Patents
Patents for C07D 305 - Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms (5,442)
03/2008
03/12/2008CN101139376A Preparation of 10-deacetyl 7-xylose baccatin or 7-xylose baccatin
03/12/2008CN101139329A Method for selectively acylating taxone C(10) hydroxy
03/12/2008CN100374429C Method for producing docetaxel using 10-deacetylpaclitaxel as raw material
03/12/2008CN100374428C Intermediary compounds for the hemisynthesis of taxanes and prepn. processes therefore
03/05/2008EP1894921A2 9, 10-Alpha, Alpha-Oh-Taxane analogs and methods for production thereof
03/05/2008EP1893594A2 Processes for the preparation of paclitaxel
03/05/2008EP1893593A1 3-phenylazetidine derivatives as dopamine agonists
03/05/2008CN101137634A Semi-synthetic taxane derivatives with antitumor activity
02/2008
02/28/2008WO2008022824A1 Method for the production of oxetane group-containing (meth)acrylates
02/28/2008WO2008006113A3 Novel belactosin derivatives as therapeutic agents/biological probes and their synthesis
02/28/2008US20080051590 Semi-Synthetic Conversion of Paclitaxel to Docetaxel
02/28/2008US20080051589 Protecting the hydroxyl of a taxane amide; reducing the amide with a transition metalcompound; removing the metal; acidolysis to form a taxane amine salt in solution;adding solvent to solidify; convert the amine salt into paclitaxel or other taxanes
02/28/2008US20080051450 Process For The Preparation Of Anhydrous And Hydrated Active Pharmaceutical Ingredients (Apis); Stable Pharmaceutical Compositions Prepared From The Same And Uses Of Said Compositions
02/27/2008EP1891033A2 Processes for the preparation of docetaxel
02/27/2008CN101130528A Process for the preparation of baccatin iii derivatives
02/27/2008CN100370980C C-2' methylated derivatives of paclitaxel for use as antitumour agents
02/26/2008USRE40120 Protecting the 7- and 10- hydroxyls and esterifying the c-13 hydroxyl with an oxazolidine 5-carboxylic acid; deprotecting and optionally acetylating the c-10 hydroxyl group; decycli-zation of the oxazolidine ring; antitumor agents
02/21/2008US20080045589 Drug Combinations with Substituted Diaryl Ureas for the Treatment of Cancer
02/21/2008US20080045584 Use of Docetaxel for Treating Hepatocellular Carcinoma
02/20/2008EP1889624A2 Combined therapy against tumors comprising substituted acryloyl distamycin derivatives, taxanes and/or antimetabolites
02/20/2008EP1615902B1 Method for production of 4,10 beta-diacetoxy-2 alpha-benzoyloxy-5 beta,20-epoxy-1,13 alpha-dihydroxy-9-oxo-19-norcyclopropa[g]tax-11-ene
02/20/2008CN101128449A Process of preparing docetaxel
02/20/2008CN101128448A Method for preparing paclitaxel
02/20/2008CN100369908C New taxane derivatives
02/20/2008CN100369907C Method for producing epoxy propane
02/19/2008US7332617 Process for the preparation of docetaxel trihydrate
02/19/2008CA2273240C Compositions and methods for treating or preventing inflammatory diseases
02/14/2008WO2008019151A1 Oxetane composition, associated method and article
02/14/2008US20080039641 Process for preparing brevifoliol
02/14/2008US20080039635 Method for the Production of a Compound, Comprising a Free Hydroxyl Group and a Hydroxyl Group Which is Protected by an Ester Function by Enzymatic Reaction
02/14/2008US20080039421 Molecular Transporters Based On Alditol Or Inositol And Processes For The Preparation Thereof
02/13/2008EP1885707A1 A process for the purification of 10-deacetylbaccatine iii from 10-de acet yl-2- debenzoyl-2-pentenoylbaccatine iii
02/12/2008CA2197467C Method for the preparation of taxol and its derivatives
02/07/2008US20080033189 Semi-Synthesis Of Taxane Intermediates And Aziridine Analogues And Their Conversion To Paclitaxel And Docetaxel
