Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
08/2006
08/17/2006WO2006086705A1 Substituted bis aryl and heteroaryl compounds as selective 5ht2a antagonists
08/17/2006WO2006085815A1 Thiazole derivatives, their process for their preparation and their use in therapy
08/17/2006WO2006085510A1 Remedy for irritable bowel syndrome
08/17/2006WO2006085108A1 Awthranilic acid derivatives and their use in treatment of diseases of lipid metabolism, in particular dyslipidaemia
08/17/2006WO2006070349A3 Novel process for preparing pramipexole and its optical isomeric mixture by reduction with sodium triacetoxyborohydride
08/17/2006WO2005107762A3 Certain chemical entities, compositions, and methods
08/17/2006WO2005037845A8 Benzothiazole and thiazole[5,5-b] pyridine compositions and their use as ubiquitin ligase inhibitors
08/17/2006US20060183918 Beta 2-adrenergic receptor agonists
08/17/2006US20060183915 reacting a 1-halo, mesylate, or tosylate-4,4-difluorobutene with a thiocyanate, giving a butenylthiocyanate; converting to a dithiocarbamate by reacting with hydrogen sulfide; condensation and cyclization with (chloro)acetaldehyde; circumvents 2-mercapto-1,3-thiazole intermediate; by-product inhibition
08/17/2006US20060183914 reacting a 1-halo, mesylate, or tosylate-4,4-difluorobutene with a thiocyanate, giving a butenylthiocyanate; converting to a dithiocarbamate by reacting with hydrogen sulfide; condensation and cyclization with (chloro)acetaldehyde; circumvents 2-mercapto-1,3-thiazole intermediate; by-product inhibition
08/17/2006US20060183913 N-[4-Methyl-5-(2-nitrooxy-ethyl)-thiazol-2-yl]-formamide for example; compound forms a naturally occurring metabolite when NO is released to slow or prevent drug tolerance; treating cardiovascular diseases, inflammation, psychiatric and neurological diseases, respiratory diseases, urogenital disorders
08/17/2006US20060183912 1,4-Bis-[4-Methyl-5-(2-nitrooxy)-ethyl)-thiazol-2-yl]-butane for example; forms a naturally occurring metabolite is formed when nitric oxide is released; treating for example cardiovascular diseases, inflammation, psychiatric and neurological diseases, respiratory diseases, urogenital disorders
08/17/2006US20060183805 Non-oxidatively metabolized compounds and compositions, synthetic pathways therefor, and uses thereof
08/17/2006US20060183783 2-[3-(2-cyclopentanecarbonyl-4-methyl-phenyl)-ureido]-thiazol-4-yl} acetic acid; 2-[3-(4-Methyl-2-[2-methylpropoxy] phenyl)-ureido]-thiazol-4-yl}-acetic acid; activators of glucokinase; treatment of metabolic disorders, hyperglycemic agent, syndrome x, anticholesterol, hypertension etc.
08/17/2006US20060183781 Novel thiazolylmethyl pyrazoles, method for the production thereof, and use thereof in dyes for keratin fibers
08/17/2006US20060183718 Thiazole-based nitric oxide donors having aryl substituent(s) and uses thereof
08/17/2006US20060183177 For detection of caspases, trypsin and tryptase; comprises luciferase and amino-modified aminoluciferin or a carboxy-terminal protected derivative; solid phase synthesis
08/17/2006CA2598429A1 Substituted bis aryl and heteroaryl compounds as selective 5ht2a antagonists
08/16/2006EP1689726A1 5-(benz- (z) -ylidene) -thiazolidin-4-one derivatives as immunosuppressant agents
08/16/2006EP1689716A1 Biaryl sulfonamides and methods for using same
08/16/2006EP1689706A2 Alpha, beta-unsaturated sulfoxides for treating proliferative disorders
08/16/2006EP1689391A2 5-phenyl-4-methyl-thiazol-2-yl-amine derivatives as inhibitors of phosphatidylinositol 3 kinase enzymes (pi3) for the treatment of inflammatory airway diseases
08/16/2006EP1689380A2 Method for treating adamts-5-associated disease
08/16/2006EP1689231A2 Insecticidal n-(heteroarylalkyl) alkanediamine derivatives
