Patents for C07D 249 - Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms (17,749) |
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09/21/2010 | US7799815 2-methyl-6-[(1R,5S/1S,5R)-3-(3-{[4-methyl-5-(4-methyl-1,3-oxazol-5-yl)-4H-1,2,4-triazol-3-yl]thio}propyl)-3-azabicyclo[3.1.0]hex-1-yl]quinoline, used to treat drug abuse and dependence, psychological disorders, urogenital disorders or as cognition activators |
09/21/2010 | CA2437950C Acylated 1,2,3,4-tetrahydronaphthyl amines and their use as pharmaceutical |
09/21/2010 | CA2428019C Estrogen receptor modulators |
09/21/2010 | CA2359948C Triazole compounds with dopamine-d3-receptor affinity |
09/16/2010 | WO2010103283A1 Bis aromatic compounds for use as ltc4 synthase inhibitors |
09/16/2010 | WO2010103021A1 Composition comprising pesticide and benzotriazole uv absorbers |
09/16/2010 | WO2010065865A3 Sulfonamide derivatives as bcl-2-selective apoptosis-inducing agents for the treatment of cancer and immune diseases |
09/16/2010 | US20100234617 process for preparation of letrozole and its intermediates |
09/16/2010 | US20100234616 Method for the preparation of rufinamide |
09/16/2010 | US20100234404 P-38 Kinase Inhibitors |
09/16/2010 | US20100234378 Alkylsulfonamide-substituted triazoles as matrix metalloprotease inhibitors |
09/16/2010 | US20100234254 Lubricating oil additive, lubricating oil composition containing the same, various low-friction sliding members, rolling bearing, and sliding bearing |
09/16/2010 | CA2754941A1 Bis aromatic compounds for use as ltc4 synthase inhibitors |
09/15/2010 | EP2228065A2 Heterocyclo inhibitors of potassium channel function |
09/15/2010 | EP2227453A2 Heteroaryl amides useful as inhibitors of voltage-gated sodium channels |
09/15/2010 | CN101830858A Preparation method of 1H-1,2,4-tolyltriazole-3-methyl formate |
09/15/2010 | CN101830857A Sodalite porous coordination polymer material as well as preparation method and application thereof |
09/14/2010 | CA2422805C Retinoids for the treatment of emphysema |
09/10/2010 | WO2010101247A1 Cyclohexane derivative having npy y5 receptor antagonism |
09/10/2010 | WO2010100199A1 Fluconazole carboxylic ester derivatives, synthesis, and use in long acting formulations |
09/10/2010 | WO2010100186A1 Fluconazole carboxylic ester derivatives, synthesis, and use in long acting formulations |
09/08/2010 | EP2226317A1 Aryl (1h-1,2,4-triazol-1-yl) compound, and process for production thereof |
09/08/2010 | EP2226316A1 Copper-catalysed ligation of azides and acetylenes |
09/08/2010 | EP2225231A1 Aminotriazole derivatives as alx agonists |
09/08/2010 | EP1693358B1 Process for producing epoxytriazole compound and intermediate therefor |
09/08/2010 | CN1819998B Optically active halohydrin derivative and process for producing optically active epoxy alcohol derivative from the same |
09/08/2010 | CN101827828A 1, 2, 4 -triazole derivatives as serotonergic modulators |
09/08/2010 | CN101824002A Water soluble triazole compound and synthesis method thereof |
09/02/2010 | WO2010098600A2 Substituted azole derivatives, pharmaceutical composition containing the derivatives, and method for treating parkinson's disease using the same |
09/02/2010 | US20100222580 Process For The Preparation Of Onium Alkylsulfates Having A Low Halide Content |
09/02/2010 | US20100222401 Compositions and methods for treating pathologic angiogenesis and vascular permeability |
09/02/2010 | US20100222400 F1F0-ATPase Inhibitors and Related Methods |
09/02/2010 | US20100222398 Novel 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors |
