Patents
Patents for C07D 233 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings (34,408)
02/1994
02/08/1994US5284963 Reacting 9-amino tetracycline derivative with haloacyl halide in mixture of polar aprotic solvent, inert solvent, base; reacting product under inert atmosphere with nucleophilic amine
02/08/1994US5284851 1-alkoxy-1,3-diazacycloalkane derivatives and their use as pesticides
02/08/1994US5284850 Terpene amino alcohols and medicinal uses thereof
02/08/1994US5284650 Process for making high solids fabric softeners using low amounts of solvents and eliminating side reactions
02/03/1994WO1994002468A1 Method of forming n-protected amino acid thiohydantoins
02/03/1994WO1994002467A1 Imidazole ethers having a ii antagonist activity
02/03/1994WO1994002452A1 Benzene derivative
02/03/1994WO1994002148A1 Novel bioactive compositions, preparation and use thereof
02/03/1994CA2140630A1 Novel bioactive compositions, preparation and use thereof
02/03/1994CA2115915A1 Benzene derivatives
02/02/1994EP0581250A2 Process for biotechnical preparation of L-thienylalanines in enantiomere pure form from 2-hydroxy-3-thienyl-acrylic acids and their use
02/02/1994EP0581003A1 Imidazolyl substituted cyclohexane derivatives
02/02/1994EP0580956A1 Process for the catalytic preparation of condensation products of formaldehyde
02/02/1994EP0378657B1 Oxazolidinone penetration enhancing compounds
02/02/1994CN1081446A 氨基酸衍生物 Amino acid derivatives
02/02/1994CN1081438A Imidazole derivatives, their method of preparation and their application in therapeutic
02/02/1994CN1023645C Novel resolution process for racemic spiro hydantoins
02/02/1994CN1023644C Antiarrhythmic drugs and the prepn. method
02/01/1994US5283341 Catalytic alkylation
02/01/1994US5283271 3,5-diphenyl or substituted 3,5-diphenyl-1-hydroxy-1,2-dihydroimidazole-2-thiones
02/01/1994US5283254 2-(imidazol-1-yl)-2-benzylethyldiene-aminoxyalkanoic acid derivatives
02/01/1994CA2101654A1 Process for the biotechnological preparation of l-thienylalanines in enantiomerically pure form from 2-hydroxy-3-thienylacrylic acids, and their use
02/01/1994CA2101311A1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles
02/01/1994CA1326669C Herbicidal oxoindanes and tetrahydronaphthalenes
01/1994
01/26/1994EP0580459A1 Substituted Phenylimidazolidins, process for their preparation, their use as medicaments and their pharmaceutical compositions containing them
01/26/1994EP0580402A2 Aminediol protease inhibitors
01/26/1994EP0580008A2 Phenylimidazolidine Derivatives, their preparation and use
01/26/1994EP0579618A1 Pyridine- and imidazole-derived agents for cardiovascular diseases
01/26/1994CN1081182A New substituted phenylimidazolidines, their preparation process, their use as medicaments and the pharmaceutical compositions containing them
01/25/1994US5281626 Benzenesulfonamide derivatives
01/25/1994US5281594 Substituted 1-(alkoxyphenyl)piperazines with ons and antihypertensive activity
01/25/1994CA1326490C Process for preparation of cimetidine
01/21/1994CA2100894A1 Aminediol protease inhibitors
01/20/1994WO1994001436A1 Dioxcyclobutene derivatives as angiotensin ii antagonists
01/20/1994WO1994001410A1 Fungicidal 2-imidazoline-5-one and 2-imidazoline-5-thione derivatives
01/20/1994WO1994001409A1 Novel intermediate for synthesis and production of amino acid derivative
01/20/1994CA2139930A1 Dioxycyclobutene derivatives as angiotensin ii antagonists
01/20/1994CA2139362A1 Novel intermediate for synthesis and production of amino acid derivative
01/20/1994CA2139346A1 Fungicide 2-imidazolin-5-ones and 2-imidazoline-5-thiones derivatives
01/19/1994EP0579277A1 Imidazole derivatives, their preparation and their use as synthetic intermediates
01/19/1994EP0579212A1 Process of preparation of 2-substituted 5-chlorimidazol-4-carbaldehydes
01/19/1994EP0579169A1 Alkylenediamine derivatives
01/19/1994EP0579071A2 Heteroaromatic compounds and plant-protecting agents containing them
01/19/1994EP0578745A1 Phosphorus containing compounds as inhibitors of retroviruses
01/19/1994CN1080930A Histamine derivatives and methods for their use as immunomodulators
01/18/1994US5280036 N-phenoxyphenyloxymethyl substituted azoles and method for controlling pests therewith
01/18/1994US5280035 Cycloalkylene azoles and their use as aromatase inhibitors
01/18/1994US5280034 Bis-heterocyclic prostaglandin analogs
01/18/1994US5280033 Substituted 1-(alkoxy-iminoalkyl) imidazole derivatives and their use in treating disease related to an enhancement of thromboxane-A2 syntheis
01/18/1994US5280032 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
