Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979) |
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08/18/2010 | EP1692109B1 Phosphodiesterase 4 inhibitors, including n-substituted diarylamine analogs |
08/18/2010 | EP1451174B1 Process for the preparation of compositions having an increased amount of pharmaceutically active salts of rotamers |
08/18/2010 | EP1400510B1 Cyclic diamine compounds having fused-ring groups |
08/18/2010 | EP0956865B2 MEDICINES COMPRISING Rho KINASE INHIBITOR |
08/18/2010 | CN1993352B Piperazine derivatives with CCR3 inhibiting activity |
08/18/2010 | CN1795193B N-acyl nitrogen heterocyles as ligands of peroxisome proliferator-activated receptors |
08/18/2010 | CN101809015A Salts of a CGRP antagonist, method for producing the same and use thereof as drugs |
08/18/2010 | CN101809014A Method for producing pyrazol-3-yl-benzamide derivative |
08/18/2010 | CN101809013A herbicide triazolylpyridine ketones |
08/18/2010 | CN101809012A Spiro substituted compounds as angiogenesis inhibitors |
08/18/2010 | CN101809001A Imidazole derivatives |
08/18/2010 | CN101808999A Quinoline derivatives as 5HT5A receptor antagonists |
08/18/2010 | CN101808996A Nicotinamide derivatives, preparation thereof and therapeutic use thereof |
08/18/2010 | CN101808994A Compounds and methods for kinase modulation, and indications therefor |
08/18/2010 | CN101808991A Acyclic derivatives as modulators of chemokine receptor activity |
08/18/2010 | CN101808990A Piperidine derivatives as modulators of chemokine receptor activity |
08/18/2010 | CN101808693A Triazine kinase inhibitors |
08/18/2010 | CN101805327A Rabeprazole sodium compound and novel preparation method thereof |
08/18/2010 | CN101805309A Benzamide derivatives useful as histone deacetylase inhibitors |
08/18/2010 | CN101250166B Thiadiazoles formamide derivative as well as synthesis and uses thereof |
08/18/2010 | CN101160128B Protective agent for retinal neuronal cell comprising indazole derivative as active ingredient |
08/18/2010 | CN101024671B 丙型肝炎病毒抑制剂 Hepatitis C virus inhibitors |
08/17/2010 | US7777051 A compound with azo containing mono and a bicyclic rings attached with an aryl or heteroaryl ring; both therapeutic and diagnostic |
08/17/2010 | US7777050 N3 alkylated benzimidazole derivatives as MEK inhibitors |
08/17/2010 | US7777049 Serotonin receptor antagonists |
08/17/2010 | US7777044 Process for the preparation of optically active derivatives of 2-(2-pyridylmethylsulfinyl)-benzimidazole via inclusion complex with 1,1′-binaphthalene-2,2′diol |
08/17/2010 | US7777041 N-(4-(5-Butyl-2-methoxyphenyl)-1,3-thiazol-2-yl)-4-((4-oxopiperidin-1-yl)carbonyl)benzamide; antiinflammatory, anticarcinogenic, antidiabetic, analgesic agents |
08/17/2010 | US7777032 N-4-[3-Chloro-4-(3-fluoro-benzyloxy)-phenyl]-N6-(3-ethyl-oxazolidin-2-ylidene)-quinazoline-4,6-diamine; use as type I receptor tyrosine kinase inhibitor; hyperproliferation diseases such as cancer; antiinflammatory agents |
08/17/2010 | US7777009 for modulation of chemokines; antiinflammatory agents; cancer |
08/17/2010 | US7776900 gamma--aminobutyric acid A (GABAA) receptor modulators such as 1-[3-(Pyridin-2-ylmethoxymethyl)-phenyl]-1H-benzoimidazole-5-carboxylic acid ethyl ester, useful in the treatment of central nervous system diseases and disorders; anxiolytic agents; side effect reduction |
08/17/2010 | US7776891 antagonists of very late antigen-4 integrin; ulcerative colitis, Crohn's disease, asthma, multiple sclerosis, rheumatoid arthritis; N-{N-[(3-Cyanobenzene)sulfonyl]-4(R)-[3,3-difluoropiperidinyl]-(L)-prolyl}-4-[(3',5'-dichloroisonicotinoyl)amino]-(L)-phenylalanine ethyl ester |
