Patents
Patents for C07D 235 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings (15,325)
02/2010
02/25/2010US20100048672 Compositions for transfection of oligonucleotides active for gene silencing and their biological and therapeutical applications
02/25/2010US20100048658 Fused heterocyclic compounds
02/25/2010US20100048656 Glyt1 transporter inhibitors and uses thereof in treatment of neurological and neuropsychiatric disorders
02/25/2010US20100048590 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
02/25/2010US20100048565 Benzimidazole derivatives
02/25/2010US20100048564 Fused bicyclic heteroaryl derivative
02/24/2010EP2155893A2 Novel nitroreductase enzymatic substrates
02/24/2010EP2155892A2 Novel peptidase substrates
02/24/2010EP2155676A2 Compounds with antiparasitic activity, applications thereof to the treatment of infectious diseases caused by apicomplexans
02/24/2010EP2154966A1 Benzimidazoles and pharmaceutical compositions thereof
02/24/2010EP1848705B1 Exo- and diastereo- selective syntheses of himbacine analogs
02/24/2010EP1542678B1 1H-1,2,4-TRIAZOLE-3-CARBOXAMIDE DERIVATIVES AS CANNABINOID-CB sb 1 /sb RECEPTOR LIGANDS
02/24/2010CN100591679C Benzimidazole, benzthiazole and benzoxazole derivatives and their use as lta4h modulators
02/18/2010WO2010018874A1 Amide compound
02/18/2010WO2010018441A2 An improved process for the preparation of substantially pure telmisartan
02/18/2010US20100041891 Amide compound
02/18/2010US20100039027 Organic electroluminescence device
02/18/2010US20100039024 New Heterocyclic bridged biphenyls
02/17/2010EP2153832A2 Heterocyclic aspartyl protease inhibitors
02/17/2010EP2152674A1 Benzimidazolone chymase inhibitors
02/16/2010US7662966 For example, 5-tert-Butyl-2-{2-[4-(1-methyl-piperidin-4-yl)-butoxy]-pyridin-4-yl}-1H-benzoimidazole; use in leukocyte recruitment inhibition, in modulating H4 receptor, and in treating conditions such as inflammation, H4 receptor-mediated conditions, and related conditions
02/16/2010US7662841 Imidazothiazole derivatives and process for producing the same
02/16/2010CA2440037C Benzimidazole derivatives for modulating the rage receptor
02/11/2010WO2010017401A1 Bi-1h-benzimidazoles as hepatitis c virus inhibitors
02/11/2010WO2010016549A1 Tricyclic compound
02/11/2010US20100035951 2-amino benzimidazole derivatives and their use as modulators of small-conductance calcium-activated potassium channels
02/10/2010EP2150532A1 Piperazine compounds for the inhibition of haematopoietic prostaglandin d synthase
02/10/2010EP1404659B1 4-aryl quinols and analogs thereof as therapeutic agents
02/09/2010US7659026 membrane electrodes; electrocatalysts; fuel cells
02/04/2010WO2010013835A2 Solid pharmaceutical composition
02/04/2010WO2010012745A2 Benzimidazoles
02/04/2010US20100029643 Heterocyclyc sulfonamides having edg-1 antagonistic activity
02/04/2010CA2732018A1 Solid pharmaceutical composition
02/03/2010CN100586936C Chemical synthesis of albendazole-sulfoxide
02/02/2010US7655683 Imidazolopyrazole derivatives useful as selective androgen receptor modulators
02/02/2010CA2485685C Calcium receptor modulating agents
02/02/2010CA2294809C Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and compositions containing same
01/2010
01/28/2010US20100022610 New Crystalline Forms
01/28/2010US20100022547 Compounds and Methods for Treating Mammalian Gastrointestinal Parasitic Infections
01/27/2010EP2146969A1 Nicotinic acid derivatives as modulators of metabotropic glutamate receptor-5
01/27/2010EP2146968A1 Urea derivatives as glutaminyl cyclase inhibitors
01/27/2010EP2146715A1 Cgrp receptor antagonists with tertiary amide, sulfonamide, carbamate and urea end groups
01/27/2010CN101633645A N3 alkylated benzimidazole derivatives as mek inhibitors
01/27/2010CN101633644A N3 alkylated benzimidazole derivatives as mek inhibitors
01/26/2010US7652053 Diaminocycloalkane MCH receptor antagonists
01/26/2010US7652020 novel hydantoin derivatives to inhibit matrix metalloproteinases (MMPs), a disintegrin and metalloproteases (ADAMs) and/or tumor necrosis factor alpha converting enzyme (TACE) and in so doing prevent the release of tumor necrosis factor alpha (TNF- alpha ); autoimmune diseases; side effect reduction
01/21/2010WO2010009405A2 Targeted nitroxide agents
01/21/2010WO2009046841A8 Piperidine and piperazine derivatives for treating tumours
01/21/2010US20100016393 Novel hydrogen sulfate salt
01/21/2010US20100016372 Benzimidazole Derivatives
01/21/2010US20100015717 Mass Tags for Quantitive Analysis
01/20/2010EP2144882A2 Tris(heterocyclyl) metal complexes as bleach catalysts
01/20/2010EP1831159B1 Tetralin and indane derivatives and uses thereof
