Patents
Patents for C07D 333 - Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom (32,883)
02/2006
02/02/2006US20060025404 Such as 1-(4-{[1-(1-methylethyl)-4-piperidinyl]oxy}phenyl)-4-{[4-(methylsulfonyl)phenyl]carbonyl}piperazine; neurodegenerative disorders including Alzheimer's disease; allergic rhinitis
02/02/2006US20060024775 Substrates for o6-alkylguanina-dna alkyltransferase
02/02/2006CA2575359A1 Piperazine derivatives useful for the treatment of gastrointestinal disorders
02/02/2006CA2574305A1 1, 1a, 5, 5a-tetrahydro-s-thia-cyclopropa'a! pentalenes: tricyclic thiophene derivatives as s1p1/edg1 receptor agonists
02/02/2006CA2573777A1 Novel cyclohexane derivative, prodrug thereof and salt thereof, and therapeutic agent containing the same for diabetes
02/02/2006CA2571587A1 Quaternary salt ccr2 antagonists
02/01/2006EP1620431A1 3-carbonylaminothiophenes and their use as fungicides
02/01/2006EP1620425A1 Substituted 3-cyanothiophene acetamides as glucagon receptor antagonists
02/01/2006EP1620424A2 Improved jasmine aromachemicals
02/01/2006EP1620397A1 Hydroxamic acids useful in the treatment of hyper-proliferative disorders
02/01/2006EP1620086A1 Compounds that modulate ppar activity and methods of preparation
02/01/2006EP1476419B1 N-biphenylmethyl aminocycloalkanecarboxamide derivatives
02/01/2006EP1370548B1 P-thienylbenzyl-amides serving as agonists of angiotensin-(1-7)-receptors, method for the production thereof, their use and pharmaceutical preparations containing the same
02/01/2006CN1729184A Preparation of heterocyclic ketones
02/01/2006CN1729183A Novel lapachone compounds and methods of use thereof
02/01/2006CN1729181A Novel tricyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them
02/01/2006CN1729158A Adamantyl acetamides as 11-beta hydroxysteroid dehydrogenase inhibitors
02/01/2006CN1729157A Substituted amino phenylacetic acids, derivatives thereof, their preparation and their use as cyclooxygenase 2 (COX-2) inhibitors
02/01/2006CN1727339A Tricyclic compounds, their production and use
02/01/2006CN1239495C Fungicides for control of take-all disease of plants
02/01/2006CN1239472C HIV integrase inhibitors
01/2006
01/31/2006US6992095 Stilbene compounds comprising an adamantyl group, compositions and methods thereof
01/31/2006CA2130723C Process for preparing y-mercaptocarboxylic acid derivatives
01/26/2006WO2006007896A1 Novel o-aminophenol derivatives and colorants containing said compounds
01/26/2006US20060020135 Long chain aliphatic alcohol derivatives and methods of making and using same
01/26/2006US20060020041 substituted ethylene diamines such as N-Geranyl-N'-(2-adamanthyl)ethane-1,2-diamine, used for the treatment of leprosy or tuberculosis caused by mycobacterial infections
01/26/2006US20060020039 E.g., 3-(2-(4-[(2-aminosulfonyl)phenyl]benzoylamino)phenoxy)benzamidine; 7-(2-(4-[(2-aminosulfonyl)phenyl]benzoylamino)-4-fluorophenoxy)1-aminoisoquinoline; and 3-(2-(4-[(2-aminosulfonyl)phenyl]phenylaminocarbonyl-4-chlorophenoxy)benzamidine; highly selective
01/26/2006US20060020019 Such as 1-(3,5-bis(trifluoromethyl)benzyloxy)-3-(dimethylamino)-2-phenylpropan-2-ol, trifluoroacetic acid salt for treating a disorder associated with aberrant levels of tachykinins or serotonin; depression, obsessive compulsive disorder, bulimia, or panic disorder
01/26/2006US20060020003 Biphenyloxy-acids
01/26/2006US20060019999 Specific inhibitors of one or more isoforms of nitric oxide synthase; 3-[[2-amino-1-phenylethyl]thio]-5-methyl-2-thiophenecarbonitrile; antiinflammatory agent; pain
01/26/2006CA2574237A1 Modulators of alpha7 nicotinic acetylcholine receptors and therapeutic uses thereof
