Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979) |
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11/09/2005 | EP1592684A1 Malonamide derivatives as gamma-secretase inhibitors |
11/09/2005 | EP1592674A1 Amino 1, 3, 5-triazines n-substituted with chiral bicyclic radicals, process for their preparation, compositions thereof and their use as herbicides and plant growth regulators |
11/09/2005 | EP1592425A2 New arylpiperazinyl compounds |
11/09/2005 | EP1592389A2 Piperazine-2-carboxamide derivatives |
11/09/2005 | EP1423378B1 Aminopyrrole compounds as antiinflammatory agents |
11/09/2005 | EP1315714B1 Quinazoline derivatives as alpha-1 adrenergic antagonists |
11/09/2005 | EP1307196A4 Inhibition of inflammatory cytokine production by cholinergic agonists and vagus nerve stimulation |
11/09/2005 | EP1212296B1 Phosphate mimics and methods of treatment using phosphatase inhibitors |
11/09/2005 | EP1163236B1 Aromatic heterocyclic compounds as anti-inflammatory agents |
11/09/2005 | EP1095016B1 Sulfur substituted sulfonylaminocarboxylic acid n-arylamides, their preparation, their use and pharmaceutical preparations comprising them |
11/09/2005 | EP1089973B1 Amidino and guanidino azetidinone tryptase inhibitors |
11/09/2005 | EP1049700B1 Chemokine receptor antagonists and methods of use therefor |
11/09/2005 | EP1019392B1 Tricyclic amides useful for inhibition of g-protein function and for treatment of proliferative diseases |
11/09/2005 | EP0943008B1 Metal mediated serine protease inhibitors |
11/09/2005 | CN1694891A Neutral metallic dendrimer complexes |
11/09/2005 | CN1694879A Isoquinoline derivatives having kinasae inhibitory activity and drugs containing the same |
11/09/2005 | CN1694875A 5-aryltetrazole compounds and uses thereof |
11/09/2005 | CN1694873A Vanilloid receptor ligands and their use in treatments |
11/09/2005 | CN1694708A Inhibitors of tgfbeta |
11/09/2005 | CN1226292C Diazesuberane derivant or its salt |
11/09/2005 | CN1226035C New use of iloperidone |
11/08/2005 | US6962996 Inhibitors of p38 |
11/08/2005 | US6962995 Phenanthroline derivatives |
11/08/2005 | US6962942 Azacycloalkanone serine protease inhibitors |
11/08/2005 | US6962936 Treating diseases such as cancer, inflammatory disorders, restenosis, |
11/08/2005 | US6962932 1-phenyl-2-heteroaryl-substituted benzimdazole derivatives, their use for the production of pharmaceutical agents as well as pharmaceutical preparations that contain these derivatives |
11/08/2005 | US6962924 Antihistamines; side effect reduction |
11/08/2005 | US6962923 Pyrazole compositions |
11/08/2005 | US6962917 E.g., (R)-2-(4-((4-fluoro-1H-benzimidazol-2-ylmethyl)-amino)-piperidin-1-yl)-1-(6- methoxyquinolin-4-yl)-ethanol; effective against both gramnegative and grampositive bacteria |
11/08/2005 | US6962913 Benzo-1,4-diazepin-2-ones as inhibitors of Aβ protein production |
11/08/2005 | CA2249222C Aminopyridine derivatives |
11/08/2005 | CA2195677C Endothelin antagonists |
11/08/2005 | CA2157288C Methods and compositions for inhibition of angiogenesis |
11/08/2005 | CA2155104C Heterocyclic-substituted alkyl amide acat inhibitors |
11/03/2005 | WO2005103043A1 2, 4, 6-substituted pyridyl derivative compounds useful as beta-secretase inhibitors for the treatment of alzheimer’s disease |
11/03/2005 | WO2005103041A2 Treatment of cns disorders using cns target modulators |
11/03/2005 | WO2005103039A1 2- (3-aminopyrrolidin-1-yl) pyridines as melanin-concentrating hormone receptor an tagonists |
11/03/2005 | WO2005103038A1 N-[6-(4-morpholinyl)-3-pyridinyl]-2-(tetrahydro-2h-pyran-4-yl)-n-[(1-{[phenyl]methyl}-4-piperidinyl)methyl] acetamide derivatives and related compounds as glyt1 transport inhibitors for the treatment of neurological disorders such as schizophrenia |
