Patents
Patents for C07D 249 - Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms (17,749)
01/2005
01/13/2005US20050009900 3-Substituted with a heterocyclic group, e.g., 2-Chloro-5-[1-(2,3-dihydroxy-propyl)-5-methyl-1H-pyrazol-3-yl]-N-(1-hydroxy-cycloheptylmethyl)-benzamide; treatment of IL-1 mediated disorders, including osteo- and rheumatoid arthritis, allergies, asthma, COPD, cancer, and reperfusion or ischemia in stroke
01/13/2005US20050009834 E.g., 3-(2-chloro-6-fluorophenyl)-1-[4-(3,5-dichloropyridin-2-yloxymethyl)phenyl]-5-methyl-1H-1,2,4-triazole and 3-(3-chloropyridin-2-yl)-1-[4-(3-chloro-5-trifluoromethylpyridin-2-yloxymethyl)phenyl]-5-methyl-1H-1,2,4-triazole; for use as pesticides, especially insecticides and acaricides
01/13/2005US20050009704 Substituted aryl ketones
01/12/2005EP1495756A1 Severe sepsis preventive therapeutic agent
01/12/2005EP1495035A1 Method for the production of bis(perfluoroalkyl)phosphinic acids and the salts thereof
01/12/2005EP1495015A1 3-aminophenol derivatives and dyes that contain these compounds while serving to dye keratin fibers
01/12/2005EP1180107A4 Novel ruthenium metal alkylidene complexes coordinated with triazolylidene ligands that exhibit high olefin metathesis activity
01/12/2005CN1184210C Methods of inhibiting corrosion using isomers of chloro-methylbenzotrazole
01/12/2005CN1184196C Substituted benzoylguanidines, method for their production, their use as medicament or diagnostic agent and mediciment containing same
01/06/2005WO2005000841A1 Preparation of n2-alkylated 1,2,3-triazoles
01/06/2005WO2005000821A1 Tachykinin receptor antagonists
01/06/2005WO2005000309A2 Chemical compounds
01/06/2005WO2005000298A2 5-membered heterocycle-based p-38 inhibitors
01/06/2005US20050004204 2-Iminopyrrolidine derivatives
01/06/2005US20050004197 Thrombin receptors antagonists; oral efficacy
01/06/2005US20050004186 Phenyl-(2-[1,3,4]thiadiazol-2-yl-phenyl)-amine and (2-[1,3,4]Oxadiazol-2-yl-phenyl)phenyl-amine derivatives; immunomodulators; inflammation, proliferative diseases
01/06/2005US20050004116 Triazole inhibitors of type 2 methionine aminopeptidase
01/06/2005US20050004115 such as 4-(4-(2-Fluorobenzyloxy)phenyl)-4-oxobutyric acid; for treatment of insulin resistance syndrome, diabetes, hyperlipidemia, fatty liver disease, cachexia, obesity, atherosclerosis and arteriosclerosis
01/06/2005CA2529109A1 Preparation of n2-alkylated 1,2,3-triazoles
01/06/2005CA2528438A1 P-38 inhibitors
01/05/2005EP1493733A2 Fungicidal heterocyclic aromatic amides, their compositions and methods of use
01/05/2005CN1561393A Inhibitors of glycogen synthase kinase-3 (GSK-3) for treating glaucoma
01/05/2005CN1183134C Tricyclic vasporessin agonists
01/04/2005US6838466 Compounds for the treatment of inflammatory disorders
01/04/2005US6838415 Substituted benzoylisoxazoles and the use thereof as herbicides
12/2004
12/30/2004US20040267025 Compounds for the treatment of metabolic disorders
12/30/2004US20040267024 Nitrogen compounds, formed by condensing carbocyclic, hydroxy ethers such as 3-(2',4'-difluorophenyl)-3,4-epoxy-2-butanol, with 1,2,4-triazole in the presence of bases; fungicides
12/30/2004US20040267012 5'-Carbamoyl-1,1-biphenyl-4-carboxamide derivatives and their use as p38 kinase inhibitors
12/30/2004US20040266848 Preparation of N2-alkylated 1,2,3-triazoles
12/30/2004US20040266831 Modulators of the glucocorticoid receptor and method
12/30/2004US20040266738 Fungicidal phenoxyphenylhydrazine derivatives
