| Patents for C07D 279 - Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms (5,149) |
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| 01/25/2005 | US6846824 E.g., ethyl 3-(4-(2-(3-oxo-2H-1,4-benzoxazin-4-yl)ethoxy)-phenyl-2-ethoxypropenoate where 1,4-benzothiazine or quinoxaline can be substituted for the benzoxazine ring; anticholesterol, diabetic agents; obesity; hyperlimpidemia |
| 01/20/2005 | US20050014747 Hypotensive agents; congestive heart failure |
| 01/20/2005 | US20050014746 compounds which bind to the interaction-domain (I-domain) of LFA-1, thus interrupting endothelial cell-leukocyte adhesion by blocking the interaction of LFA-1 with ICAM-1, ICAM-3, and other adhesion molecules |
| 01/20/2005 | US20050014744 Benzothiazine and benzothiadiazine compounds |
| 01/19/2005 | EP1498411A1 Diketohydrazine derivative compounds and drugs containing the compounds as the active ingredient |
| 01/12/2005 | CN1564817A Novel benzothiazine derivatives, their preparation and use |
| 01/11/2005 | US6841674 N-heterocyclic derivatives as NOS inhibitors |
| 01/11/2005 | US6841673 Enzyme inhibitors; antiinflammatory agents; rheumatic diseases; antidiabetic agents |
| 01/11/2005 | US6841559 Prevention or inhibition of normal pilus assembly in Gram-negative bacterium impacts the pathogenicity of the bacterium |
| 01/11/2005 | US6841550 Benzoxazine and benzothiazine derivatives and their use in medicines |
| 01/06/2005 | WO2005000406A2 Treatment of amyloid- and epileptogenesis-associated diseases |
| 01/06/2005 | US20050004112 C-fms kinase inhibitors |
| 01/06/2005 | CA2556706A1 Treatment of amyloid- and epileptogenesis-associated diseases |
| 01/05/2005 | EP1493743A1 Substituted bipiperidine intermediates and derivatives thereof |
| 12/30/2004 | US20040267011 Methods for synthesis of diarylmethanes |
| 12/29/2004 | WO2004112575A2 Gene amplification and overexpression in cancer |
| 12/29/2004 | CA2528529A1 Gene amplification and overexpression in cancer |
| 12/28/2004 | US6835495 Pentacyclic anion salts or tetrazapentalene derivatives and their uses as ionic conducting materials |
| 12/23/2004 | WO2004111022A1 3-(1,1-DIOXOTETRAHYDRO-1,2-THIAZIN-2-YL) or 3-(1,1-DOXO-ISOTHIAZOLIDIN-2YL) SUBSTITUTED BENZAMIDE COMPOUNDS AS ASP2 INHIBITORS |
| 12/23/2004 | WO2004110986A1 Benzamide derivative or salt thereof |
| 12/23/2004 | CA2526387A1 Benzamide derivative or salt thereof |
| 12/16/2004 | US20040254166 Substituted phenyl acetamides and their use as protease inhibitors |
| 12/14/2004 | US6830743 In Vivo stain compounds and methods of use to identify dysplastic tissue |
| 12/14/2004 | CA2180867C Monomeric diols and phosphate linked oligomers formed therefrom |
| 12/08/2004 | CN1178922C Substituted 1-aminoalkyl-lactams compound and their use as muscarinic receptor antagonists |
| 12/07/2004 | CA2147755C 6-(substituted methylene) penems and intermediates |
| 12/02/2004 | US20040242571 Novel benzothiazine derivatives, their preparation and use |
| 12/02/2004 | US20040242570 Conjugated psychotropic drugs and uses thereof |
| 12/02/2004 | US20040241563 Phenothiazine, phenoxazine, or phenazine derivatives; organophotoreceptor comprising electricoconductive substrate and photoconductive element; mechanical, electrostatic, and solubility properties; used with toners for quality images |
| 12/01/2004 | EP1482376A1 Charge transport materials having heteroaromatic hydrazone groups |
| 12/01/2004 | EP1481970A1 Novel herbicides |
| 12/01/2004 | EP1480986A1 Novel benzothiazine and benzothiadiazine derivatives, method for preparing same and pharmaceutical compositions containing same |
| 12/01/2004 | EP1480967A1 Novel fused ring compounds, and their use as cationic photoinitiators |
| 12/01/2004 | CN1551872A Biologically active methylene blue derivatives |