02/05/2008US7326796 Fluorinated monomers, fluorinated polymers having polycyclic groups with fused 4-membered heterocyclic rings, useful as photoresists, and processes for microlithography
01/2008
01/31/2008US20080027130 Cytotoxic agents comprising taxanes and their therapeutic use
01/30/2008CN101113143A 4,10- beta -diacetoxy-2 alpha -benzoyloxy-5 beta ,20-epoxy-1-hydroxy-9-oxo-19-norcyclopropa[g]tax-11-en-13 alpha -yl (2r,3s)-3-tert-butoxycarbonylamino-2-hydroxy-3-phenylpropionate dihydrate and its p
01/29/2008CA2226058C 8-substituted-1,3,8-triaza-spiro[4.5]decan-4-one derivatives
01/29/2008CA2215682C 10-deacetylbaccatine iii and 10-deacetyl 14.beta.-hydroxybaccatine iii derivatives, a process for the preparation thereof and pharmaceutical compositions containing them
01/24/2008US20080020148 Chromane Derivatives Method for Production and the Use Thereof
01/24/2008US20080020063 Anti-angiogenic compositions and methods of use
01/24/2008US20080020052 Vascular Embolus Of Paclitaxel-Sodium Alginate Microsphere And Its Preparation
01/23/2008CN100363354C Process for refining lipstatin
01/22/2008CA2214321C Novel taxoids, preparation thereof and pharmaceutical compositions containing same
01/17/2008DE102006039245B3 Making oxetane group-containing (meth)acrylate for use as a binder, e.g. in adhesives, paints or ink-jet ink, involves reacting ethoxylated trimethylol-propane-oxetane with (meth)acrylate using a zirconium catalyst
01/16/2008CN100361985C Paclitaxol predrug of biodegradable polymer and its synthesis method
01/15/2008US7319154 Oxidation of 17 alpha -(3-hydroxypropyl)-6 beta ,7 beta ;15 beta ,16 beta -dimethylene-androstane-3 beta ,5 beta ,17 beta -triol in the presence of a catalytic amounts of a 2,2,6,6-tetramethylpiperidine-N-oxide derivative at a pH of at least 8.0
01/10/2008WO2008006113A2 Novel belactosin derivatives as therapeutic agents/biological probes and their synthesis
01/10/2008US20080008943 Ink composition, inkjet recording method, printed material, method of producing planographic printing plate, and planographic printing plate
01/10/2008CA2657103A1 Novel belactosin derivatives as therapeutic agents/biological probes and their synthesis
01/09/2008EP1875237A2 Docetaxel immunoassay
01/09/2008EP1874753A2 Compounds, compositions and methods
01/08/2008US7317114 Process to obtain dibenzylbutyrolactonic lignans, process to obtain synthetic derivatives from lignans bearing anti-Chagas chemoprophylactic and therapeutical activities
01/08/2008US7317113 Treatment of 7-Boc-13-keto-baccatin III to give 7-Boc-13-keto-14-hydroxy-baccatin III, carbonation of the 1 and 14 hydroxyls to give 14 beta -hydroxy-7-Boc-keto-baccatin III-1,14-carbonate, and reduction of the ketone at the 13-position and cleavage of the protective group
01/03/2008WO2007078050A3 Method for preparation of amorphous, anhydrous crystalline, or hydrated crystalline docetaxel
01/02/2008EP1871753A1 Preparation of taxanes from 9-dihydro-13-acetylbaccatin iii
01/02/2008EP1608636B1 Improved process for isolation and purification of paclitaxel from natural sources
01/01/2008US7314942 Reactrting butyrolactone or valerolactone with formaldehyde;heating under critical temperature, critical pressure
12/2007
12/27/2007US20070298123 Anti-angiogenic compositions and methods of use
12/27/2007US20070298039 Immunoglobulin specific to receptor protein DR5 for treatment of cancer, inflammatory or autoimmune diseases
12/21/2007WO2007143839A1 Semi-synthetic route for the preparation of paclitaxel, docetaxel and 10-deacetylbaccatin iii from 9-dihydro-13-acetylbaccatin iii
