Patents for C07D 265 - Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms (11,132) |
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04/10/2003 | US20030069210 Especially imidazolyl- or 1,2,4-triazolyl- pyrimidine derivatives |
04/10/2003 | CA2462647A1 6-membered unsaturated heterocyclic compounds useful for selective inhibition of the coagulation cascade |
04/10/2003 | CA2462601A1 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade |
04/10/2003 | CA2462305A1 6-membered heterocyclic compounds useful for selective inhibition of the coagulation cascade |
04/10/2003 | CA2459825A1 Compounds useful as reversible inhibitors of cysteine proteases |
04/09/2003 | EP1299354A2 Factor viia inhibitory (thio)urea derivatives, their preparation and their use |
04/09/2003 | EP1003758B1 Solution phase synthesis of oligonucleotides |
04/08/2003 | US6545108 Catalysts containing N-pyrrolyl substituted nitrogen donors |
04/08/2003 | US6545049 E.g., (2E, 4E, 6E)-7-(3,5-diisopropyl-2-n-heptyloxyphenyl)-3-methylocta-2,4,6-trienoic acid, esters or amides thereof |
04/08/2003 | US6545038 Heterocyclic metalloprotease inhibitors |
04/08/2003 | CA2275323C Asymmetric synthesis of benzoxazinones |
04/03/2003 | WO2003027084A1 Improved process for the preparation of optically active phenoxazine derivatives as antidiabetic agents |
04/03/2003 | US20030065176 Anticoagulant; cardiovascular disorders |
04/03/2003 | US20030064992 N-aryl (thio) anthranilic acid amide derivatives, their preparation and their use as VEGF receptor tyrosine kinase inhibitors |
04/02/2003 | EP1296936A1 Thyroid receptor ligands, pharmaceutical compositions comprising them and their use in the treatment of disorders influenced by thyroid hormones |
04/02/2003 | EP0944609B1 Process for preparing n-alkyl ammonium acetonitrile compounds |
04/02/2003 | EP0873295B1 Dimer-selective rxr modulators and methods for their use |
04/02/2003 | CN1407977A (Hetero) aryl-substituted heterocyclic enaminones, production therof and use thereof as herbicides, acaricides and insecticides |
04/01/2003 | US6541669 Multibinding amine compounds which are beta 2 adrenergic receptor agonists useful in treatment and prevention of respiratory diseases such as asthma, bronchitis |
04/01/2003 | US6541471 Useful as a TXA2 receptor antagonist and a 5-HT2 receptor antagonist |
03/27/2003 | WO2003024949A1 Dna-pk inhibitors |
03/27/2003 | WO2003024941A1 Naphthalene compounds and use thereof as drugs |
03/27/2003 | WO2003024448A2 Inhibitors of histone deacetylase |
03/27/2003 | WO2003024401A2 Piperizinones as modulators of chemokine receptor activity |
03/27/2003 | US20030060452 N-heterocyclic derivatives as NOS inhibitors |
03/27/2003 | CA2465978A1 Inhibitors of histone deacetylase |
03/27/2003 | CA2454023A1 Dna-pk inhibitors in the treatment of retroviral mediated diseases |
03/26/2003 | EP1294704A1 Aryl phenylheterocyclyl sulfide derivatives and their use as cell adhesion-inhibiting anti-inflammatory and immune-suppressive agents |
03/26/2003 | EP1294700A2 Benzhydryl derivatives |
03/25/2003 | US6538134 Forming by reacting N-benzylethanolamine with glycoxylic acid in solvent; intermediate in synthesis of substance P receptor antagonists |
03/25/2003 | US6538024 Felbamate derived compounds |
03/20/2003 | WO2002085841A3 Substituted catechol derivatives derived from polybasic secondary amino acids, method for production and use thereof |
