Patents
Patents for C07D 333 - Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom (32,883)
01/2005
01/20/2005CA2529739A1 Aspartyl protease inhibitors
01/19/2005EP1497672A2 Ultrasonic doppler effect speed measurement
01/19/2005EP1497278A1 Heterocyclic amide derivatives as cytokine inhibitors
01/19/2005EP1497270A1 Amide compounds and methods of using the same
01/19/2005EP1497245A1 PROCESS FOR THE PREPARATION OF NONRACEMIC SYN-1-(4-HYDROXY-PHENYL)-2-(4-HYDROXY-4-PHENYL.PIPERIDIN-1Yl)-1-PROPANOL COMPOUNDS
01/19/2005EP1496896A1 Inhibitors of akt activity
01/19/2005EP1334095B1 Process for the preparation of pgd2 antagonist
01/19/2005CN1568326A Method for producing, via organometallic compounds, organic intermediate products
01/19/2005CN1568322A Pharmaceutically active sulfonamide derivatives bearing both lipophilic and ionisable moieties as inhibitors of protein junkinases
01/19/2005CN1568303A Oligofluorenylene compounds
01/19/2005CN1568298A Luminous compounds and labeling reagents using the same
01/19/2005CN1566096A Prostaglandin agonists and their use to treat bonedisorders
01/19/2005CN1185226C Intermediate for preparing benzothiophene amide derivate
01/19/2005CN1185225C Improved process for preparing nitrogen-substituted aminotetralins
01/18/2005US6844367 Benzamides and related inhibitors of factor Xa
01/18/2005US6844358 Protein tyrosine phosphatase inhibitors; benzofuran-3-yl- or benzothiophen-3-yl derivatives; containing pyridinyl, imid-azoyl, oxazoyl or thiazoyl functionality
01/13/2005WO2005003116A1 Process for preparing raloxifene hydrochloride
01/13/2005WO2005003115A1 Thiophene amino acid derivatives, process for preparing them and pharmaceutical compositions containing them
01/13/2005WO2005003114A1 5-fluoro-thiopen-compounds,the process for their preparation,the pharmaceutical compositions containing them and their use as metallopotenases inhibitors
01/13/2005US20050010058 Metallocene compounds and process for the preparation of propylene polymers
01/13/2005US20050009920 Taxol enhancer compounds
01/13/2005US20050009912 2-Amino-bicyclo[3.1.0]hexane-2,6-dicarboxylic acid derivatives; treatment of neurological or psychiatric disorders, such as anxiety disorder; greatly enhanced oral exposure
01/13/2005US20050009907 Aryl-carbaldehyde oxime derivatives and their use as estrogenic agents
01/13/2005US20050009871 Ubiquitin ligase inhibitors
01/13/2005US20050009812 Remedies for stress diseases comprising mitochondrial benzodiazepine receptor antagonists
01/13/2005US20050009804 N-heterocyclyl- or cycloalkyl-N-(2-carboxy-5-aryl-3-thiophenyl)cycloalkanecarboxamides, e.g., 5-(3-fluorophenyl)-3-[isopropyl-(4-methylcyclohexanecarbonyl)amino]-thiophene-2-carboxylic acid; especially for prevention and treatment of HVC
01/13/2005DE10328400A1 One-pot synthesis of carbocyclic or heterocyclic compounds, especially pyrimidine useful as components of natural products or drugs, from acid halide, alkyne and active hydrogen compound
01/13/2005CA2549354A1 Process for preparing raloxifene hydrochloride
01/12/2005EP1495015A1 3-aminophenol derivatives and dyes that contain these compounds while serving to dye keratin fibers
01/12/2005EP1494989A2 Compounds that modulate ppar activity and methods for their preparation
01/12/2005EP1171423B1 Carbamic acid derivatives and their use as metabotropic glutamate receptor ligands
01/12/2005EP1030851B1 Hydroxamic and carboxylic acid derivatives having mmp and tnf inhibitory activity
01/12/2005CN1564811A Acylsulfonamides as inhibitors of steroid sulfatase
01/11/2005US6841682 Prevent binding of adrenergenic receptors
01/11/2005US6841674 N-heterocyclic derivatives as NOS inhibitors
01/11/2005US6841673 Enzyme inhibitors; antiinflammatory agents; rheumatic diseases; antidiabetic agents
01/11/2005US6841669 Functionalized thiophene oligomers and their use as fluorescent markers
01/11/2005US6841569 Treatment of central nervous system disorders; anticonvulsants, antiepileptics, neuroprotective agents and muscle relaxants
01/11/2005US6841553 Contorlling fertility
01/11/2005US6841499 Homogeneous rhodium complexes bearing phosphines
01/11/2005US6840965 P-aminophenols and colorants containing said compounds
01/06/2005WO2005002288A1 Conjugate molecule, electroluminescent element using the same and electronic apparatus using the electroluminescent element
01/06/2005WO2005000839A1 Process for producing 3-acylaminobenzofuran-2-carboxylic acid derivative
01/06/2005WO2005000834A1 Pentafluoroalkanesulfinyl naphthalenes and related estrogen receptor modulators
01/06/2005WO2005000833A1 Immunosuppressant compounds and compositions
01/06/2005WO2005000829A1 Cannabinoid receptor modulator
01/06/2005WO2005000790A1 2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid derivative
01/06/2005WO2005000781A1 Biaryloxymethylarene-carboxylic acids
