Patents
Patents for C07D 241 - Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings (18,673)
01/2015
01/13/2015US8933225 Process for the synthesis of E1 activating enzyme inhibitors
01/13/2015US8933102 Pyrrolidine derived β3 adrenergic receptor agonists
01/13/2015US8933056 Soft protease inhibitors and pro-soft forms thereof
01/08/2015US20150011535 Heterocyclic compounds, medicaments containing them, use and processes for the preparation thereof
01/07/2015CN104271561A 苯丙醇类抗菌剂 Phenylpropanoid alcohol antibacterial agent
01/07/2015CN104262294A 六氟异丙醇衍生物 Hexafluoroisopropanol derivatives
01/07/2015CN104262268A 一种2-腈基喹喔啉类化合物的合成方法 A method of synthesis of the nitrile group-2- quinoxaline compounds
01/07/2015CN104262267A 用于治疗前列环素(pgi2)受体相关病症的pgi2受体调节剂 Pgi2 receptor modulator for the treatment of prostacyclin (pgi2) receptor related disorders
01/07/2015CN104262266A 一种1,4-二甲酰基-2,3,5,6-四羟基哌嗪的合成方法 A method of synthesis of 1,4-dimethoxy-2,3,5,6-tetrahydroxy-acyl piperazine
01/07/2015CN104262118A 一种二芳基衍生物的制备方法 A process for preparing diaryl derivatives
01/07/2015CN102898387B 管道化连续生产n-[(2z)-哌嗪-2-亚基]-2,2,2-三氟乙酰肼的方法 Continuous production of pipelines n - [(2z) - piperazin-2-ylidene] -2,2,2-trifluoro-acetic hydrazide method
01/07/2015CN102892758B 用于治疗cf的吡啶和吡嗪衍生物 Pyridine and pyrazine derivatives for the treatment cf
01/07/2015CN102775357B 金属卟啉催化空气氧化制备乙酰吡嗪的方法 Methods metalloporphyrin catalytic air oxidation of acetyl pyrazine preparation
01/07/2015CN102574778B 新的联苯基和苯基-吡啶酰胺类化合物 New biphenyl and phenyl - pyridine amides
01/07/2015CN102311396B 一种吡嗪类衍生物和其制备方法及在制药中的应用 A pyrazine derivatives and methods for their preparation and use in pharmacy
01/07/2015CN101805266B 有机电致发光化合物和使用该化合物的有机电致发光器件 Organic electroluminescent compounds and the use of the compounds are organic electroluminescent devices
01/06/2015US8927712 Process for the preparation of a mono-N-alkylpiperazine
01/06/2015US8927577 Quinolinyl glucagon receptor modulators
01/06/2015US8927546 Therapeutic piperazines
01/01/2015US20150005315 1-substituted 4-arylpiperazine as kappa opioid receptor antagonists
01/01/2015US20150005294 Azaheterocyclic compounds
12/2014
12/31/2014CN102924388B 一种吡嗪类化合物及其制备方法 One kind of pyrazine compounds and its preparation method
12/30/2014US8921370 Bicyclo[3.2.1]octyl amide derivatives and uses of same
12/30/2014US8920941 Pyrazine derivative, and light emitting element, display device, electronic device using the pyrazine derivative
12/30/2014CA2655159C Glycine transporter-1 inhibitors
12/30/2014CA2618479C Pyrazine derivatives and use as pi3k inhibitors
12/25/2014US20140378461 Novel compounds
12/24/2014CN104245680A 用于生产5-(二氟甲基)吡嗪-2-甲酸的方法及其生产中间体 For the production of 5- (difluoromethyl) pyrazine-2-carboxylic acid and its production method of Intermediate
12/24/2014CN104230892A 一组提高激酶活性的化合物及其应用 Kinase activity of a group of compounds improving its Application
12/24/2014CN104230743A 一种4-苄基-1-苯乙基哌嗪-2,6-二酮的制备方法 Of 4-benzyl-1-phenethyl-piperazine-2,6-dione Method
12/24/2014CN103193702B 含氮杂环化合物官能团化的方法 Nitrogen-containing heterocyclic compounds functionalized method
12/24/2014CN102464612B 含哌嗪氨基甲酸酯的二卤丙烯醚类化合物与应用 Piperazine-containing urethane dihalopropene ether compound and Applications
12/23/2014US8916593 Alkoxy-substituted 2-aminopyridines as ALK inhibitors
12/23/2014US8916561 Substituted quinoxaline compounds for the inhibition of PASK
12/23/2014US8916560 Heterocyclic compounds for the inhibition of PASK
12/23/2014US8916554 Amino-derivatives as novel inhibitors of histone deacetylase
12/18/2014US20140371232 Cajanine structure analogous compound, preparation method and use
12/18/2014US20140371228 Novel therapeutic agents
12/18/2014US20140371226 9-[4-(3-chloro-2-fluoro-phenylamino)-7-methoxy-quinazoline-6-yloxy]-1,4-diaza-spiro[5.5]undecane-5-one dimaleate, use thereof as a medicament and method for the production thereof
12/18/2014US20140371196 Diamino heterocyclic carboxamide compound
12/18/2014US20140371073 Plant growth regulating compounds
12/17/2014CN104220429A 非全身性tgr5激动剂 Non-systemic tgr5 agonist
12/17/2014CN104211650A 富马酸)11芎嗪及其制备方法以及药物组合物 Fumaric acid) 11 Gung-triazine and its preparation method and pharmaceutical compositions
12/17/2014CN103073510B 一类吡嗪基西弗碱化合物的结构、制备和用途 A class structure, preparation and use of alkali compounds pyrazine 基西弗
12/17/2014CN102675232B 4-(6-氯-喹喔啉-2-基氧基)-苯酸的合成方法 4- (6-chloro - quinoxalin-2-yloxy) - benzoic acid Synthesis of
12/16/2014US8912329 Composition for treatment of tuberculosis
12/16/2014US8912328 Formation of N-protected bis-3,6-(4-aminoalkyl)-2,5,diketopiperazine
12/16/2014US8912190 Substituted heterocyclic compounds
12/16/2014US8912188 Substituted quinoxaline carboxylic acids for the inhibition of PASK
