Patents
Patents for C07D 255 - Heterocyclic compounds containing rings having three nitrogen atoms as the only ring hetero atoms, not provided for by groups (739)
01/2012
01/12/2012WO2012003599A1 Methods for the synthesis of bis (triazacyclononane) ligands
01/12/2012WO2012003598A1 Intermediates for the synthesis of 1,2-bis(4,7-dimethyl-1,4,7-triazacyclonon-1-yl)-ethane and preparation method thereof
01/12/2012WO2011111971A3 Method for preparing (r)-3-(3-fluoro-4-(1-methyl-5,6-dihydro-1,2,4-triazin-4(1h)-yl)phenyl)-5-(substituted methyl)oxazolidin-2-one derivatives
01/12/2012US20120010200 Biaryl Heterocyclic Compounds And Methods Of Making And Using The Same
01/12/2012CA2804475A1 1,2-bis-(4,7-dimethyl-1,4,7-triazacyclonon-1-yl)-ethane and intermediate thereof
01/10/2012US8092782 Polybiotin compounds of magnetic resonance imaging and drug delivery
12/2011
12/14/2011CN102282158A 氮杂*酮衍生物 * Aza derivatives
10/2011
10/18/2011US8039642 Pyrenyloxysulfonic acid fluorescent agents
10/12/2011CN101389613B Macrocyclic factor viia inhibitors useful as anticoagulants
09/2011
09/22/2011WO2011115802A1 Conjugates of 1,4,7-triaza-cyclononanes, dinuclear metal complexes of such conjugates, and methods of use for both 1,4,7-triaza-cyclononanes and conjugates
09/22/2011CA2793179A1 Conjugates of 1,4,7-triaza-cyclononanes, dinuclear metal complexes of such conjugates, and methods of use for both 1,4,7-triaza-cyclononanes and conjugates
09/15/2011WO2011111971A2 Method for preparing (r)-3-(3-fluoro-4-(1-methyl-5,6-dihydro-1,2,4-triazin-4(1h)-yl)phenyl)-5-(substituted methyl)oxazolidin-2-one derivatives
09/13/2011US8017768 Catalitic synthesis of caged polynitramine compounds
08/2011
08/25/2011WO2011100838A1 Derivatives of 1-phenyl-1,5-dihydro-benzo[b] [1.4]diazepine-2.4-dione as inhibitors of hiv replication
08/24/2011EP2358735A1 Azepinone derivatives
07/2011
07/21/2011US20110177002 Cylic polyamines for binding phosphatidylserine
07/13/2011EP2343285A2 Peptoid compounds
05/2011
05/04/2011CN102040562A Macrocyclic aromatic-amine structured compound as well as preparation method and application thereof
04/2011
04/20/2011CN101314595B Aromatic hydrocarbons connected multi-polyamine large-ring derivants, preparation method and medical use thereof
04/19/2011US7928096 Polydiazeniumdiolated cyclic polyamines with polyphasic nitric oxide release and related compounds, compositions comprising same and methods of using same
02/2011
02/16/2011CN101977901A Linear and cyclic guanidine derivatives, method of preparation and uses thereof
02/15/2011USRE42152 FDA Orange book listed patent for plerixafor
02/15/2011CA2325937C Peptide turn mimetics
02/03/2011US20110028713 Aza compounds and production method thereof, and metal complexes as mri contrast agents
01/2011
01/25/2011US7875714 Processes for preparing certain hexaazaisowurtzitanes and their use in preparing hexanitrohexaazaisowurtzitane
01/19/2011EP2274290A2 Linear and cyclic guanidine derivatives, method of preparation and uses thereof
01/05/2011EP2269995A1 Process for production of polymers with iron complex catalyst
01/04/2011US7863440 From condensation of a urethane or urea substituted polyether, polyester, poly(ester-ether), polycarbonate, poly(carbonate-ether), polyolefin or poly(olefin-ether) endcapped with diisocyanate groups
12/2010
12/23/2010US20100322855 Bimodal ligands with macrocyclic and acyclic binding moieties, complexes and compositions thereof, and methods of using
11/2010
11/04/2010US20100278739 Targeted, nir imaging agents for therapy efficacy monitoring, deep tissue disease demarcation and deep tissue imaging
10/2010
10/07/2010WO2010114308A1 Heterocycle-amino acid derivatives for targeting cancer tissue and radioactive or non-radioactive labeled compounds thereof
10/07/2010US20100256355 Oxazolidinone derivative having 7-membered hetero ring
