Patents
Patents for C07D 271 - Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms (7,144)
07/2005
07/21/2005WO2005065683A1 Triazole, oxadiazole and thiadiazole derivative as ppar modulators for the treatment of diabetes
07/21/2005CA2549385A1 Triazole, oxadiazole and thiadiazole derivative as ppar modulators for the treatment of diabetes
07/20/2005EP1554361A1 Metallic complexes covalently bound to conjugated polymers and electronic devices containing such compositions
07/20/2005CN1211367C Prostaglandin agonists and their use to treat bone disorders
07/19/2005US6919343 N-biphenyl(substituted methyl) aminocycloalkane-carboxamide derivatives
07/14/2005WO2005063742A2 Amidino compounds as cysteine protease inhibitors
07/14/2005WO2005063705A1 Benzene compounds disubstituted with cyclic groups at the 1- and 2-positions
07/14/2005WO2005063690A1 Alpha-hydroxy amides as bradykinin antagonists or inverse agonists
07/14/2005WO2005040142B1 Novel keto-oxadiazole derivatives as cathepsin inhibitors
07/14/2005WO2005013888A3 Compounds, compositions and methods
07/14/2005US20050154211 Reacting carboxy nitriles with hydroxylamine salts, then anhydriding the chemical intermediates and cyclization to form nitrogen compounds such as ethyl 5-(2-((t-butoxy)carbonyl amino)ethyl)-1,2,4-oxadiazole-3-carboxylate
07/14/2005US20050154202 Substituted aryl amides
07/14/2005US20050153996 Compounds that modulate ppar activity and methods for their preparation
07/13/2005EP1553085A1 Cyclic amine derivatives and their use as drugs
07/13/2005CN1639141A New thiadiazoles and oxadiazoles and their use as phosphodiesterase-7 inhibitors
07/13/2005CN1639137A Substituted 3-phenyl-5-alkoxy-1, 3, 4-oxadiazol-2-ones, the production thereof and their use in medicaments
07/13/2005CN1639115A Semicarbazide derivatives and their use as antithrombotics
07/13/2005CN1638766A Use of substituted 3-phenyl-5-alkoxy-1, 3, 4-oxdiazole-2-one for producing medicaments that inhibit pancreatic lipase
07/13/2005CN1638757A 组织蛋白酶半胱氨酸蛋白酶抑制剂 Cathepsin cystatin
07/13/2005CN1210268C (Cyclo) alkyl substituted-gamma-aminobutyric acid derivatives (=GABA analogurs), their preparation and their use in the treatment of neurolog disorders
07/12/2005US6916850 Pyruvate derivatives
07/12/2005CA2238859C Amino acid derivatives, pharmaceutical compositions containing these compounds and processes for preparing them
07/06/2005EP1549624A2 Inhibitors of fatty acid amide hydrolase
07/06/2005EP1549306A1 Substituted phenylsulfonamide inhibitors of beta amyloid production
07/06/2005EP1216225B1 Novel derivatives of dicarboxylic acid having pharmaceutical properties
07/05/2005US6914158 Amidino compounds useful as nitric oxide synthase inhibitors
07/05/2005CA2230082C Amide compounds and use thereof
06/2005
06/30/2005WO2005058884A2 Cyclopropane compounds and pharmaceutical use thereof
06/30/2005WO2005058868A1 N-(4-carbamimidoyl-benzyl) -2-alkoxy-2-heterocyclyl acetamides as inhibitors of the formation of coagulation factors xa, ixa and thrombin induced by factor viia
06/30/2005WO2005058848A1 (3,4-disubstituted)propanoic carboxylates as s1p (edg) receptor agonists
06/30/2005WO2005058808A1 N-substituted-n-sulfonylaminocyclopropane compounds and pharmaceutical use thereof
06/30/2005WO2005058311A1 Heterocyclic aspartyl protease inhibitors
06/30/2005WO2005020899A3 Substituted cycloalkyamine derivatives as modulators of chemokine receptor activity
