Patents
Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619)
02/2004
02/26/2004WO2004016596A1 Condensed heterocyclic compounds as pde-iv inhibitors for the treatment of inflammatory and allergic disorders
02/26/2004WO2004016581A1 Processes for the preparation of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl]amino]benzonitrile
02/26/2004WO2004016271A1 Pyrimidones as antiviral agents
02/26/2004WO2003101444A8 Diarylurea compounds and derivatives as chk-1 inhibitors for the treatment of cancer
02/26/2004WO2003099211A3 Mitotic kinesin inhibitors
02/26/2004WO2003039549A8 Selective antibacterial agents
02/26/2004WO2003027110A3 Process for preparing 2-(4-pyridyl) amino-6-dialkyloxyphenyl-pyrido [2,3-d]pyrimidin-7-ones
02/26/2004WO2002098869A3 1,4-disubstituted benzo-fused cycloalkyl urea compounds
02/26/2004WO2002066672A3 Treatment of cns disorders using d-amino acid oxidase and d-aspartate oxidase antagonists
02/26/2004US20040039201 Functionalized compositions for improved immobilization
02/26/2004US20040039040 Urea derivative and adhesive-molecule inhibitor containing the same as active ingredient
02/26/2004US20040039034 Hydroxypropyl amides for the treatment of Alzheimer's disease
02/26/2004US20040039006 (2S)-2-(Adamantan-1-ylmethoxycarbonylamino)-3-(4-(2-(1,4,5,6-tetrahydropyrimidin-2-ylcarbamoyl)ethyl)benzoylamino)propionic acid isopropyl ester, its preparation and its use
02/26/2004US20040039005 HIV replication inhibiting pyrimidines
02/26/2004US20040039002 6,7-Dimethoxyquinazolines and therapeutic use thereof
02/26/2004US20040039001 2-guanidino-4-aryl-quinazoline
02/26/2004US20040039000 6-aminofuro(2,3-d)pyrimidines and 6-aminopyrrolo(2,3-d) pyrimidines useful in treating cancer, and secondary infections caused by Pneumocystis carinii and Toxoplasmosis gondii
02/26/2004US20040038994 Pyrimidine fused bicyclic metalloproteinase inhibitors
02/26/2004US20040038976 S,N-diarylsulfonamide derivatives; treating inflammatory diseases such as Celiac's disease, Crohn's disease or colitis.
02/26/2004US20040038969 Substituted aminopyrimidines and aminopyridazines; analgesics particularly for migraines, neuropathic pain and associated hyperalgesia and allodynia; antiinflammatory agents; treating asthma, gastrointestinal disorders, etc.
02/25/2004EP1391952A2 Salts of pentacyclic or tetrapentaline derived anions, and their uses as ionic conductive materials
02/25/2004EP1391454A1 Substituted benzamide compounds with antihypertensive activity
02/25/2004EP1391450A1 N-(heterocycle-methyl)alkylamine derivative, process for producing the same, and bactericide
02/25/2004EP1391206A1 Pharmaceutical compositions comprising arsenic for the treatment of lymphoma
02/25/2004EP1390352A1 Pyrimidine derivatives
02/25/2004EP1390351A1 Pyrimidine derivatives useful as selective cox-2 inhibitors
02/25/2004EP1390350A1 Novel compounds
02/25/2004EP1390340A1 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
02/25/2004EP1211246B1 Pyrimidine derivatives and herbicides containing the same
02/25/2004EP1165064B1 Novel inhibitors of formation of advanced glycation endproducts (age's)
02/25/2004EP1005446B1 N-aroylphenylalanine derivatives
02/25/2004CN1478085A ABCA-1 elevating compounds against coronary artery disease or atherosclerosis
02/25/2004CN1478082A Pyrimidine compounds and their use
02/25/2004CN1478078A Nitrogenous aromatic ring compounds
02/25/2004CN1477089A Substituted dicyclohexylalkyl diphenyl derivative with good low-tomp, mutual solubility, its preparation and application
02/25/2004CN1139577C Improved process for preparation of unsymmetrical 4,6-bis(aryloxy) pyrimidine compounds
