses for genetic engineering
07/08/2004WO2004056992A1 Three-dimensional structure of lipocalin-type prostaglandin d synthase and utilization of the same
07/08/2004WO2004056815A1 PYRAZOLE-DERIVATIVES AS FACTOR Xa INHIBITORS
07/08/2004WO2004056812A1 4- (pyridin-4-ylamino) -quinazoline derivatives as anti-tumor agents
07/08/2004WO2004056808A1 Novel piperidine derivatives as modulators of chemokine receptor ccr5
07/08/2004WO2004056807A1 Pyrimidine derivatives for the treatment of abnormal cell growth
07/08/2004WO2004056806A1 2-(1h-indazol-6-ylamino)-benzamide compounds as protein kinases inhibitors useful for the treatment of ophtalmic diseases
07/08/2004WO2004056805A1 Substituted 4-(4-piperidin-4-yl-piperazin-1-yl)-azepane derivatives and their use as neurokinin antagonists
07/08/2004WO2004056804A2 Solid states of pantoprazole sodium, processes for preparing them and processes for preparing known pantoprazole sodium hydrates
07/08/2004WO2004056803A1 Process for the preparation of sulphinyl derivatives by oxidation of the corresponding sulfides
07/08/2004WO2004056802A1 Complexes of e-2-methoxy-n-(3-{4-[3-methyl-4-(6-methyl-pyridin-3-yloxy)-phenylamino]-quinazolin-6-yl}-allyl)-acetamide, their method of production, and use
07/08/2004WO2004056801A1 Quinazoline derivatives
07/08/2004WO2004056800A1 Substituted 1-piperidin-4-yl-4-azetidin-3-yl-piperazine derivatives and their use as neurokinin antagonists
07/08/2004WO2004056799A2 Substituted 1-piperidin-4-yl-4-pyrrolidin-3-yl-piperazine derivatives and their use as neurokinin antagonists
07/08/2004WO2004056798A1 Phthalazine derivatives phosphodiesterase 4 inhibitors
07/08/2004WO2004056786A2 Pyrimidine derivates for the treatment of abnormal cell growth
07/08/2004WO2004056784A1 Novel carboxamides, the production and use thereof as medicaments
07/08/2004WO2004056782A1 Pyrazole compounds
07/08/2004WO2004056780A2 Tetrahydroquinoline derivatives
07/08/2004WO2004056779A2 Tetrahydroquinoline derivatives and their use as fsh receptor modulators
07/08/2004WO2004056775A1 Microsomal triglyceride transfer protein inhibitors
07/08/2004WO2004056774A2 Substituted biphenyl-4-carboxylic acid arylamide analogues as capsaicin receptor modulators
07/08/2004WO2004056773A1 Novel piperidine derivatives as modulators of chemokine receptor ccr5
07/08/2004WO2004056772A1 Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use as tachykinin antagonists
07/08/2004WO2004056770A2 Piperidine derivatives useful as ccr5 antagonists
07/08/2004WO2004056766A1 Inhibitors of tace
07/08/2004WO2004056369A1 Benzo ‘ d!azepine derivatives for the treatment of neurological disorders
07/08/2004WO2004056366A1 Phthalazine derivatives as phosphodiesterase 4 inhibitors
07/08/2004WO2004056365A2 Derivatives of aryl-quinazoline/aryl-2amino-phenyl methanone which promote the release of parathyroid hormone
07/08/2004WO2004056364A1 Substituted 1-piperidin-3-yl-4-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists
07/08/2004WO2004056319A2 Substituted n-phenyl sulfonamide bradykinin antagonists
07/08/2004WO2004048352A3 2-cyanopyrrolidines and their analogues as dpp-iv inhibitors
07/08/2004WO2004041755A3 Quinazolinone compounds as calcilytics
07/08/2004WO2004037791B1 Inhibitors of glycogen synthase kinase 3
07/08/2004WO2004037171A3 Mitotic kinesin inhibitors
07/08/2004WO2004029024A3 Radiolabeled neurokinin-1 receptor antagonists
07/08/2004WO2004024682A3 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity.