12/29/2004WO2004113394A2 Living radical polymerization initiator comprising a functional group capable of reacting with polypeptides or the like, comb polymer obtained therewith, polypeptide conjugates and drugs obtained therefrom
12/29/2004WO2004113331A1 Novel compounds that modulate pparϝ type receptors, and use thereof in cosmetic or pharmaceutical compositions
12/29/2004EP1490370A2 Triazolopyrimidines
12/29/2004EP1056729B1 N-[(substituted five-membered di- or triaza diunsaturated ring)carbonyl]guanidine derivatives for the treatment of ischemia
12/29/2004EP0986545B1 Non-steroidal (hetero) cyclically substituted acylanilides with mixed gestagen and androgen activity
12/29/2004CN1558762A Novel ligands for the HisB10 Zn2+ sites of the R-state insulin hexamer
12/29/2004CN1557808A 3-substituted piperazine triadimenol antifungal compounds and their salts
12/29/2004CN1182116C Mutilin derivatives and their use as antibacterials
12/29/2004CA2529154A1 Novel compounds that modulate ppar.gamma. type receptors, and use thereof in cosmetic or pharmaceutical compositions
12/28/2004US6835495 Pentacyclic anion salts or tetrazapentalene derivatives and their uses as ionic conducting materials
12/23/2004WO2004111015A1 Modulators of the glucocorticoid receptor and method
12/23/2004WO2004110986A1 Benzamide derivative or salt thereof
12/23/2004WO2004032875A3 Process for the preparation of tri-nitrogen containing heteroaryl-diamine derivatives useful as pharmaceutical agents and methods of producing pharmaceutical agents
12/23/2004US20040259804 (Substituted)Acyl dipeptidyl inhibitors of the ICE/ced-3 family of cysteine proteases
12/23/2004US20040259031 Specific dye compound, optical information recording medium comprising specific dye, and information recording method using this optical information recording medium
12/23/2004CA2526387A1 Benzamide derivative or salt thereof
12/22/2004EP1487843A2 Substituted phenylacetic acids
12/22/2004EP1487785A2 Novel florfenicol-type antibiotics
12/22/2004CN1181063C Beta-element-5-azacycle derivatives and its synthetic method
12/21/2004CA2241904C Substituted n-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides
12/16/2004WO2004108684A1 Novel azole derivative having antifungal activity
12/16/2004WO2003105538A8 Electroluminescent device
12/16/2004WO2003063797A8 Cycloalkyl inhibitors of potassium channel function
12/16/2004US20040254382 Imidazolyl derivatives as corticotropin releasing factor inhibitors
12/16/2004US20040254376 Cyclic amidine derivative
12/16/2004US20040254236 Antiinflammatory agents; moderate cytokine activity; bone disorders autoimmune disease; neurodegenerative diseases; viricides; asthma; antiallergens; adult respiratory distress syndrome; antiarthritic agents; antidiabetic agents
12/16/2004US20040254227 prevent reproduction of herpes c virus; viricides; antiproliferative agents; prevention infections
12/16/2004US20040254182 Enhanced propertied pharmaceuticals
12/15/2004EP1486489A2 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
12/15/2004EP1485370A1 Amino-derivatives as novel inhibitors of histone deacetylase
12/15/2004EP1485364A1 Aminocarbonyl-derivatives as novel inhibitors of histone deacetylase
12/15/2004EP1485353A1 New inhibitors of histone deacetylase
12/15/2004EP1485099A1 Inhibitors of histone deacetylase
12/15/2004EP1485088A1 Opioid receptor active 4-(3-hydroxyphenyl) or 4-(3-alkoxyphenyl)-1,2,4-triazole compounds
12/15/2004EP1337520B1 Substituted 5-aryl and 5-heteroaryl-2-(2-hydroxyphenyl)-2h-benzotriazole derivatives as uv absorbers
12/15/2004CN1555361A Butyric acid derivatives
