Patents
Patents for C07D 235 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings (15,325)
03/2006
03/08/2006CN1244583C Tiemomium azoleamine-8-carboxylic acid ester and 8-amide derivatives, its synthesizing method and application in producing anticancer preparation
03/08/2006CN1244575C Sulfonyl alkylamido hydroxyethylamino sulfonamide retroviral protease inhibitors
03/08/2006CN1244322C Use of inhibitors of sodium-hydrogen exchanging pump for production of medicine for treatment of disorders which are caused by protozoa
03/07/2006US7009060 2-oxo-benzimidazolyl substituted ethanolamine derivatives and their use as β3 agonists
03/07/2006US7008753 Optical recording medium
03/02/2006WO2006023889A2 A method for preparing irbesartan and intermediates thereof
03/02/2006WO2006023844A2 Compositions and methods comprising proteinase activated receptor antagonists
03/02/2006WO2005113542A3 N-cyclic sulfonamido inhibitors of gamma secretase
03/02/2006CA2754633A1 A method for preparing irbesartan and intermediates thereof
03/02/2006CA2576971A1 Compositions and methods comprising proteinase activated receptor antagonists
03/01/2006EP1628661A2 Modulators of vr1 receptor
03/01/2006EP1628533A2 Chemokine receptor binding heterocyclic compounds with enhanced efficacy
03/01/2006CN1243735C 2-lminopyrrolidine derivatives
03/01/2006CN1243545C DNA-cleaving antitumor agents
02/2006
02/28/2006CA2331877C Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
02/23/2006US20060041147 Coupling a 2-cyano-p-bromomethyl diphenyl with a 1,3-diazaspiro (4,4)nonane ring in the presence of a base, a reducing agent, and a phase transfer catalyst; angiotensin II receptor antagonist, treating cardiovascular ailments such as hypertension and heart failure
02/23/2006US20060041134 Silyl ethers
02/23/2006US20060040976 Thiobenzimidazole derivatives
02/22/2006EP1626964A2 New benzimidazole derivatives
02/22/2006EP1626717A2 Benzimidazoles, compositions containing such compounds and methods of use
02/22/2006EP1224187B1 Certain alkylene diamine-substituted heterocycles
02/22/2006CN1738807A Substituted aralkyl derivatives
02/22/2006CN1738799A Methods for preparing phenylalkyne derivatives
02/21/2006US7002021 Diketopyrrolopyrrole pigments
02/21/2006US7001907 Peptide-containing α-ketoamide cysteine and serine protease inhibitors
02/21/2006US7001887 Peptide derivatives
02/16/2006WO2005080317A3 Therapeutic amide derivatives
02/16/2006US20060035906 Converting hydroxyl group in 1-formyl-4-(2-hydroxyethyl) piperazine to a leaving group, reacting with 2-mercaptobenzimidazole , and removing the formyl group; formyl derivative is prepared by formylating 1-(2-hydroxyethyl)piperazine
02/16/2006US20060035884 N-cyclic sulfonamido inhibitors of gamma secretase
02/16/2006US20060035870 Carboxylic acid derivatives as IP antagonists
02/15/2006EP1010423B1 Oral pharmaceutical preparation comprising an antiulcer benzimidazole derivative, and process for its production
02/15/2006CN1733725A Process for preparing 2-iminopyrrolidine derivatives
02/15/2006CN1733722A Bis-heterocyclic compounds with antitumour and chemosensitising activity
02/15/2006CN1241916C Novel acardite compound, its preparation method and medicinal composition containing said compound
02/15/2006CN1241909C Carboxylic acid derivatives as IP antagonists
02/14/2006US6998487 Structure including at least three planar moieties, which are linearly configured such that one planar moiety is located between two neighboring planar moieties and shares an atom with each of the moieties
02/14/2006US6998486 Process for production of cyclic diamine compounds or salts thereof
02/14/2006US6998407 For prophylaxis and therapy of chronic or acute inflammatory or autoimmune diseases, those associated with aberrant lymphocyte or monocyte accumulation such as arthritis, asthma, atherosclerosis, diabetic nephropathy, inflammatory bowel disease
02/14/2006CA2241186C Benzimidazole derivatives
02/09/2006WO2006014134A1 Novel piperidine derivative for the treatment of depression
02/09/2006WO2006013210A2 2-amino benzimidazole derivatives and their use as modulators of small-conductance calcium-activated potassium channels
02/09/2006US20060030618 Vanilloid receptor ligands and their use in treatments
02/09/2006US20060030565 Amide derivatives and nociceptin antagonists
02/09/2006CA2576073A1 Novel piperidine derivative for the treatment of depression
02/09/2006CA2575882A1 2-amino benzimidazole derivatives and their use as modulators of small-conductance calcium-activated potassium channels
02/08/2006EP1622884A1 New heterocyclic amides exhibiting an inhibitory activity at the vanilloid receptor 1 (vr1).