07/08/2004WO2004012663A3 Hydantoin derivatives as inhibitors of matrix metalloproteinases and/or tnf-alpha converting enzyme
07/08/2004WO2004009017A3 Modulators of the glucocorticoid receptor and method
07/08/2004WO2003106628A3 Benzodiazepine inhibitors of mitochondial f¿1<f¿0? atp hydrolase and methods of inhibiting f¿1?f¿0? atp hydrolase
07/08/2004WO2003103663A3 Substituted pyrrolines as kinase inhibitors
07/08/2004WO2003097598A8 Compound exhibiting pgd 2 receptor antagonism
07/08/2004US20040133011 Useful for therapy of noninsulin-dependent diabetes, hyperglycemia, obesity, insulin resistance, dyslipidemia, hyperlipidemia, hypertension, Metabolic Syndrome
07/08/2004US20040133008 Amide compounds
07/08/2004US20040132993 Antiviral and antimicrobial guanidine or biguanidine derivatives
07/08/2004US20040132809 Cell adhesion inhibitors
07/08/2004US20040132804 1-aminoindane derivatives, e.g., 1-(cyclopentylcarbonylamino)-5-(4-cyclopropyl-2-(phenylsulfonyl)phenylsulfonyl)indane; exhibit anti-inflammatory and immunomodulatory activity
07/08/2004US20040132801 Therapeutic proline derivatives
07/08/2004US20040132800 aminomethyl- or ethyl-substituted indoles, tetrahydrocarbazoles and tetrahydropyrido[1,2-a]indoles
07/08/2004US20040132799 Aminoalkoxyindoles and methods of use
07/08/2004US20040132786 Differential tumor cytotoxicity compounds and compositions
07/08/2004US20040132782 Aspartyl protease inhibitors
07/08/2004US20040132781 Pyrazole compounds useful as protein kinase inhibitors
07/08/2004US20040132779 benzoyl- or pyridinoyl-amimo phenyl- or pyridinylmethylaminocarbonyl compounds, e.g., 4-[(2-acetylamino-2-phenyl-acetylamino)-methyl]-2-methylphenyl-4'-trifluoromethylbiphenyl-2-carboxamide; antiobesity and antiatherosclerosis agents
07/08/2004US20040132774 Especially (2R)-N-(1-(6-aminopyridin-2-ylmethyl)1-methyl-piperdin-4-yl)-2-((1R)-3,3, -difluorocyclopentyl)-2-hydroxy-2-phenylacetamide iodide; treating asthma, chronic obstructive pulmonary disorder and allergic or infectious rhinitis
07/08/2004US20040132772 1-carbonyl-4-carbonylaminotetrahydroquinoline derivatives; especially treating asthma and allergic rhinitis
07/08/2004US20040132758 hyterocyclylaminomethyl- or aminocarbonyl-substituted 9,10-ethanoanthracenes or their aza derivatives; treating obesity, diabetes, inflammatory and immune disorders
07/08/2004US20040132756 incorporating tartaric acid in a solid preparation having a high content of a quinolone compound, particularly sitafloxacin; reduced in fluctuations of oral absorption
07/08/2004US20040132752 cyclic ureas and triazolones; treatment or prevention of excessive weight or obesity, and for treatment of Type II diabetes, arteriosclerosis, high blood pressure, depression, anxiety, anxiety neuroses, and schizophrenia.
07/08/2004US20040132747 Novel heteroaryl derivatives and their use as medicaments
07/08/2004US20040132744 lower gastrointestinal and cardiovascular side effects; use in treatment of respiratory system disorders, as tokolitics and as antiallergics, for eye applications.
07/08/2004US20040132738 e.g., 3-[(5-benzyloxypyridin-2-yl)methylidene]-6-phenylmethylidene piperazine-2,5-dione; treating an angiogenesis-related disease.
07/08/2004US20040132736 17 Beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
07/08/2004US20040132733 Novel quinoxalinone derivatives as bradykinin B1 antagonists
07/08/2004US20040132732 Quinazolinones and derivatives thereof as factor Xa inhibitors
07/08/2004US20040132730 Inhibitors of TGFbeta
07/08/2004US20040132729 Inhibitors of p38
07/08/2004US20040132727 Quinoline and quinazoline derivatives and drugs containing the same
07/08/2004US20040132724 e.g., cis-1-Acetyl-6-ethyl-N-(4-ethylphenyl)-1,2,3,4-tetrahydro-2-methyl-4-quinolinamine; atopic dermatitis, urticaria, various allergies bullous pemphigoid, industrial sensitization, chronic transplant rejection and COPD
07/08/2004US20040132722 Glycoprotein-mediated MDR
07/08/2004US20040132721 Treatment of airway disorders
07/08/2004US20040132718 Monocyclic or bicyclic carbocycles and heterocycles as factor Xa inhibitors
07/08/2004US20040132716 CGRP antagonists
07/08/2004US20040132711 Treatment of Human Immunodeficiency Virus, organ transplant rejection, graft v. host disease, arthritis, rheumatoid arthritis, inflammatory bowel disease, atopic dermatitis, psoriasis, asthma, allergies or multiple sclerosis.
07/08/2004US20040132710 Lactams as tachkinin antagonists
07/08/2004DE10257358A1 Substituierte Pyrrole Substituted pyrroles
07/08/2004CA2511321A1 Pyrazole-derivatives as factor xa inhibitors
07/08/2004CA2511182A1 Phthalazine derivatives as phosphodiesterase 4 inhibitors
07/08/2004CA2510850A1 2-(1h-indazol-6-ylamino)-benzamide compounds as protein kinases inhibitors useful for the treatment of ophthalmic diseases
07/08/2004CA2510849A1 Solid states of pantoprazole sodium, processes for preparing them and processes for preparing known pantoprazole sodium hydrates
07/08/2004CA2510848A1 Pyrimidine derivates for the treatment of abnormal cell growth
07/08/2004CA2510846A1 New carboxylic acid amides,the preparation thereof and their use as pharmaceutical compositions
07/08/2004CA2510815A1 Microsomal triglyceride transfer protein inhibitors
07/08/2004CA2510471A1 Substituted biphenyl-4-carboxylic acid arylamide analogues as capsaicin receptor modulators
07/08/2004CA2510069A1 The gene cluster involved in safracin biosynthesis and its uses for genetic engineering
07/08/2004CA2510027A1 Piperidine derivatives useful as ccr5 antagonists
07/08/2004CA2509881A1 Substituted n-phenyl sulfonamide bradykinin antagonists
07/08/2004CA2509403A1 Pyrazole compounds