12/15/2004CN1179953C Method for producing sulfonyl-amino-carbnyl triazolinone salt
12/14/2004US6831199 Pyrimidine compounds and derivatives thereof
12/14/2004US6831177 Preparation of their intermediates, 2-acyl-5-benzylfuran derivatives and 1,2,4-triazole-3- carboxylic acid ester derivatives
12/14/2004US6831147 UV-stable polycarbonates optionally mixed with known aromatic polycarbonates, production thereof and use thereof
12/09/2004WO2004106324A1 Azolecarboxamide herbicides
12/09/2004WO2004106294A2 Triazole derivatives as inhibitors of 11-beta hydroxysteroid dehydrogenase-1
12/09/2004WO2004106285A1 Benzamide nitrile derivatives
12/09/2004WO2004061084A8 Modulation of protein functionalities
12/09/2004US20040249185 Process for the arylation of aza-heterocycles with activated aromatics in presence of caesium carbonate
12/09/2004US20040248949 carbocyclic carboxy nitriles such as 4-chloro-N-[2-({[(1S)-1-cyano-2-thien-3-ylethyl]amino}carbonyl)cyclohexyl]benzamide, used as cathepsin inhibitors; antimetastatic and antitumor agents; prophylaxis of cardiovascular and bone disorders
12/09/2004US20040248872 Safe for agricultural or gardening use; effective against insects and mammals
12/09/2004US20040248857 treatment of gram positive, gram negative and antibiotic resistant infections; 1,11-dioxo-2-naphthacenecarboxamide derivatives
12/09/2004US20040248740 for controlling undesirable plants
12/09/2004CA2527632A1 Benzamide nitrile derivatives
12/09/2004CA2526712A1 Triazole derivatives as inhibitors of 11-beta hydroxysteroid dehydrogenase-1
12/08/2004EP1483228A1 Nk1 antagonists
12/08/2004EP1482940A2 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade
12/08/2004EP1482904A1 Uv absorber compositions comprising a hydroxyphenyltriazine compound
12/08/2004EP1482896A2 Aminoalkylphosphonates and related compounds as edg receptor agonists
12/08/2004EP1482895A2 Aminoalkylphosphonates and related compounds as edg receptor agonists
12/08/2004CN1178924C Method for producing triazolinthion derivatives
12/08/2004CN1178665C Water soluble prodrugs of azole compounds
12/02/2004WO2004103366A1 Heterocyclic compounds useful to treat hcv
12/02/2004WO2004058174A3 Indane acetic acid derivatives and their use as pharmaceutical agents, intermediates, and method of preparation
12/02/2004US20040242890 Agonists of beta-adrenoceptors
12/02/2004US20040242733 Low dusting crystal transformations of 2,2'-methylenbis[4-(1,1,3,3-tetramethylbutyl)-6-benzotriazolylphenol] and mixture thereof, method for preparing them, and ultraviolet absorbent using the same
12/02/2004US20040242692 4-(3-(2,6-Dimethoxybenzyloxy)phenyl)-4-oxobutyric acid or derivatives for treatment of insulin resistance syndrome, diabetes, cachexia, hyperlipidemia, fatty liver disease, obesity, atherosclerosis or arteriosclerosis
12/02/2004US20040242627 2-Iminoimidazole derivatives (1)
12/02/2004US20040242572 New carboxamide compounds having melanin concentrating hormone antagonistic activity, pharmaceutical preparations comprising these compounds and process for their manufacture
12/02/2004DE10320326A1 New 1-benzoyl-3-(heterocyclyl-phenyl)-urea derivatives, are glycogen phosphorylase a inhibitors useful e.g. for treating type II diabetes, dyslipidemia or arteriosclerosis
12/01/2004EP1257542B1 Method for producing 2-(1,2,4-triazol-1-yl)-ethanols
12/01/2004EP1181280B1 Substituted benzoyl ketones, methods for producing them and their use as herbicides
12/01/2004EP0977745B1 Thioaryl sulfonamide hydroxamic acid compounds
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