Patents
Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619)
03/2005
03/10/2005WO2005021490A2 N-SULFONYL-α-AMINO-ACID DERIVATIVES
03/10/2005WO2005021486A1 Ester derivative and medicinal use thereof
03/10/2005WO2005020899A2 Substituted cycloalkyamine derivatives as modulators of chemokine receptor activity
03/10/2005WO2005020897A2 Compositions and methods for the treatment of disease associated with trp-p8 expression
03/10/2005WO2004112793B1 Guanidino-substituted quinazolinone compounds as mc4-r agonists
03/10/2005WO2004099148A8 Substituted pyrimidine derivatives
03/10/2005WO2004096128A3 Hiv integrase inhibitors
03/10/2005WO2004082613A3 2,4-diamino-5-[5’-substituted-benzyl] pyrimidines and 2,4-diamino-6-[5’-substituted-benzyl] quinazolines
03/10/2005US20050054819 Such as 1-benzylcyclobutyl (1S)-1-(oxo{[(1R)-1-phenylethyl]amino}acetyl)pentylcarbamate for treatment of osteoporosis
03/10/2005US20050054732 Preventives or remidies for alzheimer's disease or amyloid protein fibrosis inhibitors containing nitrogen-containing heteroaryl compounds
03/10/2005US20050054715 Vinyl phenyl derivatives as glk activators
03/10/2005US20050054662 Quinazoline derivatives as antitumor agents
03/10/2005US20050054661 Irritable bowel disorders; anxiolytic agents; antidepressants
03/10/2005US20050054660 8-Quinolinxanthine and 8-isoquinolinxanthine derivatives as PDE 5 inhibitors
03/10/2005US20050054656 Therapy for obesity, eating disorders, psychological disorders, antidepressants, central nervous system disorders
03/10/2005US20050054651 Compositions and methods for the treatment of disease associated with Trp-p8 expression
03/10/2005US20050054643 Substituted polycyclic aryl and heteroaryl pyrimidinones useful for selective inhibition of the coagulation cascade
03/10/2005US20050054638 Anticancer agents
03/10/2005US20050054626 Substituted cycloalkylamine derivatives as modulators of chemokine receptor activity
03/10/2005US20050054534 Substituted benzoylcyclohexane diones for use as herbicides
03/10/2005US20050051052 Self-assembling dyes
03/10/2005CA2536788A1 Naphthalene carboxamides and their derivatives useful as new anti-angiogenic agents
03/10/2005CA2535265A1 Compositions and methods for the treatment of disease associated with trp-p8 expression
03/09/2005EP1511730A2 Diaryl urea derivatives useful for the treatment of protein kinase dependent diseases
03/09/2005EP0906291B1 Substituted phenyl uracils
03/09/2005CN1592743A Inhibitors of glycogen synthase kinase 3
03/09/2005CN1592735A Novel alpha-oxygenated or alpha-thiolated carboxylic acid phenethylamide derivatives
03/09/2005CN1192018C Cell adhesive-inhibiting anti inflammatory and immune-suppressive compounds
03/08/2005US6864397 E.g., 1-(4-(4-pentylcyclohexyl)cyclohexyldifluoromethoxy)-4 -trifluoromethoxybenzene; preparation from difluorocyclo-hexylidenes, e.g. 1-(4-(trans-4-propylcyclohexyl)cyclohexyl-difluoromethoxy)-3,4,5 -trifluorobenzene; liquid crystals
03/08/2005US6864369 New crystal structure of lopinavir; enzyme inhibitors of human immunodeficiency virus (HIV) protease for treating HIV infections
03/08/2005US6864368 Muscle relaxants, controlling immunology, sexual disorders, rheumatic diseases
03/08/2005US6864289 Insecticides
03/08/2005US6864263 For therpay of inflammatory bowel disease, cerebral ischemia and arthritis, adult respiratory distress syndrome (ARDS) and myocarditis, as adjuvants to short term immunosuppression in transplant therapy
03/08/2005US6863838 Low melting point
03/03/2005WO2005019207A1 Fungicidal pyrimidine derivatives
03/03/2005WO2005019194A1 Derivatives of hydroxamic acid as metalloproteinase inhibitors
03/03/2005WO2005019187A1 2-substituted pyrimidines
03/03/2005WO2005019174A1 Acetylene derivatives as inhibitors of histone deacetylase
03/03/2005WO2005019151A1 Ppar modulators
03/03/2005WO2005019147A2 Pesticidally active phenol derivatives
03/03/2005WO2005003098B1 Heterocyclically substituted pentanol derivatives, method for the production thereof, and use thereof as anti-inflammatory agents
03/03/2005US20050049264 Suppressing growth of abnormal cells; gastric, brain, colon, pancreatic, lung, renal, ovarian and prostatic cancer
03/03/2005US20050049262 Substituted 2,5-dioxopurines, 2H-1,2,3-triazolyl[4,5-d]pyrimidines, or 1,2,5-thadiazolyl[3,4-d]pyrimidines; antiproliferative, antiinflammatory, and antiarthritic agents; psoriasis, asthma, multiple sclerosis, inflammatory bowel disease, lupus, graft versus host disease
03/03/2005US20050049251 Inhibitors of p38
03/03/2005US20050049247 Pyrimidines useful as modulators of voltage-gated ion channels
03/03/2005DE10207376B4 Verfahren zur Herstellung von 2-Anilino-4,6-dimethylpyrimidin A process for the preparation of 2-anilino-4,6-dimethylpyrimidine
03/03/2005CA2536313A1 Fused pyrimidine derivative and use thereof
03/03/2005CA2536089A1 Ppar modulators
03/03/2005CA2535714A1 Phenoxyacetic acid derivatives
03/03/2005CA2535350A1 Acetylene derivatives as inhibitors of histone deacetylase
03/03/2005CA2532568A1 2-substituted pyrimidines
