Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
06/2004
06/24/2004DE69233189T2 Heteroarylpiperidine-pyrrolidine und piperazine und ihre anwendung als antipsychotisches und analgetisches mittel Heteroarylpiperidines-pyrrolidine and piperazine and its application as an antipsychotic and analgesic medium
06/24/2004DE10258671A1 New bis(trifluoromethyl)amide salts of cationic heterocyles, useful e.g. as ionic liquids and as intermediates for pharmaceuticals and plant-protection agents
06/24/2004DE10258314A1 New alkoxyimino-substituted biphenylcarboxamide derivatives, useful as pesticides, antimicrobials, herbicides and antimycotics, also their new intermediates
06/24/2004CA2508608A1 Substituted piperazine compounds and their use as fatty acid oxidation inhibitors
06/23/2004EP1431285A1 Reverse hydroxamic acid derivatives
06/23/2004EP1430120A1 Inhibitors of glycogen synthase kinase-3 (gsk-3) for treating glaucoma
06/23/2004EP1430039A2 Aryl derivatives for the treatment of diabetes, hyperlipidemia, hypercholesterolemia and atherosclerosis
06/23/2004EP1429765A2 Inhibitors of histone deacetylase
06/23/2004EP1429763A2 NOVEL LIGANDS FOR THE HisB10 Zn2+ SITES OF THE R-STATE INSULIN HEXAMER
06/23/2004EP1230227B1 Benzoxa-and benzothiazolyl sulfamates and their use as steroid sulfatase inhibitors
06/23/2004EP1036075B1 Substituted thiazolidinedione and oxazolidinedione having antidiabetic, hypolipidemia and antihypertensive properties
06/23/2004CN1507436A Aryl and heteroaryl urea CHK1 inhibitors for use as radiosensitizers and chamosensitizers
06/22/2004US6753431 Production of mixed acid anhydride and amide compound
06/22/2004US6753429 1,4-disubstituted benzenes as insecticides
06/22/2004US6753426 Antiinflammatory agents; autoimmune disease
06/22/2004US6753347 Intermediates for the synthesis of benzimidazole derivatives and a process for the preparation thereof
06/22/2004US6753344 Thiophene substituted hydroxamic acid derivatives as cyclooxygenase-2 and 5-lipoxygenase inhibitors
06/22/2004US6753340 Autoimmune disease, antiarthritic agents, antiallergens, anticancer agents
06/17/2004WO2004050645A1 Substituted (thiazol-2-yl) -amide or sulfonamide as glycokinase activators useful in the treatment of type 2 diabetes
06/17/2004WO2004050623A1 Methods for preparing phenylalkyne derivatives
06/17/2004WO2004050613A2 2-substituted-3-propenamide derivatives and methods of using the same
06/17/2004WO2004050609A1 Substituted ureas and carbamates
06/17/2004WO2004050022A2 Phenylalanine derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
06/17/2004WO2004021997A3 Inhibitors of fungal invasion
06/17/2004WO2004018414A3 Antibacterial agents
06/17/2004WO2003040116A8 A process for the preparation of cephalosporins side chains
06/17/2004US20040116744 Substituted n-phenyl-phenoxy nicotinic acid-(thio)amides and their use as herbicides
06/17/2004US20040116489 (1S*,2S*,4S*,5R*,6S*) 2-Amino-4-(3-phenylthioureido)-bicyclo[3.1.0]hexane-2,6-dicarboxylic acid for treatment of neurological disorders and psychiatric disorders
06/17/2004US20040116486 Metalloproteinase inhibitors
06/17/2004US20040116485 Broad spectrum 2-(substituted-amino)-benzothiazole sulfonamide hiv protease inhibitors
06/17/2004US20040116484 comprises a mixture with fungicidally active compounds, except for cyclopropylcarboxamide derivatives and azolylmethylcycloalkanes
06/17/2004US20040116483 Glucagon antagonists/inverse agonists
06/17/2004US20040116445 Substituted thioacetamides
06/17/2004US20040116439 Serine protease inhibitors
06/17/2004US20040116424 Aryl imidazoles and related compounds as C5a receptor modulators
06/17/2004US20040116418 Compounds and methods for inhibition of HIV and related viruses
06/17/2004US20040116404 Sulphones which modulate the action of gamma secretase
06/17/2004US20040116399 for preventing or treating coagulation disorders
06/17/2004US20040116353 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same
06/17/2004CA2508487A1 Phenylalanine derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
06/17/2004CA2507875A1 Methods for preparing phenylalkyne derivatives
06/17/2004CA2507484A1 Substituted ureas and carbamates
06/17/2004CA2498089A1 Substituted (thiazol-2-yl) -amide or sulfonamide as glycokinase activators useful in the treatment of type 2 diabetes
06/16/2004EP1428820A1 Non-imidazole alkylamines as histamine H-3-receptor ligands and their therapeutic applications
06/16/2004EP1428533A2 Use of thiazolidine- or pyrrolidine-derivatives of aminoacids as antihyperglycemic agents
06/16/2004EP1428531A1 Oxyiminoalkanoic acid derivatives with hypoglycemic and hypolipidemic activity
06/16/2004EP1427712A2 Dye-azide compounds for dual phototherapy
06/16/2004EP1089963B1 Hydroxamic acid derivatives as inhibitors of the production of human cd23 and of the tnf release
06/16/2004CN1153759C Novel delta-amino-gamma-hydroxy-omega-aryl-alkane amide compounds
06/15/2004US6750351 Reacting sodium cyanide, sodium hydroxide, methanol, lower alcohol, chlorine and cyanamide to form a carbonimidic acid ester intermediate, cyclization with 2-amino mercaptoethane; high quality crystal, good yield and high purity
06/15/2004US6750255 Calcium receptor-active compounds
06/15/2004US6750238 Aralkyl ester soft drugs
06/10/2004WO2004048329A1 Antitumor benzoylsulfonamides
06/10/2004WO2004048309A1 Vitamin d receptor modulators
06/10/2004WO2004047760A2 Novel chemical compounds
06/10/2004WO2004047756A2 Propargyl-trifluoromethoxy-amino-benzothiazole derivatives
06/10/2004WO2004047744A2 3-heterocyclic benzylamide derivatives as potassium channel openers
06/10/2004WO2004024061A3 Aryl-link-aryl substituted thiazolidine-dione and oxazolidine-dione as sodium channel blockers
06/10/2004WO2004016578A3 Arylethanolamine beta2-adrenoreceptor agonist compounds
06/10/2004WO2003059265A3 Compositions and methods for treating heart failure
06/10/2004US20040110951 thiazolidinedione, oxadiazolidinedione, and triazolone compounds treating obesity, overweight condition, hyperlipidemia, glaucoma, cardiac arrhythmias, skin disorders, thyroid disease, hypothyroidism, thyroid cancer, diabetes, etc.