08/16/2006EP1583752B1 Cyclization process for substituted benzothiazole derivatives
08/16/2006EP1397488B1 Novel compounds for chemiluminescense procedures
08/16/2006EP1191019B1 Intermediates for the synthesis of benzimidazole compounds and process for the preparation thereof
08/16/2006EP1087941B1 Thiolesters and uses thereof
08/16/2006EP1019075B9 Beta 2-adrenergic receptor agonists
08/16/2006CN1269801C Amino acid derivatives and drug containing the same as the active ingredient
08/16/2006CN1269528C Application of dipeptide base peptidase IV effector for reducing blood sugar level of mammal
08/15/2006US7091380 Bradykinin B1 antagonists or inverse agonists, for prophylaxis and therapy of pain and inflammation
08/15/2006US7091360 Reacting nitrogen compounds such as benzoxazole, with grignard reagents to form chemical intermediates used to form cysteine protease inhibitors
08/15/2006US7091359 Process for the preparation of thiazolidinedione derivatives
08/15/2006US7091242 Beta-amino acid derivatives as integrin receptor antagonists
08/15/2006US7091228 4-[4'-(1,3-Benzothiazol-2-ylamino)-1,1'-biphenyl-4-yl]-2,2-dimethyl-4-oxobutanoic acid and derivatives; inhibition of DGAT-1 (diacylglycerol O-acyltransferase type 1)
08/15/2006US7091227 Serine/threonine and tyrosine kinases inhibitors
08/15/2006US7091225 Substituted oxazoles and thiazoles as hPPAR alpha agonists
08/15/2006US7091223 Autoimmune diseases; anticancer agents
08/15/2006US7091219 Administering an effective amount of bis-sulfonamide hydroxyethyl-amino derivative to a HIV patient to prevent the viral replication
08/10/2006WO2006083781A1 Antidiabetic bicyclic compounds
08/10/2006WO2006083271A2 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication
08/10/2006WO2006082952A1 Amide compound
08/10/2006WO2006082495A1 Peroxisome proliferator activated receptor modulators
08/10/2006WO2006082107A1 Thiazolidinones for use as inhibitors of polo-like kinase (plk)
08/10/2006WO2006066778A3 Novel heteroarylacetamides
08/10/2006US20060178429 2-Phenyl-3-hydrogenated furanyl, pyranyl, thiophenyl or thiopyranyl-N-heteroaromatic propionamides, e.g., 2-(3,4-Dichloro-phenyl)-3-(tetrahydro-pyran-2-yl)-N-thiazol-2-yl-propionamide; compounds increase insulin secretion in the treatment of type II diabetes.
08/10/2006US20060178410 Preparation of N-{2-[4-(3-phenyl-4-methoxyphenyl)aminophenyl]ethyl}-2-hydroxy-2-(3-hydroxymethyl-4-hydroxyphenyl)ethylamine, for example; for the treatment of pulmonary diseases such as asthma and chronic obstructive pulmonary disease
08/10/2006US20060178356 Treating oxidative stress-related conditions typically responsive to cellular enzyme modulation with a substituted phenolic compound having unsaturated groups, e.g. 1-((3-methyl-5-oxo-2-pyrazolin-1-yl), 4-(3-methoxy-4-hydroxy-phenyl)-vinyl-)benzene; skin disorders; antiischemic and cardiotonic agents
08/10/2006US20060177621 O-coordinated metal chelates and their use in optical recording media having high storage capacity
08/10/2006DE102005005813A1 New thiazolo-indazole derivatives useful as PI3 kinase inhibitors, for treating e.g. cancer and other proliferative diseases, viral infections and inflammatory, autoimmune, skin and bone diseases
08/10/2006CA2596967A1 Thiazolidinones for use as inhibitors of polo-like kinase (plk)
08/10/2006CA2593858A1 Antidiabetic bicyclic compounds
08/10/2006CA2566809A1 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication
08/09/2006EP1688138A1 Receptor function regulating agent
08/09/2006EP1687287A1 A novel process for ezetimibe intermediate
08/09/2006EP1687285A1 Thiazole and pyrazole derivatives as flt-3 kinase inhibitors
08/09/2006EP1687021A1 Method of removing transition metals, especially from metathesis reaction products
08/09/2006EP1455779B1 Indolylalkylamine derivatives as 5-hydroxytryptamine-6 ligands
