Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619) |
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10/04/2012 | WO2012135750A1 Combinations of akt inhibitor compounds and vemurafenib, and methods of use |
10/04/2012 | WO2012135697A2 Novel rho kinase inhibitors and methods of use |
10/04/2012 | WO2012135641A2 Aurora kinase inhibitors and methods of making and using thereof |
10/04/2012 | WO2012135084A1 METABOLITES OF 2-(FURAN-2-YL)-7-(2-(4-(4-(2-METHOXYETHOXY)PHENYL)PIPERAZIN-1-YL)ETHYL)-7H-PYRAZOLO[4,3-e][1,2,4]TRIAZOLO[1,5-c]PYRIMIDIN-5-AMINE AND THEIR UTILITY AS ADENOSINE A2a RECEPTOR ANTAGONISTS |
10/04/2012 | WO2012135083A1 METABOLITES OF 7-(2-(4-(6-FLUORO-3-METHYLBENZO[d]ISOXAZOL-5-YL)PIPERAZIN-1-YL)ETHYL)-2-(PROP-1-YNYL)-7H-PYRAZOLO[4,3-e][1,2,4]TRIAZOLO[1,5-c]PYRIMIDIN-5-AMINE AND THEIR UTILITY AS ADENOSINE A2a RECEPTOR ANTAGONISTS |
10/04/2012 | WO2012135009A1 Pyrimidine-4,6-diamine derivatives as pi3k inhibitors |
10/04/2012 | WO2012130882A1 Fe(iii) complexes for the treatment and prophylaxis of iron deficiency symptoms and iron deficiency anaemias |
10/04/2012 | WO2012130166A1 1-(arylmethyl)quinazoline-2,4(1h,3h)-diones as parp inhibitors and the use thereof |
10/04/2012 | WO2012129792A1 Pyrimidinone compounds, preparation methods, pharmaceutical compositions and uses thereof |
10/04/2012 | US20120253041 New phenylalanine derivatives |
10/04/2012 | US20120252830 Substituted Aminobutyric Derivatives as Neprilysin Inhibitors |
10/04/2012 | US20120252809 Substituted 3-heteroaroylamino-propionic acid derivatives and their use as pharmaceuticals |
10/04/2012 | US20120252790 Amino-Derivatives As Novel Inhibitors Of Histone Deacetylase |
10/04/2012 | CA2844699A1 Combinations of akt inhibitor compounds and abiraterone, and methods of use |
10/04/2012 | CA2831937A1 Combinations of akt inhibitor compounds and erlotinib, and methods of use |
10/04/2012 | CA2831935A1 Combinations of akt inhibitor compounds and chemotherapeutic agents, and methods of use |
10/04/2012 | CA2831932A1 Combinations of akt and mek inhibitor compounds, and methods of use |
10/04/2012 | CA2831922A1 Combinations of akt inhibitor compounds and vemurafenib, and methods of use |
10/04/2012 | CA2831015A1 1-(arylmethyl)quinazoline-2,4(1h,3h)-diones as parp inhibitors and the use thereof |
10/04/2012 | CA2829240A1 Fe(iii) complex compounds for the treatment and prophylaxis of iron deficiency symptoms and iron deficiency anemias |
10/03/2012 | EP2504319A1 Process for preparing a polymorph of the choline salt of a pyrimidin-5-yl acetic acid derivative |
10/03/2012 | EP2504318A2 Crystalline salt forms of a pyrimidin-5-yl acetic acid derivative |
10/03/2012 | EP2504314A1 Quinazoline derivatives |
10/03/2012 | EP2504309A1 Synthesis of acetoxyacetaldehyde |
10/03/2012 | CN102712602A Process for preparing 2-methyl-4-amino-5-cyanopyrimidine |
10/03/2012 | CN102712587A Novel ethane diamine hepcidin antagonists |
10/03/2012 | CN102712566A Synthesis of acetoxyacetaldehyde |
10/03/2012 | CN102702116A 4-(3-chloro-4-methoxylanilino)-6-(3-amidophenyl)quinazoline compound or pharmaceutically-acceptable salt thereof and preparation methods and applications thereof |
10/03/2012 | CN102702115A Synthetic method of 4-chloro-7-fluoro-6-nitro quinazoline |
