Patents for C07D 233 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings (34,408) |
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05/04/2010 | US7709677 e.g.3-{3-[(2-{[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino}ethyl)amino]phenyl}isonicotinic acid ; useful as agonists at atypical beta-adrenoceptors; treatment of hyperglycaemia, animal growth promoters, blood platelet aggregation inhibitors, as positive inotropic agents and antiatherosclerotic agent |
05/04/2010 | US7709657 Efficincy; using 5-(4-methyl-1H-imidazol-1-yl)benzamine as chemical intermediate for pyrimidinylamine benzamide |
05/04/2010 | US7709656 guanidinium chloride C(NR2)3+Cl- or guanidinium bromide C(NR2)3+Br, is reacted with anhydrous HF, and the guanidinium fluoride formed in situ is subsequently reacted with boron trifluoride etherate BF3*Et2O |
05/04/2010 | US7709654 Process for producing oxazole, imidazole, pyrrazole boryl compounds |
05/04/2010 | US7709517 N-methyl-4-{4-[7-(4-cyano-3 -trifluoromethylphenyl)-6,8-dioxo-5,7-diazaspiro[3.4]oct-5-yl]-phenyl}butyramide; for treatment of hormone refractory prostate cancer |
05/04/2010 | US7709515 Therapy for cardiovascular disorders; dyslipidemia; glucose metabolism disorders; Alzheimer's disease |
05/04/2010 | US7709514 benzimidazole-2-one-5-n-pentanoate; inhibiting Macrophage Migration Inhibitory Factor (MIF); rheumatoid arthritis |
05/04/2010 | US7709487 Sulfonyl-derivatives as novel inhibitors of histone deacetylase |
04/29/2010 | WO2010048207A2 Aryl gpr120 receptor agonists and uses thereof |
04/29/2010 | WO2010048170A2 Fluorination of aromatic ring systems |
04/29/2010 | WO2010047774A2 Inhibitors of mycobacterium tuberculosis malate synthase, methods of marking and uses thereof |
04/29/2010 | WO2010028032A3 Process for synthesis of imidazolium and benzimidazolium surfactants and their use in clays and nanocomposites |
04/29/2010 | US20100105922 Process for producing fused imidazole compound, reformatsky reagent in stable form, and process for producing the same |
04/29/2010 | US20100105921 N-heterocyclic carbene (nhc) catalyzed synthesis of hydroxamic acids |
04/29/2010 | US20100105904 Urea type cinnamide derivative |
04/29/2010 | US20100105894 Cyclopropane compounds and pharmaceutical use thereof |
04/29/2010 | US20100105767 Compounds, compositions and methods |
04/29/2010 | US20100105726 Imidazole derivatives that induce apoptosis and their therapeutic uses |
04/29/2010 | US20100105719 Imidazolidine carboxamide derivatives as lipase and phospholipase inhibitors |
04/29/2010 | CA2741967A1 Fluorination of aromatic ring systems |
04/29/2010 | CA2740366A1 Aryl gpr120 receptor agonists and uses thereof |
04/28/2010 | EP2180002A1 Method for producing onium salts with dialkyl phosphonate anions with low halogenide content |
04/28/2010 | EP2179984A1 Acrylamido derivatives useful as inhibitors of the mitochondrial permeability transition |
04/28/2010 | EP2178879A2 6-cycloamino-s-(pyridazin-4-yl)imidazo[1,2-b]-pyridazine and derivatives thereof preparation and therapeutic application thereof |
04/28/2010 | EP1643989B1 Cis-imidazolines as mdm2 inhibitors |
04/28/2010 | CN1852898B Ionic liquid and method of reaction using the same |
04/28/2010 | CN101698661A Noncoplanar imidazolyl aromatic diacid and preparation method thereof |
04/28/2010 | CN101698660A Imidazole-type ionic liquid containing disubstituted phenyl, and preparation method thereof |
04/27/2010 | US7705177 t-Butyl 1-[9-[1-(tert-butoxycarbonyl)cyclopropyl]-5-oxononyl]-1-cyclopropanecarboxylate; Alzheimer's Disease, Syndrome X, peroxisome proliferator activated receptor-related disorders, septicemia, thrombotic disorders, obesity, pancreatitis, hypertension, renal disease, cancer, inflammation, impotence |
