Patents
Patents for C07D 333 - Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom (32,883)
06/2000
06/13/2000US6075146 Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceuticals
06/13/2000US6075055 Excellent fungicidal activities with regard to rice blast and the like, while at the same time do not hinder desirable plant growth
06/13/2000US6075026 Certain substituted 1-aryl-3-piperazin-1'-yl propanones
06/13/2000CA2030732C Thiophene derivatives; process for preparing the same and pharmaceutical compositions containing them
06/13/2000CA1341024C Benzo-fused cycloalkane and oxa- and thia-, cycloalkane trans-1, 2-diamine derivatives
06/13/2000CA1341023C Peptide derivatives
06/08/2000WO2000032584A2 Nonsteroidal antiinflammatories
06/08/2000WO2000032582A1 Benzamide derivatives and their use as apob-100 secretion inhibitors
06/08/2000CA2353394A1 Benzamide derivatives and their use as apob-100 secretion inhibitors
06/08/2000CA2352367A1 Nonsteroidal antiinflammatories
06/07/2000EP1006107A2 Phthalamide derivatives, or salt thereof agrohorticultural insecticide, and method for using the same
06/07/2000EP1005493A1 Antiviral protease inhibitors
06/07/2000EP1005467A1 Benzothiophene derivatives as herbicides
06/07/2000EP1005340A1 Retinoid antagonists for prevention of surgical adhesions
06/07/2000CN1255491A Butyl benzene orthobenzol diacid amide derivative or its salt, garderning pesticide and its application method
06/07/2000CN1053182C Novel 9-amino-7-substituted-6-demethyl-6-deoxytetracyclines, its prepn. process and compsns. thereof
06/07/2000CN1053102C Application of benzothiophene derivative for medicines of inhibiting cartilage degradation
06/06/2000US6071970 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases
06/06/2000US6071969 Substituted aminoguanidines and methods of use thereof
06/06/2000US6071920 Bind to 5ht 1a receptors for treating disorders of the lower urinary tract; cns disorders; anxiolytic agents; antidepressants; hypotensive agents; sleep and eating disorders
06/06/2000US6071861 Dihalopropene compounds, insecticidal/acaricidal agents containing same, and intermediates for their production
06/06/2000US6071510 Modified amino acids and compositions comprising the same for delivering active agents
06/02/2000WO2000031036A1 Novel naphthalene derivatives
06/02/2000WO2000030684A1 Medicinal compositions for periodic administration
06/02/2000CA2352461A1 Pharmaceutical composition for periodic administration
05/2000
05/31/2000EP1003846A1 Protease inhibitors
05/31/2000EP1003730A1 2-benzoyl-cyclohexane-1,3-diones
05/31/2000EP1003719A2 Microbicidal n-sulfonylglycin alkynyloxyphenemethyl amide derivatives
05/31/2000EP1003495A1 Pharmaceutical compounds
05/31/2000EP0862549B1 Process for preparing optically active carboxylic acids
05/31/2000EP0751942B1 3-aryl-4-hydroxy-delta 3 -dihydrothiophenone derivatives
05/31/2000DE19856475A1 Nichtsteroidale Entzündungshemmer Nonsteroidal anti-inflammatory drugs
05/31/2000CN1255161A Protease inhibitors
05/31/2000CN1255115A Substituted 2-(3-alkenyl-benzoyl)-cyclohexane-1,3-diones
05/30/2000US6069258 Cosmetic preparations comprising photostable UV-A filters
05/30/2000US6069247 Reacting an acetylenecarboxy amide and an aryl or heterocyclyl halide or a group enhancing the electrophilicity of the atom to which it is attached for displacement; using a palladium compound catalyst, a base and an acid
05/30/2000US6069175 Administering to a mammal in need a therapeutically effective amount of a member selected from the 4-hydroxy tamoxifen, raloxifene, toremifene, centchroman, idoxifene to treat atherosclerosis
05/30/2000US6069166 Inhibitory activity against infiltration of eosionophils, and are useful as drugs for treating nasal blockage
05/30/2000US6069114 Herbicides for selectively controlling broad-leaved weeds and grass weeds in crops of useful plants
05/30/2000US6068834 Orally administering a melanins reducing oxy phenol compound to the mammal for lightening the mammalian skin; tyrosinase inhibitor
05/24/2000EP1001973A1 Compounds which inhibit leukocyte adhesion mediated by vla-4
05/24/2000EP1001927A2 Novel polyamine analogues as therapeutic and diagnostic agents
05/24/2000EP0671396B1 PROCESS FOR PRODUCING 2-SUBSTITUTED BENZO[b]THIOPHENE
05/24/2000CN1254337A N-hydroxy 4-sulfonyl butyramide compounds
05/24/2000CN1254328A Process for preparing substituted 2-3-dihydro-1-indanones
05/24/2000CN1254280A A regioselective alkylation process for preparing substituted benzo [b] thiophenes