11/03/2005 | WO2005103037A2 Selected cgrp antagonists, methods for the production thereof, and use thereof as medicaments |
11/03/2005 | WO2005103036A1 Pyrimidin-4-yl-1h-indazol-5yl-amines as chk1 kinases inhibitors |
11/03/2005 | WO2005103034A1 Novel piperidine substituted diaminothiazoles |
11/03/2005 | WO2005103033A1 1-amino-phthalazine derivatives, the preparation and the therapeutic use thereof |
11/03/2005 | WO2005103032A2 Novel alkyne compounds having an mch-antagonistic effect, and medicaments containing said compounds |
11/03/2005 | WO2005103031A1 Novel alkyne compounds with an mch-antagonistic action and medicaments containing said compounds |
11/03/2005 | WO2005103030A1 1,4-di substituted benzene compounds, process for preparing the same and use thereof |
11/03/2005 | WO2005103029A1 Novel alkyne compounds having an mch-antagonistic effect and medicaments containing said compounds |
11/03/2005 | WO2005103028A1 2-pyridyl substituted imidazoles as alk5 and/or alk4 inhibitors |
11/03/2005 | WO2005103006A1 2-pyridinylcycloalkylcarboxamide derivatives useful as fungicides |
11/03/2005 | WO2005103002A2 Novel alkyne compounds with an mch-antagonistic action and medicaments comprising said compounds |
11/03/2005 | WO2005102998A1 Novel androgens |
11/03/2005 | WO2005102997A1 3,4-disubstituted maleimides for use as vascular damaging agents |
11/03/2005 | WO2005101989A2 Piperidine derivatives as modulators of chemokine receptor ccr5 |
11/03/2005 | WO2005086871A9 Compounds, compositions and methods for inhibiting or treating hiv-1 |
11/03/2005 | WO2005011611A3 Bicyclic compounds and compositions as pdf inhibitors |
11/03/2005 | WO2005003103A3 2, 4, 6-tri-substituted 6-membered heterocycles and their use in the treatment of neurodegenerative diseases |
11/03/2005 | WO2004096131A3 Inhibitors of akt activity |
11/03/2005 | WO2002004440A9 Composition and antiviral activity of substituted indoleoxoacetic piperazine derivatives |
11/03/2005 | US20050245743 depression and/or anxiety, obesity, urinary disorder; 5-(2-Methoxyphenyl)-N-[3-(4-Piperidinyl)Phenyl]Pentanamide |
11/03/2005 | US20050245596 Derivatives of 1-(oxoaminoacetyl) pentylcarbamate as cathepsin k inhibitors for the treatment of bone loss |
11/03/2005 | US20050245593 4-Aminomethyl-1-aryl-cyclohexylamine compounds |
11/03/2005 | US20050245592 2-Iminopyrrolidine derivatives |
11/03/2005 | US20050245586 2,5-Dioxoimidazolidin-4-yl acetamides and analogues as inhibitors of metalloproteinase mmp12 |
11/03/2005 | US20050245581 3-(2-Cyanophenyl)-5-(2-methoxyphenyl)-1-phenyl-1,2-dihydropyridin-2-one; antagonists of AMPA and kainate receptors; neuroprotectants; neurodegenerative diseases; Alzheinmer's disease; antiepileptic agents; antispasmodic agents; anxiolytic agents; ddrug abuse; nervous sytem disorders; antihypoxic agents |
11/03/2005 | US20050245580 Novel substituted dihydro 3-halo-1H-pyrazole-T-carboxylates, their preparation and use |
11/03/2005 | US20050245578 Polymorphs of pantoprazole sodium salt and process for the preparation thereof |
11/03/2005 | US20050245576 Substituted pyrazoles |
11/03/2005 | US20050245574 Aminophenoxyacetic acid derivatives and pharmaceutical composition containing thereof |
11/03/2005 | US20050245572 Naphthyl ether compounds and their use |
11/03/2005 | US20050245571 Amine derivative |
11/03/2005 | US20050245565 Diamine derivatives |
11/03/2005 | US20050245555 Tri-substituted ureas as cytokine inhibitors |
11/03/2005 | US20050245554 Substituted pyrimidines |