10/03/2012 | CN102702114A Method for preparing nitro orotic acid |
10/03/2012 | CN102702113A 5-Fluorouracil derivative and preparation method and uses |
10/03/2012 | CN102702112A Preparation method of bensulfuron |
10/03/2012 | CN102702111A Processes for the preparation of 4-((4-((4-(2-cyanoethenyl)-2,6-dimethylphenyl)amino)-2-pyrimidinyl)amino)benzonitrile |
10/03/2012 | CN102702110A Preparation method of 4-amino-5, 6-dichloropyrimidine |
10/03/2012 | CN102698803A Ruthenium complex catalyst and preparation method and application thereof |
10/03/2012 | CN101863844B Synthesis method of 6,7-substituted-4-aniline quinazoline |
10/03/2012 | CN101801936B Metabolites and derivatives of ambrisentan |
10/03/2012 | CN101759653B Preparation method of 6, 7-dimethoxy quinazoline-4-ketone |
10/03/2012 | CN101687801B Ethers of naphtalene carboxylic acid amides as cancer cure |
10/03/2012 | CN101654441B Anticoagulant compound, composition and application thereof |
10/03/2012 | CN101460453B Novel sulfonamide compounds |
10/02/2012 | US8278446 reacting 4-amino-6-chloro-pyrimidine-5-carbaldehyde with 4-benzyloxy-3-chloro-phenylamine in an aqueous solvent and a catalytic amount of hydrochloric acid, to providw 4-amino-6-(4-benzyloxy-3-chloro-phenylamino)-pyrimidine-5-carbaldehyde, then oximination with (2-morpholin-4-yl-ethyl)-hydroxylamine |
10/02/2012 | US8278445 Preparation methods of azoxystrobin and its analogs |
10/02/2012 | US8278357 Derivatives of N-phenylanthranilic acid and 2-benzimidazolone as potassium channel and/or neuron activity modulators |
10/02/2012 | US8278314 Quinazoline analogs as receptor tyrosine kinase inhibitors |
10/02/2012 | US8278310 Amine salts of a CRTH2 antagonist |
10/02/2012 | US8278309 Synthetic mimetics of host defense and uses thereof |
10/02/2012 | US8278304 Substituted 4-hydroxypyrimidine-5-carboxamides |
10/02/2012 | US8277599 Compounds for placing objects by self assembling and the use thereof |
10/02/2012 | CA2575720C Pyrimidine derivatives |
09/27/2012 | WO2012129491A1 Trpv3 modulators |
09/27/2012 | WO2012128965A2 Method for preparation of 5-substituted pyrimidines |
09/27/2012 | US20120245351 Process for the preparation of lapatinib and its pharmaceutically acceptable salts |
09/27/2012 | US20120245350 Methods for the preparation of lapatinib and the salts thereof |
09/27/2012 | US20120245185 Aryl and heteroaryl sulfones as mglur4 allosteric potentiators, compositions, and methods of treating neurological dysfunction |
09/27/2012 | US20120245169 Certain chemical entities, compositions and methods |
09/27/2012 | US20120245137 Aryl sulphone derivatives as calcium channel blockers |
09/27/2012 | US20120245124 TRPV3 Modulators |
09/27/2012 | US20120244119 Anti-infective agents and uses thereof |
09/26/2012 | EP2501684A2 Process for the preparation of substituted phenylalanines |
09/26/2012 | EP2501679A1 Heterocyclic antiviral compounds |
09/26/2012 | EP2501233A1 Quinazoline compounds |
09/26/2012 | CN102695700A Pyrimidine derivatives as protein tyrosine kinase 2 inhibitors |
09/26/2012 | CN102695697A Novel multifunctional peptidase inhibitors, especially for medical use |
09/26/2012 | CN102690238A Synthesis of barbituric acid derivative as RSK2 inhibitor and application thereof |
