Patents
Patents for C07D 257 - Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms (9,612)
07/2005
07/13/2005EP1551799A1 Cyclohexyl sulphones as gamma-secretase inhibitors
07/13/2005EP1551797A1 Cyclohexyl sulphone derivatives as gamma-secretase inhibitors
07/13/2005CN1636597A Compounds for the treatment of female sexual dysfunction
07/13/2005CN1210268C (Cyclo) alkyl substituted-gamma-aminobutyric acid derivatives (=GABA analogurs), their preparation and their use in the treatment of neurolog disorders
07/13/2005CN1210263C N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
07/12/2005US6916848 Compounds for the treatment of metabolic disorders
07/12/2005US6916797 α-arylethylpiperazine derivatives as neurokinin antagonists
07/12/2005US6916461 Metal complexes that contain perfluoroalkyl, process for their production and their use in NMR diagnosis
07/12/2005CA2128378C Novel acaricidally active tetrazine derivatives
07/07/2005US20050148566 Polydiazeniumdiolated cyclic polyamines with polyphasic nitric oxide release and related compounds, compositions comprising same and methods of using same
07/07/2005US20050147563 Imaging lymph nodes with a Gadolinium complex of 10-[2-hydroxy-4-aza-5-oxo-7-aza-7-(perfluorooctylsulfonyl)-nonyl]-1,4,7-tris (carboxymethyl)-1,4,7,10-tetraazacyclododecane; in vivo contrast media in nuclear spin tomography; blood-pool agents, lymphographic agents
07/06/2005CN1209362C Tetrazolyl-phenyl acetamide glucokinase activators
06/2005
06/30/2005WO2005058884A2 Cyclopropane compounds and pharmaceutical use thereof
06/30/2005WO2005058808A1 N-substituted-n-sulfonylaminocyclopropane compounds and pharmaceutical use thereof
06/30/2005WO2005020899A3 Substituted cycloalkyamine derivatives as modulators of chemokine receptor activity
06/30/2005CA2549660A1 Cyclopropane compounds and pharmaceutical use thereof
06/30/2005CA2549598A1 N-substituted-n-sulfonylaminocyclopropane compounds and pharmaceutical use thereof
06/29/2005EP1546122A1 Process for the manufacture of valsartan
06/29/2005EP1545513A2 Compounds, compositions and methods for treating or preventing pneumovirus infection and associated diseases
06/29/2005EP1545498A2 Backbone-substituted bifunctional dota ligands, complexes and compositions thereof, and methods of using same
06/29/2005EP1480635A4 Macrocyclic module compositions
06/29/2005CN1208327C Process for preparing S, Síõ-carbonyl disulfhydryl substituted five-membered heterocyclic compound
06/28/2005US6911457 Diabetes imaging probes
06/28/2005US6911439 Alpha 4 beta 1 integrin and CD49d/ CD29 (vla-4); antiinflammatory agents
06/28/2005US6911416 Substituted N-benzoyl-n′(tetrazolylphenyl)-ureas and their use as pest control agents
06/23/2005WO2005056508A1 Method for the production of tetrahydrogeranylacetone
06/23/2005WO2005040121A3 Amides that inhibit vanilloid receptor subtype 1 (vr1) receptor
06/23/2005CA2548262A1 Method for the production of tetrahydrogeranylacetone
06/22/2005EP1542980A1 5-aryltetrazole compounds, compositions thereof, and uses therefor
06/22/2005EP1082127B1 Succinamide inhibitors of interleukin-1beta converting enzyme
06/22/2005CN1630633A N-biphenylmethyl aminocycloalkanecarboxamide derivatives with a substiituent on the methyl useful as bradykinin antagonists
06/21/2005US6908938 Heterocyclic aromatic compounds useful as growth hormone secretagogues
06/21/2005CA2247265C Process for preparing 1,4,7,10-tetraazacyclododecane and its derivatives
06/16/2005US20050131038 Process for the preparation of valsartan and intermediates thereof