09/2010
09/30/2010US20100247448 Novel lanthanide ligands and complexes, and use thereof as contrast agents
09/28/2010US7803359 UV-absorbers for ophthalmic lens materials
09/16/2010WO2010103204A1 Metal ion chelating agents, methods for preparing same and uses thereof
09/16/2010US20100234591 Biaryl heterocyclic compounds and methods of making and using the same
09/13/2010CA2658076A1 Metallic ion chelating agents, method for producing them and use of same
08/2010
08/17/2010US7777029 Protecting an amino acid compound amino group with an amino protecting group and the carboxyl with a carboxyl protecting group; reacting with cyclen; reacting the monoalkylated cyclone with an activated compound, then deprotecting
08/11/2010CN101801939A 3-substituted 1,2,3-triazin-4-one's and 3-substituted 1,3-pyrimidinone's for enhancing glutamatergic synaptic responses
08/10/2010CA2451768C Peptoid compounds
07/2010
07/27/2010US7763616 Chemokine receptor antagonists, used for the treatment of inflammatory diseases, autoimmune diseases, transplant rejection, infectious diseases, hypersensitivity responses, ophthalmic inflammation, diabetes, viral meningitis and tumors
07/01/2010US20100167995 Peptoid compounds
06/2010
06/23/2010CN101747286A Nano-aperture 30-element triphenylamine rigid macrocyclic compound and preparation method thereof
06/17/2010WO2010066051A1 Thiol-nota derivatives for kit 68ga radiolabeling
06/16/2010EP2195303A2 3-substituted 1,2,3-triazin-4-one's and 3-substituted 1,3-pyrimidinone's for enhancing glutamatergic synaptic responses
06/15/2010US7737272 Diazaphosphacycle transition metal complexes
05/2010
05/20/2010WO2010056496A1 Azepinone derivatives
05/20/2010WO2010055207A1 Chelating, chelating agents and conjugates deriver thereof
05/20/2010CA2743145A1 Azepinone derivatives
05/11/2010CA2318696C Triazepinones, process for their preparation and their therapeutic application
05/06/2010US20100111875 Trisubstituted triazamacrocyclic compounds and their use as contrast agents
04/2010
04/27/2010US7705026 Biaryl heterocyclic compounds and methods of making and using the same
03/2010
03/25/2010WO2010011367A3 Bimodal ligands with macrocyclic and acyclic binding moieties, complexes and compositions thereof, and methods of using
02/2010
02/24/2010CN101657434A Process for production of polymers with iron complex catalyst
02/18/2010US20100041880 Supramolecular Scaffolds and Methods of Making the Same
01/2010
01/28/2010US20100022500 Macrocyclic Lactams and Pharmaceutical Use Thereof
12/2009
12/30/2009WO2009113033A3 Linear and cyclic guanidine derivatives, method of preparation and uses thereof
12/23/2009CN101611019A Macrocyclic factor VIIa inhibitors useful as anticoagulants
12/09/2009EP2129664A1 Trisubstituted triazamacrocycli c compounds and their use as contrast agents
12/09/2009CN100567271C Improved purification of 4,4'(5')-di-t-butylcyclohexano-18-crown-6
11/2009
11/03/2009US7612055 Macrocyclic lactams and pharmaceutical use thereof
11/03/2009US7612036 Such as methyl (2S,5S,8R/S)-8-acetamido-2-allyl-9-[6-allyl-9-tert-butoxycarbonyl-9H-carbazol-3-yl]-3,6-diaza-5-{3-[(2,2,5,7,8-pentamethylchroman-6-sulfonyl)-guanidino]propyl}-4,7-dioxononanoate; for treatment of bacterial infections, such as those caused by vancomycin resistant microorganisms
10/2009
10/28/2009EP2111396A1 Hcv inhibiting macrocyclic phenylcarbamates
10/01/2009US20090246130 Methods and Compositions for F-18 Labeling of Proteins, Peptides and Other Molecules
09/2009
09/24/2009WO2009115644A1 Lanthanide(iii) chelates comprising beta-diketones and conjugates derived thereof
09/23/2009EP2102176A2 Macrocyclic factor viia inhibitors useful as anticoagulants
09/17/2009WO2009113148A1 Process for production of polymers with iron complex catalyst
09/17/2009WO2009113033A2 Linear and cyclic guanidine derivatives, method of preparation and uses thereof