01/19/2010US7649008 Crystal of 4-(1-((4-methylbenzothiophen-3-yl)methyl)benzimidazol-2-ylthio)butanoic acid; has chymase inhibitory activity in living body and can be used as a preventive and/or remedy for inflammatory diseases, allergic diseases, respiratory tract diseases, circulatory diseases, or bone metabolic diseases
01/19/2010US7649005 Substituted benzylaminoalkylene heterocycles
01/14/2010WO2010006238A2 Stimulus-responsive apta-chelamers
01/14/2010WO2010004385A1 Process for the preparation of pure 4'-[4-methyl-6-(1-methyl-2-benzimidazolyl)-2-propyl-1-benzimidazolyl]methyl]-2-biphenylcarboxylic acid
01/14/2010US20100010038 Tricyclic compound and pharmaceutical use thereof
01/14/2010US20100010015 Heterocyclic spiro-compounds as aldosterone synthase inhibitors
01/14/2010CA2730083A1 Stimulus-responsive apta-chelamers
01/13/2010EP2142514A1 Thiourea derivatives as glutaminyl cyclase inhibitors
01/13/2010EP2142513A1 Nitrovinyl-diamine derivatives as glutaminyl cyclase inhibitors
01/13/2010CN101624376A Substituted hydrazide compound and application thereof
01/13/2010CN100579518C Use of EP4 receptor ligands in the treatment of IL-6 involved diseases
01/12/2010US7645884 Chemical compositions for authenticatable polymers and articles, and authentication methods thereof
01/12/2010US7645785 Farnesoid-X-receptors (FXR) agonists; diabetes and dyslipidemia; 2,N-dicyclohexyl-2-(2-phenyl-benzoimidazol-1-yl)-acetamide hydrogen chloride
01/12/2010US7645784 Benzimidazole derivatives
01/12/2010US7645779 Linked biaryl compounds
01/12/2010US7645757 Derivatives of heteroaryl-alkylcarbamates, methods for their preparation and use thereof as fatty acid amido hydrolase enzyme inhibitors
01/07/2010WO2010001869A1 Tetra-substituted benzene compound and use thereof
01/07/2010US20100004285 POLYMORPH OF 4-[2-[4-[1-(2-ETHOXYETHYL)-1H-BENZIMIDAZOLE-2-YL]-1-PIPERIDINYL]ETHYL]-alpha alpha-DIMETHYL-BENZENEACETIC ACID
01/07/2010US20100004271 Heterocyclic compounds as aganist for the thyroid receptor
01/07/2010US20100004241 Non-imidazole aryloxyalkylamines
01/07/2010US20100004159 Substituted imidazolone derivatives, preparations and uses
01/06/2010EP2139866A2 Crystalline 1-(cyclohexyloxycarbonyloxy) ethyl 1-((2'-cyanobiphenyl-4-yl)methyl)-2-ethoxy-1h-benzo[d]imidazole-7-carboxylate and a process for its preparation
01/06/2010EP0934281B1 1-phenyl-benzimidazole compounds and their use as baga- a? receptor modulators
01/05/2010US7642358 Antidiabetic agents; modulate insulin drug resistance
01/05/2010US7642278 Nitrogen compounds such as 3-(5-morpholin-4-yl-1H-benz-imidazol-2-yl)-1H-indazole and/or isomers, used as immunology modulators, antidiabetic agents, antiogenesis inhibitors or for prophylaxis of Alzheimer's disease
01/05/2010US7642277 Non-nucleoside reverse transcriptase inhibitors
01/05/2010US7642275 Histone deacetylase inhibitors
01/05/2010US7642265 Benzimidazoles and analogs thereof as antivirals
01/05/2010CA2426457C Aryl or heteroaryl fused imidazole compounds as anti-inflammatory and analgesic agents
01/05/2010CA2318192C .beta.2-adrenergic receptor agonists
12/2009
12/31/2009US20090326029 Non-cyclic substituted benzimidazole thiophene benzyl ether compounds
12/31/2009US20090326027 N-Phenyl-2-0X0-1,4-Diazaspiro [4.5] Dec-3-EN-1-YL Acetamide Derivatives And Their Use As Glycine Transporter Inhibitors
12/31/2009US20090325993 GLYT1 Transporter Inhibitors and Uses Thereof in Treatment of Neurological and Neuropsychiatric Disorders
12/31/2009US20090325962 Tyrosine derivative
12/31/2009US20090325944 Methods and Compositions for Modulating Glycosylation
12/30/2009WO2009130422A3 N-acylthiourea and n-acylurea inhibitors of the hedgehog protein signalling pathway
12/30/2009WO2009120874A3 INHIBITORS OF ANTIGEN RECEPTOR-INDUCED NF-кB ACTIVATION
12/30/2009EP2138484A1 Fused bicyclic heteroaryl derivatives
12/30/2009EP1608352B1 Polyamine compounds for treating chemokine receptor mediated diseases
12/30/2009CN101613321A Mono- and bicyclic azole derivatives that inhibit the interaction of ligands with rage
12/30/2009CA2729227A1 2-heterocyclylaminoalkyl-(p-quinone) derivatives for treatment of oxidative stress diseases
12/29/2009US7638513 inhibitors of matrix metalloproteinases, aggrecanases, tumor necrosis factor-alpha converting enzyme, and tumor necrosis factors
12/24/2009US20090318514 Novel Pharmaceutical Compositions
12/24/2009US20090318445 Pdf inhibitors
12/23/2009EP1879564B1 Compounds to treat amyloidosis and prevent death of beta-cells in type 2 diabetes mellitus
12/23/2009EP1523475B1 Heterocyclically substituted benzoylureas, method for their production and their use as medicaments
12/23/2009CN101611018A Heterocyclyc sulfonamides having Edg-I antagonistic activity
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