Patents
Patents for C07D 309 - Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings (12,815)
04/2003
04/03/2003US20030064935 Amino acid complexes of C-aryl glucosides for treatment of diabetes and method
04/02/2003EP1298115A1 Process for the preparation of polyhydric alcohols
04/02/2003EP1296716A2 New formulation
04/02/2003EP0807617B1 Process for preparing 1,5-pentanediol derivative
04/02/2003CN1407990A C-aryl glucoside sgltz inhibitors
04/02/2003CN1406938A Lactonization in course of preparing lovastatin or similarities
04/01/2003US6541655 Catalytic compositions and methods for asymmetric allylic alkylation
04/01/2003US6541511 Treatment and prophylaxis of hypercholesterolemia and of various cardiac disorders.
04/01/2003US6541489 Excellent inhibitory activity of one or more matrix metalloprotease (MMP) enzymes, such as MMP-2, MMP-9, and MMP-13, while exhibiting substantially less inhibition at least of MMP- 1
03/2003
03/27/2003WO2003024975A1 Laulimalide-derivatives, their use and process for the production of laulimalide and laulimalide-derivatives
03/27/2003WO2003024949A1 Dna-pk inhibitors
03/27/2003WO2003024529A1 Simplified sarcodictyn derivatives as anti-tumor agents
03/27/2003WO2002098854A3 Process for preparing chiral diol sulfones and dihydroxy acid hmg coa reductase inhibitors
03/27/2003WO2002060859A3 Cyclic derivatives as modulators of chemokine receptor activity
03/27/2003US20030060633 Asymmetric synthesis of kavalactones
03/27/2003CA2460244A1 Simplified sarcodictyn derivatives as anti-tumor agents
03/27/2003CA2454023A1 Dna-pk inhibitors in the treatment of retroviral mediated diseases
03/26/2003EP1295886A1 Laulimalide-derivates, their use and process for the production of laulimalide and laulimalide-derivates
03/26/2003EP1294706A1 A process for lactonization to produce simvastatin
03/26/2003EP0882113B1 Process for preparing compositions useful as intermediates for preparing lubricating oil and fuel additives and derivatives thereof
03/26/2003CN1406283A Method of purifying a fermentation broth
03/25/2003US6537527 Skin lightening compositions
03/20/2003WO2003022841A1 Intermediates for preparing neuraminidase inhibitor conjugates
03/20/2003WO2003022787A1 Method for preparing unsaturated fatty hydroxy-acids and esters thereof, their use in pharmaceutical and/or cosmetic compositions
03/20/2003US20030055246 Serine protease inhibitors
03/20/2003US20030055035 Useful in hyperpolarizing cell membranes, opening potassium channels, relaxing smooth muscle cells, and inhibiting bladder contractions
03/20/2003CA2459760A1 Method for preparing unsaturated fatty hydroxy-acids and esters thereof, their use in pharmaceutical and/or cosmetic compositions
03/19/2003EP1292555A2 Catalytic hydrogenation of ketones and aldehydes
03/19/2003EP0799228B1 3-aryl-tetronic acid derivatives, the production thereof and the use thereof as anti-parasitic agents
03/18/2003CA2238377C Cyclohexenone oxime ether metal salts
03/13/2003WO2003020684A1 (alpha)-haloenamine reagents
03/13/2003WO2002078625A3 Therapeutic combinations for cardiovascular and inflammatory indications
03/13/2003WO2002024194A3 Use of statins (hmg-coa reductase inhibitors) for the preparation of medicament as a novel type of immunomodulator, immunosuppressor and anti-inflammatory agent
03/13/2003US20030050482 Process of lactonization in the preparation of statins
03/13/2003CA2458859A1 (alpha)-haloenamine reagents
03/12/2003EP1289972A1 Serine protease inhibitors
03/11/2003US6531299 Incubating proteins comprising polyketide synthase, butyryl Coenzyme A, and thioester of butyric acid
03/06/2003WO2003018570A1 Process of lactonization in the preparation of statins
03/06/2003WO2003018553A1 Oral antidiabetic agents
03/06/2003WO2003018552A2 Aromatic and heteroaromatic acid halides for synthesizing polyamides
03/06/2003WO2003018535A2 Novel aminobenzoephenones
03/06/2003WO2002083066A3 Amino acid complexes of c-aryl glucosides for treatment of diabetes and method
03/06/2003US20030044644 4-dicyanomethylene-2-p-dimethylaminostyryl-6-methyl-4H-pyran derivatives with modified electron withdrawing groups and electron donating groups
03/06/2003CA2458621A1 Oral antidiabetic agents
03/06/2003CA2458616A1 Aromatic and heteroaromatic acid halides for synthesizing polyamides
03/05/2003EP1288212A1 Process of lactonization in the preparation of statins
03/05/2003EP1286967A1 Cyclohexane derivatives and their use as therapeutic agents
03/05/2003EP1286956A1 Phenyl-substituted 2-enamino-keto nitriles
03/05/2003EP0627433B1 Process for producing imidazopyridine derivative and intermediate
