Patents
Patents for C07D 263 - Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings (20,978)
10/1995
10/10/1995US5457109 Use of thiazolidinedione derivatives and related antihyperglycemic agents in the treatment of disease states at risk for progressing to noninsulin-dependent diabetes mellitus
10/04/1995EP0675114A1 Oxazolinone derivative having intracellular phospholipase a 2? inhibitor activity
10/04/1995EP0674630A1 7-HALO- AND 7$g(b),8$g(b)-METHANO-TAXOLS, ANTINEOPLASTIC USE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
10/04/1995EP0674626A1 Novel selective aromatase inhibiting compounds
10/04/1995EP0674618A1 Asymmetric process for preparing florfenicol, thiamphenicol, chloramphenicol and oxazoline intermediates
10/03/1995US5455353 4-(benzyl-2-oxo-oxazolidin-5 ylmethyl)N tertbutyl-decahydroisoquinoline-3-carboxamides
10/03/1995US5455260 Anticholesterol agents; reduction of serum cholesterol without reducing mevalonic metabolite synthesis; side effect
09/1995
09/28/1995WO1995025727A1 Naphthylamides as central nervous system agents
09/28/1995DE19510454A1 New aryloxy-phenoxy alkyl- and aryloxy-phenyl-1,3-dioxolan-4-one derivs.
09/27/1995EP0673933A1 Aminoalkyl benzoxazolinones and benzothiazolinones process for their preparation and compositions containing them
09/27/1995EP0673370A1 Tropone-substituted phenyloxazolidinone antibacterial agents
09/27/1995CN1109054A Oxazolidin-2-one derivatives
09/26/1995US5453508 Manufacture of 4-aryl-2-perfluoroalkyl-3-oxazolin-5-one from arylglycine
09/26/1995US5453488 Amino-substituted heterocycles as renin inhibitors
09/24/1995CA2145257A1 Thiazolidine and oxazolidine derivatives, their preparation and their medical use
09/23/1995CA2145026A1 Aminoalkyl benzoxazolinones and benzothiazolinones; process for preparing the same and pharmaceutical compositions containing them
09/21/1995WO1995025106A1 Oxazolidinone derivatives and pharmaceutical compositions containing them
09/21/1995WO1995025104A1 Novel heterocyclic ethanolamine derivatives with beta-adrenoreceptor agonistic activity
09/21/1995WO1995025099A1 2-cyano-1,3-dione derivatives useful as herbicides
09/20/1995EP0672038A1 Herbicides
09/20/1995EP0672034A1 Benzimidazole compounds which inhibit platelet aggregation
09/20/1995EP0672029A1 SELECTIVE PRECIPITATION OF $g(a)-ARYL CARBOXYLIC ACID SALTS
09/20/1995EP0671911A1 Carboxy-peptidyl derivatives as antidegenerative active agents
09/20/1995EP0563358B1 9-substituted bicyclo [3.3.0]octane derivatives, for use as txa2 antagonists
09/19/1995US5451681 Process for preparing nematicidal benzoxazole and benzthiazole compounds
09/19/1995US5451596 Cycloalkyl amine bis-aryl squalene synthase inhibitors
09/19/1995US5451594 Nematocides, insecticides, miticides and fungicides
09/19/1995US5451394 Quaternary salts of para-dialkylamino benzamide derivatives
09/14/1995WO1995024403A1 (4,4-difluorobut-3-enylthio)-substituted heterocyclic or carbocyclic ring compounds having pesticidal activity
09/14/1995WO1995024397A1 3,5-disubstituted and 3,5,6-trisubstituted 2-isoxazolines and isoxazoles, process for preparing the same and their use as medicaments
09/14/1995WO1995024385A1 Sulphonamide derivatives as aspartyl protease inhibitors
09/14/1995WO1995024382A1 L-n6-(1-iminoethyl)lysine derivatives useful as nitric oxide synthase inhibitors
09/14/1995WO1995024379A1 Benzamide analogs, useful as parp (adp-ribosyltransferase, adprt) dna repair enzyme inhibitors
09/14/1995DE4408084A1 3,5-Disubstituierte und 3,4,5-trisubstituierte 2-Isoxazoline und Isoxazole, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel 3,5-Disubstituted and 3,4,5-trisubstituted 2-isoxazolines and isoxazoles, to processes for their preparation and their use as medicaments
09/14/1995CA2350941A1 Benzamide analogues as parp dna repair enzyme inhibitors
09/14/1995CA2185004A1 3,5-disubstituted and 3,4,5-trisubstituted 2-isoxazolines and isoxazoles, process for preparing the same and their use as medicaments
09/14/1995CA2183653A1 Sulphonamide derivatives as aspartyl protease inhibitors
09/14/1995CA2182520A1 (4,4-difluorobut-3-enylthio)-substituted heterocyclic or carbocyclic ring compounds having pesticidal activity
09/13/1995EP0671654A1 Photographic material containing a new type of hydrazide
09/13/1995EP0671160A1 Use of sulphonic acids as antiageing agents in cosmetic and/or dermatological compositions
09/13/1995EP0541706B1 Process and intermediate for the preparation of 2-hydroxy-3-sulfido-3-phenyl propanoic acids
09/13/1995EP0541593B1 Cyclopentane derivatives, process for producing them and their pharmaceutical use
09/13/1995EP0401286B1 Process for preparing n-(hydroxyalkyl)-2-unsaturated amides and 2-alkenyl oxazolines
09/13/1995CN1108252A Oxazoline derivative, process for preparing the same and agricultural and horticultural chemical for controlling noxious organisms containing the same
09/12/1995US5449782 Orally active antiviral compounds
09/12/1995US5449686 4-phenylcyclohexanone derivatives; inhibit production of tumor necrosis factor and phosphodiesterase V
09/08/1995WO1995023797A1 Process for making an epoxide
09/07/1995DE4407135A1 New heterocyclyl substd. aryl-cycloalkyl:amine derivs.
