Patents for C07D 249 - Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms (17,749) |
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01/13/2005 | US20050009900 3-Substituted with a heterocyclic group, e.g., 2-Chloro-5-[1-(2,3-dihydroxy-propyl)-5-methyl-1H-pyrazol-3-yl]-N-(1-hydroxy-cycloheptylmethyl)-benzamide; treatment of IL-1 mediated disorders, including osteo- and rheumatoid arthritis, allergies, asthma, COPD, cancer, and reperfusion or ischemia in stroke |
01/13/2005 | US20050009834 E.g., 3-(2-chloro-6-fluorophenyl)-1-[4-(3,5-dichloropyridin-2-yloxymethyl)phenyl]-5-methyl-1H-1,2,4-triazole and 3-(3-chloropyridin-2-yl)-1-[4-(3-chloro-5-trifluoromethylpyridin-2-yloxymethyl)phenyl]-5-methyl-1H-1,2,4-triazole; for use as pesticides, especially insecticides and acaricides |
01/13/2005 | US20050009704 Substituted aryl ketones |
01/12/2005 | EP1495756A1 Severe sepsis preventive therapeutic agent |
01/12/2005 | EP1495035A1 Method for the production of bis(perfluoroalkyl)phosphinic acids and the salts thereof |
01/12/2005 | EP1495015A1 3-aminophenol derivatives and dyes that contain these compounds while serving to dye keratin fibers |
01/12/2005 | EP1180107A4 Novel ruthenium metal alkylidene complexes coordinated with triazolylidene ligands that exhibit high olefin metathesis activity |
01/12/2005 | CN1184210C Methods of inhibiting corrosion using isomers of chloro-methylbenzotrazole |
01/12/2005 | CN1184196C Substituted benzoylguanidines, method for their production, their use as medicament or diagnostic agent and mediciment containing same |
01/06/2005 | WO2005000841A1 Preparation of n2-alkylated 1,2,3-triazoles |
01/06/2005 | WO2005000821A1 Tachykinin receptor antagonists |
01/06/2005 | WO2005000309A2 Chemical compounds |
01/06/2005 | WO2005000298A2 5-membered heterocycle-based p-38 inhibitors |
01/06/2005 | US20050004204 2-Iminopyrrolidine derivatives |
01/06/2005 | US20050004197 Thrombin receptors antagonists; oral efficacy |
01/06/2005 | US20050004186 Phenyl-(2-[1,3,4]thiadiazol-2-yl-phenyl)-amine and (2-[1,3,4]Oxadiazol-2-yl-phenyl)phenyl-amine derivatives; immunomodulators; inflammation, proliferative diseases |
01/06/2005 | US20050004116 Triazole inhibitors of type 2 methionine aminopeptidase |
01/06/2005 | US20050004115 such as 4-(4-(2-Fluorobenzyloxy)phenyl)-4-oxobutyric acid; for treatment of insulin resistance syndrome, diabetes, hyperlipidemia, fatty liver disease, cachexia, obesity, atherosclerosis and arteriosclerosis |
01/06/2005 | CA2529109A1 Preparation of n2-alkylated 1,2,3-triazoles |
01/06/2005 | CA2528438A1 P-38 inhibitors |
01/05/2005 | EP1493733A2 Fungicidal heterocyclic aromatic amides, their compositions and methods of use |
01/05/2005 | CN1561393A Inhibitors of glycogen synthase kinase-3 (GSK-3) for treating glaucoma |
01/05/2005 | CN1183134C Tricyclic vasporessin agonists |
01/04/2005 | US6838466 Compounds for the treatment of inflammatory disorders |
01/04/2005 | US6838415 Substituted benzoylisoxazoles and the use thereof as herbicides |
12/30/2004 | US20040267025 Compounds for the treatment of metabolic disorders |
12/30/2004 | US20040267024 Nitrogen compounds, formed by condensing carbocyclic, hydroxy ethers such as 3-(2',4'-difluorophenyl)-3,4-epoxy-2-butanol, with 1,2,4-triazole in the presence of bases; fungicides |
12/30/2004 | US20040267012 5'-Carbamoyl-1,1-biphenyl-4-carboxamide derivatives and their use as p38 kinase inhibitors |
12/30/2004 | US20040266848 Preparation of N2-alkylated 1,2,3-triazoles |
12/30/2004 | US20040266831 Modulators of the glucocorticoid receptor and method |
12/30/2004 | US20040266738 Fungicidal phenoxyphenylhydrazine derivatives |