08/17/2010 | US7776885 Benzimidazolone compounds having 5-HT4 receptor agonistic activity |
08/17/2010 | US7776884 Cyclic derivatives as modulators of chemokine receptors activity |
08/17/2010 | US7776883 Quinolin-4-ones as inhibitors of retroviral integrase for the treatment of HIV, AIDS and AIDS related complex (ARC) |
08/17/2010 | US7776876 administering cyclic Glycyl-2-Allyl Proline as as neuroprotectants, for the prophylaxis of nervous system disorders |
08/17/2010 | US7776874 Cycloalkylcarbonyl-3H-spiro[2-benzofuran-1,3'-pyrrolidin]-3-ones: N-methyl-5-[4-(1-{[3-oxo-1'H,3H-spiro[2-benzofuran-1,3'-pyrrolidin]-1'-yl]carbonyl}cyclopropyl)phenyl]pyridine-2-carboxamide; 11- beta hydroxyl steroid dehydrogenase type 1 inhibitors; mineralcorticoid receptor antagonists; diabetes |
08/17/2010 | US7776872 Diaminopyrimidines as P2X3 and P2X2/3 modulators |
08/17/2010 | US7776862 Pyridyl and phenyl substituted piperazine-piperidines with CXCR3 antagonist activity |
08/17/2010 | US7776861 Cycloheteroalkenyl compounds used as analgesics and for treating incontinence, inflammatory bowel disease, Parkinson's disease, amyotrophic lateral sclerosis, dementia, epilepsy, retinopathy, pruritus, psychoses, Huntington's disease, headaches, vomiting, dyskinesia or as anxiolytics and antidepressants |
08/17/2010 | US7776182 8-Oxyl-7,7,9,9-tetramethyl-1,3,8-triaza-spiro[4.5]decane-2,4-dione; antiyellowing agents for lignin |
08/17/2010 | CA2605854C Novel pyridine derivative and pyrimidine derivative (3) |
08/17/2010 | CA2545092C Quinolonecarboxylic acid compounds having 5-ht4 receptor agonistic activity |
08/17/2010 | CA2481535C Use of ep4 receptor ligands in the treatment of il-6 involved diseases |
08/17/2010 | CA2461963C Cyclic amine compounds |
08/17/2010 | CA2438991C Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
08/17/2010 | CA2412854C Vitronectin receptor antagonist pharmaceuticals for use in combination therapy |
08/17/2010 | CA2407208C Process for producing optically active sulfoxide derivative |
08/17/2010 | CA2378165C Dihydrobenzodiazepines and their use in the treatment of dyslipidaemia |
08/17/2010 | CA2377236C Pyrazole derivative, production process thereof, and pest control agent containing the same as active ingredient |
08/17/2010 | CA2370412C Pharmaceutical compounds |
08/17/2010 | CA2325471C Piperididinyl and n-amidinopiperidinyl derivatives |
08/12/2010 | WO2010091209A1 Pyridine compounds as subtype selective modulators of alpha2b and/or alpha 2c adrenergic receptors |
08/12/2010 | WO2010091104A1 Glucosylceramide synthase inhibitors |
08/12/2010 | WO2010090875A1 Derivatives of n2-(3-pyridil or phenyl)-n4-(4-piperidyl)-2,4-pyrimidinediamine useful in the treatment of inflammatory, autoimmune or proliferative diseases |
08/12/2010 | WO2010090347A1 Dihydroquinolinone derivatives |
08/12/2010 | WO2010090344A1 Hydrazide compound and use of the same in pest control |
08/12/2010 | WO2010090299A1 A novel cyanopyrimidine derivative |
08/12/2010 | WO2010090290A1 Aminopyrazine derivative and medicine |
08/12/2010 | WO2010090198A1 Process for preparing 1-(4-piperidinyl)benzimidazolone derivatives |
08/12/2010 | WO2010090009A1 Indoline derivatives |
08/12/2010 | WO2010089327A2 Indole derivatives as anticancer agents |
08/12/2010 | WO2010089127A1 Substituted spiro-amides as b1r modulators |
08/12/2010 | WO2010089119A1 Heterocyclic derivatives as m-glu5 antagonists |
08/12/2010 | WO2010089084A1 Substituted indole compounds as bradykinin receptor 1 modulators |