02/24/2004US6696487 Fungicidal phenyl(thio)urea and phenyl(thio)carbamate derivatives
02/24/2004US6696482 Formulations for hydrophobic pharmaceutical agents
02/24/2004US6696472 Substituted N-phenoxy-N-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
02/24/2004US6696456 Carbocyclic acids and salts such as (2s,3r)-3-ethylsulfanyl-2-(4'-fluoro-biphenyl-4-sulfonylamino)-3- phenylpropionic acid, used as metalloenzyme antagonists for the prophylaxis of degenerative joint disease and as wound healing agents
02/24/2004US6696455 Nitrogen compounds such as 6-chloro-2-methyl-4-oxo-pyrido (3,2-d)pyrimidine used as anticarcinogenic agents and/or for prophylaxis of infections caused by pneumocystis or toxoplasma
02/24/2004US6696452 Glycogen synthase kinase-3 and aurora-2 a serine/threonine protein kinase inhibitors; antidiabetic and anticancer agents and alzheimer's disease treatments
02/24/2004US6696451 Dihydropyrimidines
02/24/2004US6696445 Neuropeptide y receptor antagonists comprising heterocyclic nitrogen compounds and/or prodrugs used for prophylaxis of eating and cardiovascular disorders
02/24/2004US6696442 Carbocyclic and heterocyclic substituted semicarbazones and thiosemicarbazones and the use thereof
02/24/2004US6696435 For treating atherosclerosis, other coronary artery diseases; 3-((3-(3-trifluoromethoxyphenoxy)phenyl)((3-(1,1,2,2-tetrafluoroethoxy) -phenyl)methyl) amino)-1,1,1-trifluoro-2-propanol for example
02/19/2004WO2004014916A1 Pyrimidine fused bicyclic metalloproteinase inhibitors
02/19/2004WO2004014873A1 4-substituted quinazoline-8-carboxyamide derivative and pharmaceutically acceptable addition salt thereof
02/19/2004WO2004014872A1 Process for preparing the calcium salt of rosuvastatin
02/19/2004WO2004014871A1 Vanilloid receptor ligands and their use in treatments
02/19/2004WO2004014870A1 Fluorinated phenyl-naphthalenyl-urea compounds as inhibitors of cytokines involved in inflammatory processes
02/19/2004WO2004014869A2 5,6-fused 3,4-dihydropyrimidine-2-one derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014868A2 Pyrimidine-2,4-dione derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014867A2 Matrix metalloproteinase inhibitors and methods for identification of lead compounds
02/19/2004WO2004014847A1 Mcp-1 receptor antagonists and method of use thereof
02/19/2004WO2004014844A2 Aryl and heteroaryl compounds and methods to modulate coagulation
02/19/2004WO2004014825A1 Cannabinoid receptor ligands
02/19/2004WO2004014384A2 Cyclic compounds containing zinc binding groups as matrix metalloproteinase inhibitors
02/19/2004WO2004014381A2 Matrix metalloproteinase inhibitors and methods for identification of lead compounds
02/19/2004WO2003027234A9 Small organic molecule regulators of cell proliferation
02/19/2004US20040034251 Such as 2-(4,6-dimethoxypyrimidine-2-ylcarbonyl)acetanilide; for use as intermediate in production of agricultural chemicals and medicines
02/19/2004US20040034242 Compounds containing a specific branched chain end terminal group, which is isopropyl, sec.-butyl, or tert.-butyl; a polar leading group, and long chain aliphatic, non-cyclic, saturated or nonsaturated linking groups
02/19/2004US20040034190 Preparation of supramolecular polymers by copolymerization of monomers containing quadruple hydrogen bonding units with regular monomers
02/19/2004US20040034104 2,2-Diphenylbutanamide derivatives and medicines containing the same
02/19/2004US20040034084 Side effect reduction; for treatment of AIDS, cancer and arthritis