01/26/2006CA2574217A1 Diamine derivative, process of preparation thereof, and fungicide comprising diamine derivative as an active ingredient
01/26/2006CA2572753A1 Novel o-aminophenol derivatives and colorants containing said compounds
01/25/2006EP1618087A2 Antibacterial agents
01/25/2006EP1618084A1 Bioreductively activated stilbene prodrugs
01/25/2006EP1097158B1 Ligands for metals and metal-catalyzed processes
01/25/2006CN1726204A Enantiomers of thiophene hydroxamic acid derivatives and their use as hdac inhibitors
01/25/2006CN1726201A Substituted piperazines,(1,4) diaszepines, and 2,5-diazabicyclo (2.2.1)iieptanes as histamine h1 and/or h3 antagonists or histamine h3 reverse antagonists
01/25/2006CN1238337C Pesticide
01/24/2006US6989402 Thyroid receptor ligands and method II
01/24/2006US6989384 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
01/19/2006US20060014836 e.g. 1-(Benzofuran-2-carbonyl-3-(3-phenoxy-phenyl)-thiourea;viricides; hepatitis virus
01/19/2006US20060014830 2-amino-2-oxoethyl 1-(4'-fluoro-1,1'-biphenyl-4-yl)cyclopropylmethylcarbamate and 2-(methylamino)-2-oxoethyl 1-(4'-fluoro-1,1'-biphenyl-4-yl)cyclopropylmethylcarbamate; fatty acid amide (FAAH) hyrdrolase inhibitors; analgesics; neuropathic pain;psychological disorders; anticarcinogenic agents; AIDS
01/19/2006US20060014822 1,2,4-Triaminobenzene derivatives useful for treating disorders of the central nervous system
01/19/2006US20060014806 Dihalo-allyloxy-phenol derivatives having pesticidal activity
01/19/2006US20060014803 Diarylselenide compounds and their use in human or veterinary medicine and in cosmetics
01/19/2006US20060014797 [2-(2-Dimethylamino-ethyl)-benzo[b]thiophen-3-yl]-(4-fluoro-phenyl)-methanone; for inhibiting one or more histamine receptors, such as the histamine H1 receptor; improved selectivity, a quicker onset of action, a shorter half-life and/or the ability to penetrate the CNS
01/19/2006US20060014794 CXCR1 and CXCR2 chemokine antagonists
01/19/2006US20060014779 3-Aryloxy/thio-3-substituted propanamines and their use in inhibiting serotonin and norephinephrine reuptake
01/19/2006US20060014752 Heterocyclic anti-epileptogenic agents and methods of use thereof
01/19/2006US20060014743 Methods of preventing bacterial infections with florfenicol-type antibiotics
01/18/2006EP1616865A1 Inhibition of p38 kinase using symmetrical and unsymmetrical diphenyl ureas
01/18/2006EP1615907A1 5-amino-2-carbonylthiophene derivatives for use as p38 map kinase inhibitors in the treatment of inflammatory diseases
01/18/2006EP1615904A2 Substituted benzosulphonamide as potentiators of glutamate receptors
01/18/2006EP1615892A2 Benzamide 2-hydroxy-3-diaminoalkanes
01/18/2006EP1268096B1 Extrusion die
01/18/2006EP1210327B1 New vitamin d derivatives with cyclic substructures in the side chains, method and intermediates for their production and their use in the preparation of medicaments
01/18/2006CN1723207A Inhibitors of histone deacetylase
01/18/2006CN1723192A Arylene-carboxylic acid (2-amino-phenyl)-amide derivatives as pharmaceutical agents
01/18/2006CN1723010A Novel skin lightening agents, compositions and methods
01/18/2006CN1237059C Novel process for preparing 5-aminomethyl-2-thiophenecarbonitrile HC1 by one-pot reaction
01/18/2006CN1237051C Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
01/12/2006WO2006003194A1 Process for preparing amines and a carboxamide thereof
01/12/2006WO2006003096A1 Condensed thiophene derivatives and their use as cyclic glp-1 agonists
01/12/2006WO2005094810A3 Novel pharmaceutical compositions
01/12/2006US20060009528 Cannabinoid receptor ligands
