Patents
Patents for C07D 333 - Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom (32,883)
05/2001
05/16/2001EP0798288B1 Triciclic compounds
05/16/2001EP0695300B1 Novel 1,3-benzodioxole and 1,2-dialkoxybenzene derivatives as ocular hypotensive agents
05/16/2001CN1295569A Process for producing benzothiophenecarboxylic acid amide derivatives
05/16/2001CN1295548A Novel tricyclic compound
05/16/2001CN1295471A Antagonists for treatment of CD11/CD18 adhesion receptor mediated disorders
05/16/2001CN1295065A Phenyl heterocyclic compound used as epoxy enzyme -2 inhibitor
05/16/2001CN1295064A Novel tricyclic compound and medicine composition containing the same
05/16/2001CN1294913A Pharmaceutical use of compound
05/15/2001US6232467 Biosynthesis of an amine with ketone and boron compound; compoundlibraries
05/15/2001US6232342 Protease inhibitors
05/15/2001US6232322 Biphenyl oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia
05/15/2001US6232314 Arylalkylpiperazine compounds as antioxidants
05/15/2001US6232089 CD23 processing enzyme preparation
05/10/2001WO2001032646A2 Sulfonamide derivatives
05/10/2001WO2001032604A1 Activators of soluble guanylate cyclase
05/10/2001WO2001032602A1 Diaryl-enynes
05/10/2001DE19953804A1 Novel tetrahydrothiophene compounds such as 5-propyl-tetrahydrothiophene-2-carboxylic acid-(4-(5-undecyl-pyrimidine-2-yl)-phenyl)-ester are useful as dopants for improving the properties of liquid crystal mixtures
05/10/2001CA2389773A1 Activators of soluble guanylate cyclase
05/10/2001CA2387660A1 Diaryl-enynes as glycine transport inhibitors
05/09/2001EP1097382A2 Imidazoline receptor binding compounds
05/09/2001EP1097158A2 Ligands for metals and metal-catalyzed processes
05/09/2001EP1097129A1 N-benzocycloalkyl-amide derivatives and their use as medicaments
05/09/2001EP1097128A1 Imidamide derivatives
05/09/2001EP1097117A2 Aryl vinyl ether derivatives and their use as herbicides
05/09/2001CN1294577A 钾通道抑制剂 Potassium channel inhibitors
05/09/2001CN1065528C Thiol and sulfur-contg. O-(meth) acrylate compound and use thereof
05/08/2001US6228942 Dehydration to esterify or amidate surface of oxidized or aminated carbon powder or fiber suspended in solution containing a monomer or polymer having amine, hydroxy, and/or viny ether groups
05/08/2001US6228881 Aromatic heterocyclic compounds and their use as anti-inflammatory agents
05/08/2001US6228878 Administering indolin-5-one derivatives; inhibiting formation of abnormally phosphorylated paired helical filament epitopes
05/08/2001US6228848 3-(1-propen-3-oxo)-5,6-dihydronaphthalene derivatives; side effect reduction
05/08/2001CA2167040C New alkylated (hetero)cyclic compounds; process for preparing the same and pharmaceutical compositions containing them
05/08/2001CA2032330C Benzyl-substituted rhodanine derivatives for treating inflammatory bowel disease
05/03/2001WO2001030333A2 Tissue factor antagonists and methods of use thereof
05/03/2001WO2001030149A1 Novel succinic acid metallo-beta-lactamase inhibitors and their use in treating bacterial infections
05/03/2001WO2001030148A1 Novel substituted succinic acid metallo-beta-lactamase inhibitors and their use in treating bacterial infections
05/03/2001WO2000066546A3 Monofluoroalkyl derivatives
05/03/2001CA2388077A1 Novel succinic acid metallo-beta-lactamase inhibitors and their use in treating bacterial infections
05/03/2001CA2387857A1 Tissue factor antagonists and methods of use thereof
05/02/2001EP1095654A2 Use of raloxifene and its analogs for the manufacture of a medicament for the Inhibition of LDL oxidation and atherosclerosis
05/02/2001EP1095016A1 Sulfur substituted sulfonylaminocarboxylic acid n-arylamides, their preparation, their use and pharmaceutical preparations comprising them
05/02/2001EP1095015A2 Sulfonylamino carboxylic acid n-arylamides as guanylate cyclase activators
05/02/2001EP0984959A4 Aromatic sulfonyl alpha-hydroxy hydroxamic acid compounds
05/02/2001EP0983257A4 Aromatic sulfonyl alpha-cycloamino hydroxamic acid compounds
05/02/2001EP0973392A4 Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds
05/02/2001CN1293666A Benzenesulfonamide-derivatives and their use as medicaments
05/02/2001CN1293192A New benzothiophene, benzofuran and indole compounds, preparation method therefor and medicine composition containing same
05/01/2001US6225346 Tyrphostin like compounds
05/01/2001US6225336 For therapy of systemic mastocytosis and disorder of systemic mast cell activation as well as tracheal contraction, asthma, allergic rhinitis, allergic conjunctivitis, urticaria, ischemic reperfusion injury, and inflammation
05/01/2001US6225334 Glyoxylic acid derivatives
05/01/2001US6225328 Adamantyl-substituted retinoids and pharmaceutical/cosmetic compositions comprised thereof
05/01/2001US6225312 Piperazine and piperidine compounds
04/2001
04/26/2001WO2001029024A2 Method for preparing a thiophene derivative