09/26/2012 | CN102690237A Method for synthesizing high-purity azoxystrobin |
09/26/2012 | CN102174025B Isotope labeling reagent as well as preparation method and application thereof |
09/26/2012 | CN101808992B 1,1,1-trifluoro-2-hydroxy-3-phenylpropane derivatives |
09/26/2012 | CN101367767B Room temperature solvent-free synthesis of 3,4-dihydropyrimidine-2-ketone |
09/26/2012 | CN101119965B Tetralin and indane derivatives and uses thereof |
09/25/2012 | US8273897 Method for producing 2,2-difluoroethylamine derivative by amide hydrogenation |
09/25/2012 | US8273879 Triazolo pyrimidine compounds |
09/25/2012 | US8273878 Process for the preparation of pyrimidine compounds |
09/25/2012 | US8273767 Bicyclic-substituted amines as histamine-3 receptor ligands |
09/25/2012 | US8273758 Substituted tricyclic derivatives |
09/25/2012 | US8273751 Organic compounds |
09/25/2012 | US8273747 tert-Butyl (4-((4'-cyano-4-methoxy-biphenyl-3-ylmethyl)-amino)-cyclohexyl)-methyl-carbamate; hedgehog pathway agonists; alopecia; angiogenesis; wound healing; alzheimer's disease; inhibit aging effects on skin |
09/25/2012 | CA2667285C New sulfonamide derivatives as bradykinin antagonists |
09/20/2012 | WO2012125993A1 Solid state forms of rilpivirine base, and rilipivirine salts |
09/20/2012 | WO2012125521A1 Quinazolinediones and their use |
09/20/2012 | WO2012124696A1 Guanidine compound |
09/20/2012 | WO2012123467A1 Pyrimidine amide compounds |
09/20/2012 | WO2012122707A1 Quaternary ammonium salt compounds, preparation method, pharmaceutical composition and use thereof |
09/20/2012 | US20120238578 Compositions useful as inhibitors of voltage-gated sodium channels |
09/20/2012 | US20120238575 Antiproliferative pyrimidyl, fused pyrimidyl and pyrimidyl hydrazones |
09/20/2012 | US20120238570 Inhibitors of the hedgehog pathway |
09/20/2012 | CA2830157A1 Guanidine compound |
09/20/2012 | CA2829123A1 Quinazolinediones and their use |
09/19/2012 | EP2499118A2 Processes for the preparation of erlotinib hydrochloride form a and erlotinib hydrochloride form b |
09/19/2012 | CN102686570A Mesoionic pesticides |
09/19/2012 | CN102686569A Phenoxy-substituted pyrimidines as opioid receptor modulators |
09/19/2012 | CN102675418A Luteinizing hormone-releasing hormone (LHRH) antagonist derivative, preparation method of LHRH antagonist derivative and application of LHRH antagonist derivative |
09/19/2012 | CN102675315A Substitutive benzene alkyl contained purine compounds and preparation method and application thereof |
09/19/2012 | CN102675226A 3-substituted-1-methyl-quinazoline-2,4-dione compounds, preparation method and application thereof |
09/19/2012 | CN102675225A Synthesis method of erlotinib hydrochloride |
09/19/2012 | CN102675224A 2-substituent-7-fluorine-4-aromatic mixed base quinazoline derivant and preparation method and use thereof |
09/19/2012 | CN102675223A Preparation method for polysubstitution quinazoline and heterocyclic ring pyrimidine derivative |
09/19/2012 | CN102675222A Method for preparing multi-substituted quinazoline and heterocyclic pyrimidine derivative |
09/19/2012 | CN102675221A Intermediate in method for preparing pyrimidinedione derivative |
09/19/2012 | CN102675220A Etravirine preparing method and intermediate of etravirine |