03/20/2003 | US20030055093 For therapy of cardiovascular diseases, stable or unstable angina pectoris, coronary heart disease, stable or unstable angina pectoris, coronary heart disease, Prinzmetal angina, acute coronary syndrome, heart failure, myocardial infarction |
03/20/2003 | US20030055076 Novel compounds, their preparation and use |
03/19/2003 | EP1292584A1 Process for the synthesis of (2r, 2-alpha-r, 3a)-2- 1-(3,5-bis(trifluoromethyl)phenyl)ethoxy]-3-(4-fluorophenyl)-1,4-oxazine |
03/19/2003 | EP1292583A1 Process for the synthesis of (2r, 2-alpha-r)-4-benzyl-2- 1-(3,5-bis(trifluoromethyl)phenyl)ethoxy]-1,4-oxazin-3-one |
03/19/2003 | EP1292582A1 4-benzyl-2-hydroxy-1,4-oxazin-3-one and polymorphic forms thereof |
03/18/2003 | US6534535 Inhibitors of factor Xa |
03/13/2003 | WO2003020709A1 1,2-oxazin-3-one derivatives as antibacterial agents |
03/13/2003 | WO2003020688A1 Selective protein tyrosine phosphatase inhibitors |
03/13/2003 | WO2002078625A3 Therapeutic combinations for cardiovascular and inflammatory indications |
03/13/2003 | US20030050309 A gelatinase inhibitor for modulating the activity of a dopamine, serotonin, or norepinephrine receptor or transporter |
03/13/2003 | US20030050298 A sulfonamide substituted diphenyl thiourea compounds treating a chemokine mediated disease |
03/12/2003 | EP1289965A1 Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists |
03/12/2003 | EP1289964A1 Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists |
03/12/2003 | EP0874830B1 A metalloproteinase inhibitor, a pharmaceutical composition containing it and the pharmaceutical use and method useful for the preparation thereof |
03/12/2003 | CN1401639A Process for synthesis of azacyclic compounds |
03/11/2003 | US6531610 Intermediate acylating carbonate |
03/11/2003 | US6531596 S(-)-2-methoxy-3-(4-(2-(phenoxazin-10-yl)methoxy) phenyl)propionic acid; benzylating p-hydroxybenzaldehyde or tyrosine; reaction with phenoxazinyl mesylate |
03/11/2003 | US6531471 Morpholinone and morpholine derivatives and uses thereof |
03/06/2003 | WO2003018566A1 New piperidinyl derivates as modulators of chemokine receptor activity |
03/06/2003 | WO2003018565A1 Method for synthesizing oxazinones |
03/06/2003 | WO2003018535A2 Novel aminobenzoephenones |
03/05/2003 | EP1288205A1 Novel phenylalanine derivatives |
03/05/2003 | EP1286978A1 Cyclohexyl derivatives and their use as therapeutic agents |
03/05/2003 | EP1286967A1 Cyclohexane derivatives and their use as therapeutic agents |
03/05/2003 | EP1286956A1 Phenyl-substituted 2-enamino-keto nitriles |
03/05/2003 | EP1140923B1 Method for preparing (r)- (+) -3 1- 2-( 4-benzoyl- 2-(3,4- difluorophenyl)morpholin- 2-yl)ethyl]- 4-phenylpiperidin -4-yl -1,1- dimethylurea, its salts solvates and/or hydrates |
03/04/2003 | US6528627 Bridged aromatic substituted amine ligands with donor atoms |
03/04/2003 | US6528507 Arginine salt of 3-(4-(2-(phenoxazin-10-yl)ethoxy) phenyl)-2-ethoxypropanoic acid |
02/27/2003 | WO2003016292A1 Ultraviolet light absorbers |
02/27/2003 | WO2003000181A3 Dipeptidyl peptidase inhibitors for the treatment of diabetes |
02/27/2003 | CA2454080A1 Ultraviolet light absorbers |
02/26/2003 | EP1284724A1 Method of preparing alkylated salicylamides via a dicarboxylate intermediate |
02/26/2003 | CN1399639A New oxabispidine compound useful in treatment of cardiac arrhythmias |
02/25/2003 | US6525072 Prevention and treatment of cellular disorders such as cancer |
02/25/2003 | US6525036 Compounds and compositions as protease inhibitors |