08/09/2006CN1816532A Heterocyclically-substituted pentanol derivatives, process for their production and their use as anti-inflammatory agents
08/09/2006CN1816531A Preparation and use of aryl alkyl acid derivatives for the treatment of obesity
08/08/2006US7087761 Cyclic thiourea and acetylthiourea derivatives of benzothiazole for drugs
08/08/2006US7087644 Cardiovascular disorders; stimulant of guanylate cyclase ; therapy for liver fibrosis
08/08/2006US7087623 Thiazole and other heterocyclic ligands for mammalian dopamine, muscarinic and serotonin receptors and transporters, and methods of use thereof
08/08/2006US7087614 Pyrimidine inhibitors of phosphodiesterase (PDE) 7
08/08/2006US7087610 Aids therapy
08/08/2006US7087604 Antiarthritic agents;multiple sclerosis; anticholesterol agents; cardiovascular disorders
08/08/2006US7087593 Psychological disorder treatments that increase the activity of cholinergic receptors
08/08/2006US7087229 Releasable polymeric conjugates based on aliphatic biodegradable linkers
08/08/2006CA2200707C Novel prostaglandin synthase inhibitors
08/08/2006CA2188835C Novel compounds and methods for synthesis and therapy
08/03/2006WO2006081165A1 Improved process for preparing (dihalopropenyl)phenylakeyl substituted benzoxazoles
08/03/2006WO2006080407A1 Ppar-activating compound
08/03/2006WO2006080406A1 Tricyclic compounds
08/03/2006WO2005060456A8 Method for treating adamts-5-associate disease
08/03/2006WO2003072033A3 Common ligand mimics: thiazolidinediones and rhodanines
08/03/2006US20060173190 Nematicidal thiazoline-containing fluorobutenes
08/03/2006US20060173075 P-(sulfonyl) aryl and heteroarylamines-as anti-inflammatory agents
08/03/2006US20060173044 Substituted propargylamines
08/03/2006US20060173013 Piperidinyl cyclopentyl aryl benzylamide modulators of chemokine receptor activity
08/03/2006US20060172990 Antibacterial agents
08/03/2006US20060172936 e.g. hexahydrofuro[2,3-b]furan-3-yl N-((1S,2R)-1-benzyl-3-(cyclopentyloxy)[(3-[2-(dimethylamino)ethyl]aminophenyl)sulfonyl]amino-2-hydroxypropyl)carbamate; against human immunodeficiency virus, chronic and acute viral infections
08/03/2006CA2593803A1 Thiazole-amide compounds and compsitions as protein kinase inhibitors
08/02/2006EP1686114A1 Process for producing optically active 2-alkylcysteine, derivative thereof, and processes for production
08/02/2006EP1685119A1 N-acylsulfonamide apoptosis promoters
08/02/2006EP1685118A2 Compounds having beta2 adrenergic receptor agonist and muscarinic receptor antagonist activity
08/02/2006EP1685095A1 Method for the production of organic salts containing bis(perfluoroalkyl)phosphinate anions
08/02/2006EP1684762A2 Urea derivatives as kinase modulators
08/02/2006EP1684745A2 Hepatitis c virus inhibitors
08/02/2006EP0986551B1 Sulfonamide derivatives, their production and use
08/02/2006CN1812978A Phenyl substituted carboxylic acids as inhibitors of protein tyrosine phosphatase-1b
08/02/2006CN1812977A Substituted carboxylic acids
08/02/2006CN1812966A N-alkynyl-2- (substituted aryloxy) alkylthioamide derivatives as fungicides
08/02/2006CN1812959A Method for producing difluoro-acetyl-acetic acid alkylesters
08/02/2006CN1812956A Biaryloxymethylarenecarboxylic acids as glycogen synthase activator
08/02/2006CN1810791A Synthesis process of medicine for treating hemopathy
08/02/2006CN1267418C Diarylselenide compounds and their use in human or veterinary medicine and in cosmetics
08/01/2006US7084170 Antitumor agents for treating a tumor of the colon or rectum in a mammal; N-[2,4-dichlorobenzoyl]-5-bromothiophene-2-sulfonamide sodium salt
08/01/2006US7084166 Such as 1,1-di-(N-benzyl-indol-3-yl)-1-butene; for drug resistant tumors
08/01/2006US7084162 Substituted acid derivatives useful as antidiabetic and antiobesity agents and method