05/24/2000CN1254255A Methods for reducing fibrinogen
05/23/2000US6066756 Phenylacetic acid derivatives, preparation thereof and intermediates therefor, and compositions containing them
05/18/2000WO2000027840A1 Process for racemization
05/18/2000WO2000027790A1 Mutilin compounds
05/18/2000WO2000004892A3 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions
05/17/2000EP1000934A2 Pesticidal and parasiticidal use of 1-aryl-1-(substituted thio, sulfinyl and sulfonyl)-2-nitroethane compounds
05/17/2000EP1000930A2 Tachykinin antagonists
05/17/2000EP1000619A2 Method for treating glaucoma
05/17/2000EP1000066A1 Fused 1,2,4-thiadiazine derivatives, their preparation and use
05/17/2000EP1000054A1 Oligo-thiophenes useful as antimetastatic agents, a preparation thereof and pharmaceutical compositions containing them
05/17/2000EP1000047A1 1-(n-phenylaminoalkyl)-piperazine derivatives substituted at position 2 of the phenyl ring
05/17/2000EP1000018A2 Urokinase inhibitors
05/17/2000EP0999834A1 Antithrombotic agents
05/17/2000EP0848701B1 O-benzyl oxime ether derivatives and their use in crop protection compositions
05/17/2000CN1253560A Sulfonamides for treatment of endothelin-mediated disorders
05/17/2000CN1253559A Sulfonyl divalent aryl alpha-hydroxamic acid compounds
05/17/2000CN1253556A Process for preparing benzothiophenes
05/17/2000CN1253555A Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and pharmaceutical compositions containing same
05/17/2000CN1253500A Polythiophene anti-tumor agents
05/17/2000CN1253474A Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds
05/17/2000CN1253019A Method for preparing medicine composition capable of inhibiting post infective virus proteinase
05/17/2000CN1052474C Process for preparing sulfamide
05/16/2000US6063956 Aryl and heteroarylcyclopropyl oxime ethers and their use as fungicides and insecticides
05/16/2000US6063798 Substituted N-methylenethioureas as pesticides
05/16/2000CA2289827A1 Pesticidal and parasiticidal use of 1-aryl-1-(substituted thio, sulfinyl and sulfonyl)-2-nitroethane
05/16/2000CA2126752C Benzopyran and related ltb4 antagonists
05/11/2000WO2000026219A1 Oxime derivatives and the use thereof as latent acids
05/10/2000EP0797578B1 Fungicides for the control of take-all disease of plants
05/10/2000CN1252799A N-heterocyclic derivatives as NOS inhibitor
05/10/2000CN1252790A N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
05/10/2000CN1252717A Intermediates and process for preparing benzo (b) thiophenes
05/10/2000CN1252713A N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
05/10/2000CN1052240C Method for preparing inhibitor of retroinfection viral protease
05/10/2000CN1052234C Fungicides for the control of take-all disease of plants
05/09/2000US6060508 Benzylamine derivatives, their preparation and their application in therapeutics
05/09/2000US6060492 Side effect reduction
05/09/2000US6060476 α- and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
05/04/2000WO2000024738A1 Process for preparing 3-(substituted phenyl)-5-thienyl or furyl)-1,2,4-triazoles and novel intermediates utilized therein
05/04/2000WO2000024732A1 Method of lithiating five-membered heterocycles
05/04/2000WO2000024710A1 N-(2-aryl-propionyl)-sulfonamides and pharmaceutical preparations containing them
05/04/2000WO2000006085A3 Compounds and methods
05/03/2000EP0997460A1 Benzothiophene compounds as antithrombotic agents and intermediates
05/03/2000EP0997459A1 Intermediates for preparing retroviral protease inhibiting compounds
05/03/2000EP0997458A1 Novel tricyclic compounds having saturated rings and medicinal compositions containing the same
05/03/2000EP0997455A1 Restricted 9-cis retenoids
05/03/2000EP0997147A1 Amino acid derivatives
05/03/2000EP0996614A1 Acrylonitrile compounds, process for their production and pesticides containing them
05/03/2000EP0996439A1 $g(b)-ALKOXYACRYLATES AGAINST MALARIA
05/03/2000EP0996434A1 Kappa agonist anti-pruritic pharmaceutical formulations and method of treating pruritus therewith
05/03/2000EP0861233B1 N-protected/n-substituted-beta-amino hydroxy sulfonates
05/03/2000EP0779884B1 Imidic acid derivatives and their use as pesticides
05/03/2000CN1252053A Cetp activity inhibitors
05/03/2000CN1051994C Isohydroxy oximino acid derivatives, preparation thereof and use as bactericide
05/03/2000CN1051990C Method for preparing ring-substituted 2-amino-1,2,3,4-tetra-hydronaphthalenes