Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979) |
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12/30/2009 | EP1608632B1 Quinazolines useful as modulators of ion channels |
12/30/2009 | EP1608352B1 Polyamine compounds for treating chemokine receptor mediated diseases |
12/30/2009 | EP1487444B1 Use of pyridyl amides as inhibitors of angiogenesis |
12/30/2009 | CN101616910A Modulators of interleukin-1 receptor-associated kinase |
12/30/2009 | CN101616909A Substituted isoquinoline and isoquinolinone derivatives as inhibitors of Rho-kinase |
12/30/2009 | CN101616908A Carboxamide compounds and their use as calpain inhibitors |
12/30/2009 | CN101613343A Caderofloxacin lactate crystals I and II and preparation method thereof |
12/30/2009 | CN101613321A Mono- and bicyclic azole derivatives that inhibit the interaction of ligands with rage |
12/30/2009 | CN100575346C Pyrimidinone derivaties as therapeutic agents against acute and chronic inflammatory, ischaemic and remodelling processes |
12/30/2009 | CN100575345C Pyridone derivative having affinity for cannabinoid 2-type receptor |
12/30/2009 | CN100575341C Tetrahydro-indolone derivative and tetrahydro-indazolone derivatives and their use |
12/30/2009 | CN100574750C Rapidly-disintegrating formulation for releasing active ingredients |
12/30/2009 | CA2766328A1 New therapeutic agents |
12/30/2009 | CA2729546A1 Compounds and compositions as kinase inhibitors |
12/30/2009 | CA2729327A1 Organic compounds |
12/30/2009 | CA2729275A1 5- and 6-membered heterocyclic compounds |
12/30/2009 | CA2729259A1 1,2-disubstituted heterocyclic compounds |
12/30/2009 | CA2729220A1 Di-substituted phenyl compounds |
12/30/2009 | CA2729115A1 Substituted triazinone derivatives |
12/30/2009 | CA2729108A1 Organic compounds |
12/30/2009 | CA2728806A1 Squaric acid derivatives as inhibitors of the nicotinamide phosphoribosyltransferase |
12/30/2009 | CA2728730A1 Novel tetramethyl substituted piperidine derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
12/30/2009 | CA2728680A1 Substituted n-oxide pyrazine derivatives |
12/30/2009 | CA2728283A1 Isoquinolinone derivatives as nk3 antagonists |
12/30/2009 | CA2728210A1 Synthesis and use of heterocyclic antibacterial agents |
12/30/2009 | CA2728016A1 Novel substituted pyridin-2-ones and pyridazin-3-ones |
12/30/2009 | CA2727573A1 Diaryl compounds and uses thereof |
12/30/2009 | CA2727455A1 Heteroaryl compounds and uses thereof |
12/29/2009 | USRE41065 Such as (6,7-dimethoxyquinazolin-4-yl)-(3-ethynylphenyl)-amine for treatment of hyperproliferative diseases |
12/29/2009 | US7638638 Antiinflamamtory agents; autoimmune disease; immunosuppressants;multiple sclerosis; antiarthritic agents |
12/29/2009 | US7638634 Amorphous esomeprazole hydrate |
12/29/2009 | US7638633 Process for synthesis of proton pump inhibitors |
12/29/2009 | US7638631 Methylene dipiperidine derivatives |
12/29/2009 | US7638630 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as VLA-4 inhibitors |
12/29/2009 | US7638629 4-Isopropylphenyl)-2-[4-(trifluoromethyl)phenyl]piperidin-4-yl}acetic acid; modulators of gamma secretase isoforms, 1-42; antifibrillatory agents; neurodegenerative diseases; modulating activity of gamma -secretase as opposed to suppressing it to reduced risk of side effects; beta secretase inhibitors |