12/29/2004 | WO2004113394A2 Living radical polymerization initiator comprising a functional group capable of reacting with polypeptides or the like, comb polymer obtained therewith, polypeptide conjugates and drugs obtained therefrom |
12/29/2004 | WO2004113331A1 Novel compounds that modulate pparϝ type receptors, and use thereof in cosmetic or pharmaceutical compositions |
12/29/2004 | EP1490370A2 Triazolopyrimidines |
12/29/2004 | EP1056729B1 N-[(substituted five-membered di- or triaza diunsaturated ring)carbonyl]guanidine derivatives for the treatment of ischemia |
12/29/2004 | EP0986545B1 Non-steroidal (hetero) cyclically substituted acylanilides with mixed gestagen and androgen activity |
12/29/2004 | CN1558762A Novel ligands for the HisB10 Zn2+ sites of the R-state insulin hexamer |
12/29/2004 | CN1557808A 3-substituted piperazine triadimenol antifungal compounds and their salts |
12/29/2004 | CN1182116C Mutilin derivatives and their use as antibacterials |
12/29/2004 | CA2529154A1 Novel compounds that modulate ppar.gamma. type receptors, and use thereof in cosmetic or pharmaceutical compositions |
12/28/2004 | US6835495 Pentacyclic anion salts or tetrazapentalene derivatives and their uses as ionic conducting materials |
12/23/2004 | WO2004111015A1 Modulators of the glucocorticoid receptor and method |
12/23/2004 | WO2004110986A1 Benzamide derivative or salt thereof |
12/23/2004 | WO2004032875A3 Process for the preparation of tri-nitrogen containing heteroaryl-diamine derivatives useful as pharmaceutical agents and methods of producing pharmaceutical agents |
12/23/2004 | US20040259804 (Substituted)Acyl dipeptidyl inhibitors of the ICE/ced-3 family of cysteine proteases |
12/23/2004 | US20040259031 Specific dye compound, optical information recording medium comprising specific dye, and information recording method using this optical information recording medium |
12/23/2004 | CA2526387A1 Benzamide derivative or salt thereof |
12/22/2004 | EP1487843A2 Substituted phenylacetic acids |
12/22/2004 | EP1487785A2 Novel florfenicol-type antibiotics |
12/22/2004 | CN1181063C Beta-element-5-azacycle derivatives and its synthetic method |
12/21/2004 | CA2241904C Substituted n-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides |
12/16/2004 | WO2004108684A1 Novel azole derivative having antifungal activity |
12/16/2004 | WO2003105538A8 Electroluminescent device |
12/16/2004 | WO2003063797A8 Cycloalkyl inhibitors of potassium channel function |
12/16/2004 | US20040254382 Imidazolyl derivatives as corticotropin releasing factor inhibitors |
12/16/2004 | US20040254376 Cyclic amidine derivative |
12/16/2004 | US20040254236 Antiinflammatory agents; moderate cytokine activity; bone disorders autoimmune disease; neurodegenerative diseases; viricides; asthma; antiallergens; adult respiratory distress syndrome; antiarthritic agents; antidiabetic agents |
12/16/2004 | US20040254227 prevent reproduction of herpes c virus; viricides; antiproliferative agents; prevention infections |
12/16/2004 | US20040254182 Enhanced propertied pharmaceuticals |
12/15/2004 | EP1486489A2 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation |
12/15/2004 | EP1485370A1 Amino-derivatives as novel inhibitors of histone deacetylase |
12/15/2004 | EP1485364A1 Aminocarbonyl-derivatives as novel inhibitors of histone deacetylase |
12/15/2004 | EP1485353A1 New inhibitors of histone deacetylase |
12/15/2004 | EP1485099A1 Inhibitors of histone deacetylase |
12/15/2004 | EP1485088A1 Opioid receptor active 4-(3-hydroxyphenyl) or 4-(3-alkoxyphenyl)-1,2,4-triazole compounds |
12/15/2004 | EP1337520B1 Substituted 5-aryl and 5-heteroaryl-2-(2-hydroxyphenyl)-2h-benzotriazole derivatives as uv absorbers |