12/11/2014US20140359951 Novel oxidation dye precursors
12/10/2014CN104203916A 作为杀线虫剂的n-环酰胺 As nematicides n- cyclic amide
12/10/2014CN104193699A 一种小分子化合物及其合成方法和应用 A small molecule compounds and synthetic methods and applications
12/10/2014CN104193690A 3,4,5-三羟基没食子酰胺苯磺酰胺类衍生物及其制备方法和应用 3,4,5-trihydroxy gallic acid amide benzene sulfonamide derivatives, preparation method and application
12/10/2014CN104193686A N-没食子酰胺-嘧啶基苯磺酰胺类衍生物及其制备方法和应用 N- gallic acid amide - benzene sulfonamides pyrimidine derivatives and preparation method and application
12/10/2014CN102863397B 喹喔啉酮酰胺类化合物、其制备方法与应用 -quinoxalinone Amides, their preparation and use
12/09/2014US8907088 Methods of making cyclic, N-amino functional triamines
12/09/2014US8907087 Substituted pyrazino[2,3-b]pyrazines as mTOR kinase inhibitors
12/09/2014US8906926 Substituted diketopiperazine analogs for use as drug delivery agents
12/04/2014US20140357632 Benzopiperazine derivatives as cetp inhibitors
12/04/2014US20140356430 Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-((trans)-4-methoxycyclohexyl)-3,4-dihydropyrazino [2,3-b]pyrazin-2(1h)-one, a solid form thereof and methods of their use
12/04/2014US20140356360 Piperazinyl derivatives for the treatment of cancer
12/02/2014US8901302 Pyrazino[2,3-D]isoxazole derivative which is useful as a production intermediate of pyrazine carboxamide derivative
12/02/2014US8901295 Inhibitors of cyclophilins and uses thereof
12/02/2014US8901129 Methods of facilitating neural cell survival using GDNF family ligand (GFL) mimetics or RET signaling pathway activators
12/02/2014US8901126 Substituted imidazo[1,5-A]quinoxalin-4-ones are useful for preventing or treating storage dysfunction, voiding dysfunction and bladder/urethral diseases
12/02/2014US8901119 Peptide deformylase inhibitors
12/02/2014US8901116 Method for treating pain, anxiety or depression using carbamoyloxy alkanoyl piperazine compound
12/02/2014US8900550 Catalytic radiofluorination
11/2014
11/27/2014US20140350030 Bicarbocyclic and tricarbocyclic ethynyl derivatives and uses of same
11/27/2014US20140350024 Antimicrobial agents
11/25/2014US8895776 Modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto
11/25/2014US8895739 Acylation of hindered amines and functionalized bis-peptides obtained thereby
11/25/2014US8895589 Pyridinyl amides as P2X3 and P2X2/3 inhibitors
11/25/2014US8895572 Fused heterocyclic indane carboxamide CGRP receptor antagonists
11/25/2014US8895564 Biguanide derivative compound
11/25/2014US8895560 Opioid antagonists
11/25/2014US8895559 Quinoxalines derivatives and pharmaceutical compositions and kits
11/25/2014US8895554 Compounds, compositions and methods for the treatment of amyloid diseases and synucleinopathies such as Alzheimer's disease, type 2 diabetes, and Parkinson's disease
11/25/2014US8895474 Herbicidally active cyclopentanediones and derivatives thereof, and their use in controlling weeds
11/20/2014US20140343068 Certain chemical entities, compositions, and methods
11/18/2014US8889863 Stereoselective methods, catalysts and intermediates for the synthesis of (−)-Nutlin-3 and related compounds
11/18/2014US8889693 Fibrosis inhibitor
11/18/2014US8889692 Pyrazinone derivatives, pharmaceutically acceptance salts thereof and their uses
11/18/2014US8889683 Substituted quinoxalines as inhibitors of fatty acid binding protein
11/18/2014US8889667 Therapeutic compounds and compositions
11/18/2014US8889664 Phosphatidylinositol 3-kinase inhibitors and methods of their use
11/18/2014US8889099 Methods and compositions for delivering peptides
11/13/2014US20140336375 Allosteric modulators of 5-hydroxytryptamine 2c receptor (5-ht2cr)
11/13/2014US20140336198 Amine Derivatives as Potassium Channel Blockers
11/11/2014US8884015 Process for the preparation of a mono-N-alkypiperazine
11/11/2014US8884009 Process for making bortezomib and intermediates for the process
11/11/2014US8883861 Iminic monomers and polymers thereof
11/11/2014US8883796 Biphenyl derivatives, pharmaceutical composition comprising the same, and preparation method thereof
11/11/2014US8883786 Glucocorticoid receptor antagonists
11/11/2014US8883778 Cyclic inhibitors of 11 beta-hydroxysteroid dehydrogenase 1
11/11/2014US8883432 Coelenterazine analogues and coelenteramide analogues
11/06/2014US20140329837 Arylpyrazinones such as but not limited to 3-(4-chlorophenyl-1-ethylpyrazin-2-(1h0)-one
11/06/2014US20140329821 Novel Substituted Bicyclic Aromatic Compounds as S-Nitrosoglutathione Reductase Inhibitors
11/04/2014US8877971 Method for preparing formamide compounds
11/04/2014US8877760 Substituted pyrazine-2-carboxamide kinase inhibitors
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