Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979) |
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12/28/2010 | US7858641 melanocortin-4 receptor (MC4-R) agonists such as (3R,5S)-N-(2-{2-[2-fluoro-4-(methyloxy)phenyl]ethyl}-1-oxo-1,2-dihydroisoquinolin-6-yl)-3,5-dimethyl-N'-[(1S,2S,3S,5R)-2,6,6-trimethylbicyclo[3.1.1]hept-3-yl]piperazine-1-carboximidamide, used for the treatment of obesity or diabetes |
12/28/2010 | US7858633 Cycloalkyl substituted pyrimidinediamine compounds and their uses |
12/28/2010 | US7858631 such as (3R,5S)-N-(3-{2-[2-fluoro-4-(methyloxy)phenyl]ethyl}-4-oxo-3,4-dihydropyrido[2,3-d]pyrimidin-7-yl)-3,5-dimethyl-N'-[(1S,2S,3S,5R)-2,6,6-trimethylbicyclo[3.1.1]hept-3-yl]piperazine-1-carboximidamide, used as melanocortin-4 receptor (MC4-R) agonists, for the treatment of obesity or diabetes |
12/28/2010 | US7858624 such as methyl 2-((R)-((R)-1-((2S,3S)-5-(butylamino)-1-cyclohexyl-3-hydroxy-5-oxopentan-2-ylcarbamoyl)piperidin-3-yl)(3-chlorophenyl)methoxy)ethylcarbamate, used as hypotensive agents or for the treatment of cardiovascular disorders, vision defects, aldosteronism and obesity |
12/28/2010 | US7858622 calcitonin gene related peptide antagonists such as [(3-[4-amino-3-chloro-5-(trifluoromethyl)phenyl]-1-[4-[1-(3-ethoxy-3-oxopropyl)piperidin-4-yl]piperidin-1-yl]-1-oxopropan-2-yl]4-(3-oxo-5-phenyl-1H-1,2,4-triazol-2-yl)piperidine-1-carboxylate; headaches; diabetes; irritable bowel syndrome; hot flashes |
12/28/2010 | US7858621 Compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist; and pharmaceutical compositions containing the same |
12/28/2010 | US7858619 Improved solubility, lower tendency to bind to plasma proteins and greater activity especially in serum-based assay systems; remodeling of heart after myocardial infarction; atherosclerosis; 2-[4-(4-Fluorophenoxy)benzenesulfonyl]-6-(2-piperidin-1-ylethoxy)-1,2,3,4-tetrahydroisoquinoline-1-carboxylic acid |
12/28/2010 | US7858615 (S)-(-)-1-(4-fluoroisoquinolin-5-Yl)Sulfonyl-2-methyl-1,4-homopiperazine hydrochloride dihydrate |
12/28/2010 | US7858614 Therapeutic pyrazolonaphthyridine derivatives |
12/28/2010 | US7858211 Organic electroluminescent device |
12/23/2010 | WO2010148314A2 Preparation of esomeprazole and its pharmaceutically acceptable salts |
12/23/2010 | WO2010147917A1 Disubstituted phthalazine hedgehog pathway antagonists |
12/23/2010 | WO2010147302A2 Novel intermediates of voriconazole and preparation method of voriconazole using the same |
12/23/2010 | WO2010146881A1 Substituted isoquinoline derivative |
12/23/2010 | WO2010146488A1 Bicyclic and tricyclic compounds as kat ii inhibitors |
12/23/2010 | WO2010146428A1 An improved process for the preparation of rabeprazole |
12/23/2010 | WO2010146395A1 Pyrazine carboxamides as inhibitors of dgat1 |
12/23/2010 | WO2010146236A1 Urea substituted sulphonamide derivatives |
12/23/2010 | WO2010146083A1 Anthelmintic agents and their use |
12/23/2010 | WO2010145186A1 Peptide deformylase inhibitor containing 2,5-dihydropyrrole and synthesis method thereof |
12/23/2010 | WO2010128528A3 Piperidine derivatives useful for treatment of diebetes |
12/23/2010 | WO2010126626A3 Dual mechanism inhibitors for the treatment of disease |
12/23/2010 | WO2010091876A3 Small molecule bradykinin b1 receptor antagonists |