02/08/2006EP1622878A2 Compounds, compositions and methods
02/08/2006EP1318978B1 N-acylsulfonamide apoptosis promoters
02/08/2006EP1183243B1 Short-acting benzodiazepines
02/08/2006CN1732161A 1,3-diamino-2-hydroxypropane pro-drug derivatives
02/08/2006CN1732146A Cycloalkyl inhibitors of potassium channel function
02/08/2006CN1730482A A temodar synthesis method
02/08/2006CN1240702C Process for extracting tetrodosin with high output rate
02/07/2006US6995181 hyterocyclylaminomethyl- or aminocarbonyl-substituted 9,10-ethanoanthracenes or their aza derivatives; treating obesity, diabetes, inflammatory and immune disorders
02/07/2006US6995154 Catalyst for joining, breaking of Dna; antitumor, anticancer agents
02/02/2006WO2006010968A1 New aryloxy acetic acid amide derivatives
02/02/2006US20060025596 Method for deuteration or tritiation of heterocyclic ring
02/02/2006US20060025464 Benzimidazole derivatives as therapeutic agents
02/02/2006US20060025402 Benzimidazolidinone derivatives as muscarinic agents
02/01/2006EP1620434A1 Fused bicyclic-substituted amines as histamine-3 receptor ligands
02/01/2006EP1620391A2 Cyclic derivatives as modulators of chemokine receptor activity
02/01/2006EP1341774B1 Fused heteroaromatic glucokinase activators
02/01/2006EP1080078B1 Heterocyclic compounds and methods to treat cardiac failure and other disorders
02/01/2006CN1729188A Synthesis of heteroaryl acetamides
02/01/2006CN1727339A Tricyclic compounds, their production and use
02/01/2006CN1239485C Benzophenones as inhibitors of IL-1 beta and TNF-alpha
02/01/2006CN1239478C 3,4-dibidro-1H-anphthalene derivatives used as high selectivity inhibitor of cyclooxygenase-2
01/2006
01/26/2006WO2005121102A3 Factor viia inhibitor
01/26/2006US20060020146 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex
01/26/2006US20060018825 Probe for diseases with amyloid accumulation, amyloid-staining agent, remedy and preventive for diseases with amyloid accumulation and diagnostic probe and staining agent for neurofibrillary change
01/26/2006CA2574625A1 Process for the preparation of (2r, 3r)-2-hydroxy-3-amino-3-aryl-propionamide and (2r, 3r)-2-hydroxy-3-amino-3-aryl-propionic acid alkyl ester
01/26/2006CA2574217A1 Diamine derivative, process of preparation thereof, and fungicide comprising diamine derivative as an active ingredient
01/26/2006CA2570968A1 Gonadotropin releasing hormone receptor antagonists
01/25/2006EP1618087A2 Antibacterial agents
01/25/2006EP0978392B1 Optical recording media
01/25/2006CN1726214A Enantiomer (-) of tenatoprazole and the therapeutic use thereof
01/25/2006CN1726194A Novel compounds
01/25/2006CN1726031A 8-trialkylsiloxy-2-methyl-9-phenyl-7-oxo-7,8,9,10-tetrahydroimidazo[1,2-h][1,7]naphthyridines
01/25/2006CN1238340C Alkylthio-and aryl (heteroyl) thio substituted p-phenylenediamines their manufacture and their use in rubber
01/19/2006US20060014963 2-Oxo-benzimidazolyl substituted ethanolamine derivatives and their use as beta3 agonists
01/19/2006US20060014787 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
01/19/2006US20060014781 Thiazole, imidazole and oxazole compounds and treatments of disorders associated with protein aging
01/18/2006EP1615896A1 Novel benzimidazole derivatives and pharmaceutical compositions comprising these compounds
01/18/2006EP1615636A1 Bicyclic compounds as nr2b receptor antagonists
01/18/2006EP1268096B1 Extrusion die
01/18/2006EP1210327B1 New vitamin d derivatives with cyclic substructures in the side chains, method and intermediates for their production and their use in the preparation of medicaments
01/18/2006EP1194410B1 Benzimidazole derivatives and pharmaceutical compositions comprising these compounds
01/18/2006CN1723208A Magnesium salt of imidazole derivative
01/18/2006CN1723022A inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 and type 2
01/18/2006CN1721411A Benzimidazole derivatives as modulators IgE
01/18/2006CN1721401A Inhibitors of LFA-1 binding to ICAMS and uses thereof
01/12/2006WO2006004924A2 Imidazolo-related compounds, compositions and methods for their use
01/12/2006WO2005092066A3 Imidazole compounds
01/12/2006US20060009461 Acetamides and benzamides that are useful in treating sexual dysfunction
01/12/2006CA2572316A1 Imidazolo-related compounds, compositions and methods for their use
01/11/2006EP1614680A2 Process for preparing 2-iminopyrrolidine derivatives
01/11/2006EP1614678A2 Sulfur substituted sulfonylaminocarboxylic acid N-heteroarylamides, their preparation, their use and pharmaceutical preparations comprising them
01/11/2006EP1613618A2 BENZIMIDAZOLE DERIVATIVES AND THEIR USE FOR MODULATING THE GABA- sb A /sb RECEPTOR COMPLEX
01/11/2006EP1613368A2 Carboxamide spirohydantoin cgrp receptor antagonists
01/11/2006EP1613313A1 2-phenyl-benzimidazol and 2-phenyl-imidazo-4,5!-pyridine derivatives as checkpoint kinase cds1 (chk2) inhibitors for the treatment of cancer
1 ... 52 53 54 55 56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 ... 154