04/26/2001WO2001029019A1 Method for preparing a benzofuran or benzothiophene compound
04/26/2001WO2001029017A2 N-SUBSTITUTED 3-AMINO-2,2-DI-C-ALKYL-1,4-BUTYROLACTONES AND 1,4-THIOBUTYROLACTONES FOR USE AS PROMOTER OF η-AMINOBUTYRIC ACID ACTIVITY AND FOR TREATING NERVOUS DISORDERS AND PREPARATION METHOD
04/26/2001WO2001028987A1 Benzylcycloalkyl amines as modulators of chemokine receptor activity
04/26/2001WO2001028974A2 Intermediates for making a benzofuran or benzothiophene derivative nitrated in position 5 and uses thereof
04/26/2001WO2001028537A2 Bissulfonamide derivatives as enzyme inhibitors
04/26/2001WO2000061574A3 Method for producing thiophenyl-amidines
04/26/2001WO2000055125A3 N-cyanomethyl amides as protease inhibitors
04/26/2001US20010000511 Treatment of skin disorders, inflammation, nerve system disorders, cancer
04/26/2001CA2387974A1 N-substituted 3-amino-2,2-di-c-alkyl-1,4-butyrolactones and 1,4-thiobutyrolactones for use as promoter of .gamma.-aminobutyric acid activity and for treating nervous disorders andpreparation method
04/26/2001CA2387713A1 Intermediates for making a benzofuran or benzothiophene derivative nitrated in position 5 and uses thereof
04/26/2001CA2387593A1 Enzyme inhibitors
04/26/2001CA2384240A1 Benzylcycloalkyl amines as modulators of chemokine receptor activity
04/25/2001EP1093456A2 Naphtho- and dihydrobenzo-thiophene derivatives as cytotoxic antitumor agents
04/25/2001CN1292779A Halogenated amidino amino acid derivatives useful as nitric oxide synthase inhibitors
04/25/2001CN1292698A Glycine transport inhibitors
04/24/2001US6222048 Diaryl-2-(5H)-furanones as Cox-2 inhibitors
04/24/2001US6222034 As serotinin receptor antagonists; for therapy of depression, central nervous system disorders
04/24/2001US6221914 Sulfonamide bridging compounds that inhibit tryptase activity
04/24/2001US6221902 Biphenyl sulfonyl aryl carboxylic acids useful in the treatment of insulin resistance and hyperglycemia
04/24/2001US6221898 Anticoagulants
04/24/2001US6221889 Interleukin antagonist; skin disorders, respiratory system disorders, rheumatic disorders
04/24/2001US6221869 N-aminoalkyldibenzothiophenecarboxamides new dopamine receptor subtype specific ligands
04/24/2001US6221865 Inhibitors of protein farnesyltransferase and protein geranylgeranyltransferase.
04/24/2001US6221838 Administering an analog of an obesity protein.
04/24/2001CA2078520C Trimetazidine derivatives, process for preparing same and pharmaceutical compositions containing same
04/19/2001WO2001027099A2 Bicyclic compounds composition and method for stabilizing the same
04/19/2001WO2001027084A1 Beta disubstituted metalloprotease inhibitors
04/19/2001WO2001027068A1 Biaryl ether derivatives useful as monoamine reuptake inhibitors
04/19/2001WO2001026807A1 Supported ferrocene-based catalysts for selective aldehyde hydrogenation
04/19/2001CA2386485A1 Beta disubstituted metalloprotease inhibitors
04/19/2001CA2383653A1 Supported ferrocene-based catalysts for selective aldehyde hydrogenation
04/18/2001EP1092716A2 Derivatives of benzothiophenes, benzofurans and indoles, method for their preparation and pharmaceutical compositions containing them
04/18/2001EP1092714A2 Process for the synthesis of benzo[b]thiophenes
04/18/2001EP1091952A1 Thiophene and furan 2,5-dicarboxamides useful in the treatment of cancer
04/18/2001EP0771201B1 Use of 2-phenyl-3-aroylbenzothiophenes for the preparation of a medicament for inhibiting primary endometrial hyperplasia
04/18/2001EP0765321B1 2-amino-3-aroyl-benzo beta thiophenes and method of making the same
04/18/2001CN1291981A Thiophene nitrone compounds
04/18/2001CN1291973A N-sulphonyl and N-sulphinyl phenylglycinamide
04/18/2001CN1064674C Alkoxyaryl compounds, their process of preparation and pharmaceutical compositions which contain them
04/17/2001US6218429 Tricyclic compounds, their production and use
04/17/2001US6218426 For therapy of mammalian reproductive disorders and steroid hormone-dependent tumors as well as for regulating fertility, where suppression of gonadotropin release is indicated
04/17/2001US6218425 Useful in the treatment of estrogen-related disorders such as osteoporosis, hyperlipidemia, estrogen-related breast cancer, uterine fibrosis, endometriosis, and restenosis
04/17/2001US6218394 4-Aryl-1-(indanmethyl, dihydrobenzofuranmethyl or dihydrobenzothiophene-methyl) piperazines
04/17/2001CA2196054C Dihydrobenzofuran and related compounds useful as anti-inflammatory agents
04/12/2001WO2001025208A1 Pyridinium derivatives for the management of aging-related and diabetic vascular complications, process for their preparation and therapeutic uses thereof
04/12/2001WO2001025198A1 Method for improving the solubility of tricyclic amino alcohol derivatives
04/12/2001WO2001025197A1 Antifungal enediynes
04/12/2001WO2001025190A1 Novel diarylamide derivatives and use thereof as medicines