06/30/2005US20050143426 Osteoporosis, bone disorders, or diseases associated with excessive secretion of PTH, such as hyperparathyroidism; reduce or inhibit parathyroid hormone (PTH) secretion
06/30/2005CA2549825A1 N-(4-carbamimidoyl-benzyl) -2-alkoxy-2-heterocyclyl acetamides as inhibitors of the formation of coagulation factors xa, ixa and thrombin induced by factor viia
06/30/2005CA2549660A1 Cyclopropane compounds and pharmaceutical use thereof
06/30/2005CA2549598A1 N-substituted-n-sulfonylaminocyclopropane compounds and pharmaceutical use thereof
06/30/2005CA2548388A1 Heterocyclic aspartyl protease inhibitors
06/30/2005CA2547198A1 (3,4-disubstituted)propanoic carboxylates as s1p (edg) receptor agonists
06/29/2005EP1546089A2 Aryl and heteroaryl compounds and methods to modulate coagulation
06/29/2005CN1633410A Substituted methylene amide derivatives as modulators of protein tyrosine phosphatases(ptps)
06/29/2005CN1208327C Process for preparing S, Síõ-carbonyl disulfhydryl substituted five-membered heterocyclic compound
06/23/2005US20050137212 Hppars activators
06/23/2005US20050137200 Potassium channel modulators; antiarrhythmia agents
06/23/2005US20050137168 inhibit the formation of coagulation factors Xa, IXa and thrombin induced by factor VIIa and tissue factor; for treatment and/or prevention of arterial and venous thrombosis, deep vein thrombosis, pulmonary embolism, unstable angina pectoris, cardiac infarction, stroke
06/22/2005CN1630633A N-biphenylmethyl aminocycloalkanecarboxamide derivatives with a substiituent on the methyl useful as bradykinin antagonists
06/21/2005US6908938 Heterocyclic aromatic compounds useful as growth hormone secretagogues
06/21/2005US6908937 Heterocyclic fluoroalkenyl thioethers (II)
06/21/2005US6908935 Calcium receptor modulating agents
06/21/2005US6908492 Cationic hair dyes; colorfastness, photostability
06/16/2005WO2005032550A3 Peptide deformylase inhibitors
06/16/2005WO2005003081A3 Sulfonimide containing compounds and their use in polymer electrolyte membranes for electrochemical cells
06/14/2005US6906072 Central nervous system disorders
06/14/2005US6906006 Applying to plants, environment
06/14/2005CA2304967C 4(3)substituted-4(3)-aminomethyl-(thio)pyran or -piperidine derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
06/09/2005WO2005051932A1 Arylheterocycle derivative and agricultural or horticulrual bactericide and insecticide
06/09/2005WO2005040142A9 Novel keto-oxadiazole derivatives as cathepsin inhibitors
06/09/2005US20050124656 Substituted methylene amide derivatives as modulators of protein tyrosine phosphatases(ptps)
06/09/2005US20050124654 Compounds and methods of use
06/09/2005US20050124631 For example, 2-amino-7-chloro-6-hydroxy-4-methylbenzothiazole; compounds that prevent the formation of polyglutamine containing protein aggregates; treatment of spinal and bulbar muscular atrophy, dentatorubal pallidoluysian atrophy, spinocerebellar ataxia, Alzheimers disease
06/08/2005EP1537077A2 4-(3,3-dihalo-allyloxy) phenol derivatives having pesticidal properties
06/08/2005EP1536790A2 Oxadiazoles as modulators of metabotropic glutamate receptor-5
06/08/2005EP1536784A1 Hetero biaryl derivatives as matrix metalloproteinase inhibitors
06/08/2005EP1373231B1 3-heterocyclyl-propano-hydroxamic acid as pcp inhibitors
06/08/2005EP0849256B1 Amide compounds and use of the same
06/08/2005CN1205185C Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