12/23/2010 | WO2009133572A3 Process for the preparation of amorphous raberazole sodium |
12/23/2010 | US20100324298 Novel Process for the Preparation of Esomeprazole and Salts Thereof |
12/23/2010 | US20100324297 Method for producing 1, 2-dihydropyridine-2-one compound |
12/23/2010 | US20100324093 Ccr9 inhibitors and methods of use thereof |
12/23/2010 | US20100324092 Pyridyl and pyrimidinyl derivatives as histone deacetylase inhibitors |
12/23/2010 | US20100324091 Pyrazolone Derivative |
12/23/2010 | US20100324088 Fused Pyridone M1 Receptor Positive Allosteric Modulators |
12/23/2010 | US20100324084 Urea derivatives of tropane, their preparation and their therapeutic application |
12/23/2010 | US20100324076 Novel sEH Inhibitors and their Use |
12/23/2010 | US20100324070 Indole, indazole and benzimidazole arylamides as p2x3 and p2x2/3 antagonists |
12/23/2010 | US20100324066 Crystalline forms of 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methyl-1-piperazinyl)propoxy]-3-quinolinecarbonitrile and methods of preparing the same |
12/23/2010 | US20100324064 Novel analogs of choline for neuroprotection and cognitive enhancement in neurodegenerative disorders |
12/23/2010 | US20100324061 Enantiomerically pure aminoheteroaryl compounds as protein kinase inhibitors |
12/23/2010 | US20100324058 thrombin function compounds and pharmaceutical compositions based on them |
12/23/2010 | US20100324053 Trisubstituted 1,2,4 triazoles |
12/23/2010 | US20100324049 Diaryl ketimine derivative having antagonism against melanin-concentrating hormone receptor |
12/23/2010 | US20100324048 Disubstituted phthalazine hedgehog pathway antagonists |
12/23/2010 | US20100324046 4-carboxybenzylamino derivatives as histone deacetylase inhibitors |
12/23/2010 | US20100324045 Cyclic urea inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
12/23/2010 | US20100324043 Bicyclic And Tricyclic Compounds As KAT II Inhibitors |
12/23/2010 | US20100324042 Heterocyclic compounds and their use as glycogen synthase kinase 3 inhibitors |
12/23/2010 | US20100324030 5-Quinoline derivatives having an anti-bacterial activity |
12/23/2010 | US20100324028 Novel compounds |
12/23/2010 | US20100324025 Antibacterial Agents |
12/23/2010 | US20100324024 Quinolizidinone M1 Receptor Positive Allosteric Modulators |
12/23/2010 | US20100324017 Acylguanidine derivative |
12/23/2010 | US20100324016 Heteroaromatic and aromatic piperazinyl azetidinyl amides as monoacylglycerol lipase inhibitors |
12/23/2010 | US20100324015 Heteroaromatic and aromatic piperazinyl azetidinyl amides as monoacylglycerol lipase inhibitors |
12/23/2010 | US20100324013 Azetidinyl diamides as monoacylglycerol lipase inhibitors |
12/23/2010 | US20100324012 Azetidinyl diamides as monoacylglycerol lipase inhibitors |
12/23/2010 | US20100324011 Azetidinyl diamides as monoacylglycerol lipase inhibitors |
12/23/2010 | US20100324010 Amide compounds and use of the same |
12/23/2010 | US20100324009 Substituted Sulfonamide Compounds |
12/23/2010 | US20100323965 Thrombopoietin Mimetics |
12/23/2010 | US20100323887 Mesoionic pesticides |
12/23/2010 | US20100322980 Pyrimidine derivatives useful for the treatment of diseases mediated by crth2 |
12/23/2010 | US20100322901 5, 6-ring annulated indole derivatives and use thereof |
12/23/2010 | CA2765130A1 Anthelmintic agents and their use |