06/16/2005US20050130949 Antiproliferative agents; ATP-ase activity; e.g. 5,9,14-Trimethyl-4-undecyl-1,5,9,14-tetraazacycloheptadecan-2-one; budmunchiamine compounds
06/16/2005US20050130941 Methods of treating alzheimer's disease
06/15/2005EP1539691A2 Compounds, compositions and methods for treating or preventing pneumovirus infection and associated diseases
06/15/2005EP1311504B1 Tetrazolyl-phenyl acetamide glucokinase activators
06/15/2005CN1628106A Salts of valsartan
06/14/2005US6905804 Charge transport material comprising a fluorenone hydrazone having a) least two fluorenone alkylsulfonylphenylhydrazone groups, b) at least two fluorenone pyrrolylhydrazone groups, c) at least two fluorenone benzotriazolylhydrazone groups, d)
06/14/2005CA2304967C 4(3)substituted-4(3)-aminomethyl-(thio)pyran or -piperidine derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
06/09/2005WO2005051930A1 Modified-protein formation inhibitor
06/09/2005WO2005051929A1 Conversion of aromatic nitriles into tetrazoles
06/09/2005WO2005051928A1 Process for production of tetrazolyl compounds
06/09/2005WO2005051893A2 Vitamin d receptor modulators
06/09/2005WO2005021535A3 A method of removing the triphenylmethane protecting group
06/09/2005US20050124671 Benzylcycloalkyl amines as modulators of chemokine receptor activity
06/09/2005US20050123849 Electrophotographic organophotoreceptors with novel charge transport materials
06/08/2005EP1537077A2 4-(3,3-dihalo-allyloxy) phenol derivatives having pesticidal properties
06/08/2005EP1537075A2 Diarylurea derivatives and their use as chloride channel blockers
06/08/2005EP1536784A1 Hetero biaryl derivatives as matrix metalloproteinase inhibitors
06/08/2005EP1465854A4 Chalcone derivatives and their use to treat diseases
06/08/2005EP1220831B1 Biaryl ether derivatives useful as monoamine reuptake inhibitors
06/07/2005US6903218 Substituted or unsubstituted aryl-1-hydroxyethylaminocarbonylalkyl-chroman-sulfonamide compounds are useful in the treatment of beta-3 receptor mediated conditions
06/07/2005US6903088 Compounds which inhibit leukocyte adhesion mediated by VLA-4
06/02/2005WO2005049588A1 Process for isolation of valsartan
06/02/2005WO2005049587A1 Process for preparation of biphenyl tetrazole
06/02/2005WO2005049586A1 Process for production of (s) -n-pentanoyl-n-[[2’-(1h-tetrazole-5yl) [1,1’-biphenyl]-4-yl]methyl]-l-valine
06/02/2005WO2005048810A2 Sigma-2 receptor radiotracers for imaging the proliferative status of solid tumors
06/02/2005US20050119488 Phenyltetrazole compounds
06/01/2005EP1535914A1 Processes for producing epoxytriazole derivative and intermediate therefor
06/01/2005EP1115695B1 (r)-chiral halogenated 1-substitutedamino-(n+1)-alkanols useful for inhibiting cholesteryl ester transfer protein activity
06/01/2005EP0991625B1 Inhibitors of factor xa with a neutral p1 specificity group
06/01/2005CN1203899C Compounds with chelation affinity and selectivity for first transition series elements, and their use in medical therapy
06/01/2005CN1203898C Perfluoroalkyl-containing metal complexes, its preparing method and use in NMR diagnostics
05/2005
05/31/2005US6900207 N-containing five-membered ring compounds and pharmaceutical agents comprising the same as active ingredient
05/31/2005CA2324343C C11 oxymyl and hydroxylamino prostaglandins useful as medicaments
05/26/2005WO2005047236A1 Sulfoxide and bis-sulfoxide compounds and compositions for cholesterol management and related uses