01/17/1994CA2100308A1 Heteroaromatic compounds and crop protection agents containing them
01/15/1994CA2100376A1 Alkylenediamine derivatives
01/12/1994EP0578516A1 Optionally substituted phenylimidazolidins, process for their preparation, their use as medicaments and the pharmaceutical compositions containing them
01/12/1994EP0578080A2 3,9-disubstituted-spiro (5.5)undecanes active on the cardiovascular system, process for their preparation and pharmaceutical composition containing same
01/12/1994EP0578002A1 Imidazolyl substituted phenylpropionic and cinnamic acid derivatives
01/12/1994CN1080635A Process for preparing methylolhydantoins
01/12/1994CN1023476C Process of preparing trifluoromethylvinyl derivatives starting with appropriate halogenovinyl derivatives
01/11/1994US5278182 Azole-1-carboxylic acid ester derivatives and fungicidal compositions
01/11/1994US5278177 Enzyme inhibitory
01/11/1994US5278166 4-amino-3-heteroaryl butyric acid compounds, compositions, and their use for treating disorders involving a dysfunction of GABAB receptors
01/11/1994US5278148 Hypotensive agents
01/09/1994CA2097248A1 Substituted phenylimidazolidines, a process for their preparation, their application as medicaments and pharmaceutical compositions containing them
01/09/1994CA2097247A1 Phenylimidazolidines, substituted or not, a process for their preparation, their application as medicaments and pharmaceutical compositions containing them
01/06/1994WO1994000420A1 Novel tight-binding inhibitors of leukotriene a4 hydrolase
01/06/1994WO1994000120A1 Chemical compounds
01/06/1994WO1993022376A3 Amino compounds as processing stabilisers for thermoplastic materials
01/05/1994EP0577025A2 Angiotensin-II-receptorantagonist for the treatment and prophylaxis of coronary heart diseases
01/05/1994EP0577023A2 Angiotensin-II receptor-antagonists for the treatment of arrhythmices
01/05/1994EP0576766A1 Propanolamine derivatives, their preparation and use
01/05/1994DE4222063A1 New 4-hetero-aryl-benzyl alcohol or halide cpds. - used as intermediates for drugs, esp. angiotensin II antagonists, prepd. e.g. from boronic acid cpd. and hetero-aryl halide
01/04/1994US5276247 Contains cationic or anionic surfactants; treating with laminar mineral
01/04/1994US5276049 Cyclic urea derivatives, pharmaceutical compositions containing these compounds and methods of using the same
01/04/1994US5276048 4-(1H-pyrrol-1-yl)imidazoles with angiotensin II antagonist activity
01/04/1994US5276034 Substituted imidazolyl-alkyl-piperazine and -diazepine derivatives
01/04/1994CA1325808C Fungicidal azolyl-derivatives
01/02/1994CA2099447A1 Angiotensin ii receptor antagonists for the treatment and prophylaxis of coronary heart disease
01/02/1994CA2099425A1 Angiotensin ii receptor antagonists for the treatment of disturbances in cardiac rhythm
12/1993
12/29/1993EP0575844A2 Hydroxamic acid derivatives and pharmaceutical compositions thereof
12/29/1993EP0575490A1 GnRH ANALOGS
12/29/1993CN1079908A Histamine derivatives and methods for their use as immunomodulators
12/29/1993CN1023318C Process for preparing 1-hydroxyalkyl-5-nitro imidazoles
12/29/1993CN1023317C Method for controlling weeds
12/28/1993US5274104 N-substituted heterocyclic derivatives useful in the treatment of cardiovascular disorders
12/28/1993US5274095 A 4-(4-(julolid-9-yl)imidazol-2-yl-2,6-ditert-butyl-phenol derivative
12/28/1993US5273993 Compounds having one or more aminosulfonyloxy radicals useful as pharmaceuticals
12/28/1993US5273991 Imidazole-containing compositions and methods of use thereof analogs of distamycin
12/28/1993US5273984 Salts formed between basic histamine H2 -receptor antagonists and bismuth complexes
12/28/1993CA1325637C Fungicide azolyl-derivatives
12/27/1993CA2099078A1 Imidazolyl-substituted cyclohexane derivatives
12/27/1993CA2099068A1 Imidazolyl-substituted phenylpropionic and cinnamic acid derivatives
12/26/1993CA2098166A1 Hydroxamic acid derivatives
12/23/1993WO1993025549A1 Process for preparing 1,3-dioxolane derivatives
12/23/1993WO1993025536A1 1,2,3-triazole and imidazole compounds and their antitumor use
12/23/1993DE4220069A1 Prodn. of 5-hydroxy-2-imino-4-imidazolinone - by reaction of methyl glyoxylate hemiacetal and guanidine carbonate in presence of alcohol
12/22/1993EP0574758A1 Hydroxamic acid derivatives as collagenase inhibitors
12/22/1993CN1079649A Imidazolyl-alkenoic acids
12/22/1993CN1079648A Imidazolyl-alkenoic acids
12/22/1993CN1023221C Process for preparing 1-alkyl-5-nitroimidazoles
12/22/1993CN1023220C Process for preparing 1-hydroxyalkyl-2-methyl-5-nitro imidazoles
12/22/1993CN1023219C Substituted imidazole derivatives and their preparation and use