| 12/01/2004 | CN1550496A Acetylenic alpha-amino acid-based sulfamide hydroxamic acid TACE inhibitors |
| 11/30/2004 | US6825193 Heterocyclic amines such as 4-(3,4-dichlorophenyl)-2-(2-(4-methylpiperazin-1-yl)-benzylidene) -thiomorpholin-3-one, used as antiserotonine agents |
| 11/25/2004 | WO2004101559A1 Fused bicyclic-substituted amines as histamine-3 receptor ligands |
| 11/25/2004 | WO2004101539A1 Cyclic sulfonamides for inhibition of gamma-secretase |
| 11/25/2004 | WO2004101538A1 Cyclohexyl sulphones as gamma-secretase inhibitors |
| 11/25/2004 | US20040235666 Substituted imidates as pesticidal agents |
| 11/18/2004 | US20040230054 Cyclic sulfonamides for inhibition of gamma-secretase |
| 11/18/2004 | US20040229819 Hemiasterlin derivatives and uses thereof |
| 11/17/2004 | EP1477186A1 Antipruritics |
| 11/17/2004 | EP1210333B1 p-Tolyl-heterocycles as herbicides |
| 11/16/2004 | US6818645 2-amino-trihydroindole or tetrahydronapthalene-2-yl derivatives, useful for disease state associated with smooth muscle disorders, such as gastrointestinal and urogenital disorders |
| 11/16/2004 | US6818640 2-imino-1,3-thiazine derivatives |
| 11/16/2004 | US6818327 Organic electroluminescence device |
| 11/11/2004 | WO2004096795A2 C-fms kinase inhibitors |
| 11/11/2004 | US20040224953 Fused bicyclic-substituted amines as histamine-3 receptor ligands |
| 11/11/2004 | US20040224952 e.g., 4-{2-[2-(2-(R)-Methyl-pyrrolidin-1-yl)-ethyl]-benzothiazol-5-yl}-benzonitrile; useful for treating conditions and disorders related to memory and cognition processes, neurological processes, cardiovascular function, and body weight. |
| 11/11/2004 | CA2536964A1 C-fms kinase inhibitors |
| 11/10/2004 | EP1475372A1 Nile red type compound emitting red light, process for producing the same, and luminescent element utilizing the same |
| 11/10/2004 | CN1545425A Light-stabilized in vivo stain composition and method of manufacture |
| 11/10/2004 | CN1544945A Inhibition of Tau-Tau-association |
| 11/09/2004 | US6815094 Diphenyl anthracene derivatives and organic electroluminescent device employing the same |
| 11/09/2004 | US6815090 Organic electroluminescence device |
| 11/04/2004 | WO2004094396A2 Dihydrothiazine prodrugs of thiazolium agents |
| 11/04/2004 | WO2004094382A1 Muscarinic agonists |
| 11/04/2004 | CA2522756A1 Dihydrothiazine prodrugs of thiazolium agents |
| 11/04/2004 | CA2518324A1 Muscarinic agonists |
| 11/03/2004 | EP1472219A1 Novel benzothiazine and benzothiadiazine derivatives, method for preparing same and pharmaceutical compositions containing same |
| 11/03/2004 | CN1542002A Inhibitors of metalloproteinase, pharmaceutical compositions containing them, their pharmaceutical application and methods and intermediate compounds for their preparation |
| 11/03/2004 | CN1173947C 2,4,5-trisubstituted phenylketo-enols for use as pesticides and herbicides |
| 11/02/2004 | US6812227 Acetylenic α-amino acid-based sulfonamide hydroxamic acid tace inhibitors |
| 10/28/2004 | WO2004092116A1 Bicyclic compounds having bradykinin receptors affinity and pharmaceutical compositions thereof |
| 10/28/2004 | WO2004091613A2 Substituted phenyl acetamides and their use as protease inhibitors |
| 10/28/2004 | US20040214043 Acenaptho(1,2-k)fluoranthene derivatives; color purity, efficient light emission, durability |
| 10/28/2004 | US20040213736 Introducing into the subject a ligand capable of labelling aggregated paired helical filament (PHF) tau protein, determining the presence and\or amount of ligand bound to extracellular aggregated PHF tau in the medial temporal lobe of the brain, correlating the result of the determination |
| 10/28/2004 | CA2521937A1 Bicyclic compounds having bradykinin receptors affinity and pharmaceutical compositions thereof |