04/27/2010 | US7705053 Benzamide derivative |
04/27/2010 | US7705050 Amides, useful in the inhibition of IL-8-induced chemotaxis of neutrophils |
04/27/2010 | US7705030 2-Amino-5-[3-(2fluoropyridin-3-yl)phenyl]-3methyl-5-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]-3,5-dihydro-4H-imidazol-4-one; Alzheimer's disease, cognitive impairment, Down's Syndrome, senile dementia, cerebral amyloid angiopathy, neurofibrillary tangles, beta -amyloid deposits |
04/27/2010 | US7704998 Sulfonyl-derivatives as novel inhibitors or histone deacetylase |
04/27/2010 | US7704992 methyl((1S)-1-(((2S)-2-(5-(9-(2-((2S)-1-((2S)-2-((methoxycarbonyl)amino)-3-methylbutanoyl)-2-pyrrolidinyl)-1H-imidazol-5-yl)-6-methyl-6,7-dihydro-5H-dibenzo[c,e]azepin-3-yl)-1H-imidazol-2-yl)-1-pyrrolidinyl)carbonyl)-2-methylpropyl)carbamate; inhibit the function of the non-structural proteins (NS5A) |
04/27/2010 | CA2493667C Vanilloid receptor ligands and their use in treatments |
04/22/2010 | WO2010045580A1 Sphingosine-1-phosphate receptor antagonists |
04/22/2010 | WO2010043000A1 S1p receptors modulators and their use thereof |
04/22/2010 | WO2010012442A3 Insecticidal benzenedicarboxamide derivative |
04/22/2010 | US20100099727 Amino acid and peptide conjugates of arylalkylic acids for cosmetic use |
04/22/2010 | US20100099682 Acetylene derivatives |
04/22/2010 | CA2740783A1 Sphingosine-1-phosphate receptor antagonists |
04/22/2010 | CA2740484A1 S1p receptors modulators and their use thereof |
04/21/2010 | EP2176234A2 Novel crystals and process of making 5-({[2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy- benzoic acid |
04/21/2010 | EP2176233A1 Gamma secretase modulators |
04/21/2010 | EP2176232A1 1-(azolin-2-yl)amino-1,2-diphenylethane compounds for combating animal pests |
04/21/2010 | EP1620082B1 Medical use of inhibitors of glutaminyl and glutamate cyclases for treating alzheimer's disease and down syndrome |
04/21/2010 | EP1610780B1 Cyclic protein tyrosine kinase inhibitors |
04/21/2010 | CN1978462B Imidazoline modified amino acid, and its synthesizing method and use for polypeptide marking |
04/20/2010 | USRE41254 Synthesis procedure for biphenylimidazolyl-(1)-phenylmethane and related compounds |
04/20/2010 | US7700785 Process for preparation of dialkyl carbonate |
04/20/2010 | US7700775 Drug delivery |
04/20/2010 | US7700585 Derivatives of N-[phenyl(pyrrolidine-2-YL)methyl]benzamide and N-[(azepan-2-YL) phenylmethyl]benzamide, preparation method thereof and application of same in therapeutics |
04/20/2010 | CA2630009C Novel carboxylic acid derivatives and process for producing the same |
04/20/2010 | CA2418744C Novel aminocyclohexane derivatives |
04/20/2010 | CA2393159C Methods of treating tumors |
04/15/2010 | WO2010041767A1 Process for producing alpha-hydroxyketone compound |
04/15/2010 | WO2010041614A1 2-benzyl-4-(2,4-dichlorophenyl)-5-methylimidazole compound |
04/15/2010 | WO2009152906A3 Use of ionic liquids with tetracyanoborate anions as a solvent for extraction of alcohols from aqueous solutions |
04/15/2010 | WO1998051902A9 Low toxicity corrosion inhibitor |
04/15/2010 | US20100093809 Therapeutic substituted thiazolidinones, oxazolidinones, and related compounds |
04/14/2010 | EP2174969A1 Resin composition |
04/14/2010 | EP2173720A2 2-imidazolines having a good affinity to the trace amine associated receptors (taars) |
04/14/2010 | EP2173719A1 4-imidazolines and their use as antidepressants |