06/07/2005US6903216 Antiarrhythmic agents for the treatment and prophylaxis of atrial arrhythmias, atrial fibrillation (AF) or atrial flutter; potassium channel modulators, beta-blocker
06/02/2005US20050119332 Substituted thiophene compounds as modulators of protein tyrosine phosphatases (PTPases)
06/02/2005US20050119316 Semicarbazide derivatives and the use thereof as antithrombotics
06/02/2005US20050119312 Lipid lowering agents; hypotensive agents; obesity
06/01/2005EP1535909A2 Cyclic amine derivatives and their use as drugs
06/01/2005EP1534671A2 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
06/01/2005EP1534259A2 Sulfonamides as potassium channel blockers
06/01/2005EP0946499B1 N-(aryl/heteroaryl/alkylacetyl) amino acid amides, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds
05/2005
05/31/2005US6900233 Substituted 3-phenyl-5-alkoxy-3H-(1,3,4)-oxadiazol-2-ones, pharmaceutical composition and method for treating obesity thereof
05/31/2005US6900218 Reducing oxidation stresses; central nervous system disorders; antiinflammatory agents
05/31/2005US6900207 N-containing five-membered ring compounds and pharmaceutical agents comprising the same as active ingredient
05/26/2005US20050113451 7-acetamidinyl derivatives
05/26/2005US20050113440 Compounds that modulate PPAR activity and methods for their preparation
05/26/2005US20050113428 2-{3,5-bis[(3-chlorobenzyl)oxy]benzyl}-1,2,4-oxadiazolidine-3,5-dione to treat disorders associated with elevated PAI-1(Plasminogen activator inhibitor) levels
05/26/2005US20050112407 Organic electroluminescent device
05/25/2005EP1533292A1 Dibenzylamine compound and medicinal use thereof
05/25/2005EP1531810A2 Substituted heterocyclic derivatives useful as antidiabetic and antiobesity agents and method
05/25/2005CN1620424A Compounds for the treatment of inflammatory disorders
05/24/2005US6897306 3-heterocyclylpropanohydroxamic acids
05/24/2005US6897237 MMP-12 inhibitors
05/24/2005US6897220 Antiproliferative agents
05/24/2005CA2155840C Hydroxymethyl furazane carboxylic acid derivatives and their use in the treatment of cardio-vascular conditions
05/19/2005US20050107616 Alpha-ketoamide derivatives as cathepsin k inhibitors
05/19/2005US20050107444 E.g., 2-(3-{3-[(2-chloro-3-(trifluoromethyl)-benzyl)-(2,2-diphenylethyl)-amino]-propoxy}phenyl)-1-morpholin-4-yl-ethanone; agonists of the nuclear receptors, LXR alpha and LXR beta used to increase ABCA1, ABCG1, and apolipoprotein E expression and inhibiting cholesterol absorption
05/19/2005US20050107354 Preventive or therapeutic agent for kidney disease
05/18/2005EP1265860B1 Amidino compound and salts thereof useful as nitric oxide synthase inhibitors
05/18/2005CN1617852A Alpha-(n-sulphonamido)acetamide derivatives as beta-amyloid inhibitors
05/18/2005CN1617850A Dibenzylamine compound and medicinal use thereof
05/18/2005CN1616592A White light-emitting compound, process for producing the same, and luminescent element utilizing the same
05/18/2005CN1202095C Heteroaromatic ring compounds
05/18/2005CN1202094C 1,2,4-oxdiazoline containing substituent of aryl group in 3 position and its solid phase synthesis method
05/17/2005US6894072 Compounds as NS3-serine protease inhibitors of hepatitis C virus
05/17/2005US6894054 Central nervous system disorders; muscular disorders
05/17/2005US6893650 Fungicides; locus infestation; such as N,N-dimethyl-N'-(4-(3-trifluoromethylbenzylthio)-2,5-xylyl)formamidine
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