Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
08/2011
08/18/2011CA2789298A1 Preparation process of the sodium salt of esomeprazole
08/18/2011CA2787823A1 Arylmethoxy isoindoline derivatives and compositions comprising and methods of using the same
08/17/2011EP2357182A1 Inhibitors of tyrosine kinases
08/17/2011EP2357181A1 2,4-Diaminopyrimidines as inhibitors of cell cycle kinases
08/17/2011EP2357176A1 Amidoacridine derivatives useful as selective inhibitors of ubiquitin specific protease 7
08/17/2011EP2357175A1 isoquinoline derivatives AND THEIR USE IN INCREASING ENDOGENEOUS ERYTHROPOIETIN
08/17/2011EP2357173A1 New alkyne compounds with MCH-antagonistic activity and medicaments containing them
08/17/2011EP2357169A1 Isoindolone compounds and their use as metabotropic glutamate receptor potentiators
08/17/2011EP2356109A2 Compositions and methods for treating alcohol use disorders, pain and other diseases
08/17/2011EP2356108A1 Carbamate derivatives of alkyl-heterocycles, preparation thereof and therapeutic use thereof
08/17/2011EP2356107A1 Substituted (pyridyl)-azinylamine derivatives as fungicides
08/17/2011EP2356106A1 Biaryl spiroaminooxazoline analogues as alpha2c adrenergic receptor modulators
08/17/2011EP2356105A1 ( pyrrolidin-2 -yl) phenyl derivatives for use in the treatment of pain
08/17/2011EP2356104A1 Fungicide heterocyclyl-triazinyl-amino derivatives
08/17/2011EP2356103A1 Novel pyrazolone-derivatives and their use as pd4 inhibitors
08/17/2011EP2356102A1 Substituted (pyridyl)-azinylamine derivatives as plant protection agents
08/17/2011EP2356101A1 Pyrimidine and triazine sulfonamide derivates as b1 bradykinin receptor (b1r) inhibitors for treating pain
08/17/2011EP2356094A1 Novel phenyl amide or pyridil amide derivatives and their use as gpbar1 agonists
08/17/2011EP2356093A1 Carbazole compounds and therapeutic uses of the compounds
08/17/2011EP2355817A1 Heterocyclic gamma secretase modulators
08/17/2011EP2355659A1 Fused heterocyclic m1 receptor positive allosteric modulators
08/17/2011EP2225231B1 Aminotriazole derivatives as alx agonists
08/17/2011EP2190836B1 2-heteroarylamino-pyrimidine derivatives as kinase inhibitors
08/17/2011EP2188268B1 Substituted piperazinyl pyrazines and pyridines as 5-ht7 receptor antagonists
08/17/2011EP2094656B1 P<0}{0pyrrol derivatives, preparation and use of the same in therapy<0}
08/17/2011EP2091919B1 Derivatives of 18-amino substituted analogs of the geldamycin hydroquinon with cytotoxic activity for the treatment of cancer
08/17/2011EP1904475B1 N-thio-anthranilamid compounds and their use as pesticides
08/17/2011EP1896422B1 Tyrosine kinase inhibitors
08/17/2011EP1797069B1 Hiv inhibiting 5-heterocyclyl pyrimidines
08/17/2011EP1797048B1 Hiv inhibiting 5-carbo- or heterocyclic substituted pyrimidines
08/17/2011EP1781619B1 Sigma receptor inhibitors
08/17/2011EP1773775B1 Six-membered heterocycles useful as serine protease inhibitors
08/17/2011EP1771441B1 Novel carboxamides for use as xa inhibitors
08/17/2011EP1761505B1 Pyrimidine urea derivatives as kinase inhibitors
08/17/2011EP1687295B1 Bipiperidinyl derivatives useful as inhibitors of chemokine receptors
08/17/2011EP1379507B1 HETEROARYL UREAS CONTAINING NITROGEN HETERO-ATOMS AS p38 KINASE INHIBITORS
08/17/2011EP1246808B1 1,2-diaryl benzimidazoles for treating illnesses associated with a microglia activation
08/17/2011EP0853618B1 Substituted (sulfinic acid, sulfonic acid, sulfonylamino or sulfinylamino) n- (aminoiminomethyl)phenylalkyl -azaheterocyclylamide compounds
08/17/2011CN1933836B Heteroaryl piperidine glycine transporter inhibitors
08/17/2011CN1913886B 杂环天冬氨酰蛋白酶抑制剂 Heterocyclic aspartyl protease inhibitors
08/17/2011CN1894236B Amino-benzimidazoles derivatives as inhibitors of respiratory syncytial virus replication
08/17/2011CN1878766B Methods for synthesizing quinolinone compounds
08/17/2011CN1549717B Cysteine protease inhibitors with 2-cyano-4-amino-pyrimidine structure and cathepsin k inhibitory activity, and pharmaceutical uses
08/17/2011CN102159568A 2-[1H-Benzimidazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides and 2-[benzothiazol-2(3H)-ylidene]-2-(pyrimidin-2-yl)acetamides as kinase inhibitors
08/17/2011CN102159567A Process for the preparation of esomeprazole magnesium in a stable form
08/17/2011CN102159566A Pyridone and pyridazone analogues as gpr119 modulators
08/17/2011CN102159565A Benzimidazole compound in crystal form and salt thereof
08/17/2011CN102159554A Substituted 6- (1-piperazinyl) -pyridazines as 5-ht6 receptor antagonists
08/17/2011CN102159547A Heterocyclic carboxamide compounds
08/17/2011CN102159546A Aminopyridine kinase inhibitors