09/02/2010 | US20100221176 Methods and compositions for protein labelling |
09/02/2010 | CA2751343A1 Substituted azole derivatives, pharmaceutical composition containing the derivatives, and method for treating parkinson's disease using the same |
09/01/2010 | EP2224013A1 Methods for the determination of telomerase activity using click chemistry |
09/01/2010 | EP2223922A2 Inhibitors of human phosphatidyl-inositol 3-kinase delta |
09/01/2010 | EP1720546B1 Novel, sustained-action beta-2-agonists and their use as medicaments |
09/01/2010 | EP1379508B1 N-(aryl)-2-arylethenesulfonamides and therapeutic uses thereof |
09/01/2010 | EP1028942B1 Dipeptide nitriles |
09/01/2010 | CN101820759A Fungicidal n-cycloalkyl-benzyl-thiocarboxamides or n-cycloalkyl-benzyl-n' -substituted-amidine derivatives |
09/01/2010 | CN101817793A S-triazolyl alpha-mercaptoacetanildes as inhibitors of HIV reverse transcriptase |
09/01/2010 | CN101817792A Bistriazolone, bistriadimenol compounds with antimicrobial activity, and salts, synthesis method and uses thereof |
09/01/2010 | CN101817784A Ethylene derivatives and pesticides containing said derivatives |
09/01/2010 | CN101239932B Preparation of 3,5-di(2-cyano-isopropyl)-toluene |
08/31/2010 | US7786156 reacting [2-(5-Hydrazinomethyl-1H-indol-3-yl)-ethyl]-dimethyl-amine with a 1,2,4-triazolyl forming reagent such as 1,3,5-triazine, formamidine, formamidinium salts or formamide, to obtain (3-[2-(dimethylamino)ethyl]-5-(1,2,4-triazol-1-ylmethyl)indole) |
08/31/2010 | US7786122 use to treat Alzheimer's Disease; (2R)-2-[N-(4-Chlorobenzenesulfonyl)-N-(4-methoxybenzyl)amino]-4-methylpentanoic acid amide for example |
08/31/2010 | CA2269399C Ocular devices manufactured with free radical-polymerizable latent ultra-violet absorbers |
08/26/2010 | WO2010094289A1 Allosteric binding compounds |
08/26/2010 | WO2010076033A9 Toluidine sulfonamides and their use |
08/26/2010 | US20100216984 Novel chromophoric silyl protecting groups and their use in the chemical synthesis of oligonucleotides |
08/26/2010 | US20100216815 N-substituted oxindoline derivatives as calcium channel blockers |
08/25/2010 | CN101812028A 5-chlorol-2-hydroxyl-3-(4-substituted-1H-1,2,3-triazole) benzoic acid compound as well as preparation method and application thereof |
08/25/2010 | CN101323600B Triadimefon and triadimenol compounds having antimicrobial activity, salts, synthetic methods and uses thereof |
08/24/2010 | US7781471 cannabinoid receptor antagonists, used for treating psychological disorders, neurodegenerative diseases, gastrointerstinal disorders, eating disorders, non-insulin dependent diabetes, drug abuse and dependence, headaches, obesity, sleep disorders and dyslipidemia |
08/24/2010 | US7781463 Enzyme inhibitors |
08/24/2010 | US7781462 1-(3,4,5-trimethoxy-phenyl)-5-(4-bromo-phenyl)-1H-[1,2,3]triazole; 1-(2-hydroxy-4-methoxy-5-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-5-(4-bromo-phenyl)-1H-[1,2,3]triazole; inhibits tubulin polymerization in a cell; cancer |
08/24/2010 | CA2423103C N-acylsulfonamide apoptosis promoters |
08/19/2010 | WO2010093845A1 Triazole and imidazole derivatives for use as tgr5 agonists in the treatment of diabetes and obesity |
08/19/2010 | WO2010092180A1 Aminotetraline derivatives, pharmaceutical compositions containing them, and their use in therapy |
08/19/2010 | WO2010091543A1 Novel hydrazino-cyclobut-3-ene-1, 2-dione derivatives as cxcr2 antagonists |
08/19/2010 | WO2010023685A3 Crystalline form of 2-(2-hydroxy phenyl)benz[e][1,3]oxazin-4-one, process for the same and use for producing 4-(3,5-bis(2-hydroxyphenyl)-1h-1,2,4-triazol-1-yl)benzoic acid |