03/05/2003CN1102588C Process for manufacturing simwastatin from lovastatin or mevinolinic acid
03/04/2003US6528510 HIV protease inhibitors
02/2003
02/27/2003WO2003016317A1 Processes for preparing calcium salt forms of statins
02/27/2003WO2002092588A3 Aromatic sulfone hydroxamates and their use as protease inhibitors
02/27/2003WO2002053517A3 Process for stereoselective synthesis of prostacyclin derivatives
02/27/2003WO2002017911A1 Parathyroid hormone production inhibitors containing vitamin d3 derivatives
02/27/2003US20030040084 Macrolide analogs
02/27/2003CA2420759A1 Parathyroid hormone production inhibitors containing vitamin d3 derivatives
02/25/2003US6525206 Compounds with high monoamine transporter affinity
02/25/2003US6525205 Lactonization process
02/25/2003US6525052 Compounds useful as reversible inhibitors of cysteine proteases
02/20/2003WO2003014102A1 Certain substituted polyketides, pharmaceutical compositions containing them and their use in treating tumors
02/20/2003WO2003013542A1 Asymmetric synthesis of kavalactones
02/20/2003WO2003013502A1 Compounds which mimic the chemical and biological properties of discodermolide
02/20/2003WO2002032842A9 Compounds with high monoamine transporter affinity
02/20/2003WO2002030882A9 Sulfoxide and bis-sulfoxide compounds and compositions for cholesterol management and related uses
02/20/2003WO2002030860A9 Ketone compounds and compositions for cholesterol management and related uses
02/20/2003CA2456720A1 Asymmetric synthesis of kavalactones
02/20/2003CA2456553A1 Compounds which mimic the chemical and biological properties of discodermolide
02/20/2003CA2454081A1 Certain substituted polyketides, pharmaceutical compositions containing them and their use in treating tumors
02/19/2003EP1284264A1 Process for producing simvastatin
02/19/2003EP1144360A4 A method for the synthesis of compounds of formula 1 and derivatives thereof
02/19/2003CN1398189A Combination therapy of radiation and COX-2 inhibitor for treatment of neoplasia
02/19/2003CN1101809C Processes for preparing 3-arylsulfur hydroxamic acids
02/19/2003CN1101805C key intermediates in mfg. of simvastatin
02/18/2003US6521762 Process for purifying lovastatin and simvastatin with reduced levels of dimeric impurities
02/18/2003US6521650 Amines as pharmaceutical agents
02/13/2003WO2002040462A3 Cysteine protease inhibitors
02/12/2003EP1282415A2 Compounds and methods for regulating bacterial growth and pathogenesis
02/12/2003EP0871623B1 3-azetidinylalkylpiperidines or -pyrrolidines as tachykinin antagonists
02/12/2003CN1396919A Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-pyran-2-one
02/12/2003CN1396807A 除草组合物 Herbicidal compositions
02/12/2003CN1396262A Preparation method of epoxyinalool or mixture containing epoxy inalool
02/11/2003US6518460 Processes for preparing 3-arylsulfur hydroxamic acids
02/11/2003US6518326 Open chain alkoxyamine compounds and their use as polymerization regulators
02/11/2003US6518303 Selectively inhibit COX-2 in preference to COX-1 and are useful in the treatment of COX-2 mediated diseases, such as inflammation, pain, fever and asthma with fewer side effects
02/11/2003US6518289 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
02/10/2003WO2002014250A1 Derivatives of 4-(trifluoromethyl)-phenol and 4-(trifluoromethylphenyl)-2-(tetrahydropyranyl) ether and method for producing the same
02/10/2003CA2418749A1 Derivatives of 4-(trifluoromethyl)-phenol and 4-(trifluoromethylphenyl)-2-(tetrahydropyranyl) ether and method for producing the same
02/06/2003WO2003010130A1 Amino acid derivatives
02/05/2003EP1280770A1 C 2? phenyl-substituted cyclic keto-enols used as pesticides and herbicides
02/05/2003EP0745087B1 Novel cytotoxic macrolides, their isolation from a marine sponge and their use as antitumor agents
02/05/2003CN1394855A Substituted heterocyclic compound
02/04/2003US6515117 C-aryl glucoside SGLT2 inhibitors and method
02/03/2003WO2002016312A2 Novel compounds inhibiting factor xa activity
02/03/2003CA2418283A1 Novel compounds inhibiting factor xa activity
01/2003
01/30/2003WO2003007954A2 Sulfonyl aryl hydroxamates and their use as matrix metalloprotease inhibitors
01/30/2003WO2003007878A2 Antifungal agents of sordarin derivatives
01/30/2003US20030022865 Sulfoxide and bis-sulfoxide compounds and compositions for cholesterol management and related uses
01/30/2003CA2453613A1 Sulfonyl aryl hydroxamates and their use as matrix metalloprotease inhibitors
01/29/2003EP1278747A1 Pyrano, piperidino, and thiopyrano compounds and methods of use
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