08/17/2011CN102159544A Pyridyl modulators of gamma-secretase
08/17/2011CN102159207A Substituted pyrrolidine-2-carboxamides
08/17/2011CN102159079A Heterocyclic compounds used as pesticides
08/17/2011CN102154005A Stilbene two-photon fluorescence probe for detecting zinc ion in cell
08/17/2011CN102153544A Preparation method and application of novel tyrosine kinase inhibitors
08/17/2011CN102153541A Bispyridyl benzimidazole compounds and synthesis method thereof
08/17/2011CN102153540A Chemokine receptor binding heterocyclic compounds with enhanced efficacy
08/17/2011CN102153539A 3-aminopyrrolidine derivatives as modulators of chemokine receptors
08/17/2011CN102153538A Benzocyclodirivative
08/17/2011CN102153508A 3,5-(E)-dibenzylidene-N-cyclopropyl piperidine-4-ketone and application of the 3,5-(E)-dibenzylidene-N-cyclopropyl piperidine-4-ketone in preparing antitumour drugs
08/17/2011CN102153502A Carbazole derivative and light-emitting element and light-emitting apparatus using carbazole derivative
08/17/2011CN102151273A 2,4,6-triamino-1,3,5-triazine derivative
08/17/2011CN102151270A Pyrimidine derivatives for the prevention of HIV infection
08/17/2011CN101407496B Method for synthesizing 3,5-disubstituted pyrazole
08/17/2011CN101184728B Peptide deformylase (PDF) inhibitors 4
08/17/2011CN101045724B Coupling method for preparing quinolone intermediate
08/17/2011CN101010296B Piperazine derivatives of alkyhydroxy indole
08/16/2011US7999110 Crystalline 2[[(4-methoxy-3-methyl-2-pyridinyl)-methyl]sulfinyl]-5-(1H-pyrrol-1-yl)-1H-benzimidazole (ilaprazole) having x-ray powder diffraction peak at 15.8 degrees; inhibiting gastric acid secretion; gastrointestinal inflammatory disorders; flowability, storage stability; dissolution rate
08/16/2011US7999100 Method for chiral inversion of (S)-(+)-and (R)-(−)-10,11-dihydro-10-hydroxy-5H-dibenz/b,f/azepine-5-carboxamide and optically enriched mixtures thereof
08/16/2011US7998986 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors
08/16/2011US7998985 1,5-diphenyl-3-pyridinylamino-1,5-dihydropyrrolidin-2-one as CB1 receptor modulator
08/16/2011US7998984 2-pyridone derivatives for the treatment of disease or condition in which inhibition of neutrophil elastase activity is beneficial
08/16/2011US7998981 Aminoaryl sulphonamide derivatives as functional 5-HT6 ligands
08/16/2011US7998979 Antibacterial quinoline derivatives
08/16/2011US7998969 Non-nucleoside reverse transcriptase inhibitors
08/16/2011US7998963 Arylpiperazine derivatives and uses thereof
08/16/2011US7998962 Enantiomers of 2'-Fluoralky1-6-nitroquipazine as serotonin transporter positron emission tomography imaging agents and antidepressant therapeutics
08/16/2011CA2624749C Pyrimidine amide compounds as pgds inhibitors
08/16/2011CA2590261C Aminopyrazine analogs for treating glaucoma and other rho kinase-mediated diseases and conditions
08/16/2011CA2557163C Substituted 1,2,3,4-tetrahydroisoquinoline derivatives
08/16/2011CA2556653C Tetrahydroquinolinones and their use as antagonists of metabotropic glutamate receptors
08/16/2011CA2482655C Substituted indoles
08/16/2011CA2400639C Compounds with 5-ht1a activity useful for treating disorders of the outer retina
08/11/2011WO2011097526A1 Compounds and compositions as protein kinase inhibitors
08/11/2011WO2011096461A1 Quinoline derivative
08/11/2011WO2011095997A1 Benzamide compounds as glucokinase activators and their pharmaceutical application
08/11/2011WO2011095984A1 A process for the preparation of amorphous esomeprazole
08/11/2011WO2011095885A1 An improved process for the preparation of piperaquine
08/11/2011WO2011095835A1 Highly pure imatinib or a pharmaceutically acceptable salt thereof
08/11/2011WO2011095625A1 1,2,4-triazine-4-amine derivatives
08/11/2011WO2011095459A1 Pyridazine derivatives, process for their preparation and their use as fungicides
08/11/2011WO2011095452A1 Aryl benzylamine compounds
08/11/2011WO2011095450A1 Cyclohexyl amide derivatives as crf receptor antagonists
08/11/2011WO2011095045A1 Pyridinone amide derivatives, preparation methods and medical uses thereof
08/11/2011WO2011042910A3 Optical resolution of substituted 2-(2- pyridinylmethylsulphinyl)-1h-benzimidazoles
08/11/2011WO2011012269A3 Method and substances for preparation of n-substituted pyridinium compounds
08/11/2011WO2010143170A3 Compounds useful for treating premature aging and in particular progeria
08/11/2011US20110196157 Optically active cyclic alcohol compound and method for preparing the same
08/11/2011US20110196153 Processes of synthesizing dihydropyridophthalazinone derivatives
08/11/2011US20110196150 Arylmethoxy Isoindoline Derivatives and Compositions Comprising and Methods of Using the Same