08/19/2010 | US20100210854 Cyclopropenones and the Photochemical Generation of Cyclic Alkynes Therefrom |
08/19/2010 | CA2750793A1 Aminotetraline derivatives, pharmaceutical compositions containing them, and their use in therapy |
08/18/2010 | EP2217577A2 Novel compounds and compositions and methods of use |
08/18/2010 | EP2217565A1 Compounds which modulate the cb2 receptor |
08/18/2010 | CN101808995A Novel glucokinase activators and methods of using same |
08/18/2010 | CN101808988A Piperidine and piperazine derivatives |
08/18/2010 | CN101805303A Substituted hydroxylamine derivatives with anti-inflammatory activity and preparation method and application thereof |
08/18/2010 | CN101805302A 2-(4-phenyl-3-aryloxy-1,2,4-triazole-5-sulfenyl) acetamide and synthesis and application thereof |
08/18/2010 | CN101805301A Method for preparing chiral flutriafol |
08/18/2010 | CN101805300A Method for preparing chiral hexaconazole |
08/18/2010 | CN101307018B Diethylene triaminepentaacetic acid carboxyl active ester or analogues, method for synthesizing same and use |
08/17/2010 | US7776898 Opioid receptor active compounds |
08/17/2010 | US7776897 such as 3-[1-(5-chloro-2-thienyl)cyclopenty]-5,6,7,8,9,10-hexahydro [1,2,4]triazolo[4,3-a]azocine, having a strong 11 beta -hydroxysteroid dehydrogenase type 1inhibitory activity and exhibiting an excellent blood-glucose level-lowering action, used for the therapy of diabetes and insulin resistance |
08/17/2010 | CA2397734C Water soluble prodrugs of azole compounds |
08/12/2010 | WO2010090094A1 Aromatic amino compound manufacturing method |
08/12/2010 | US20100204472 Indane acetic acid derivatives and their use as pharmaceutical agents, intermediates, and method of preparation |
08/12/2010 | US20100204280 Cinnamoyl inhibitors of transglutaminase |
08/12/2010 | US20100204206 Di(hetero)arylcyclohexane derivatives, their preparation, their use and pharmaceutical compositions comprising them |
08/12/2010 | US20100200842 Surface modifying agent, laminated structure and transistor including the same, and method of manufacturing the laminated structure |
08/11/2010 | EP2215065A1 Ccr10 antagonists |
08/11/2010 | EP2215052A1 Desferrioxamine conjugates, derivatives and analogues |
08/11/2010 | EP2215049A1 P2x3, receptor antagonists for treatment of pain |
08/11/2010 | CN101798298A Imidazole derivatives |
08/11/2010 | CN101798290A Method for synthesizing chiral cyproconazole |
08/10/2010 | CA2488592C 11-beta-hydroxysteroid dehydrogenase 1 inhibitors useful for the treatment of diabetes, obesity and dyslipidemia |
08/10/2010 | CA2483159C Triazole derivatives as tachykinin receptor antagonists |
08/10/2010 | CA2237099C Sulfonylaminocarboxylic acids |
08/05/2010 | WO2010087419A2 Ester compound and use thereof |
08/05/2010 | US20100197911 Nitrogen-Containing Aromatic Derivatives |
08/05/2010 | US20100197871 Ligands for copper-catalyzed azide-alkyne cycloaddition reactions |
08/05/2010 | US20100197806 Method Involving 1-Benzotriazolyl Carbonate Esters of Polymers |
08/05/2010 | US20100197749 Chemical compounds |
08/05/2010 | US20100197696 Pesticidal heterocyclic dihaloallyl compounds |
08/05/2010 | US20100197644 Chemical Compounds 572 |
08/04/2010 | EP2212301A1 An improved process for preparation of letrozole and its intermediates |
08/04/2010 | EP1638947B1 Triazole derivatives as inhibitors of 11-beta hydroxysteroid dehydrogenase-1 |
08/04/2010 | CN101796034A Novel 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors |
08/04/2010 | CN101792438A Method for synthesizing 1-substituted-1,2,3-tolyltriazole |