05/26/2005US20050113580 2-(3-{3-[[2-chloro-3-(trifluoromethyl)benzyl](2,2-dephenylethyl)amino]propoxy}phenyl)-ethanol; agonists of the nuclear receptors, LXR alpha and LXR beta used to increase ABCA1, ABCG1, and apolipoprotein E expression and inhibiting cholesterol absorption
05/26/2005CA2534342A1 Amino acid prodrugs
05/25/2005EP1533305A1 A process for the preparation of valsartan and intermediates thereof
05/25/2005EP1533292A1 Dibenzylamine compound and medicinal use thereof
05/25/2005EP1531879A1 Use of organic compounds
05/25/2005EP1531822A1 1-aryl-4-substituted piperazine derivatives for use as ccr1 antagonists for the treatment of inflammation and immune disorders
05/25/2005CN1203047C Biaryl ether derivatives useful as monoamine reuptake inhibitors
05/24/2005US6897237 MMP-12 inhibitors
05/19/2005US20050107421 Nitrogen compounds such as 2-Butyl-1-(2-methylpropyl)-1H-tetrazolo[1,5-a]imidazo[4,5-c][1,8]naphthyridine, used to induce biosynthesis of cytokines such as interferons and tumor necrosis factors, or for prophylaxis of viral diseases
05/19/2005US20050107398 benzamide compounds labeled with detectable radionuclides that selectively bind to cancer cells, used for medical diagnosis such as tomography
05/19/2005US20050107345 Aminoalkylphosphonates and related compounds as edg receptor agonists
05/19/2005DE10348023A1 Neue Alanyl-Aminopeptidasen-Inhibitoren zur funktionellen Beeinflussung unterschiedlicher Zellen und zur Behandlung immunologischer, entzündlicher, neuronaler und anderer Erkrankungen New alanyl aminopeptidase inhibitors for functional interference of different cells and for the treatment of immunological, inflammatory, neuronal and other diseases
05/18/2005CN1617852A Alpha-(n-sulphonamido)acetamide derivatives as beta-amyloid inhibitors
05/18/2005CN1617850A Dibenzylamine compound and medicinal use thereof
05/18/2005CN1616453A Antivirally active heterocyclic azahexane derivatives
05/17/2005US6894165 Imidazonaphthyridines
05/17/2005US6894151 Lithium complexes of N-(1-hydroxymethyl-2,3-dihydroxypropyl)-1,4,7-triscarboxymethyl-1,4,7,10-tetraazacyclododecane, their production and use
05/17/2005US6893650 Fungicides; locus infestation; such as N,N-dimethyl-N'-(4-(3-trifluoromethylbenzylthio)-2,5-xylyl)formamidine
05/12/2005WO2005041867A2 2-(3,4-dimethylphenyl)-4-{[2-hydroxy-3’(1h-tetrazol-5-yl)biphenyl-3-yl]-hydrazono}-5-methyl-2,4-dihydropyrozol-3-one choline
05/12/2005US20050101652 New salt hydrates
05/12/2005CA2543216A1 2-(3,4-dimethylphenyl)-4-{[2-hydroxy-3'(1h-tetrazol-5-yl)biphenyl-3-yl]-hydrazono}-5-methyl-2,4-dihydropyrozol-3-one choline
05/11/2005EP1528921A2 Methods for treatment and prevention of gastrointestinal conditions
05/11/2005CN1200933C Substituted N-benzoyl-N'-(tetrazolylphenyl)-ureas and their use as pest control agents
05/11/2005CN1200704C Appliance of probucol monoesters for treatment of cardiovascular and inflammatory disease
05/10/2005US6890956 Cyclohexyl sulphones as gamma-secretase inhibitors
05/06/2005WO2005040121A2 Amides that inhibit vanilloid receptor subtype 1 (vr1) receptor
05/06/2005CA2539967A1 Amides that inhibit vanilloid receptor subtype 1 (vr1) receptor
05/04/2005EP1528055A2 Sulphonamide Derivatives
05/04/2005EP1526851A2 Compounds useful for the treatment of diseases responsive to antiangiogenetic therapy
05/04/2005CN1612866A Amorphous and crystalline forms of losartan potassium and process for their preparation
05/03/2005US6887877 Viricide for hepatitis virus
05/03/2005CA2149886C Process for preparing tetrazolyl-benzopyranones
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