09/01/2009US7582753 Reacting [5-cyclohexyl-1-(2-cyclopentyl-2-oxo-ethyl)-2-oxo-1,2-dihydro-benzo[e][1,2,4]triazepin-3-yl]-acetic acid with thionyl chloride in situ, in acetonitrile; for production of gastrin and cholecystokinin receptor ligands
09/01/2009US7582280 Conjugates of antioxidants with metal chelating ligands for use in diagnostic and therapeutic applications
07/2009
07/23/2009WO2008096001A8 Hcv inhibiting macrocyclic phenylcarbamates
07/15/2009EP2006283A9 Process for production of amides or lactams
07/14/2009US7560592 N-halo-4-carboxybenzene sulfonamides; soap, lotion, wipe, or swab; minimal side effects; bactericide, pesticide, fungicide, deodorizing; also bovine teat cleaners, drugs for cultured fish, soap biocides, stain removal agents, and paint fungicides
07/09/2009WO2009038752A3 3-substituted 1,2,3-triazin-4-one's and 3-substituted 1,3-pyrimidinone's for enhancing glutamatergic synaptic responses
06/2009
06/18/2009US20090156801 Biomolecule labeling reactants based on azacycloalkanes and conjugates derived thereof
06/09/2009US7544828 oxidizing N-[4-cyano-3-(trifluoromethyl) phenyl]-3-[(4-fluorophenyl) thio]-2-hydroxy-2-methyl propanamide with potassium permanganate in water and water miscible solvent such as acetonitrile, acetone, acetic acid etc. crystallizing bicalutamide from a mixture of ethyl acetate and petroleum ether
06/04/2009WO2009069833A1 Aza compounds and production method thereof, and metal complexes as mri contrast agents.
05/2009
05/19/2009CA2336634C Antiviral macrocyclic compounds
05/07/2009US20090118502 organic or inorganic salt of N-{3-[4'-(4-Aminomethyl-[1,2,3]triazol-1-ylmethyl)-2-fluoro-biphenyl- 4-yl]-2-oxo-oxazolidin-5-(S)-ylmethyl}-acetamide; anti-infective, anti-proliferative, anti-inflammatory, and prokinetic agents
04/2009
04/28/2009US7524837 Benzotriazapinone salts and methods for using same
04/08/2009CN101405276A Compositions and methods for the inhibition of phospholipase A2
03/2009
03/26/2009WO2009038752A2 3-substituted 1,2,3-triazin-4-one's and 3-substituted 1,3-pyrimidinone's for enhancing glutamatergic synaptic responses
03/26/2009CA2700158A1 3-substituted 1,2,3-triazin-4-one's and 3-substituted 1,3-pyrimidinone's for enhancing glutamatergic synaptic responses
03/25/2009CN101395143A Aza heterocyclics for the treatment of malaria or aids
03/24/2009CA2342616C Method of treating a textile
03/18/2009CN101389613A Macrocyclic factor viia inhibitors useful as anticoagulants
03/18/2009CN101389599A Modified amino acids
03/12/2009WO2008079836A4 Macrocyclic factor viia inhibitors useful as anticoagulants
03/12/2009US20090068248 Polydiazeniumdiolated cyclic polyamines with polyphasic nitric oxide release and related compounds, compositions comprising same and methods of using same
03/05/2009US20090062311 Macrocylic inhibitors of hepatitis c virus
03/04/2009EP1064300B1 Peptide turn mimetics
03/03/2009US7498432 Method of synthesis of 1, 4, 7, 10, 13, 16, 21, 24-octaazabicyclo [8.8.8] hexacosane (1) and 1, 4, 7, 10, 13, 16, 21, 24-octaazabicyclo [8.8.8] hexacosa, 4, 6, 13, 15, 21, 23-hexaene (2)
02/2009
02/19/2009US20090048222 Triaza Compound Immunoregulatory Agents
02/12/2009US20090042764 Cleaning Agent Comprising Complexes with Bleach Catalytic Activity
02/11/2009EP2022787A1 Process for the preparation of N-1 protected N ring nitrogen containing cyclic polyamines and products thereof
02/11/2009CN101365336A Methods to enhance chemotherapy
01/2009
01/29/2009WO2009014730A1 Macrocyclic serine protease inhibitors
01/21/2009EP2016060A1 Biomolecule labeling reactants based on azacycloalkanes and conjugates derived thereof
01/15/2009WO2008079836A3 Macrocyclic factor viia inhibitors useful as anticoagulants
12/2008
12/24/2008EP2006283A2 Process for production of amides or lactams
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