| Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621) |
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| 02/16/2010 | US7662644 Use of specified fluorescent dyes to conjugate to antibody; detecting binding of an antibody to an antigen; antibody conjugate |
| 02/16/2010 | CA2478183C Substituted amides |
| 02/16/2010 | CA2442882C Sulphones which modulate the action of gamma-secretase |
| 02/16/2010 | CA2402436C Amidino compound and salts thereof useful as nitric oxide synthase inhibitors |
| 02/16/2010 | CA2385081C Carboxylic acid compound and a medicament comprising it |
| 02/16/2010 | CA2343883C An improved process for the preparation of thiazolidine-2,4-dione derivatives |
| 02/11/2010 | WO2010015655A1 Cyclohexyl amide derivatives and their use as crf-1 receptor antagonists |
| 02/11/2010 | US20100035944 Compounds and methods for modulating g protein-coupled receptors |
| 02/11/2010 | US20100035898 Organic compounds |
| 02/11/2010 | CA2732887A1 Cyclohexyl amide derivatives and their use as crf-1 receptor antagonists |
| 02/10/2010 | EP2151438A1 Pharmaceutical containing ppar agonist |
| 02/10/2010 | EP2151435A1 Pharmaceutical composition for treatment of alzheimer's disease |
| 02/10/2010 | EP2150532A1 Piperazine compounds for the inhibition of haematopoietic prostaglandin d synthase |
| 02/10/2010 | EP1833805B1 New 3-phenylpropionic acid derivatives for the treatment of diabetes |
| 02/10/2010 | EP1747196B1 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication |
| 02/10/2010 | EP1404659B1 4-aryl quinols and analogs thereof as therapeutic agents |
| 02/10/2010 | CN101643457A Artificial sulfamethylthiazole antigen and preparation method and application thereof |
| 02/09/2010 | US7659404 Broad spectrum 2-(substituted-amino)-benzothiazole sulfonamide HIV protease inhibitors |
| 02/09/2010 | US7659297 improved selectivity and pharmacokinetic properties; 6-Fluoro-1-[(1 H-indazol-4-yl)amino]-4,4-dimethyl-2-(trifluoromethyl)-1,2,3,4-tetrahydronaphthalene-2,5-diol; cyclization of imines |
| 02/09/2010 | US7659295 Therapeutic substituted thiazolidinones, oxazolidinones, and related compounds |
| 02/09/2010 | US7659270 (1R)-2-((2S)-2-(5-(6-(4-(2-((2S)-1-((2R)-2-(dimethylamino)-2-phenylacetyl)-2-pyrrolidinyl)-1H-imidazol-5-yl)phenyl)-3-pyridinyl)-1H-imidazol-2-yl)-1-pyrrolidinyl) -N,N-dimethyl-2-oxo-1-phenylethanamine; inhibit the function of the non-structural proteins (NS5A) |
| 02/09/2010 | US7659228 Synergistic insecticide mixtures |
| 02/09/2010 | CA2440760C Substituted pyrazolopyrimidines and thiazolopyrimidines used as analgesics |
| 02/09/2010 | CA2413061C Serine protease inhibitors |
| 02/09/2010 | CA2315646C Inhibition of raf kinase using symmetrical and unsymmetrical substituted diphenyl ureas |
| 02/09/2010 | CA2291065C Raf kinase inhibitors |
| 02/09/2010 | CA2274201C Di-or triaza-spiro[4,5]decane derivatives |
| 02/09/2010 | CA2201863C Substituted 4-biarylbutyric or 5-biarylpentanoic acids and derivatives as matrix metalloprotease inhibitors |
| 02/09/2010 | CA2192092C Arylsulfonamido-substituted hydroxamic acids as matrix metalloproteinase inhibitors |
| 02/04/2010 | WO2010014611A1 Cycloalkylidene and heterocycloalkylidene histone deacetylase inhibitor compounds |
| 02/04/2010 | WO2010014586A1 Asymmetric process for making substituted 2-amino-thiazolones |
| 02/04/2010 | WO2010013567A1 Amide derivative, pest control agent containing the amide derivative and pest controlling method |
| 02/04/2010 | WO2010012795A1 Fungicidal n-(2-phenoxyethyl)carboxamide derivatives and their aza, thia and sila analogues |
| 02/04/2010 | WO2010012794A1 Fungicide n-cycloalkyl-n-biphenylmethyl-carboxamide derivatives |
| 02/04/2010 | WO2010012793A1 Fungicide aminothiazole derivatives |
| 02/04/2010 | WO2010012107A1 Selective glycosidase inhibitors and uses thereof |
| 02/04/2010 | US20100029733 Bicyclic nitrogen-containing heterocyclic compounds |