06/10/2004US20040110832 management, treatment and/or control of diseases caused in intrinsic clotting pathway utilizing factor IX such as stroke, myocardial infarction, aneurysm surgery, and deep vein thrombosis associated with surgical procedures etc
06/10/2004US20040110810 e.g., 2-(2-methyl-5-amino)phenyl-4-(3-pyridyl)-thiazole; c-kit inhibitors; treating cell proliferative, metabolic, allergic, and degenerative disorders.
06/10/2004US20040110809 di- and tricycle-substituted imidazolidine-, oxazolidine- and thiazolidine diones and thiones, e.g., 5-[p-(quinolin-3-yl)-alpha-hydroxybenzyl]-5-methylimidazolidinedione
06/10/2004US20040110808 Acylamino-substituted heteroaromatic compounds and their use as pharmaceuticals
06/10/2004US20040110807 Thiazole derivatives
06/10/2004US20040110802 Antibacterial benzoic acid derivatives
06/10/2004US20040110801 Prevention of degenerative joint diseases, rheumatoid arthritis, osteoarthritis, ulcerative colitis, irritable colon and Crohn's diseas, antitumor agents; drug mixture for transdermal drug delivery, sustained release; chemical synthesis
06/10/2004US20040110753 Tyrosine derivatives
06/10/2004US20040110752 2-amino-5-((hetero)aryl)-thiazole derivatives; treatment of disorders such as cancer, immunologic disorders and allergic disorders, optionally in combination with other drugs such as immunosuppressants
06/10/2004CA2507414A1 Propargyl-trifluoromethoxy-amino-benzothiazole derivatives
06/10/2004CA2507256A1 Thiazolidine compounds in the treatment of anemic conditions
06/09/2004EP1426366A1 Thiazolidine derivative and medicinal use thereof
06/09/2004EP1426360A1 2-phenyl-3-heteroarylpropionic acid derivative or salt thereof and medicine containing the same
06/09/2004EP1426046A1 Novel use of tricyclic compound
06/09/2004EP1425265A1 Derivatives of c2-substituted indan-1-ol systems, methods for the production thereof and their use as medicaments
06/09/2004EP1425258A2 Hydroxyeicosenoic acid analogs
06/09/2004EP1425030A2 Non-oxidatively metabolized compounds and compositions, synthetic pathways therefor, and uses thereof
06/09/2004DE10255660A1 New macrocycles useful for the treatment of cancer
06/09/2004CN1503790A Heterocyclic sulfonamide inhibitors of beta amyloid production
06/09/2004CN1503788A Novel azoles having an insecticidal action
06/09/2004CN1503786A Large conductance calcium-activated k channel opener
06/09/2004CN1503774A Carboxylic acid derivative and thereof
06/09/2004CN1502613A Polymorph of a pharmaceutical and prepation
06/08/2004US6747146 Method of producing nitroguanidine- and nitroenamine derivatives
06/08/2004US6747053 Heteroaryl nitriles
06/08/2004US6747041 Heterocyclic dicarboxylic acid diamide derivatives, agricultural/horticultural insecticides and method of using the same
06/08/2004US6747023 Sulfonyl derivatives
06/08/2004CA2079692C Novel 7-substituted-9-substituted amino-6-demethyl-6-deoxytetracyclines
06/03/2004WO2004046170A2 Tubulysins, method for producing the same and tubulysin preparations
06/03/2004WO2004046162A2 Non-steroidal fxr agonists
06/03/2004WO2004046095A1 Substituted aryl thioureas and related compounds; inhibitors of viral replication
06/03/2004WO2004045536A2 Method and compositions for temporarily incapaciting subjets
06/03/2004WO2004045533A2 Method and compositions for treating persistent pulmonary hypertension using aralkyl ester soft drugs
06/03/2004WO2004033418A3 Sulfonylamino-acetic derivatives and their use as orexin receptor antagonists
06/03/2004WO2004022060A8 (1h-benzoimidazol-2-yl)-(piperazinyl)-methanone derivatives and related compounds as histamine h4-receptor antagonists for the treatment of inflammatory and allergic disorders
06/03/2004WO2003051842A3 Compositions decreasing activity of hormone-sensitive lipase
06/03/2004US20040106802 Novel compounds and therapeutic uses thereof
06/03/2004US20040106663 Inhibitors of fungal invasion
06/03/2004US20040106658 Heterocyclic fluoroalkenyl thioethers and the use thereof as pesticides(III)