01/12/2006US20060009511 N-(2-arylethyl) benzylamines as antagonists of the 5-ht6 receptor
01/12/2006US20060006365 Derivatives of SBF and the corresponding radical anions for use in components for molecular electronics, in particular for the molecular-based computational systems, for the OLEDs and for non-linear optics
01/12/2006US20060005320 N-alkylheteroaryl secondary para-phenylenediamine and composition comprising such a para-phenylenediamine
01/11/2006EP1614678A2 Sulfur substituted sulfonylaminocarboxylic acid N-heteroarylamides, their preparation, their use and pharmaceutical preparations comprising them
01/11/2006EP1614676A1 Compound inhibiting in vivo phosphorus transport and medicine containing the same
01/11/2006EP1613622A1 Oxime derivatives and their use as pharmaceutically active agents
01/11/2006EP1613612A2 Bioreductively-activated prodrugs
01/11/2006EP1613303A1 Substituted p-diaminobenzene derivatives
01/11/2006EP1412347B1 Process for the preparation of heterocyclic pentalene derivatives
01/11/2006EP1338596B1 processes for the preparation of carbapenem-type antibacterial agents
01/11/2006EP1256342B1 Hypoglycemics comprising organic zinc (ii) complexes
01/11/2006EP1056732B1 4-aminothiazole derivatives, their preparation and their use as inhibitors of cyclin-dependent kinases
01/11/2006CN1720332A Substrates for O6-alkylguanine-DNA alkyltransferase
01/11/2006CN1720245A Oxime ester photoinitiators with heteroaromatic groups
01/11/2006CN1720242A Synthetic lactone formulations and method of use
01/11/2006CN1235870C Novel use of phenyl hetero alkylamine derivatives
01/10/2006US6984738 Reduction, catalytic hydrogenation
01/10/2006US6984737 Di(het)arylaminothiophene derivatives
01/10/2006US6984660 To treat and/or prevent hypertension, cardiac hypertrophy, cardiac insufficiency, coronary heart diseases such as angina pectoris, and endothelial dysfunction or endothelial damage as a consequence of atherosclerotic processes or diabetes
01/10/2006US6984647 Antiinflammatory agents; analgesics; antiarthritic agents
01/10/2006US6984637 Cyclic amine derivatives-CCR-3 receptor antagonists
01/10/2006US6984462 Organic electroluminescent devices using double-spiro organic compounds
01/10/2006CA2383332C Benzisoxazolyl-, pyridoisoxazolyl- and benzthienyl-phenoxy derivatives useful as d4 antagonists
01/05/2006WO2006000323A1 Novel hexafluoroisopropanol derivatives
01/05/2006WO2006000288A1 Phenylcarboxylic acid derivatives and use thereof for the treatment of diabetes
01/05/2006US20060004220 by phosgenation of an aminobenzoylsulfamic acid amide intermediate; prepared from a p-nitrobenzoyl chloride or benzoate and a sulfamic acid amide and reducing the nitrobenzoylsulfamic acid amide; isocyanates are crop protection agents
01/05/2006US20060004093 obesity; antidiabetic agents; Alzheimer's disease; Huntington's disease;schizophrenia; anticancer agents; psoriasis; antiepileptic agents; strokes
01/05/2006US20060004068 Novel hexafluoroisopropanol derivatives
01/05/2006US20060004066 Method for treating ADAMTS-5-associated disease
01/05/2006US20060004063 Inhibitors of HCV NS5B polymerase
01/05/2006US20060004062 Compounds for inhibiting insulin secretion and methods related thereto
01/05/2006US20060004048 Novel biaromatic compounds which activate PPARgamma type receptors and cosmetic/pharmaceutical compositions comprised thereof
01/05/2006US20060004016 Administering (-)3-((S)-((2S,5R)-4-allyl-2,5-dimethyl-1-piperazinyl)(3-thienyl)methyl)phenol or a pharmaceutically acceptable salt thereof for reducing ischemic damage
01/05/2006US20060002853 Stilbene derivatives and their use for binding and imaging amyloid plaques