| 02/04/2010 | US20100029730 such as N-acetyl-N-(4'-bromo-1,1'-biphenyl-2-yl)-4-(difluoromethyl)-2-methyl-1,3-thiazole-5-carboxamide, used for controlling unwanted phytopathogenic fungi; microbiocides |
| 02/04/2010 | US20100029690 Nitrogen-containing heterocyclic compounds |
| 02/04/2010 | US20100029689 Phosphodiesterase 4 inhibitors |
| 02/04/2010 | US20100029639 Ion channel modulating compounds and uses thereof |
| 02/04/2010 | US20100029588 Substituted phenylamidines and the use thereof as fungicides |
| 02/04/2010 | CA2794350A1 Amide derivative, pest control agent containing the amide derivative, and pest controlling method |
| 02/04/2010 | CA2737348A1 Amide derivative, pest control agent containing the amide derivative, and pest controlling method |
| 02/04/2010 | CA2732336A1 Selective glycosidase inhibitors and uses thereof |
| 02/04/2010 | CA2731323A1 Cycloalkylidene and heterocycloalkylidene histone deacetylase inhibitor compounds |
| 02/04/2010 | CA2731200A1 Fungicidal n-(2-phenoxyethyl)carboxamide derivatives and their aza, thia and sila analogues |
| 02/04/2010 | CA2731198A1 Fungicide n-cycloalkyl-n-biphenylmethyl-carboxamide derivatives |
| 02/04/2010 | CA2730711A1 Asymmetric process for making substituted 2-amino-thiazolones |
| 02/03/2010 | CN101641342A Thiazolidine derivatives |
| 02/03/2010 | CN101638396A Production process for rubber accelerator 2-thiol group benzothiazole |
| 02/03/2010 | CN101638395A Heterocyclic analog of diphenylethlene compound and application thereof |
| 02/02/2010 | US7655804 Diketohydrazine derivative compounds and drugs containing the compounds as the active ingredient |
| 02/02/2010 | US7655684 1-(Urea-, thiourea- and cyanoguanidine-methylene)benzyl)imidaoles, treatment of neuronal disorders, especially Alzheimer's disease, Down Syndrome, Parkinson's disease and Huntington's disease |
| 02/02/2010 | US7655680 (E)-3-[2-(3,4-diethoxyphenyl)thiazole-4-yl]-1-(2-methoxyphenyl)propenone; inhibiting the activity of phosphodiesterase 4, the production of tumor necrosis factor alpha, and the production of interleukin 4; atopic dermatitis |
| 02/02/2010 | US7655676 Selective activity against propionibacterium acne; minimum inhibitory concentration (MIC) against Propionibacterium acnes strains both sensitive and resistant to erythromycin and clindamycin and against a series Staphylococcus strains |
| 02/02/2010 | US7655641 3-(4-{2-[(5-Fluoro-3- methyl-benzo[b]thiophene-2- sulfonyl)-propyl- amino]-ethylsulfanyl}- 2-methyl-phenyl)- propionic acid; peroxisome proliferator activated receptor (PPAR); syndrome X, type II diabetes, hyperglycemia, hyperlipidemia, obesity, hypertension, arteriosclerosis and cardiovascular diseases |
| 02/02/2010 | US7655621 Cross-linked glycopeptide-cephalosporin antibiotics |
| 02/02/2010 | US7655600 1-(azolin-2-yl)amino-1,2-diphenylethane compounds for combating insects, arachnids and nematodes |
| 02/02/2010 | US7655380 Polymeric material containing a latent acid, i.e. a compound which is not an acid but which can be converted to an acid by the influence of laser irradiation |
| 02/02/2010 | CA2294809C Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and compositions containing same |
| 01/28/2010 | WO2010011926A2 A novel betaine cocrystal of epalrestat |
| 01/28/2010 | WO2010011922A2 Novel crystalline salts of epalrestat |
| 01/28/2010 | WO2010010797A1 Pharmaceutical composition comprising dyrk-inhibiting compound |
| 01/28/2010 | WO2010010435A2 Fused oxazole and thiazole derivatives as trpms modulators |
| 01/28/2010 | WO2010010288A2 Alkylthiazol carbamate derivatives, preparation thereof and therapeutic use thereof |
| 01/28/2010 | WO2009132452A8 Diaryl-cyclylalkyl derivatives as calcium channel blockers |
| 01/28/2010 | US20100022773 Apoptosis promoters |
| 01/28/2010 | US20100022605 N-hydroxyamide derivatives possessing antibacterial activity |
| 01/28/2010 | US20100022596 Epothilone analogues |