08/12/2010 | WO2010067085A3 Synthesis of 9-(arylalkyl)-1,2,3,4-tetrahydro-υ-carboline and analogues and intermediates |
08/12/2010 | WO2010042758A3 Oxazole-pyridazine-oxazole alpha-helix mimetic |
08/12/2010 | WO2010042489A3 Aminoquinoline derived heat shock protein 90 inhibitors, methods of preparing same, and methods for their use |
08/12/2010 | WO2009109616A8 1-benzyl-3-hydroxymethylindazole derivatives and use thereof in the treatment of diseases based on the expression of mcp-1, cx3cr1 and p40 |
08/12/2010 | US20100204479 Crystalline forms of dexlansoprazole |
08/12/2010 | US20100204478 Improved process for amophous rabeprazole sodium |
08/12/2010 | US20100204472 Indane acetic acid derivatives and their use as pharmaceutical agents, intermediates, and method of preparation |
08/12/2010 | US20100204470 method for salt preparation |
08/12/2010 | US20100204282 Reverse indoles as 5-lipoxygenase-activating protein (FLAP) inhibitors |
08/12/2010 | US20100204280 Cinnamoyl inhibitors of transglutaminase |
08/12/2010 | US20100204279 Therapeutic Salt Compositions and Methods |
08/12/2010 | US20100204276 Indole compounds, a process for their preparation and pharmaceutical compositions containing them |
08/12/2010 | US20100204275 N-piperidin-4-ylmethyl-amide derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
08/12/2010 | US20100204274 Piperidinyl derivatives as modulators of chemokine receptor activity |
08/12/2010 | US20100204273 Quinoline and Quinazoline Derivatives Having Affinity for 5HT1-Type Receptors |
08/12/2010 | US20100204272 Compounds which have activity at M1 receptor and their uses in medicine |
08/12/2010 | US20100204260 synthesis of new class of nonsteroidal antiinflammatory and antibacterial agent for use treating septic shock, asthma, arthritis, cancer; e.g. 1-Benzyl-2,4,5-triphenyl-4,5-dihydro-1H-imidazole-4-carboxylic acid |
08/12/2010 | US20100204255 Bicyclic derivatives as modulators of ion channels |
08/12/2010 | US20100204246 5-aminopyrazol-3-yl-3h-imidazo (4,5-b) pyridine derivatives and their use for the treatment of cancer |
08/12/2010 | US20100204245 Amino-pyridines As Inhibitors Of Beta-secretase |
08/12/2010 | US20100204241 New pyridazin-3(2h)-one derivatives |
08/12/2010 | US20100204236 Substituted imidazoles as bombesin receptor subtype-3 modulators |
08/12/2010 | US20100204228 Aryl Sulfonamides Useful for Modulation of the Progesterone Receptor |
08/12/2010 | US20100204227 Isoindoline compounds and methods of their use |
08/12/2010 | US20100204226 Quinazolinones as prolyl hydroxylase inhibitors |
08/12/2010 | US20100204216 PHARMACEUTICAL COMPOSITION FOR INHIBITING AMYLOID-beta PROTEIN ACCUMULATION |
08/12/2010 | US20100204208 Protein kinase c inhibitors and uses thereof |
08/12/2010 | US20100204207 Compounds and Methods for Treating Dyslipidemia |
08/12/2010 | US20100204200 Inhibitors of cathepsin s |
08/12/2010 | US20100204199 Cyclic 11-beta hydroxysteroid dehydrogenase type i inhibitors |
08/12/2010 | US20100203645 Novel zwitterionic dyes for labeling in proteomic and other biological anaylses |
08/12/2010 | US20100203613 Aminopyridine Dimer Compounds, Compositions and Related Methods for Neuronal Nitric Oxide Synthase Inhibition |
08/12/2010 | US20100200054 Compound for organic photoelectric device and organic photoelectric device including the same |
08/12/2010 | US20100199443 Yello anionic disazo dyes |
08/12/2010 | CA2751695A1 Aminopyrazine derivatives and medicines |
08/12/2010 | CA2751651A1 Pyridine compounds as subtype selective modulators of alpha2b and/or alpha 2c adrenergic receptors |