02/20/2003 | US20030036558 Useful in the treatment of chronic complications arising from diabetes, such as neuropathy; may also contain an angiotensin converting enzyme inhibitor. |
02/19/2003 | EP1283829A1 Method for making acylamides by synthesizing and acylating benzoxazines |
02/19/2003 | CN1397547A Novel benzene amine compound, its prepn. process and medicinal compsns. contg. them |
02/18/2003 | WO2002016329A1 Novel phenylalanine derivatives |
02/18/2003 | US6521666 Inhibitors of α4 mediated cell adhesion |
02/18/2003 | US6521633 Treating NIDDM with RXR agonists |
02/13/2003 | WO2003011931A1 Use of aromatic polyamines to enhance thermal properties of benzoxazine polymers |
02/13/2003 | WO2003011834A1 Novel vinyl n-(2-benzoylphenyl)-l-tyrosine derivatives and their use as antidiabetics etc |
02/13/2003 | WO2003011298A1 Antibacterial oxazinones and methods for their use and synthesis |
02/13/2003 | US20030032644 Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity |
02/13/2003 | US20030032635 Heterocyclic esters and amides |
02/12/2003 | EP1283199A1 Melanin-concentrating hormone antagonist |
02/12/2003 | EP1282610A1 Benzoxazine and benzothiazine derivatives and the use thereof in medicaments |
02/12/2003 | EP1282414A2 Felbamate derived compounds |
02/11/2003 | US6518310 Non-peptidic; inhibits trypsin-like protease, thrombin and embolus formation; anticoagulant |
02/06/2003 | US20030027821 Administering 2-oxy substituted benzoxazin-5-one derivative to a human or animal for the prevention or treatment of obesity or an obesity related disorder |
02/06/2003 | US20030027794 N-heterocyclic derivatives as NOS inhibitors |
02/06/2003 | US20030027238 Optical molecular sensors for cytochrome P450 activity |
02/05/2003 | EP1280784A2 Biologically active 4h-benzo 1,4]oxazin-3-ones |
02/05/2003 | EP1280783A2 Methods of treatment using benzoxazinones as peroxisome proliferator activated receptor gamma modulators |
02/05/2003 | EP1280782A2 Novel benzoxazinones as peroxisome proliferator activated receptor gamma modulators and method of treatment |
02/05/2003 | CN1395467A Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binding agents |
02/05/2003 | CN1394855A Substituted heterocyclic compound |
02/05/2003 | CN1100777C N-heterocyclic derivatives as NOS inhibitor |
02/05/2003 | CN1100754C Method for producing trifluoroacetoacetic acid anilides |
02/05/2003 | CN1100540C Protein tyrosine kinase aryl and heteroaryl quinazoline compounds having selective inhibition of HER-2 autophosphorylation properties |
02/04/2003 | US6514990 Pharmaceutically active compounds and methods of use |
02/04/2003 | US6514687 Screening a candidate compound for activity as a Cytochrome P450 enzyme substrate by contacting the compound, enzyme, and a reagent chromogen comprising the ether of a phenolic dye such as a coumarin, resofurin or fluorescein dye |
01/30/2003 | WO2003008397A1 An improved process for the preparation of antidiabetic phenoxazine compounds |
01/30/2003 | WO2003008396A1 Optically active oxazine derivative |
01/30/2003 | US20030023007 Enhancement of thermal properties of benzoxazine polymers by use of aromatic polyamines to incorporate internal benzoxazine groups within the monomer |
01/30/2003 | US20030022895 2-Amino-benzoxazinones for the treatment of viral infections |
01/29/2003 | EP1278803A2 Sulfonated 8,9]benzophenoxazine dyes and the use of their labelled conjugates |