02/19/2004US20040034076 Such as methyl-3-azido-2-((4,6-dimethoxy-2-pyrimidinyl)oxy) 3,3-diphenylpropionate; for treatment of high blood pressure
02/19/2004US20040034048 Didepsipeptide-based endoparasiticides, new didepsipeptides and process for preparing the same
02/19/2004US20040034044 Quinazoline derivatives and drugs
02/19/2004US20040034043 Positively-charged peptide nucleic acid analogs with improved properties
02/19/2004US20040034034 Novel piperazine derivatives
02/19/2004US20040034032 Quinoline and quinazoline compounds useful in therapy
02/19/2004US20040034025 Having a high residual activity, greater activity at lower application rates, curative activity, and a broader spectrum of efficacy; heterocyclic aromatic amides having a hydroxy group adjacent to the amide functionality
02/19/2004US20040034022 Polymorphic forms/hydrates of n-[4-(3-chloro-4-fluorophenylamino)-7-(3-morpholin-4-ylpropoxy)-quinazolin-6-yl]-acrylamide dihydrochloride
02/19/2004US20040034018 2-amino-trihydroindole or tetrahydronapthalene-2-yl derivatives, useful for disease state associated with smooth muscle disorders, such as gastrointestinal and urogenital disorders
02/19/2004CA2497656A1 Pyrimidine-2,4-dione derivatives as matrix metalloproteinase inhibitors
02/19/2004CA2495067A1 Mcp-1 receptor antagonists and method of use thereof
02/19/2004CA2494827A1 Cannabinoid receptor ligands
02/19/2004CA2494824A1 Fluorinated phenyl-naphthalenyl-urea compounds as inhibitors of cytokines involved in inflammatory processes
02/19/2004CA2493008A1 Aryl and heteroaryl compounds and methods to modulate coagulation
02/18/2004EP1389461A1 Pyrimidones with antiviral properties
02/18/2004EP1389205A1 Quinazoline and quinazoline-like compounds for the treatment of integrin-mediated disorders
02/18/2004EP1389194A2 Inhibitors of bace
02/18/2004EP1389189A2 Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues
02/18/2004EP1389183A1 Sulfonamide derivatives
02/18/2004EP1389103A2 Synthesis and evaluation of novel phthalimide mimics as anti-angiogenic agents
02/18/2004EP1216248B1 Triazolopyrimidine derivatives
02/18/2004EP1178958B1 N-cyanomethyl amides as protease inhibitors
02/18/2004EP0968192B1 Substituted tetrahydropyrimidine derivatives and their use as polymerization inhibitors for vinyl aromatic compounds
02/18/2004CN1138780C Thienopyrimidines
02/18/2004CN1138778C Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation
02/18/2004CN1138763C Di-or tri-fluoromethanesulfonyl anilide derivs, process for preparation of them and herbicides contg. them as active ingredient
02/18/2004CN1138760C Preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and TACE inhibitors
02/18/2004CN1138546C Certain 1,4,5-tri-substituted imidazole compounds useful as cytokine
02/17/2004US6693196 Bis(2,4-diaminophenoxy)pyridines and pyrimidines
02/17/2004US6693195 Process for preparing 4,6-dihydroxypyrimidine (DHP)
02/17/2004US6693194 By reacting 4,6-dichloro-2-(methylthio)pyrimidine in an inert organic solvent with an alkali metal methoxide, transferring to an aqueous acid medium and oxidation; using the product to prepare 7-((4,6-
02/17/2004US6693137 Sulphonamide derivatives
02/17/2004US6693123 (4-(3-pyridylaminomethylene)-2-phenylbenzoyl)-n -methylmethionine, methyl ester for example; restenosis, hyperplasia
02/17/2004US6693105 Using xanthinyl derivatives to reduce treatment induced toxicity; inhibiting cellular signaling through second messenger pathway; reducing cellular level of nonarachi-donate phosphatidic acid and diacylglycerol
02/17/2004US6693103 1,2,3,4-tetrahydro-2-thioxo-quinolinyl and 1,2,3,4-tetrahydro-2-oxo-quinolinyl derivatives as progesterone receptor modulators