04/14/2010 | EP2173717A2 Novel glucokinase activators and methods of using same |
04/14/2010 | EP2173707A1 Pleuromutilin derivatives and their use as antimicrobials |
04/14/2010 | EP1694410B1 Cyclopropane derivatives and pharmaceutical use thereof |
04/14/2010 | EP1551799B1 Cyclohexyl sulphones as gamma-secretase inhibitors |
04/14/2010 | EP1400515B1 Cyclic diamine compound having five-membered cyclic group |
04/14/2010 | EP1335901B1 Pharmaceutically active sulfanilide derivatives |
04/14/2010 | CN101694867A Organic light emitting devices having carrier blocking layers comprising metal complexes |
04/14/2010 | CN101693694A Preparation method of glyoxaline formic ether and derivative thereof |
04/14/2010 | CN101693693A Method for preparing 2-propyl imidazole |
04/14/2010 | CN101693692A Hybrid ionic liquid hydrate, preparation process and application thereof |
04/14/2010 | CN101692832A Composition for controlling harmful bio-organisms and method for controlling harmful bio-organisms using the same |
04/14/2010 | CN101104603B Method for producing phentolamine |
04/13/2010 | US7696379 Acetylene derivatives |
04/13/2010 | US7696233 Method for controlling particular insect pests by applying anthranilamide compounds |
04/13/2010 | CA2336807C Sulfur substituted sulfonylaminocarboxylic acid n-arylamides, their preparation, their use and pharmaceutical preparations comprising them |
04/08/2010 | WO2010039719A1 Crystalline form of an alkoxyimidazol-1-ylmethyl biphenyl carboxylic acid |
04/08/2010 | WO2010039238A1 Compounds for inflammation and immune-related uses |
04/08/2010 | WO2009146024A8 Etomidate analogues with improved pharmacokinetic and pharmacodynamic properties |
04/08/2010 | US20100087657 Enantioselective synthesis of (+) and (-)-2-[1-(2,6-dichlorophenoxy)-ethyl]-1,3-diazacyclopent-2-3ene |
04/08/2010 | US20100087656 Compositions Containing Fatty Acids and/or Derivatives Thereof and a Low Temperature Stabilizer |
04/08/2010 | US20100087655 Method for production of n-(2-amino-1,2-dicyanovinyl)imidates, method for production of n-(2-amino-1,2-dicyanovinyl)formamidine, and method for production of aminoimidazole derivatives |
04/08/2010 | US20100087478 HIF-1 Inhibitors |
04/08/2010 | US20100087442 Diketohydrazine derivative compounds and drugs containing the compounds as the active ingredient |
04/08/2010 | US20100087438 New Potassium Channel Blockers |
04/08/2010 | US20100087428 Novel Potassium Channel Blockers |
04/08/2010 | CA2739303A1 Compounds for inflammation and immune-related uses |
04/08/2010 | CA2736102A1 Crystalline form of an alkoxyimidazol-1-ylmethyl biphenyl carboxylic acid |
04/07/2010 | EP2172462A1 Method for production of 3-hydroxypropan-1-one compound, method for production of 2-propen-1-one compound, and method for production of isoxazoline compound |
04/07/2010 | EP2172450A1 Novel malonic acid sulfonamide derivative and pharmaceutical use thereof |
04/07/2010 | EP2170823A1 N-(2-(hetaryl)aryl)arylsulfonamides and n-(2-(hetaryl)hetaryl)arylsulfonamides |
04/07/2010 | EP2170814A2 Antibacterial agents |
04/07/2010 | EP2170260A1 Azo derivatives containing a pyrazolinone unit for dyeing keratin fibres |
04/07/2010 | EP1590340B1 Inhibitors of histone deacetylase |
04/07/2010 | CN1934090B Substituted N-cyclohexyl imidazolinones having an MCH-modulatory effect |
04/07/2010 | CN101691358A Application and synthesis method of caffeidine nitrate |
04/07/2010 | CN101691357A Novel disubstituted imidazolone anti-tumor compounds and preparation method thereof |
04/06/2010 | US7692007 Process for the preparation of onium salts having a low chloride content |