| 01/28/2010 | US20100022594 thiophene sulfonamide derivatives such as 5-Chloro-N-[(S)-2-hydroxy-1-phenylethyl]thiophene-2-sulfonamide, that inhibit the production of beta amyloid protein from amyloid precursor protein; capable of passing through the blood-brain barrier, used for treatment of Alzheimer's disease and Down's syndrome |
| 01/28/2010 | US20100022570 Novel microbiocides |
| 01/28/2010 | US20100022547 Compounds and Methods for Treating Mammalian Gastrointestinal Parasitic Infections |
| 01/28/2010 | US20100022542 Compounds exhibiting thrombopoietin receptor agonism |
| 01/28/2010 | US20100022491 4-hydroxy-2-oxo-2,3-dihydro-1,3-benzothiazol-7yl compounds for modulation of b2-adrenoreceptor activity |
| 01/28/2010 | US20100021388 Benzothiazole derivative compounds, compositions and uses |
| 01/28/2010 | CA2731789A1 Alkyl thiazole carbamate derivatives, preparation thereof, and use thereof as faah enzyme inhibitors |
| 01/27/2010 | EP2146974A1 N- hydroxy-4-{5-[4-(5-isopropyl-2-methyl-1,3-thiazol-4-yl)phenoxy]pentoxy} benzamidine 2 ethansulfonic acid salt, process for the preparation thereof and pharmaceutical composition comprising the same |
| 01/27/2010 | EP1438298B1 Piperazine derivatives with ccr1 receptor antagonist activity |
| 01/27/2010 | CN100584842C Thiazole derivative |
| 01/27/2010 | CN100584833C Ritonavir analogous compound useful as retroviral protease inhibitor, preparation of the ritonavir analogous compound and pharmaceutical composition for the ritonavir analogous compound. |
| 01/26/2010 | US7652146 Reacting an amide with a thiourea; inflammatory and immune conditions |
| 01/26/2010 | US7652045 Activator of peroxisome proliferator-activated receptor δ |
| 01/26/2010 | US7652044 P-38 inhibitors |
| 01/26/2010 | US7652036 Carbamic acid compounds comprising a bicyclic heteroaryl group as HDAC inhibitors |
| 01/26/2010 | US7652021 (2S)-4,4-difluoro-1-{N-[3-(pyrimidin-2-ylamino)-1-adamantyl]glycyl}pyrrolidine-2-carbonitrile; dipeptidyl peptidase IV enzyme inhibitors; non-insulin dependent diabetes mellitus |
| 01/26/2010 | US7652020 novel hydantoin derivatives to inhibit matrix metalloproteinases (MMPs), a disintegrin and metalloproteases (ADAMs) and/or tumor necrosis factor alpha converting enzyme (TACE) and in so doing prevent the release of tumor necrosis factor alpha (TNF- alpha ); autoimmune diseases; side effect reduction |
| 01/26/2010 | US7652018 4-[2-(3,5,5-Trimethyl-2-oxoimidazolidin-1-yl)-1,3-thiazol-4-yl]benzonitrile; 1-[4-(4-Bromophenyl)-1,3-thiazol-2-yl]-3-methylimidazolidin-2-one; contraception, fibroids, endometriosis, dysfunctional bleeding, uterine leiomyomata, polycystic ovary syndrome, or hormone-dependent carcinomas |
| 01/26/2010 | CA2430579C Isoindolin-1-one glucokinase activators |
| 01/26/2010 | CA2422889C Method for the treatment of neurological and neuropsychological disorders |
| 01/21/2010 | WO2010009120A2 Novel salts and polymorphs of desazadesferrithiocin polyether analogues as metal chelation agents |
| 01/21/2010 | WO2010008729A2 Process for making substituted 2-amino-thiazolones |
| 01/21/2010 | WO2010008522A2 Nucleophilic fluorination of aromatic compounds |
| 01/21/2010 | WO2010007482A2 Thiazole derivatives as stearoyl coa desaturase inhibitors |
| 01/21/2010 | WO2010007389A1 5 -amidothiazole derivatives and their use as checkpoint kinase inhibitors |
| 01/21/2010 | WO2010007318A2 Novel imidazo[1,2-a]pyrimidine derivatives, method for the preparation thereof, use thereof as medicaments, pharmaceutical compositions and novel use in particular as met inhibitors |
| 01/21/2010 | WO2010007317A1 Novel imidazo[1,2-a]pyridine derivatives, method for the preparation thereof, use thereof as medicaments, pharmaceutical compositions and novel use in particular as met inhibitors |
| 01/21/2010 | WO2010007316A2 Novel triazolo(4,3-a)pyridine derivatives, process for the preparation thereof, use thereof as medicaments, pharmaceutical compositions and novel use, in particular as met inhibitors |
| 01/21/2010 | WO2010007060A1 Azolin-2-ylamino compounds for combating animal pests |
| 01/21/2010 | WO2010007046A2 Organic compounds |