12/29/2009 | US7638627 Imatinib hydrochloride; reacting N-(2-methyl-5-aminophenyl-4-(3-pyridyl)-2-pyrimidineamine with 4-(4-methyl-piperazinomethyl)benzoyl chloride; improved reduction step to simplify, increase yield, improve purity |
12/29/2009 | US7638546 Imidazolyl derivatives |
12/29/2009 | US7638537 Pyrazole compounds as transforming growth factor (TGF) inhibitors |
12/29/2009 | US7638527 4-[(4-N,N-diethylaminocarbonyl)phenyl]-spiro[2H,1-benzopyran-2,4'-piperidine; ligands of delta opioid receptor; analgesic, anxiolitic, antidepressant, analgesic; gastrointestinal disorders, neurodegenerative diseases; side effect reduction |
12/29/2009 | US7638521 3-guanidinocarbonyl-1-heteroaryl-indole derivatives, preparation process, their use as medicaments, and pharmaceutical compositions comprising them |
12/29/2009 | US7638520 Pyrimidine compounds |
12/29/2009 | US7638518 3-(Benzimidazol-2-yl)pyrazole derivatives; inhibitors of ATP and protein kinase interactions; diabetes, rheumatoid arthritis, Crohn's disease, septic shock, cachexia, pancreatitis, Alzheimer's disease, Parkinson's disease; antimetastasis, anticarcinogenic, antitumor, antidepressant, antiallergen agents |
12/29/2009 | US7638514 Agriculture |
12/29/2009 | US7638513 inhibitors of matrix metalloproteinases, aggrecanases, tumor necrosis factor-alpha converting enzyme, and tumor necrosis factors |
12/29/2009 | CA2524043C 1-(2h-pyrazol-3-yl)-3-{4-'1-(benzoyl)-piperidin-4-ylmethyl!-phenyl}-urea derivatives and related compounds as inhibitors of p38 kinase and/or tnf inhibitors for the treatment of inflammations |
12/29/2009 | CA2478799C Di-aryl substituted tetrazole modulators of metabotropic glutamate receptor-5 |
12/29/2009 | CA2447521C Delivery of antihistamines through an inhalation route |
12/29/2009 | CA2429720C Tricyclic compounds useful for the inhibition of farnesyl protein transferase |
12/29/2009 | CA2429440C Dehalogeno-compounds |
12/29/2009 | CA2428133C Indolylmaleimide derivatives as protein kinase c inhibitors |
12/29/2009 | CA2424522C Substituted benzene derivatives or salts thereof |
12/29/2009 | CA2423296C N-(4-aryloxypiperidin-1-ylalkyl) cinnamic amides as ccr33 receptor antagonists |
12/29/2009 | CA2387013C 6-position substituted indolinones, the preparation thereof and their use as pharmaceutical compositions |
12/29/2009 | CA2370250C Di-aryl acid derivatives as ppar receptor ligands |
12/29/2009 | CA2351488C Substituted 4-amino-2-arylcyclopenta[d]pyrimidines, their preparation, their use and pharmaceutical preparations comprising them |
12/29/2009 | CA2287214C Substituted benzopyran derivatives for the treatment of inflammation |
12/24/2009 | US20090318692 Process of making imatinib |
12/24/2009 | US20090318684 Rock inhibitors and uses thereof |
12/24/2009 | US20090318668 Water-Soluble CC-1065 Analogs and Their Conjugates |
12/24/2009 | US20090318592 Process for the Synthesis of Amine Ethers |
12/24/2009 | US20090318504 Use of GAL3 receptor antagonists for the treatment of depression and/or anxiety and compounds useful in such methods |
12/24/2009 | US20090318503 Bis-quaternary ammonium salts and methods for modulating neuronal nicotinic acetylcholine receptors |
12/24/2009 | US20090318500 4-(2, 6-Dichloro-benzoylamino)-1H-pyrazole-3-carboxylic acid (1-methanesulphonyl-piperidin-4-yl)-amide for the Treatment of Cancer |