11/03/2005 | US20050245552 N-substituted pyridinone and pyrimidinone derivatives for use as lp-pla2 inhibitors in the treatment of artherosclerosis |
11/03/2005 | US20050245551 Amide derivatives |
11/03/2005 | US20050245547 6-((6,7-Bis(methoxy)-4-quinolinyl)oxy)-N-(3-methylphenyl)-1-benzofuran-3-carboxamide;antiproliferative; -metastasis; -carcinogenic; -tumor; -inflammatory; -arthritic agents;hypotensive agents; myocardium necrosis; rheumatic diseases; tyrosine kinase inhibitors; antiallergens; asthma |
11/03/2005 | US20050245542 Pyridazine, pyrimidine and pyrazine ethyne compounds |
11/03/2005 | US20050245538 Dipeptidyl peptidase inhibitor; antidiabetic agents; obesity; viricides; anticancer agents; oral diseases; autoimmune disease |
11/03/2005 | US20050245536 N-Pyridyl-7-substituted-2-indolecarboxamides, e.g., 1-Methyl-7-[2-(4-methyl-piperazin-1-yl)-pyrimidin-4-yloxy]-1H-indole-2-carboxylic acid (2-tert-butyl-5-methoxy-pyridin-4-yl)-amide; used to treat chronic inflammatory diseases |
11/03/2005 | US20050245530 Monocyclic heterocycles as kinase inhibitors |
11/03/2005 | US20050245529 Alkyne compounds with MCH antagonistic activity and medicaments comprising these compounds |
11/03/2005 | US20050245527 Nitrogen containing heterocyclic compounds and medicines containing the same |
11/03/2005 | US20050245526 Beta-agonists, methods for the preparation thereof and their use as pharmaceutical compositions |
11/03/2005 | US20050245525 Compounds useful for inhibiting CHK1 |
11/03/2005 | US20050245523 Heteroaryl derivatives and their use as medicaments |
11/03/2005 | US20050245521 3-[-2-(Piperazin-1-yl)benzyl]pyrrolidin-2-one derivatives; antidepressants, anxiolytic agents; obsessive compulsive disorder, psychological disorders, phobias; 5-HT1 agonist or antagonists; side effect reduction, in particular cardiac QTc prolongation; hydrogenation |
11/03/2005 | US20050245520 2-Phenylpyridin-4-yl derivatives as alk5 inhibitors |
11/03/2005 | US20050245515 Indolyl derivatives as liver-X-receptor (LXR) modulators |
11/03/2005 | US20050245513 Hetero-bridge substituted 8-arylquinoline pde4 inhibitors |
11/03/2005 | US20050245511 Novel compounds that inhibit tryptase activity |
11/03/2005 | US20050245505 Novel heterocyclic compounds, method for preparing same and use thereof as medicines, in particular as antibacterial agents |
11/03/2005 | US20050245503 Therapeutic heterocycles |
11/03/2005 | US20050245501 Succinoylamino lactams as inhibitors of A-beta protein production |
11/03/2005 | US20050245500 Beta-ketoamide compounds with MCH antagonistic activity |
11/03/2005 | US20050245499 Heterocyclic protein kinase inhibitors and uses thereof |
11/03/2005 | US20050245485 Novel indole derivatives as selective androgen receptor modulators (SARMS) |
11/03/2005 | US20050245399 Pyrazole derivatives as herbicidal compositions containing them |
11/03/2005 | US20050244807 Two-photon absorption heteroaromatic chromophores and compositions thereof |
11/03/2005 | DE19910403B4 3-Hydroxy-1,2,3,3a-tetrahydro-benzo[b]cyclopent[e]azepin-4,10(5H,10aH)-dion-Derivate enthaltende Arzneimittel 3-hydroxy-1,2,3,3a-tetrahydro-benzo [b] cyclopent [e] azepine-4,10 (5H, 10AH) -dione derivatives of drugs containing |
11/03/2005 | DE102004018796A1 Ausgewählte CGRP-Antagonisten, Verfahren zu deren Herstellung sowie deren Verwendung als Arzneimittel Selected CGRP antagonists, processes for their preparation and their use as medicaments |
11/03/2005 | DE102004017935A1 Neue Alkin-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel New alkyne compounds with MCH-antagonistic activity and pharmaceutical compositions containing them |