09/07/1995DE4407134A1 New heterocyclyl substd. benzyl-piperazine derivs.
09/06/1995EP0670318A2 Acetamides with analgesic and neuroprotective activity
09/06/1995EP0670305A1 Process for producing 3-amino-2-hydroxy-1-propanol derivative
09/06/1995EP0669915A1 Method for the preparation of 1,3-oxazolidin 5-carboxylic acid.
09/05/1995CA1336911C Serotonin antagonists
09/04/1995CA2143691A1 Acetamides
08/1995
08/30/1995EP0669323A1 Utilization of benzazols as UV-absorbers, new benzazoles and process for their preparation
08/30/1995EP0668859A1 Processes for preparing 2,4-oxazolidinediones.
08/30/1995CN1107468A Preparation of novel heterocyclic nonionic contrast medium for radiophotograph
08/29/1995US5446205 Functionalized fluoropolyethers
08/29/1995US5446170 Process for the manufacture of insecticidal arylpyrroles via oxazole amine intermediates
08/29/1995US5446166 Reacting isocyanoacetate with prophosphatrane and acyl halide or acid anhydride
08/29/1995US5446158 Process for synthesis of FK-506 and tricarbonyl intermediates
08/29/1995US5445934 Selective photoremovable groups on surface
08/24/1995WO1995022546A1 Intracellular signalling mediators
08/24/1995WO1995022533A1 Process for producing 3-isoxazolecarboxylic acid
08/24/1995WO1995022523A1 Cyclic nitrogenous compound and herbicide
08/24/1995WO1995022326A1 Cholinesterase activator
08/24/1995WO1995021154A3 Phenyl acetic acid derivatives, process and intermediate products for their production and agents containing them
08/24/1995CA2183562A1 Intracellular signalling mediators
08/24/1995CA2183426A1 Process for producing 3-isoxazolecarboxylic acid
08/24/1995CA2182882A1 Cholinesterase activator
08/23/1995CN1107277A Novel compound with platelet aggregation inhibitor activity
08/23/1995CN1107148A Method for the preparation of 2-perflouoroalkyl-3-oxazolin-5-one
08/22/1995US5444079 Arthropodicidal oxazolines
08/22/1995US5444075 Penetration enhancers for transdermal delivery of systemic agents
08/22/1995US5443986 Enzymatic analysis using substrates that yield fluorescent precipitates
08/22/1995US5443948 Reacting silver nitrate with alkali metal halide or ammonium halide to form silver halide, purification of grains by ultrafiltration in combination with spectral sensitization
08/17/1995WO1995021837A1 Potassium salt of biphenylmethane derivative and medicine containing the same
08/17/1995WO1995021833A1 Substituted oxazacycloalkenes, intermediate products and use as fungicides
08/17/1995DE4404373A1 Substituierte Oxazacycloalkene Substituted Oxazacycloalkene
08/17/1995CA2181260A1 Potassium salt of biphenylmethane derivative and medicine containing the same
08/16/1995EP0666857A1 Method for preparing taxane derivatives
08/16/1995CN1106806A Adhesion receptor antagonists
08/16/1995CN1106803A Fungicidal optically active 2-imidazolin-5-one and 2-imidazoline-5-thione derivatives
08/15/1995US5441975 Anticholesterol agent
08/10/1995WO1995021154A2 Phenyl acetic acid derivatives, process and intermediate products for their production and agents containing them
08/10/1995WO1995021153A1 Phenyl acetic acid derivatives, process and intermediate products for their production and agents containing them
08/10/1995CA2182529A1 Phenylacetic acid derivatives, preparation thereof and intermediates therefor, and compositions containing them
08/10/1995CA2182407A1 Phenylacetic acid derivatives, preparation thereof and intermediates therefor, and compositions containing them
08/09/1995EP0666254A1 2-Aroylcydohexanediones, process for their preparation and their use as herbicide or as plant growth regulating agent
08/09/1995EP0425650B1 Anti-inflammatory 4-aminophenol derivatives
08/08/1995US5439932 Substituted amine derivatives having anti-hyperlipemia activity
08/08/1995US5439927 For potassium channel opening, hypotensive agents, broncho- or vasodilators, gastrointestinal disorders
08/08/1995US5439908 Diazinyl butyric acid amides and esters
08/08/1995CA2141763A1 2-aroylcyclohexanediones, their preparation and their use as herbicides or plant growth-regulating agents
08/08/1995CA1336597C Azacycloalkane derivatives, absorption promoters containing the derivatives as the effective ingredient and external preparations containing the absorption promoters
08/02/1995EP0664792A1 Fibrinogen receptor antagonists
08/02/1995EP0664791A1 Process for the preparation of oxime derivatives, certain intermediates and the use of the oxime derivatives as fungicides
08/02/1995CN1106008A 4-aryloxy-and 4-arylthiopiperidine derivatives
08/01/1995US5438148 Simultaneous addition of boron tribromide and solution of dimethyl ether of desired product in methylene chloride to methylene chloride while maintaining constant ratio
08/01/1995US5438074 3-aryl-2-hydroxypropionic acid derivatives and analogs as hypoglycemic agents