| 10/27/2004 | CN1172920C Process for producing 2-(4-alkyl-1-piperazyl)-benzaldehyde and-benzal compound |
| 10/26/2004 | US6809095 Novel antitobesity and hypocholesterolemic compounds lower total cholesterol; increase high density lipoprotein (hdl) and decrease low denstiy lipoprotein |
| 10/21/2004 | US20040209873 Arylcycloalkyl derivatives having branched side chains, processes for their preparation and their use as pharmaceuticals |
| 10/21/2004 | US20040208822 technetium labelled complexes; for the treatment or diagnosis of pathologies caused by attack on human cartilage, arthritis |
| 10/20/2004 | EP1289964B1 Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists |
| 10/13/2004 | EP1466899A1 Hydroxamic acid derivative and mmp inhibitor containing the same as active ingredient |
| 10/13/2004 | CN1537016A Remedies for psychoneurosis |
| 10/07/2004 | WO2004085431A1 Prostaglandin analogs as ep4 receptor antagonists |
| 10/07/2004 | WO2004085430A1 Prostaglandin analogs as ep4 receptor agonists |
| 10/07/2004 | US20040198701 EP4 receptor agonist, compositions and methods thereof |
| 10/06/2004 | EP1135379B1 Antitumor dibenzofluorene derivatives |
| 10/06/2004 | CN1534076A Red light emitted compound used for organic electroluminous device and orgainic electroluminous device using same |
| 10/05/2004 | US6800656 Tricyclic compounds and method of treating herpes virus |
| 10/05/2004 | US6800618 Phenothiazine or iminodibenzyl derivatives as antimalarial agents |
| 09/29/2004 | CN1533278A Naphtothiazine positive allosteric AMPA receptor modulators (PAARM) |
| 09/23/2004 | US20040186098 Method for preventing and treating hearing loss using sensorineurotrophic compounds |
| 09/23/2004 | US20040186093 Cyclizing a sulfamide acyclic compound with a deprotonating agent in an aprotic solvent; forming an intermediates for the preparation of naphthyridine carboxamide compounds which are HIV integrase enzyme inhibitors; commercial available starting materials alkanesulfonyl halides, haloalkylamine |
| 09/21/2004 | US6794383 Heart muscular cell apoptosis inhibitors and remedies/preventives for heart diseases |
| 09/21/2004 | US6794373 Contraceptive methods using benzimidazolones |
| 09/15/2004 | EP1456189A1 Benzothia(dia)zine derivatives and their use as ampa modulators |
| 09/15/2004 | EP1185526B1 Novel quaternary ammonium derivatives, method for preparing same and pharmaceutical use |
| 09/15/2004 | EP0986384A4 Inhibitors of protein isoprenyl transferases |
| 09/15/2004 | CN1529756A Steroselective preparation of cyclic L-amino acids |
| 09/10/2004 | WO2004076402A1 Arylcycloalkyl derivatives with branched side chains as ppar receptor modulators, method for their production and their use as medicaments |
| 09/10/2004 | CA2516626A1 Arylcycloalkyl derivatives with branched side chains as ppar receptor modulators, method for their production and their use as medicaments |
| 09/09/2004 | US20040176426 farnesoid X receptor; to mitigate and thereby treat hypercholesterolemia; antagonists, which block the negative feedback downregulation of cyp7a expression produced by certain cholic acids |
| 09/09/2004 | US20040176364 Aryl substituted thiazinidinones and the use thereof |
| 09/09/2004 | DE10308352A1 Arylcycloalkylderivate mit verzweigten Seitenketten, Verfahren zu ihrer Herstellung und ihre Anwendung als Arzneimittel Arylcycloalkylderivate with branched side chains, to processes for their preparation and their use as medicaments |
| 09/08/2004 | EP1453789A2 N,n'-substituted-1,3-diamino-2-hydroxypropane derivatives |
| 09/08/2004 | EP1165505B1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds |
| 09/08/2004 | CN1526689A Diphenyl anthracene derivate and organic electroluminescent apparatus using diphenyl anthracene derivate |