12/24/2009 | US20090318499 Compounds having analgesic and/or immunostimulant activity |
12/24/2009 | US20090318498 Piperidyl acrylamide antagonists of ccr2 |
12/24/2009 | US20090318497 Substituted pyridylmethyl bicycliccarboxyamide compounds |
12/24/2009 | US20090318493 Aryl pyrrolidinyl and piperidinyl ketone derivatives and uses thereof |
12/24/2009 | US20090318489 Aporphine compounds and pharmaceutical use thereof |
12/24/2009 | US20090318483 3-{[4-(4-acetyl-3-hydroxy-2-propylphenoxymethyl)-phenyl]-(S)-hydroxymethyl}-benzoic acid; anxiolytic, neuroleptic agent and antidepressant as glutamate receptor agonist; antiinflammatory agent as leukotriene receptor agonist; |
12/24/2009 | US20090318481 Potentiators Of Glutamate Receptors |
12/24/2009 | US20090318478 Quinazoline derivatives |
12/24/2009 | US20090318474 Pyridine and pyrimidine derivatives as mglur 2 antagonists |
12/24/2009 | US20090318473 5,6-bisaryl-2-pyridine-carboxamide derivatives, preparation and application thereof in therapeutics as urotensin ii receptor antagonists |
12/24/2009 | US20090318472 Aminopyrazine derivatives and compositions |
12/24/2009 | US20090318467 Novel heteroaryl carboxamide derivatives |
12/24/2009 | US20090318466 Compounds useful as pesticides |
12/24/2009 | US20090318463 Indolylmaleimide Derivatives |
12/24/2009 | US20090318452 INHIBITORS OF p38 |
12/24/2009 | US20090318448 Inhibitors of Bruton's Tyrosine Kinase |
12/24/2009 | US20090318447 N-[6-(4-morpholinyl)-3-pyridinyl]-2-(tetrahydro-2h-pyran-4-yl)-n-[(1--4-piperidinyl) methyl] acetamide derivatives and related compounds as glyt1 transport inhibitors for the treatment of neurological disorders such as schizophrenia |
12/24/2009 | US20090318446 4-(1H-Indol-3-yl)-Pyrimidin-2-Ylamine Derivatives and Their Use in Therapy |
12/24/2009 | US20090318438 Heterocyclic compounds and their use as anticancer agents |
12/24/2009 | US20090318407 Inhibitors of protein kinases |
12/24/2009 | US20090318406 Substituted oxindole derivatives and their use as vasopressin and/or oxytocin receptor ligands |
12/24/2009 | US20090318373 Receptor-type kinase modulators and methods of use |
12/24/2009 | US20090317359 2,6-disubstituted quinazolines, quinoxalines, quinolines and isoquinolines and methods of their use as inhibitors of raf kinase |
12/23/2009 | WO2009155362A1 Small molecule hematopoietic growth factor mimetic compounds and their uses |
12/23/2009 | WO2009155121A2 Inhibitors of pi3 kinase |
12/23/2009 | WO2009155001A2 Wnt protein signalling inhibitors |
12/23/2009 | WO2009154190A1 Pyridone compound |
12/23/2009 | WO2009153721A1 Nicotinamide derivatives |
12/23/2009 | WO2009153589A1 Pyridine compounds |
12/23/2009 | WO2009153569A2 Cb1 receptor modulators |
12/23/2009 | WO2009153313A1 2 -arylaminoquinazolines for treating proliferative diseases |
12/23/2009 | WO2009153215A1 Method for producing an intermediate product of dabigatran etexilate |
12/23/2009 | WO2009153191A1 Novel Microbiocides |
12/23/2009 | WO2009153182A1 Novel heteroaryl carboxamide derivatives |
12/23/2009 | WO2009153180A1 Heteroaromatic monoamides as orexinin receptor antagonists |
12/23/2009 | WO2009153179A1 Pyrrolidine derivatives as nk2 receptor antagonists |
12/23/2009 | WO2009153178A2 Aryl ketone as mri |