03/02/2005EP1509574A1 Yellow anionic disazo dyes
03/02/2005EP1509537A2 Cellular accumulation of phosphonate analogs of hiv protease inhibitor compounds and the compounds as such
03/02/2005EP1509507A2 Mitotic kinesin inhibitors
03/02/2005EP1509497A1 Calcium receptor modulating arylalkylamines
03/02/2005EP1509218A1 Peptide deformylase inhibitors
03/02/2005EP1509213A2 Acetamides and benzamides that are useful in treating sexual dysfunction
03/02/2005EP1183091A4 Optimization of ligand affinity for rna targets using mass spectrometry
03/02/2005EP1086082B9 Arylsubstituted olefinic amines and their use as cholinergic receptors agonists
03/02/2005EP0871448B1 Aryl and heteroaryl quinazoline compounds which inhibit csf-1r receptor tyrosine kinase
03/02/2005CN1589153A Preventives/remedies for urinary disturbance
03/02/2005CN1589149A Reduced toxicity cisplatin formulations and methods for using the same
03/02/2005CN1589145A αv整联蛋白受体拮抗剂 αv integrin receptor antagonists
03/02/2005CN1191248C 1-(2-naphthyl) and 1(2-azanaphthyl)-4-(1-phenylmethyl)piperazines being dopamine D4 receptor subtype lignds
03/01/2005US6861423 Methods of treating p38 kinase-mediated disorders with pyrido[2,3-d]pyrimidin-7-one compounds
02/2005
02/24/2005WO2005016914A1 Chemical compounds
02/24/2005WO2005016911A1 4-pyrimidone derivatives and their use as peptidyl peptidase inhibitors
02/24/2005WO2005016895A1 Novel compound of 6-methyl-3-phenethyl-3,4-dihydro-1h-quinazoline-2-thinone, its preparation and a depigmentation compositon containing the same as an effective component
02/24/2005WO2005016894A1 2, 4-pyrimidinediamines useful in the treatment of neoplastic diseases, inflammatory and immune system disorders
02/24/2005WO2005016886A1 Sulfonyl substituted n-(biarylmethyl) aminocyclopropanecarboxamides
02/24/2005WO2005016862A1 Substituted arylalkanoic acid derivative and use thereof
02/24/2005WO2005016346A1 Quinazoline analogs as receptor tyrosine kinase inhibitors
02/24/2005WO2005016344A1 Piperazine derivatives for the treatment of hiv infections
02/24/2005WO2005016264A2 Diamine derivatives of quinone and uses thereof
02/24/2005WO2004087056A3 BI-CYCLIC PYRIMIDINE INHIBITORS OF TGFβ
02/24/2005US20050043397 Derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them
02/24/2005US20050043392 Moderators of mnocyte chemoattractant protein; therapy for asthma; multiple sclerosis, antiarthritic agents, atherosclerosis
02/24/2005US20050043358 Aminoalcohol derivatives and their use as beta 3 adrenergic agonists
02/24/2005US20050043338 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
02/24/2005US20050043336 Quinazoline derivatives as antitumor agents
02/24/2005US20050043334 Such as N6-(4,5-dihydrooxazol-2-yl)-N4-[3-methyl-4-(6-methylpyridin-3-yloxy)-phenyl]-quinazoline-4,6-diamine; for treatment of hyperproliferative disorders such as cancer
02/24/2005US20050043333 Quinazolinone derivative
02/24/2005US20050043322 For therapy of hypertension
02/24/2005US20050043307 Novel heterocycle as agonist or antagonist for nervous systems which can contain double or triple bonds with nitrogen, oxygen or sulfur with carbon or azo groups and or salts and as modulators or receptors with carriers
02/24/2005US20050043305 Aryl substituted pyridines, pyrimidines, pyrazines and triazines and the use thereof
02/24/2005US20050043300 Piperazine derivatives
02/24/2005US20050042771 Identifying non-drug targets; use in drug design for improving knowledge of drug-target and drug-non-target interactions, so that drug adverse reactions can be reduced or eliminated in drugs such as troglitazone, rosiglitazone, pioglitazone, methotrexate, atorvastatin, celecoxib, rofecoxib, cerivastatin
02/24/2005US20050042676 Contacting sample with lysine selective agent to cap epsilon -amino group, digesting sample to produce peptide fragments, deactivating cleavage reagent, deblocking/deprotecting, then recovering fragments; solid phase synthesis; kits
02/24/2005CA2535665A1 Substituted arylalkanoic acid derivative and use thereof
02/24/2005CA2535619A1 4-pyrimidone derivatives and their use as peptidyl peptidase inhibitors
02/24/2005CA2534866A1 Piperazine derivatives for the treatment of hiv infections
02/23/2005EP1507775A1 Heterocyclic compounds which inhibit leukocyte adhesion mediated by alpha4 integrins
02/23/2005EP1507768A1 Aryl-alkyne compounds as herbicides
02/23/2005EP1507756A1 Ccr9 inhibitors and methods of use thereof
02/23/2005EP1507533A2 Heteroaryl compounds which inhibit leukocyte adhesion mediated by alpha-4 integrins
02/23/2005EP1507528A2 Methods for using jnk inhibitors for treating or preventing disease-related wasting
02/23/2005EP1507504A1 Cycloalkyl inhibitors of potassium channel function
02/23/2005EP1318146B1 Process for producing pyrimidine derivative and intermediate thereof
02/23/2005EP1226128B1 New pyrimidine-2,4,6-trione derivatives, processes for their production and pharmaceutical agents containing these compounds
02/23/2005EP0876337B1 New lh-rh antagonists with improved effectiveness