12/23/2010 | CA2764542A1 Disubstituted phthalazine hedgehog pathway antagonists |
12/23/2010 | CA2764124A1 Substituted isoquinoline derivative |
12/23/2010 | CA2764013A1 Pyrazine carboxamides as inhibitors of dgat1 |
12/23/2010 | CA2763960A1 Bicyclic and tricyclic compounds as kat ii inhibitors |
12/22/2010 | EP2264032A2 Hiv protease inhibiting sulfonamides |
12/22/2010 | EP2264030A1 Substituted cyclic hydroxamates as inhibitors of matrix metalloproteinases |
12/22/2010 | EP2264028A1 Pyrazole compounds useful as protein kinase inhibitors |
12/22/2010 | EP2264026A1 Alkylaminopyridine derivative |
12/22/2010 | EP2264025A1 Method to produce a crystalline form of compounds (II') |
12/22/2010 | EP2264024A1 Process for the preparation of enantiomerically enriched proton pump inhibitors |
12/22/2010 | EP2264023A1 Method for producing pyrimidine compound |
12/22/2010 | EP2264022A1 Cyano anthranilamide insecticides |
12/22/2010 | EP2264021A1 Process for producing an anthranilamide compound |
12/22/2010 | EP2264014A1 Substituted pyridazines as anti-inflammatory agents and protein kinase inhibitors |
12/22/2010 | EP2264009A1 Pyridylaminoacetic acid compound |
12/22/2010 | EP2263672A1 Novel pharmaceutically acceptable salts of 4-(1H-imidazol-4-ylmethyl)pyridine and their therapeutical uses |
12/22/2010 | EP2262795A1 Muscarinic receptor agonists, compositions, methods of treatment thereof, and processes for preparation thereof |
12/22/2010 | EP2262794A1 Sulfonamide compounds and their use as fungicide |
12/22/2010 | EP2262793A2 Nilotinib hci crystalline forms |
12/22/2010 | EP2262792A1 Substituted sulfonamide derivatives |
12/22/2010 | EP2262791A2 Substituted sulfonamide derivatives |
12/22/2010 | EP2262790A1 Crystal of benzimidazole compound |
12/22/2010 | EP2262789A1 2-aminoquinolines |
12/22/2010 | EP2262778A2 1-benzyl-3-hydroxymethylindazole derivatives and use thereof in the treatment of diseases based on the expression of mcp-1, cxcr1 and p40 |
12/22/2010 | EP2262777A2 1-benzyl-3-hydroxymethylindazole derivatives and use thereof in the treatment of diseases based on the expression of mcp-1, cx3cri |
12/22/2010 | EP2262773A1 2-aminoquinoline derivatives |
12/22/2010 | EP2262772A1 Quinoline derivatives as axl kinase inhibitors |
12/22/2010 | EP2262771A1 A method for the preparation of dabigatran |
12/22/2010 | EP2262770A1 2-trifluoromethylnicotinamide derivatives as hdl-cholesterol raising agents |
12/22/2010 | EP2262767A1 Novel triaryl derivatives useful as modulators of nicotinic acetylcholine receptors |
12/22/2010 | EP2094684B1 1,5-diphenyl-3-benzylamino-1,5-dihydropyrrolidin 2-ones as cb1 receptor modulators |
12/22/2010 | EP2061774B1 Arylpiperazine derivatives and uses thereof |
12/22/2010 | EP1915345B1 Fluoro substituted 2-oxo azepan derivatives |
12/22/2010 | EP1784396B1 Pyrazole-substituted aminoheteroaryl compounds as protein kinase inhibitors |
12/22/2010 | EP1758869B1 Pyridazin-3(2h)-one derivatives and their use as pde4 inhibitors |
12/22/2010 | EP1453805B1 4-piperidinyl alkylamine derivatives as muscarinic receptor antagonists |
12/22/2010 | CN1988907B Dual small molecule inhibitors of cancer and angiogenesis |
12/22/2010 | CN1886380B Benzoimidazole compounds |
12/22/2010 | CN1812973B Indazole compounds useful as protein kinase inhibitors |