12/15/2004 | CN1555361A Butyric acid derivatives |
12/15/2004 | CN1179953C Method for producing sulfonyl-amino-carbnyl triazolinone salt |
12/14/2004 | US6831199 Pyrimidine compounds and derivatives thereof |
12/14/2004 | US6831177 Preparation of their intermediates, 2-acyl-5-benzylfuran derivatives and 1,2,4-triazole-3- carboxylic acid ester derivatives |
12/14/2004 | US6831147 UV-stable polycarbonates optionally mixed with known aromatic polycarbonates, production thereof and use thereof |
12/09/2004 | WO2004106324A1 Azolecarboxamide herbicides |
12/09/2004 | WO2004106294A2 Triazole derivatives as inhibitors of 11-beta hydroxysteroid dehydrogenase-1 |
12/09/2004 | WO2004106285A1 Benzamide nitrile derivatives |
12/09/2004 | WO2004061084A8 Modulation of protein functionalities |
12/09/2004 | US20040249185 Process for the arylation of aza-heterocycles with activated aromatics in presence of caesium carbonate |
12/09/2004 | US20040248949 carbocyclic carboxy nitriles such as 4-chloro-N-[2-({[(1S)-1-cyano-2-thien-3-ylethyl]amino}carbonyl)cyclohexyl]benzamide, used as cathepsin inhibitors; antimetastatic and antitumor agents; prophylaxis of cardiovascular and bone disorders |
12/09/2004 | US20040248872 Safe for agricultural or gardening use; effective against insects and mammals |
12/09/2004 | US20040248857 treatment of gram positive, gram negative and antibiotic resistant infections; 1,11-dioxo-2-naphthacenecarboxamide derivatives |
12/09/2004 | US20040248740 for controlling undesirable plants |
12/09/2004 | CA2527632A1 Benzamide nitrile derivatives |
12/09/2004 | CA2526712A1 Triazole derivatives as inhibitors of 11-beta hydroxysteroid dehydrogenase-1 |
12/08/2004 | EP1483228A1 Nk1 antagonists |
12/08/2004 | EP1482940A2 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade |
12/08/2004 | EP1482904A1 Uv absorber compositions comprising a hydroxyphenyltriazine compound |
12/08/2004 | EP1482896A2 Aminoalkylphosphonates and related compounds as edg receptor agonists |
12/08/2004 | EP1482895A2 Aminoalkylphosphonates and related compounds as edg receptor agonists |
12/08/2004 | CN1178924C Method for producing triazolinthion derivatives |
12/08/2004 | CN1178665C Water soluble prodrugs of azole compounds |
12/02/2004 | WO2004103366A1 Heterocyclic compounds useful to treat hcv |
12/02/2004 | WO2004058174A3 Indane acetic acid derivatives and their use as pharmaceutical agents, intermediates, and method of preparation |
12/02/2004 | US20040242890 Agonists of beta-adrenoceptors |
12/02/2004 | US20040242733 Low dusting crystal transformations of 2,2'-methylenbis[4-(1,1,3,3-tetramethylbutyl)-6-benzotriazolylphenol] and mixture thereof, method for preparing them, and ultraviolet absorbent using the same |
12/02/2004 | US20040242692 4-(3-(2,6-Dimethoxybenzyloxy)phenyl)-4-oxobutyric acid or derivatives for treatment of insulin resistance syndrome, diabetes, cachexia, hyperlipidemia, fatty liver disease, obesity, atherosclerosis or arteriosclerosis |
12/02/2004 | US20040242627 2-Iminoimidazole derivatives (1) |
12/02/2004 | US20040242572 New carboxamide compounds having melanin concentrating hormone antagonistic activity, pharmaceutical preparations comprising these compounds and process for their manufacture |
12/02/2004 | DE10320326A1 New 1-benzoyl-3-(heterocyclyl-phenyl)-urea derivatives, are glycogen phosphorylase a inhibitors useful e.g. for treating type II diabetes, dyslipidemia or arteriosclerosis |
12/01/2004 | EP1257542B1 Method for producing 2-(1,2,4-triazol-1-yl)-ethanols |
12/01/2004 | EP1181280B1 Substituted benzoyl ketones, methods for producing them and their use as herbicides |
12/01/2004 | EP0977745B1 Thioaryl sulfonamide hydroxamic acid compounds |