12/21/2007WO2007124700A3 Pharmaceutical composition containing taxane derivative destined for the preparation of an infusion solution, method of preparation thereof and use thereof
12/20/2007US20070293687 Semi-synthetic route for the preparation of paclitaxel, docetaxel, and 10-deacetylbaccatin iii from 9-dihydro-13-acetylbaccatin iii
12/19/2007EP1165068B1 C10 heterosubstituted acetate taxanes as antitumor agents
12/19/2007CN101088994A Process of synthesizing taxol and docetaxel
12/19/2007CN100355740C Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-pyran-2-ketone
12/18/2007CA2209001C Hydrophobic taxane derivatives
12/13/2007WO2007142236A1 3-ethyloxethane compound having hydroxyl group and method for producing the same
12/12/2007EP1747209A4 A facile method for synthesizing baccatin iii compounds
12/12/2007CA2549951A1 Semi-synthetic route for the preparation of paclitaxel, docetaxel and 10-deacetylbaccatin iii from 9-dihydro-13-acetylbaccatin iii
12/11/2007US7307176 Inclusion complex of taxol with 2-hydroxypropyl-beta-cyclodextrin
12/06/2007WO2007137513A1 A TYPE OF NOVEL 2'-α-HYDROXYALKYL TAXEL COMPOUNDS AND THE PREPARATION METHODS THEREOF
12/05/2007CN101081841A Novel 2'-alpha-hydroxyalkyl taxone compound and preparation method thereof
12/04/2007US7304093 Ketone compounds and compositions for cholesterol management and related uses
12/04/2007CA2418125C Beta-lactams useful in the preparation of substituted isoserine esters
11/2007
11/29/2007WO2007135954A1 2-oxetanone derivative and process for production thereof
11/29/2007WO2007014247A3 Novel compounds, pharmaceutical compositions containing same, and methods of use for same
11/28/2007EP1858870A1 Semi-synthetic taxane derivatives with antitumor activity
11/28/2007EP1534674A4 Cytotoxic agents containing novel potent taxanes and their therapeutic use
11/28/2007CN100351246C Process for selective derivatization of taxanes
11/27/2007US7300604 Tetrahydroxybenzene tetraester derivative and polymer thereof
11/27/2007CA2100218C Preparation and polymerization of perfluoroalkoxy alkylene oxides to prepare hydrophobic polyethers
11/22/2007WO2007106576A3 Methods and materials for immunization against cancer
11/22/2007US20070270482 Cytotoxic Agents Comprising New C-2 Modified Taxanes
11/21/2007EP1856216A1 Sprayable coating composition
11/21/2007EP1856081A1 Method for preparing paclitaxel
11/21/2007EP1856080A1 Method for preparing docetaxel
11/21/2007EP1856079A1 Spiro-heterocyclic chromans, thiochromans and dihydroquinolines
11/21/2007EP1301500B1 Nitrosated and nitrosylated taxanes, compositions and methods of use
11/21/2007CN101076523A (meth) acryloyl group-containing oxetane compound and production method thereof
11/21/2007CN101074219A Method for separating and extracting 10-deacetylbakedin III from taxicatin
11/21/2007CN101074218A Cephalotamannine derivative, its production, its medicinal composition and use
11/21/2007CN100349882C Method for preparing derivatives of baccatin iii
11/15/2007WO2007076160A3 C-10 carbamates of taxanes
11/15/2007US20070265180 3-Methyl Oxetanemethanol Derivatives and Their Use in Perfume Compositions
11/15/2007CA2651212A1 Hydrolytically-resistant boron-containing therapeutics and methods of use
11/14/2007CN100348580C Taxol enhancer compounds
11/08/2007WO2007126893A2 A convergent process for the synthesis of taxane derivatives
11/08/2007WO2007124700A2 Pharmaceutical composition containing taxane derivative destined for the preparation of an infusion solution, method of preparation thereof and use thereof
11/08/2007CA2649335A1 Pharmaceutical composition containing a taxane derivative, destined for the preparation of an infusion solution, method of preparation thereof and use thereof
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