01/06/2005WO2005000406A2 Treatment of amyloid- and epileptogenesis-associated diseases
01/06/2005WO2005000309A2 Chemical compounds
01/06/2005US20050004252 Light emitting polymer
01/06/2005US20050004251 Light emitting polymer
01/06/2005US20050004212 Antitumor/cancer activity; topoisomerase I inhibitors
01/06/2005US20050004211 Inhibiting topoisomerase I; blocking S or G2/M phase of tumor and/or cancer cells
01/06/2005US20050004115 such as 4-(4-(2-Fluorobenzyloxy)phenyl)-4-oxobutyric acid; for treatment of insulin resistance syndrome, diabetes, hyperlipidemia, fatty liver disease, cachexia, obesity, atherosclerosis and arteriosclerosis
01/06/2005CA2672071A1 Process for preparing 3-acylaminobenzofuran-2-carboxylic acid derivative
01/06/2005CA2556706A1 Treatment of amyloid- and epileptogenesis-associated diseases
01/06/2005CA2531020A1 Cannabinoid receptor modulator
01/06/2005CA2530377A1 Process for preparing 3-acylaminobenzofuran-2-carboxylic acid derivative
01/06/2005CA2530309A1 Process for the preparation of insulin sensitizer and intermediate compound thereof
01/06/2005CA2529875A1 Biaryloxymethylarene-carboxylic acids
01/06/2005CA2524048A1 Immunosuppressant compounds and compositions
01/05/2005EP1493743A1 Substituted bipiperidine intermediates and derivatives thereof
01/05/2005EP1493742A1 Amine and amide derivatives as ligands for the neuropeptide Y Y5 receptor useful in the treatment of obesity and other disorders
01/05/2005EP1493741A2 Benzo[b]thiophene compounds, intermediates, processes, compositions and methods
01/05/2005EP1493740A1 5-fluoro-thiophene compounds, the process for their prepartion, the pharmaceutical compositions containing them and their use as metalloproteinases inhibitors
01/05/2005EP1493739A1 Thiophene derivatives of aminoacids, process for the preparation thereof and compositions containing them
01/05/2005EP1492795A1 1- or 3-thia-benzonaphthoazulenes as inhibitors of tumour necrosis factor production and intermediates for the preparation thereof
01/05/2005EP1492794A1 Piperazine substituted aryl benzodiazepines and their use as dopamine receptor antagonists for the treatment of psychotic disorders
01/05/2005EP1492783A1 4,5,6,7-tretrahydrobenzo(b) thiophene derivatives and methods for medical intervention against mycrobacterial infections
01/05/2005EP1492781A1 N,n'-disubstituted piperazine compounds and the use of the same as analgesics
01/05/2005EP1492534A1 Carbamic acid compounds comprising a piperazine linkage as hdac inhibitors
01/05/2005EP1027051B1 Antithrombotic agents
01/05/2005CN1183126C Dihydrobenzofuran and related compounds useful as anti-inflammatory agents
01/05/2005CN1183119C Arylpiperzines as metalloproteinase inhibiting agents (MMP) and their use
01/05/2005CN1183107C Alkynyl containing hydroxamic acid compounds as TACE inhibitors
01/05/2005CN1183098C 3-amino-3-aryl-1-alcohol derivatives and preparation and use thereof
01/04/2005US6838584 Estrogen receptor modulators
01/04/2005US6838483 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
01/04/2005US6838472 Substituted urea retinoid agonists
12/2004
12/30/2004US20040267025 Compounds for the treatment of metabolic disorders
12/30/2004US20040266857 11,12-dehydro-naphtho[1,2-b]thioxane-9,10-dione derivatives; antiproliferative agents; psoriasis, cancer
12/30/2004US20040266856 Biaryloxymethylarenecarboxylic acids as glycogen synthase activator
12/30/2004US20040266827 Convergent asymmetric route to produce a key intermediate towards the synthesis of a garft inhibitor
12/30/2004US20040266789 Substituted amino carboxylic acids
12/30/2004US20040266782 Cyclic amine derivatives-CCR-3 receptor antagonists
12/30/2004US20040266764 Hydroxamic acid derivatives
12/29/2004WO2004113331A1 Novel compounds that modulate pparϝ type receptors, and use thereof in cosmetic or pharmaceutical compositions
12/29/2004WO2004113328A1 Convergent asymmetric synthesis route to produce a key intermediate towards the synthesis of a garft inhibitor
12/29/2004WO2004113289A2 Glycosidase inhibitors and methods of synthesizing same
12/29/2004WO2004113282A1 Therapeutic agents
12/29/2004WO2004113281A1 Tricyclic derivatives or pharmaceutically acceptable salts thereof, their preparations and pharmaceutical compositions containing them
12/29/2004WO2004113273A1 Pesticidally active ketone and oxime derivatives
12/29/2004WO2004113258A1 Carbon-carbon bond forming reaction
12/29/2004WO2004099175A3 Blockers of the quorum sensing system of gram-negative bacteria
12/29/2004WO2004002940A8 Inhibitors of hcv ns5b polymerase
12/29/2004EP1491538A1 Anti-mitotic agents which inhibit tubulin polymerization
12/29/2004EP1491190A1 Decomposition inhibitor for extracellular matrix of cartilage
12/29/2004EP1490339A1 Novel chalcone derivatives and uses thereof
12/29/2004EP1490317A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof